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Bulletin 2011/10 - European Patent Office

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(A01N) I.1(1)<br />

(25) En (26) En<br />

(21) 09747197.3 (22) 06.05.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/042951 06.05.2009<br />

(87) WO 2009/140111 2009/47 19.11.2009<br />

(30) 15.05.2008 US 127807<br />

(54) • ANGIOTENSIN-II-REZEPTORANTAGONIS-<br />

TEN<br />

• ANGIOTENSIN II RECEPTOR ANTAGO-<br />

NISTS<br />

• ANTAGONISTES DU RÉCEPTEUR DE<br />

L'ANGIOTENSINE LL<br />

(71) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065, US<br />

Nicox S.A., Taissounières HB4 1681 route<br />

des Dolines BP 313, 06560 Sophia Antipolis<br />

- Valbonne, FR<br />

(72) ALI, Amjad, Rahway NJ 07065-0907, US<br />

LO, Michael, Man-chu, Rahway NJ 07065-<br />

0907, US<br />

SEBHAT, Iyassu, K., Rahway NJ 07065-<br />

0907, US<br />

FRANKLIN, Chris, Rahway NJ 07065-0907,<br />

US<br />

ALMIRANTE, Nicoletta, F-06560 Valbonne,<br />

FR<br />

STEFANINI, Silvia, F-06560 Valbonne, FR<br />

BIONDI, Stefano, F-06560 Valbonne, FR<br />

ONGINI, Ennio, F-06560 Valbonne, FR<br />

(74) Hussain, Deeba, et al, Merck & Co., Inc.<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

A01N 43/40 → (51) A61K 31/44<br />

(51) A01N 43/42 (11) 2 291 077 A1*<br />

(25) En (26) En<br />

(21) 09767252.1 (22) 21.05.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/044889 21.05.2009<br />

(87) WO 2009/154940 2009/52 23.12.2009<br />

(30) 18.06.2008 US 73695<br />

(54) • HERSTELLUNGSVERFAHREN FÜR RHO-<br />

KINASEHEMMERVERBINDUNGEN<br />

• PROCESS FOR THE PREPARATION OF<br />

RHO-KINASE INHIBITOR COMPOUNDS<br />

• PROCESSUS DE PRÉPARATION DE COM-<br />

POSÉS INHIBITEURS DE RHO-KINASE<br />

(71) Inspire Pharmaceuticals, Inc., 4222 Emperor<br />

Boulevard, Suite 200, Durham, NC 27703,<br />

US<br />

(72) SHE, Jin, Durham, NC 27703, US<br />

DECAMP, Jonathan, Bryan, Raleigh, NC<br />

27615, US<br />

WATSON, Paul, S., Carrboro, NC 275<strong>10</strong>, US<br />

SLADE, David, J., Durham, NC 27713, US<br />

(74) Schüssler, Andrea, Kanzlei Huber &<br />

Schüssler Truderinger Strasse 246, 81825<br />

München, DE<br />

(51) A01N 43/50 (11) 2 291 078 A1*<br />

A01N 43/76 A61K 31/42<br />

(25) En (26) En<br />

(21) 09747248.4 (22) 08.05.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/043299 08.05.2009<br />

(87) WO 2009/140163 2009/47 19.11.2009<br />

(30) 15.05.2008 US 127770 P<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(54) • OXAZOLBENZIMIDAZOLDERIVATE<br />

• OXAZOLOBENZIMIDAZOLE DERIVATIVES<br />

• DÉRIVÉS D'OXAZOLOBENZIMIDAZOLE<br />

(71) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065, US<br />

(72) BRNARDIC, Edward, J., Rahway NJ 07065-<br />

0907, US<br />

CONVERSO, Antonella, Rahway NJ 07065-<br />

0907, US<br />

FRALEY, Mark, E., Rahway NJ 07065-0907,<br />

US<br />

GARBACCIO, Robert, M., Rahway NJ 07065-<br />

0907, US<br />

HUANG, Shaei, Y., Rahway NJ 07065-0907,<br />

US<br />

(74) Buchan, Gavin MacNicol, et al, Merck Sharp<br />

& Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

A01N 43/50 → (51) A01N 43/40<br />

A01N 43/76 → (51) A01N 43/50<br />

(51) A01N 43/78 (11) 2 291 079 A2*<br />

A61K 31/425<br />

(25) En (26) En<br />

(21) 09747191.6 (22) 06.05.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/042924 06.05.2009<br />

(87) WO 2009/140<strong>10</strong>5 2009/47 19.11.2009<br />

(88) 07.01.20<strong>10</strong><br />

(30) 14.05.2008 US 127630<br />

(54) • FORMULIERUNGEN FÜR CATHEPSIN-K-<br />

HEMMER<br />

• FORMULATIONS FOR CATHEPSIN K INHI-<br />

BITORS<br />

• PRÉPARATIONS POUR INHIBITEURS DE<br />

LA CATHEPSINE K<br />

(71) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065, US<br />

(72) FAN, Haihong, Rahway New Jersey 07065-<br />

0907, US<br />

MAHJOUR, Majid, Rahway New Jersey<br />

07065-0907, US<br />

MOSER, Justin, Rahway New Jersey 07065-<br />

0907, US<br />

REGE, Bhagwant, Rahway New Jersey<br />

07065-0907, US<br />

(74) Hussain, Deeba, et al, Merck & Co., Inc.<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

(51) A01N 43/82 (11) 2 291 080 A1*<br />

A61K 31/41<br />

(25) En (26) En<br />

(21) 09762826.7 (22) 14.05.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/003014 14.05.2009<br />

(87) WO 2009/151529 2009/51 17.12.2009<br />

(30) 14.05.2008 US 127603<br />

14.05.2009 US 465767<br />

(54) • NEUE MODULATOREN VON SPHINGO-<br />

SINPHOPHATREZEPTOREN<br />

• NOVEL MODULATORS OF SPHINGOSINE<br />

PHOSPHATE RECEPTORS<br />

• NOUVEAUX MODULATEURS DES RÉCEP-<br />

TEURS DE LA SPHINGOSINE PHOSPHATE<br />

(71) The Scripps Research Institute, <strong>10</strong>550 North<br />

Torrey Pines Road, La Jolla, CA 92037, US<br />

(72) ROBERTS, Edward, La Jolla California<br />

92037, US<br />

17<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>10</strong>/<strong>2011</strong>) 09.03.<strong>2011</strong><br />

ROSEN, Hugh, La Jolla California 92037, US<br />

BROWN, Steven, La Jolla California 92037,<br />

US<br />

GUERRERO, Miguel A., La Jolla California<br />

92037, US<br />

PENG, Xuemei, La Jolla California 92037, US<br />

PODDUTOORI, Ramulu, La Jolla California<br />

92037, US<br />

(74) Lumsden, Stuart Edward Henry, Marks &<br />

Clerk LLP 90 Long Acre, GB-London WC2E<br />

9RA, GB<br />

(51) A01N 45/00 (11) 2 291 081 A1*<br />

A61K 31/56<br />

(25) En (26) En<br />

(21) 09762915.8 (22) <strong>10</strong>.06.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/003521 <strong>10</strong>.06.2009<br />

(87) WO 2009/151619 2009/51 17.12.2009<br />

(30) 15.12.2008 US 201854<br />

12.06.2008 US 129222<br />

(54) • POVIDON-IOD, EIN NEUES ALTERNATIVES<br />

KONSERVIERUNGSMITTEL FÜR OPH-<br />

THALMISCHE ZUSAMMENSETZUNGEN<br />

• POVIDONE IODINE, A NOVEL ALTERNA-<br />

TIVE PRESERVATIVE FOR OPHTHALMIC<br />

COMPOSITIONS<br />

• LA POVIDONE IODÉE, NOUVEAU<br />

CONSERVATEUR INNOVANT POUR COM-<br />

POSITIONS OPHTALMIQUES<br />

(71) Foresight Biotherapeutics, Inc., 50 W. 57th<br />

Street, 15th Floor, New York, NY <strong>10</strong>019, US<br />

(72) CAPRIOTTI, Joseph, A., New York NY <strong>10</strong>025,<br />

US<br />

LIANG, Bo, East Brunswick NJ 08816, US<br />

SAMSON, C., Michael, New York NY <strong>10</strong>016,<br />

US<br />

STEIN, Jason, New York NY <strong>10</strong>162, US<br />

WEISER, Michael, New York NY, US<br />

(74) Vossius & Partner, Siebertstrasse 4, 81675<br />

München, DE<br />

(51) A01N 53/00 (11) 2 291 082 A2*<br />

A01P 7/04<br />

(25) Fr (26) Fr<br />

(21) 09784228.0 (22) 24.06.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) FR 2009/000770 24.06.2009<br />

(87) WO 20<strong>10</strong>/007239 20<strong>10</strong>/03 21.01.20<strong>10</strong><br />

(30) 25.06.2008 FR 0803577<br />

(54) • VERFAHREN ZUR BEKÄMPFUNG VON<br />

BODENINSEKTEN<br />

• METHOD FOR CONTROLLING SOIL<br />

INSECTS<br />

• PROCEDE DE LUTTE CONTRE LES<br />

INSECTES DU SOL<br />

(71) Sbm Developpement S.A.S., 42, chemin<br />

Moulin Carron Le Norly, 69130 Eculy, FR<br />

(72) PEYRON, Xavier, 13011 Marseille, FR<br />

(74) Santarelli, 146, rue Paradis, 13294 Marseille<br />

Cedex 6, FR<br />

(51) A01N 53/00 (11) 2 291 083 A2*<br />

A01P 7/04<br />

(25) Fr (26) Fr<br />

(21) 09784229.8 (22) 24.06.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) FR 2009/000771 24.06.2009

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