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Bulletin 2011/10 - European Patent Office

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(C07C) I.1(1)<br />

A61P 29/00<br />

(25) En (26) En<br />

(21) 09732683.9 (22) 14.04.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/040538 14.04.2009<br />

(87) WO 2009/129246 2009/43 22.<strong>10</strong>.2009<br />

(30) 14.04.2008 US 44886<br />

28.07.2008 PCT/US2008/071392<br />

12.03.2009 US 159778<br />

(54) • ZUSAMMENSETZUNGEN UND VERFAH-<br />

REN ZU IHRER HERSTELLUNG UND VER-<br />

WENDUNG<br />

• COMPOSITIONS AND METHODS FOR<br />

PREPARING AND USING SAME<br />

• COMPOSITIONS ET LEURS PROCÉDÉS DE<br />

PRÉPARATION ET D UTILISATION<br />

(71) Ardea Biosciences, Inc., 4939 Directors<br />

Place, San Diego, CA 92121, US<br />

(72) QUART, Barry, D., Encinitas CA 92024, US<br />

ROWLINGS, Colin, Edward, Encinitas CA<br />

92024, US<br />

(74) Williams, Paul Howard, Bayer Schering<br />

Pharma AG <strong>Patent</strong>s and Licensing Müllerstrasse<br />

178, 13342 Berlin, DE<br />

C07C 323/22 → (51) C07C 405/00<br />

(51) C07C 323/60 (11) 2 291 351 A1*<br />

C07D 231/40 C07D 241/20<br />

C07D 263/56 C07D 277/64<br />

C07D 285/135 A61K 31/16<br />

A61K 31/165 A61K 31/415<br />

A61K 31/423 A61K 31/428<br />

A61K 31/433 A61K 31/53<br />

A61P 3/04 A61P 3/<strong>10</strong><br />

(25) En (26) En<br />

(21) 08750117.7 (22) 07.05.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) EP 2008/055594 07.05.2008<br />

(87) WO 2009/135526 2009/46 12.11.2009<br />

(54) • ALPHA-MERCAPTOAMIDE<br />

• ALPHA-MERCAPTO-AMIDES<br />

• ALPHA-MERCAPTOAMIDES<br />

(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(72) NAPOLETANO, Mauro, I-20127 Milano, IT<br />

HAACK, Thomas, I-22<strong>10</strong>0 Como, IT<br />

TSCHINKE, Vincenzo, CH-4<strong>10</strong>2 Binningen,<br />

CH<br />

JELAKOVIC, Stjepan, 79<strong>10</strong>0 Freiburg, DE<br />

MAH, Robert, CH-4132 Muttenz, CH<br />

(74) von Sprecher, Georg, et al, Novartis Pharma<br />

AG <strong>Patent</strong> Department, 4002 Basel, CH<br />

(51) C07C 335/26 (11) 2 291 352 A2*<br />

C07C 275/54 C07D 213/81<br />

C07D 307/68 C07D 317/68<br />

C07D 319/18 C07D 333/38<br />

A61K 31/17 C07D 209/06<br />

C07D 235/14 A61P 3/<strong>10</strong><br />

A61P 25/00<br />

(25) Fr (26) Fr<br />

(21) 09733789.3 (22) 16.04.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) FR 2009/000442 16.04.2009<br />

(87) WO 2009/130422 2009/44 29.<strong>10</strong>.2009<br />

(88) 30.12.2009<br />

(30) 24.04.2008 FR 0802302<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(54) • N-ACYLTHIOHARNSTOFF- UND N-ACYL-<br />

HARNSTOFFVERBINDUNGEN ALS INHIBI-<br />

TOREN DES HEDGEHOG-PROTEIN-<br />

SIGNALPFADES<br />

• N-ACYLTHIOUREA AND N-ACYLUREA<br />

INHIBITORS OF THE HEDGEHOG PROTEIN<br />

SIGNALLING PATHWAY<br />

• N-ACYLTHIOUREES ET N-ACYLUREES<br />

INHIBITEURS DE LA VOIE DE SIGNALI-<br />

SATION DES PROTEINES HEDGEHOG<br />

(71) Centre National de la Recherche Scientifique,<br />

3, rue Michel-Ange, 75016 Paris, FR<br />

(72) RUAT, Martial, F-91400 Orsay, FR<br />

FAURE, Hélène, F-91190 Gif-sur-Yvette, FR<br />

TRAIFFORT, Elisabeth, F-75013 Paris, FR<br />

SCHOENFELDER, Angèle, F-67450 Lampertheim,<br />

FR<br />

MANN, André, F-67540 Ostwald, FR<br />

TADDEI, Maurizio, I-53035 Monteriggioni, IT<br />

SOLINAS, Antonio, I-53<strong>10</strong>0 Siena, IT<br />

MANETTI, Fabrizio, I-53019 Castelnuovo<br />

Berardenga, IT<br />

(74) Mena, Sandra, et al, Cabinet Orès 36, rue de<br />

St Pétersbourg, F-75008 Paris, FR<br />

(51) C07C 405/00 (11) 2 291 353 A1*<br />

C07D 295/088 C07D 333/38<br />

C07C 323/22 C07C 225/22<br />

C07D 213/70 C07D 417/12<br />

C07D 307/68 A61K 31/192<br />

A61K 31/4439 A61K 31/44<br />

A61K 31/38 A61P 27/06<br />

(25) En (26) En<br />

(21) 09751196.8 (22) 13.05.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/043700 13.05.2009<br />

(87) WO 2009/142967 2009/48 26.11.2009<br />

(30) 20.05.2008 US 54682<br />

(54) • THERAPEUTISCHE PROSTAGLANDINVER-<br />

BINDUNGEN ALS WIRKSTOFFE GEGEN<br />

OKULÄRE HYPOTONIE<br />

• THERAPEUTIC PROSTAGLANDIN COM-<br />

POUNDS USED AS OCULAR HYPOTEN-<br />

SIVE AGENTS<br />

• COMPOSÉS PROSTAGLANDINES THÉRA-<br />

PEUTIQUES UTILISÉS EN TANT<br />

QU'AGENTS HYPOTENSIFS OCULAIRES<br />

(71) Allergan, Inc., 2525 Dupont Drive, T2-7H,<br />

Irvine, CA 92612, US<br />

(72) OLD, David W., Irvine California 92620, US<br />

NGO, Vinh X., Huntington Beach California<br />

92646, US<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastraße 4, 81925 München, DE<br />

C07D 207/26 → (51) C07D 409/12<br />

C07D 209/06 → (51) C07C 335/26<br />

(51) C07D 213/06 (11) 2 291 354 A1*<br />

C07D 213/127 C07D 213/30<br />

C07D 401/<strong>10</strong> C07D 405/<strong>10</strong><br />

C07D 213/643 H01L 51/05<br />

(25) En (26) En<br />

(21) 0975<strong>10</strong>96.0 (22) 23.04.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) US 2009/041491 23.04.2009<br />

(87) WO 2009/142867 2009/48 26.11.2009<br />

(30) 22.05.2008 US 125296<br />

(54) • PHENYLPYRIDINEINHEITEN ENTHAL-<br />

TENDE VERBINDUNG<br />

56<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>10</strong>/<strong>2011</strong>) 09.03.<strong>2011</strong><br />

• COMPOUND COMPRISING PHENYL PYR-<br />

IDINE UNITS<br />

• COMPOSÉ COMPRENANT DES UNITÉS<br />

PHÉNYLPYRIDINES<br />

(71) General Electric Company, 1 River Road,<br />

Schenectady, NY 12345, US<br />

(72) LIANG, Yangang, Shanghai 201208, CN<br />

LIU, Shengxia, Shanghai 200123, CN<br />

CHICHAK, Kelly, Scott, Clifton Park NY<br />

12065, US<br />

YE, Qing, Schenectady NY 12309, US<br />

LIU, Jie, Niskayuna NY 12309, US<br />

(74) Szary, Anne Catherine, London <strong>Patent</strong><br />

Operation GE International Inc 15 John Adam<br />

Street, GB-London WC2N 6LU, GB<br />

C07D 213/127→ (51) C07D 213/06<br />

C07D 213/30 → (51) C07D 213/06<br />

C07D 213/643→ (51) C07D 213/06<br />

C07D 213/70 → (51) C07C 405/00<br />

C07D 213/75 → (51) C07C 233/80<br />

C07D 213/81 → (51) C07C 335/26<br />

(51) C07D 215/00 (11) 2 291 355 A2*<br />

C07D 215/02 C07D 215/12<br />

C07D 215/233<br />

(25) En (26) En<br />

(21) 09701340.3 (22) 02.01.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) IN 2009/000002 02.01.2009<br />

(87) WO 2009/087684 2009/29 16.07.2009<br />

(88) 04.11.20<strong>10</strong><br />

(30) 04.01.2008 IN DE00412008<br />

(54) • NEUARTIGE TETRAHYDROCHINOLINE ALS<br />

AROMATASEHEMMER<br />

• NOVEL TETRAHYDROQUINOLINES AS<br />

AROMATASE INHIBITORS<br />

• NOUVELLES TÉTRAHYDROQUINOLÉINES<br />

EN TANT QU'INHIBITEURS D'AROMATASE<br />

(71) Panjab University, Chandigarh 160 014, IN<br />

Kakatiya University, Warangal 506 009, IN<br />

(72) AKKINEPALLY, Raghuram, Rao, Chandigarh<br />

160 014, IN<br />

JAVALI, Narashima, Murthy, Warangal 506<br />

009, IN<br />

(74) Grosset-Fournier, Chantal Catherine, et al,<br />

Grosset-Fournier & Demachy 54, rue Saint-<br />

Lazare, 75009 Paris, FR<br />

C07D 215/02 → (51) C07D 215/00<br />

C07D 215/12 → (51) C07D 215/00<br />

C07D 215/12 → (51) C07D 491/04<br />

C07D 215/14 → (51) C07D 491/04<br />

C07D 215/20 → (51) C07D 491/04<br />

C07D 215/233→ (51) C07D 215/00<br />

(51) C07D 217/02 (11) 2 291 356 A1*<br />

(25) En (26) En<br />

(21) 09750840.2 (22) 22.05.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

AL BA RS<br />

(86) PL 2009/000053 22.05.2009<br />

(87) WO 2009/142521 2009/48 26.11.2009

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