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Bulletin 2011/10 - European Patent Office

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(C07D) I.1(2)<br />

(54) • Pyrazolderivat, Zwischenprodukt davon<br />

und Herbizid, das dieses als aktiven<br />

Inhaltsstoff umfasst<br />

• Pyrazole derivative, its intermediate, and<br />

herbicide containing the same as active<br />

ingredient<br />

• Dérivé du pyrazole, son intermédiaire et<br />

herbicide contenant celui-ci en tant que<br />

principe actif<br />

(71) SAGAMI CHEMICAL RESEARCH CENTER,<br />

2743-1, Hayakawa, Ayase-shi, Kanagawa<br />

252-1193, JP<br />

KAKEN PHARMACEUTICAL CO., LTD., 28-8,<br />

Honkomagome 2-chome, Bunkyo-ku, Tokyo<br />

113-8650, JP<br />

(72) Hirai, Kenji, Sagamihara-shi Kanagawa 228-<br />

0821, JP<br />

Uchida, Atsushi, Machida-shi Tokyo 194-<br />

0033, JP<br />

Watanabe, Atsuko, Yokohama-shi Kanagawa<br />

241-0021, JP<br />

Abe, Taeko, Sagamihara-shi Kanagawa 228-<br />

0802, JP<br />

Ueda, Takuya, Abiko-shi Chiba 270-1158, JP<br />

Sakurai, Hiroshi, Fujieda-shi Shizuoka 426-<br />

0041, JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastraße 4, 81925 München, DE<br />

(62) 02712451.0 / 1 362 852<br />

C07D 233/00 → (51) A61K 9/14<br />

C07D 233/58 → (51) C07C 323/00<br />

(51) C07D 233/61 (11) 2 292 607 A2<br />

(25) En (26) En<br />

(21) <strong>10</strong>171942.5 (22) 07.06.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(30) 09.06.2005 US 688976 P<br />

(54) • Verfahren zur Herstellung von organischen<br />

Verbindungen<br />

• Process for the synthesis of organic<br />

compounds<br />

• Procédé de synthèse de composés organiques<br />

(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(84) BE BG CH CY CZ DE DK EE ES FI FR GB GR<br />

HU IE IS IT LI LT LU LV MC NL PL PT RO SE<br />

SI SK TR<br />

(71) Novartis Pharma GmbH, Brunner Strasse 59,<br />

1230 Wien, AT<br />

(84) AT<br />

(72) Abel, Stephan, 79576, Weil am Rhein, DE<br />

Acemoglu, Murat, 4052, Basel, CH<br />

Erb, Bernhard, 5073, Gipf-Oberfrick, CH<br />

Krell, Christoph, 4057, Basel, CH<br />

Sclafani, Joseph, Ledgewood, NJ 07852, US<br />

Meisenbach, Mark, 68480, Durmenach, FR<br />

Prashad, Mahavir, Montville, NJ 07045, US<br />

Shieh, Wen-Chung, Berkeley, NJ 07922, US<br />

Xue, Song, Parsippany, NJ 07054, US<br />

(74) Roth, Peter Richard, Novartis Pharma AG<br />

<strong>Patent</strong> Department, 4002 Basel, CH<br />

(62) 06772447.6 / 1 896 426<br />

C07D 239/26 → (51) C07C 237/20<br />

C07D 239/30 → (51) C07D 239/52<br />

C07D 239/34 → (51) C07D 239/52<br />

C07D 239/36 → (51) C07D 239/52<br />

(51) C07D 239/52 (11) 2 292 608 A1<br />

A01N 43/50 C07D 239/545<br />

C07D 239/36 C07D 239/34<br />

C07D 239/30<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(25) De (26) De<br />

(21) <strong>10</strong>182907.5 (22) 02.03.1998<br />

(84) BE CH DE DK ES FR GB IT LI NL<br />

(27) 02.03.1998 EP 05002366<br />

(30) 14.03.1997 DE 197<strong>10</strong>609<br />

(54) • Zwischenprodukte zur Herstellung von<br />

substituierten Aminosalicylsäureamiden<br />

mit funizider Wirkung<br />

• Intermediates for the preparation of substituted<br />

Aminosalicylic acid amides with<br />

fungicidal activity<br />

• Produits intermèdiaires destinés à la préparation<br />

d'amines d'acide aminosalicylique<br />

substituées à action fongicide<br />

(71) Bayer CropScience AG, Gebäude 6<strong>10</strong>0<br />

Alfred-Nobel-Straße 50, 40789 Monheim, DE<br />

(72) Seitz, Thomas Dr., 40764 Langenfeld, DE<br />

Stelzer, Uwe Dr., 51399 Burscheid, DE<br />

Wolfrum, Peter Dr., 40789 Monheim, DE<br />

Stenzel, Klaus Dr., 40595 Düsseldorf, DE<br />

(62) 05002366.2 / 1 533 303<br />

98913618.9 / 0 970 057<br />

C07D 239/545→ (51) C07D 239/52<br />

C07D 239/62 → (51) C07C 223/06<br />

C07D 239/66 → (51) C07C 223/06<br />

C07D 239/94 → (51) A61K 31/517<br />

C07D 241/20 → (51) A61K 31/4965<br />

(51) C07D 249/04 (11) 2 292 609 A1<br />

A61K 31/4192 A61P 25/00<br />

(25) En (26) En<br />

(21) <strong>10</strong>170757.8 (22) 26.07.20<strong>10</strong><br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

BA ME RS<br />

(30) 04.08.2009 IT MI20091412<br />

(54) • Kristalline Formen von Rufinamide<br />

• Crystalline forms of rufinamide<br />

• Formes crystallines de rufinamide<br />

(71) Dipharma Francis S.r.l., Via Bissone, 5,<br />

20021 Baranzate (MI), IT<br />

(72) Razzetti, Gabriele, 20099 Sesto San Giovanni<br />

(MI), IT<br />

Vladiskovic, Chiara, 20146 Milano, IT<br />

Allegrini, Pietro, 20097 S. Donato Milanese<br />

(MI), IT<br />

(74) Minoja, Fabrizio, Bianchetti Bracco Minoja S.<br />

r.l. Via Plinio 63, 20129 Milano, IT<br />

C07D 263/14 → (51) C07F 9/09<br />

C07D 263/24 → (51) C07C 237/20<br />

C07D 277/06 → (51) C07C 237/20<br />

C07D 277/22 → (51) C07C 323/00<br />

C07D 295/16 → (51) C07C 323/00<br />

C07D 295/185→ (51) C07C 237/20<br />

C07D 307/<strong>10</strong> → (51) C07C 323/40<br />

C07D 307/52 → (51) C07C 311/21<br />

C07D 307/66 → (51) C07C 223/06<br />

(51) C07D 313/00 (11) 2 292 6<strong>10</strong> A1<br />

C07D 405/14 C07D 407/06<br />

C07D 493/<strong>10</strong> C07D 493/04<br />

A61K 31/335 A61K 31/336<br />

A61K 31/4427 A61K 31/4523<br />

223<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>10</strong>/<strong>2011</strong>) 09.03.<strong>2011</strong><br />

A61K 31/455 A61K 31/4025<br />

A61P 35/00<br />

(25) En (26) En<br />

(21) <strong>10</strong>182752.5 (22) 01.02.2002<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

(30) 01.02.2001 JP 200<strong>10</strong>25458<br />

(54) • Makroliden mit VEGF Transkription hemmender<br />

Wirkung<br />

• Macrolides with VEGF transcription suppression<br />

activity<br />

• Macrolides comme inhibiteurs de la transcription<br />

de VEGF<br />

(71) MERCIAN CORPORATION, 5-8, Kyobashi 1chome,<br />

Chuo-ku, Tokyo <strong>10</strong>4-8305, JP<br />

Eisai R&D Management Co., Ltd., 6-<strong>10</strong>,<br />

Koishikawa 4-chome, Bunkyo-ku, Tokyo<br />

112-8088, JP<br />

(72) Mizui, Yoshiharu, Tsukuba-shi Ibaraki 305-<br />

0051, JP<br />

Sakai, Takashi, Tsukuba-shi Ibaraki 305-<br />

0035, JP<br />

Yamamoto, Satoshi, Moriya-shi Ibaraki 302-<br />

0124, JP<br />

Komeda, Keisuke, Tsukuba-shi Ibaraki 305-<br />

0031, JP<br />

Fujita, Masanori, Ushiku-shi Ibaraki 300-<br />

1206, JP<br />

Okuda, Akifumi, Tsukuba-shi Ibaraki 305-<br />

0035, JP<br />

Kishi, Kumiko, Tsukuba-shi Ibaraki 305-<br />

0035, JP<br />

Niijima, Jun, Tsukuba-shi Ibaraki 305-0035,<br />

JP<br />

Nagai, Mitsuo, Tsukuba-shi Ibaraki 305-<br />

0035, JP<br />

Okamoto, Kiyoshi, Tsukuba-shi Ibaraki 305-<br />

0856, JP<br />

Iwata, Masao, Tsukuba-shi Ibaraki 305-0045,<br />

JP<br />

Kotake, Yoshihiko, Tsuchiura-shi Ibaraki<br />

300-0832, JP<br />

Uenaka, Toshimitsu, Ushiku-shi Ibaraki 300-<br />

1233, JP<br />

Asai, Naoki, Tsukuba-shi Ibaraki 305-0047,<br />

JP<br />

Matsufuji, Motoko, Komae-shi Tokyo 201-<br />

0005, JP<br />

Sameshima, Tomohiro, Fujisawa-shi Kanagawa<br />

251-0052, JP<br />

Kawamura, Naoto, Yamato-shi Kanagawa<br />

242-0007, JP<br />

Dobashi, Kazuyuki, Hadano-shi Kanagawa<br />

257-0013, JP<br />

Nakashima, Takashi, Fujisawa-shi Kanagawa<br />

251-0021, JP<br />

Yoshida, Masashi, Chigasaki-shi Kanagawa<br />

253-0017, JP<br />

Tsuchida, Toshio, Yamato-shi Kanagawa<br />

242-0007, JP<br />

Takeda, Susumu, Yakohama-shi Kanagawa<br />

232-0071, JP<br />

Yamada, Tomonari, Yaidu-shi Shizuoka 425-<br />

0086, JP<br />

Norihisa, Koji, Iwata-shi Shizuoka 438-0078,<br />

JP<br />

Yamori, Takao, Tokyo 162-0836, JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastraße 4, 81925 München, DE<br />

(62) 02711280.4 / 1 380 579<br />

C07D 317/58 → (51) C07C 311/21<br />

C07D 331/04 → (51) C07C 323/52<br />

C07D 333/08 → (51) C07C 323/40<br />

C07D 333/24 → (51) C07C 237/20

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