Bulletin 2011/10 - European Patent Office

(C07D) I.1(1)
• GAMMA-LACTAMES SUBSTITUÉS EN
TANT QU AGENTS THÉRAPEUTIQUES
(71) Allergan, Inc., 2525 Dupont Drive, T2-7H,
Irvine, CA 92612, US
(72) OLD, David, W., Irvine CA 92620, US
DINH, Danny, T., Garden Grove CA 92840,
US
(74) HOFFMANN EITLE, Patent- und Rechtsanwälte
Arabellastraße 4, 81925 München, DE
C07D 409/12 → (51) C07D 231/56
(51) C07D 409/14 (11) 2 291 369 A1*
A61K 31/416 A61K 31/4439
A61P 11/00 A61P 29/00
C07D 407/12 C07D 407/14
(25) En (26) En
(21) 09750866.7 (22) 20.05.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK TR
AL BA RS
(86) SE 2009/000267 20.05.2009
(87) WO 2009/142571 2009/48 26.11.2009
(30) 20.05.2008 US 54616
14.07.2008 US 80312
15.01.2009 US 144776
(54) • PHENYL- ODER BENZODIOXINYLSUBSTI-
TUIERTE INDAZOLDERIVATE
• PHENYL AND BENZODIOXINYL SUBSTI-
TUTED INDAZOLES DERIVATIVES
• DÉRIVÉS D'INDAZOLES À SUBSTITU-
TIONS PHÉNYLE ET BENZODIOXINYLE
(71) AstraZeneca AB, 151 85 Södertälje, SE
(72) BAYER SCHERING PHARMA AG, D-13353
Berlin, DE
BERGER, Markus, D-13353 Berlin, DE
DAHMEN, Jan, S-221 87 Lund, SE
EDMAN, Karl, S-431 83 Mölndal, SE
ERIKSSON, Anders, S-221 87 Lund, SE
HANSSON, Thomas, S-221 87 Lund, SE
HEMMERLING, Martin, S-221 87 Lund, DE
HOSSAIN Nafizal, S-221 87 Lund, SE
KLINGSTEDT, Tomas, S-221 87 Lund, SE
LEPISTÖ, Matti, S-221 87 Lund, SE
NILSSON, Stinabritt, S-221 87 Lund, SE
REHWINKEL, Hartmut, D-13353 Berlin, DE
C07D 409/14 → (51) C07D 231/56
C07D 409/14 → (51) C07D 401/04
(51) C07D 413/10 (11) 2 291 370 A1*
C07D 413/14 A61K 31/5355
A61P 19/10
(25) En (26) En
(21) 09739190.8 (22) 30.04.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK TR
AL BA RS
(86) US 2009/002633 30.04.2009
(87) WO 2009/134387 2009/45 05.11.2009
(30) 01.05.2008 US 49650 P
25.07.2008 US 137148 P
25.07.2008 PCT/US2008/009017
04.02.2009 US 206817 P
(54) • CYCLISCHE INHIBITOREN VON 11BETA-
HYDROXYSTEROIDDEHYDROGENASE 1
• CYCLIC INHIBITORS OF 11BETA-HYDRO-
XYSTEROID DEHYDROGENASE 1
• INHIBITEURS CYCLIQUES DE LA 11-BÊTA-
HYDROXYSTÉROÏDE DÉHYDROGÉNASE 1
(71) Vitae Pharmaceuticals, Inc., 502 West Office
Center Drive, Fort Washington, PA 19034,
US
Europäisches Patentblatt
European Patent Bulletin
Bulletin européen des brevets
Boehringer Ingelheim International GmbH,
Binger Straße 173, 55216 Ingelheim am
Rhein, DE
(72) CLAREMON, David, A., Maple Glen PA
19002, US
ZHUANG, Linghang, Chalfont PA 18914, US
LEFTHERIS, Katerina, Skillman NJ 08558,
US
TICE, Colin, M., Ambler PA 19002, US
YE, Yuanjie, Ambler PA 19002, US
SINGH, Suresh, B., Kendall Park NJ 08824,
US
HIMMELSBACH, Frank, 55216 Ingelheim Am
Rhein, DE
(74) Simpson, Mark Geoffrey, Potter Clarkson
LLP Park View House 58 The Ropewalk,
Nottingham NG1 5DD, GB
(51) C07D 413/10 (11) 2 291 371 A1*
C07D 413/14 A61K 31/5355
A61P 19/10 C07D 417/10
C07D 417/14
(25) En (26) En
(21) 09739195.7 (22) 30.04.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK TR
AL BA RS
(86) US 2009/002641 30.04.2009
(87) WO 2009/134392 2009/45 05.11.2009
(30) 01.05.2008 US 49650 P
25.07.2008 PCT/US2008/009017
25.07.2008 US 137148 P
04.02.2009 US 206775 P
(54) • CYCLISCHE INHIBITOREN VON 11BETA-
HYDROXYSTEROIDDEHYDROGENASE 1
• CYCLIC INHIBITORS OF 11BETA-HYDRO-
XYSTEROID DEHYDROGENASE 1
• INHIBITEURS CYCLIQUES DE LA 11-BÊTA-
HYDROXYSTÉROÏDE DÉHYDROGÉNASE 1
(71) Vitae Pharmaceuticals, Inc., 502 West Office
Center Drive, Fort Washington, PA 19034,
US
Boehringer Ingelheim International GmbH,
Binger Straße 173, 55216 Ingelheim am
Rhein, DE
(72) CLAREMON, David, A., Maple Glen PA
19002, US
ZHUANG, Linghang, Chalfont PA 18914, US
LEFTHERIS, Katerina, Skillman NJ 08558,
US
TICE, Colin, M., Ambler PA 19002, US
XU, Zhenrong, Horsham PA 19002, US
YE, Yuanjie, Ambler PA 19002, US
SINGH, Suresh, B., Kendall Park NJ 08824,
US
CACATIAN, Salvacion, Blue Bell PA 19422,
US
ZHAO, Wei, Eagleville PA 19403, US
HIMMELSBACH, Frank, 55216 Ingelheim Am
Rhein, DE
ECKHARDT, Matthias, 55216 Ingelheim Am
Rhein, DE
(74) Simpson, Mark Geoffrey, Potter Clarkson
LLP Park View House 58 The Ropewalk,
Nottingham NG1 5DD, GB
C07D 413/12 → (51) C07D 231/56
C07D 413/14 → (51) C07D 401/04
C07D 413/14 → (51) C07D 413/10
C07D 413/14 → (51) C07D 417/14
(51) C07D 417/00 (11) 2 291 372 A2*
(25) En (26) En
(21) 09751378.2 (22) 19.05.2009
59
Anmeldungen
Applications
Demandes (10/2011) 09.03.2011
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK TR
AL BA RS
(86) US 2009/044511 19.05.2009
(87) WO 2009/143150 2009/48 26.11.2009
(88) 14.01.2010
(30) 19.05.2008 US 54326
(54) • MODULATOREN DER ALKALISCHEN
PHOSPHATASE AUS DARM UND ANWEN-
DUNGEN DAVON
• INTESTINAL ALKALINE PHOSPHATASE
MODULATORS AND USES THEREOF
• MODULATEURS DE LA PHOSPHATASE
ALCALINE INTESTINALE ET LEURS UTI-
LISATIONS
(71) Burnham Institute for Medical Research,
10901 N. Torrey Pines Road, La Jolla, CA
92037, US
(72) MILLAN, Jose, Luis, La Jolla, CA 92037, US
NARISAWA, Sonoko, La Jolla, CA 92037, US
SERGIENKO, Eduard, La Jolla, CA 92037, US
(74) Elbel, Michaela, Pateris Patentanwälte Partnerschaft
Altheimer Eck 13, 80331 München,
DE
C07D 417/10 → (51) C07D 413/10
C07D 417/12 → (51) C07C 405/00
(51) C07D 417/14 (11) 2 291 373 A1*
C07D 413/14 A61K 31/5355
A61P 19/10
(25) En (26) En
(21) 09739187.4 (22) 30.04.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK TR
AL BA RS
(86) US 2009/002629 30.04.2009
(87) WO 2009/134384 2009/45 05.11.2009
(30) 25.07.2008 PCT/US2008/009017
01.05.2008 US 49650 P
04.02.2009 US 206825 P
25.07.2008 US 137148 P
(54) • CYCLISCHE INHIBITOREN VON 11BETA-
HYDROXYSTEROIDDEHYDROGENASE 1
• CYCLIC INHIBITORS OF 11BETA-HYDRO-
XYSTEROID DEHYDROGENASE 1
• INHIBITEURS CYCLIQUES DE LA 11-BÊTA-
HYDROXYSTÉROÏDE DÉHYDROGÉNASE 1
(71) Vitae Pharmaceuticals, Inc., 502 West Office
Center Drive, Fort Washington, PA 19034,
US
(72) CLAREMON, David, A., Maple Glen PA
19002, US
ZHUANG, Linghang, Chalfont PA 18914, US
LEFTHERIS, Katerina, Skillman NJ 08558,
US
TICE, Colin, M., Ambler PA 19002, US
YE, Yuanjie, Ambler PA 19002, US
SINGH, Suresh, B., Kendall Park NJ 08824,
US
(74) Simpson, Mark Geoffrey, Potter Clarkson
LLP Park View House 58 The Ropewalk,
Nottingham NG1 5DD, GB
C07D 417/14 → (51) C07D 413/10
(51) C07D 453/02 (11) 2 291 374 A1*
(25) En (26) En
(21) 09750841.0 (22) 22.05.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK TR
AL BA RS
(86) PL 2009/000054 22.05.2009