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Bulletin 2011/10 - European Patent Office

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(C07D) II.1(1)<br />

(54) • TRIAZA- UND TETRAAZA-ANTHRAZEN-<br />

DIONDERIVATE, IHRE HERSTELLUNG<br />

UND VERWENDUNG ALS PHARMAZEU-<br />

TIKA<br />

• TRIAZA- AND TETRAAZA-ANTHRACENE-<br />

DIONE DERIVATIVES, THEIR PREPAR-<br />

ATION AND THEIR USE AS<br />

PHARMACEUTICALS<br />

• DERIVES DE TRIAZA- ET TETRAAZA-<br />

ANTHRACENEDIONES, LEURS PREPARA-<br />

TION ET UTILISATION COMME PHARMA-<br />

CEUTIQUES<br />

(73) Sanofi-Aventis Deutschland GmbH,<br />

Brüningstraße 50, 65929 Frankfurt am Main,<br />

DE<br />

(72) WEICHERT, Andreas, 22846 Norderstedt, DE<br />

STROBEL, Hartmut, 65835 Liederbach, DE<br />

WOHLFART, Paulus, 64625 Bensheim, DE<br />

PATEK, Marcel, Tucson, AZ 85704, US<br />

SMRCINA, Martin, Tucson, AZ 85737, US<br />

WEICHSEL, Aleksandra, sanofi-aventis, Tucson,<br />

AZ 85737-9525, US<br />

(51) C07D 473/04 (11) 2 007 766 B1<br />

(25) En (26) En<br />

(21) 07754689.3 (22) 28.03.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 31.12.2008<br />

(86) US 2007/008205 28.03.2007<br />

(87) WO 2007/120538 2007/43 25.<strong>10</strong>.2007<br />

(30) 11.04.2006 US 79<strong>10</strong>12 P<br />

(54) • NARKOTINREINIGUNGSVERFAHREN<br />

• NARCOTINE PURIFICATION PROCESS<br />

• PROCÉDÉ DE PURIFICATION DE LA NAR-<br />

COTINE<br />

(73) MALLINCKRODT, INC., 675 McDonnell<br />

Boulevard, Hazelwood, MO 63042, US<br />

(72) TOMAZI, Keith, G., Florissant, Missouri<br />

63031, US<br />

LOVE JR., Leroy, St. Louis, Missouri 63034,<br />

US<br />

HAAR JR., Joseph P., Edwardsville, Illinois<br />

62025, US<br />

(74) Adam, Holger, et al, Kraus & Weisert <strong>Patent</strong>und<br />

Rechtsanwälte Thomas-Wimmer-Ring<br />

15, 80539 München, DE<br />

(51) C07D 487/04 (11) 1 753 765 B1<br />

A61K 31/5025 A61P 37/02<br />

(25) En (26) En<br />

(21) 05738153.5 (22) 26.04.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

(43) 21.02.2007<br />

(86) GB 2005/001583 26.04.2005<br />

(87) WO 2005/116033 2005/49 08.12.2005<br />

(30) 26.05.2004 GB 0411770<br />

(54) • IMMUNOINHIBITORISCHE HETEROCYCLI-<br />

SCHE VERBINDUNGEN<br />

• IMMUNO INHIBITORY HETEROCYCLIC<br />

COMPOUNDS<br />

• COMPOSES HETEROCYCLIQUES<br />

IMMUNO-INHIBITEURS<br />

(73) MediGene AG, Lochhamer Strasse 11, 82152<br />

Martinsried, DE<br />

(72) MATTHEWS, Ian Richard, Oxfordshire OX14<br />

4RX, GB<br />

(74) Bösl, Raphael Konrad, Isenbruck Bösl<br />

Hörschler LLP <strong>Patent</strong>anwälte Prinzregentenstrasse<br />

68, 81675 München, DE<br />

(51) C07D 487/04 (11) 1 836 206 B1<br />

A61K 31/437 A61P 3/<strong>10</strong><br />

(25) En (26) En<br />

(21) 05855291.0 (22) 23.12.2005<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 26.09.2007<br />

(86) US 2005/046706 23.12.2005<br />

(87) WO 2006/071752 2006/27 06.07.2006<br />

(30) 29.12.2004 US 640135 P<br />

(54) • DIPEPTIDYLPEPTIDASE-IV-INHIBITOREN<br />

AUF AZOLOPYRIMIDINBASIS UND VER-<br />

FAHREN<br />

• AZOLOPYRIMIDINE-BASED INHIBITORS<br />

OF DIPEPTIDYL PEPTIDASE IV AND<br />

METHODS<br />

• INHIBITEURS AZOLOPYRIMIDINIQUES DE<br />

LA DIPEPTIDYL-PEPTIDASE IV, ET PRO-<br />

CEDES CORRESPONDANTS<br />

(73) Bristol-Myers Squibb Company, Route 206<br />

and Province Line Road P.O. Box 4000,<br />

Princeton NJ 08543-4000, US<br />

(72) MENG, Wei, Pennington, NJ 08534, US<br />

HAMANN, Lawrence G., Cherry Hill, NJ<br />

08003, US<br />

BRIGANCE, Robert Paul, Levittown, PA<br />

19054, US<br />

(74) Reitstötter - Kinzebach, <strong>Patent</strong>anwälte<br />

Sternwartstrasse 4, 81679 München, DE<br />

(51) C07D 487/04 (11) 1 838 712 B1<br />

A61K 31/519 A61P 35/00<br />

(25) En (26) En<br />

(21) 05818622.2 (22) 12.12.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 03.<strong>10</strong>.2007<br />

(86) GB 2005/004770 12.12.2005<br />

(87) WO 2006/064196 2006/25 22.06.2006<br />

(30) 14.12.2004 EP 04292982<br />

30.05.2005 EP 05291158<br />

(54) • PYRAZOLOPYRIMIDINVERBINDUNGEN<br />

ALS ANTITUMORMITTEL<br />

• PYRAZOLOPYRIMIDINE COMPOUNDS AS<br />

ANTITUMOR AGENTS<br />

• COMPOSES DE PYRAZOLOPYRIMIDINE<br />

EN TANT QU`AGENTS ANTITUMORAUX<br />

(73) AstraZeneca AB, 151 85 Södertälje, SE<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU<br />

(72) BARLAAM, Bernard Christophe, AstraZeneca<br />

Reims, F-51689 Reims, FR<br />

DUCRAY, Richard, AstraZeneca Reims, F-<br />

51689 Reims, FR<br />

KETTLE, Jason Grant, AstraZeneca R & D<br />

Alderley, Macclesfield Cheshire SK<strong>10</strong> 4TG,<br />

GB<br />

C07D 487/04 → (51) C07D 471/14<br />

(51) C07D 487/06 (11) 2 079 747 B1<br />

A61K 31/55 A61P 3/00<br />

A61P 43/00<br />

(25) En (26) En<br />

(21) 07825335.8 (22) 03.<strong>10</strong>.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

RS<br />

(43) 22.07.2009<br />

(86) IB 2007/003027 03.<strong>10</strong>.2007<br />

(87) WO 2008/044127 2008/16 17.04.2008<br />

(30) 13.<strong>10</strong>.2006 US 829419 P<br />

(54) • ALS ANABOLE MITTEL FÜR VIEH GEEIG-<br />

NETE HETEROZYKLISCHE VERBINDUN-<br />

GEN<br />

• HETEROCYCLIC COMPOUNDS USEFUL AS<br />

ANABOLIC AGENTS FOR LIVESTOCK ANI-<br />

MALS<br />

589<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>10</strong>/<strong>2011</strong>) 09.03.<strong>2011</strong><br />

• COMPOSÉS HÉTÉROCYCLIQUES UTILES<br />

EN TANT QU'AGENTS ANABOLIQUES<br />

POUR LE BÉTAIL<br />

(73) Pfizer Limited, Ramsgate Road, Sandwich,<br />

Kent CT13 9NJ, GB<br />

(72) BOYLE, Jessica, Sandwich Kent CT13 9NJ,<br />

GB<br />

FENWICK, Ashley, Edward, Sandwich Kent<br />

CT13 9NJ, GB<br />

GETHIN, David, Morris, Sandwich Kent CT13<br />

9NJ, GB<br />

McCUSKER, Catherine Frances, Shawlands,<br />

Glasgow, G41 4 AN, GB<br />

(74) Lane, Graham Mark Hamilton, et al, Pfizer<br />

Limited <strong>European</strong> <strong>Patent</strong> Department,<br />

Ramsgate Road Sandwich CT13 9NJ, GB<br />

(51) C07D 489/00 (11) 1 730 151 B1<br />

C07D 489/08<br />

(25) En (26) En<br />

(21) 05730345.5 (22) 30.03.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

AL BA HR LV MK YU<br />

(43) 13.12.2006<br />

(86) US 2005/0<strong>10</strong>666 30.03.2005<br />

(87) WO 2005/097801 2005/42 20.<strong>10</strong>.2005<br />

(30) 30.03.2004 US 557492 P<br />

13.08.2004 US 601534 P<br />

18.<strong>10</strong>.2004 US 620072 P<br />

31.01.2005 US 648625 P<br />

<strong>10</strong>.02.2005 US 651778 P<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

OXYCODONHYDROCHLORID MIT WENI-<br />

GER ALS 25 PPM 14-HYDROXYCODEINON<br />

• PROCESS FOR PREPARING OXYCODONE<br />

HYDROCHLORIDE HAVING LESS THAN 25<br />

PPM 14-HYDROXYCODEINONE<br />

• PROCEDE DE PREPARATION D'HYDRO-<br />

CHLORURE D'OXYCODONE PRESENTANT<br />

MOINS DE 25 PPM DE 14-HYDROXYCO-<br />

DEINONE<br />

(73) EURO-CELTIQUE S.A., 2, avenue Charles de<br />

Gaulle, 1653 Luxembourg, LU<br />

(72) CHAPMAN, Robert, Downingtown, PA<br />

19335, US<br />

RIDER, Lonn, S., Foster, RI 02825, US<br />

HONG, Qi, Sharon, MA 02607, US<br />

KYLE, Donald, Newtown, PA 18940, US<br />

KUPPER, Robert, East Greenwich, RI 02818,<br />

US<br />

(74) Maiwald <strong>Patent</strong>anwalts GmbH, Elisenhof<br />

Elisenstrasse 3, 80335 München, DE<br />

(60) <strong>10</strong>011787.8<br />

<strong>10</strong>011788.6<br />

<strong>10</strong>011791.0<br />

<strong>10</strong>011792.8<br />

<strong>10</strong>011793.6<br />

C07D 489/08 → (51) C07D 489/00<br />

(51) C07D 491/052 (11) 2 <strong>10</strong>9 615 B1<br />

C07D 491/16 C07D 495/16<br />

A61K 31/436 A61P 1/00<br />

A61P 25/00<br />

(25) En (26) En<br />

(21) 08713287.4 (22) 25.01.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 21.<strong>10</strong>.2009<br />

(86) US 2008/00<strong>10</strong>42 25.01.2008<br />

(87) WO 2008/094476 2008/32 07.08.2008<br />

(30) 31.01.2007 US 898602 P<br />

08.03.2007 US 905690 P<br />

(54) • SUBSTITUIERTE PYRANO [2, 3 - B]<br />

PYRIDINDERIVATE ALS CANNABINOID-1<br />

REZEPTORMODULATOREN

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