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Bulletin 2011/10 - European Patent Office

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(C07D) I.1(1)<br />

C07D 277/64 → (51) C07C 323/60<br />

C07D 285/135→ (51) C07C 323/60<br />

C07D 295/088→ (51) C07C 405/00<br />

(51) C07D 301/32 (11) 2 291 363 A1*<br />

(25) En (26) En<br />

(21) 09713275.7 (22) 20.02.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/00<strong>10</strong>95 20.02.2009<br />

(87) WO 2009/<strong>10</strong>5252 2009/35 27.08.2009<br />

(30) 23.02.2008 US 70992<br />

(54) • VERBESSERTES VERFAHREN ZUR RÜCK-<br />

GEWINNUNG VON ETHYLENOXID<br />

• IMPROVED ETHYLENE OXIDE RECOVERY<br />

PROCESS<br />

• PROCÉDÉ AMÉLIORÉ DE RÉCUPÉRATION<br />

D'OXYDE D'ÉTHYLÈNE<br />

(71) Ozero, Brian, P.O. Box 768, Westhampton<br />

Beach, NY 11978, US<br />

(72) Ozero, Brian, Westhampton Beach, NY<br />

11978, US<br />

(74) Richards, John, et al, Ladas & Parry LLP<br />

Dachauerstrasse 37, 80335 München, DE<br />

C07D 301/32 → (51) C07C 29/12<br />

C07D 307/48 → (51) C07C 51/48<br />

C07D 307/68 → (51) C07C 335/26<br />

C07D 307/68 → (51) C07C 405/00<br />

(51) C07D 307/78 (11) 2 291 364 A2*<br />

A61K 31/343<br />

(25) En (26) En<br />

(21) 09762685.7 (22) 12.06.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) KR 2009/003165 12.06.2009<br />

(87) WO 2009/151299 2009/51 17.12.2009<br />

(88) 01.04.20<strong>10</strong><br />

(30) 12.06.2008 KR 20080055307<br />

(54) • STYRYLBENZOFURANDERIVATE ALS<br />

INHIBITOREN DER BILDUNG VON BETA-<br />

AMYLOID-FIBRILEN UND VERFAHREN ZU<br />

DEREN HERSTELLUNG<br />

• STYRYLBENZOFURAN DERIVATIVES AS<br />

INHIBITORS FOR BETA-AMYLOID FIBRIL<br />

FORMATION AND PREPARATION METHOD<br />

THEREOF<br />

• DÉRIVÉS DE STYRYLBENZOFURANE<br />

COMME INHIBITEURS DE LA FORMATION<br />

DE FIBRILLES D AMYLOÏDE BÊTA ET<br />

LEUR PROCÉDÉ DE PRÉPARATION<br />

(71) Korea Institute of Science and Technology,<br />

39-1, Hawolgok-2-dong Seongbuk-gu, Seoul<br />

136-791, KR<br />

Hanmi Holdings Co., Ltd, No 45, Bangidong,<br />

Songpa-gu Seoul 138-828, KR<br />

(72) KIM, Dong Jin, Seoul 139-242, KR<br />

YOO, Kyung Ho, Seoul 132-040, KR<br />

BYUN, Ji Hun, Seoul 135-0<strong>10</strong>, KR<br />

KIM, YoungSoo, Yongin-si Gyeonggi-do<br />

446-561, KR<br />

KIM, Hye Yun, Seoul 135-280, KR<br />

LEE, Gwan Sun, Seoul 138-739, KR<br />

KIM, Maeng Sup, Seoul 134-060, KR<br />

AHN, Young Gil, Seongnam-si Gyeonggi-do<br />

463-785, KR<br />

LEE, Ji Hoon, Seoul 140-911, KR<br />

LEE, Myoung-Hwan, Seoul 157-876, KR<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

HWANG, Hana, Anyang-si Gyeonggi-do 431-<br />

762, KR<br />

RYU, Jiyeon, Seoul 138-912, KR<br />

(74) Goddar, Heinz J., Forrester & Boehmert<br />

Pettenkoferstrasse 20-22, 80336 München,<br />

DE<br />

C07D 317/38 → (51) C07C 29/12<br />

C07D 317/68 → (51) C07C 335/26<br />

C07D 319/18 → (51) C07C 335/26<br />

C07D 333/20 → (51) C07C 59/64<br />

C07D 333/38 → (51) C07C 335/26<br />

C07D 333/38 → (51) C07C 405/00<br />

C07D 333/40 → (51) C07C 59/72<br />

(51) C07D 401/04 (11) 2 291 365 A1*<br />

C07D 401/14 C07D 405/14<br />

C07D 409/14 C07D 413/14<br />

A61K 31/4525 A61P 35/00<br />

(25) En (26) En<br />

(21) 09755262.4 (22) 28.05.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/003258 28.05.2009<br />

(87) WO 2009/145899 2009/49 03.12.2009<br />

(30) 30.05.2008 US 130445<br />

(54) • 5-SUBSTITUIERTE ISOINDOLIN-VERBIN-<br />

DUNGEN<br />

• 5-SUBSTITUTED ISOINDOLINE COM-<br />

POUNDS<br />

• COMPOSÉS CONSISTANT EN ISOINDOLI-<br />

NES SUBSTITUÉES EN POSITION 5<br />

(71) CELGENE CORPORATION, 86 Morris Avenue,<br />

Summit, NJ 07901, US<br />

(72) MULLER, George, W., Rancho Santa Fe, CA<br />

92067 , US<br />

CHEN, Roger, S., C., Edison NJ 08820, US<br />

RUCHELMAN, Alexander, L., Cream Ridge<br />

NJ 08514, US<br />

ZHANG, Weihong, Highland Park, NJ 08904,<br />

US<br />

MAN, Hon-Wah, Princeton, NJ 08540, US<br />

KHALIL, Ehab, M., Whitenhouse Station, NJ<br />

08889, US<br />

(74) Ritter, Thomas Kurt, et al, Jones Day<br />

Prinzregentenstraße 11, 80538 München, DE<br />

C07D 401/<strong>10</strong> → (51) C07D 213/06<br />

C07D 401/12 → (51) C07D 231/56<br />

C07D 401/14 → (51) C07D 231/56<br />

C07D 401/14 → (51) C07D 401/04<br />

C07D 403/02 → (51) C07D 403/<strong>10</strong><br />

C07D 403/08 → (51) C07D 403/<strong>10</strong><br />

(51) C07D 403/<strong>10</strong> (11) 2 291 366 A2*<br />

C07D 403/08 C07D 403/02<br />

(25) En (26) En<br />

(21) 09763190.7 (22) 20.05.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/044587 20.05.2009<br />

(87) WO 2009/151899 2009/51 17.12.2009<br />

58<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>10</strong>/<strong>2011</strong>) 09.03.<strong>2011</strong><br />

(88) 25.02.20<strong>10</strong><br />

(30) 26.05.2008 IN CH12852008<br />

18.09.2008 US 98003 P<br />

(54) • HERSTELLUNG VON IMATINIB-MESYLAT<br />

• PREPARATION OF IMATINIB MESYLATE<br />

• PRÉPARATION DE MÉSYLATE D IMATINIB<br />

(71) Dr. Reddy's Laboratories, Ltd., 7-1-27<br />

Ameerpet, Hyderabad 500 016 AP, IN<br />

Dr. Reddy's Laboratories Inc., 200 Somerset<br />

Corporate Boulevard, 7th Floor, Bridgewater,<br />

NJ 08807, US<br />

(72) KADABOINA, Rajasekhar, Andhra Pradesh,<br />

IN<br />

NARIYAM, Munaswamy, Sekhar, Hyderabad<br />

500 072 Andhra Pradesh, IN<br />

PATEL, Vijay, Bhailalbhai, Hyderabad 500<br />

072 Andhra Pradesh, IN<br />

(74) Bates, Philip Ian, et al, Reddie & Grose 16<br />

Theobalds Road, London WC1X 8PL, GB<br />

C07D 403/<strong>10</strong> → (51) C07D 231/56<br />

C07D 403/12 → (51) C07D 231/56<br />

C07D 405/<strong>10</strong> → (51) C07D 213/06<br />

C07D 405/14 → (51) C07D 401/04<br />

C07D 407/12 → (51) C07D 409/14<br />

C07D 407/14 → (51) C07D 231/56<br />

C07D 407/14 → (51) C07D 409/14<br />

(51) C07D 409/06 (11) 2 291 367 A1*<br />

A61K 31/403<br />

(25) En (26) En<br />

(21) 09735602.6 (22) 22.04.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/041398 22.04.2009<br />

(87) WO 2009/132097 2009/44 29.<strong>10</strong>.2009<br />

(30) 24.04.2008 US 475<strong>10</strong> P<br />

(54) • SUBSTITUIERTE GAMMA-LACTAME ALS<br />

THERAPEUTISCHE MITTEL<br />

• SUBSTITUTED GAMMA LACTAMS AS<br />

THERAPEUTIC AGENTS<br />

• GAMMA LACTAMES SUBSTITUÉS EN<br />

TANT QU'AGENTS THÉRAPEUTIQUES<br />

(71) Allergan, Inc., 2525 Dupont Drive, T2-7H,<br />

Irvine, CA 92612, US<br />

(72) OLD, David, W., Irvine CA 92620, US<br />

DINH, Danny, T., Garden Grove CA 92840,<br />

US<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastraße 4, 81925 München, DE<br />

C07D 409/06 → (51) C07D 409/12<br />

(51) C07D 409/12 (11) 2 291 368 A1*<br />

C07D 207/26 C07D 409/06<br />

A61K 31/4015 A61P 27/06<br />

(25) En (26) En<br />

(21) 09734653.0 (22) 22.04.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/041389 22.04.2009<br />

(87) WO 2009/132088 2009/44 29.<strong>10</strong>.2009<br />

(30) 24.04.2008 US 47501 P<br />

(54) • SUBSTITUIERTE GAMMA-LACTAME ALS<br />

THERAPEUTISCHE MITTEL<br />

• SUBSTITUTED GAMMA LACTAMS AS<br />

THERAPEUTIC AGENTS

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