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Document 135. (a) Fong TM, Yu H, Cascieri MA, Underwood D, Swain CJ, Strader CD. J Biol Chem 1994; 269:14957–14961; (b) Fong TM, Yu H, Cascieri MA, Underwood D, Swain C, Strader CD. J Biol Chem 1994; 269:2728–2732; (c) Fong TM, Cascieri MA, Yu H, Bansai A, Swain CJ, Strader CD, Nature 1993; 362:30–353; (d) Gether Y, Johansen TE, Snider RM, Lowe JA, Kakanishi S, Schwartz TW. Nature 1993; 362:345–348. 136. (a) Beinborn M, Lee Y-M, McBridde EW, Quinn SM, Kopin AS. Nature 1993; 362:348–350; (b) Kopin AS, McBride EW, Quinn SM, Kolakowski LF, Beinborn M. J Biol Chem 1995; 270:5019–5023; (c) Silvente-Poirot S, Wank SA. J Biol Chem 1996; 271:14698–14706. 137. (a) Surratt CK, Johnson PS, Moriwaski A, et al. J Biol Chem 1994; 269:20548–20553; (b) Kong H, Raynor K, Yusuda K, et al. J Biol Chem 1993; 268:23055–23058; (c) Kong H, Raynor K, Yano H, Takeda J, Bell GI, Reisine T. Proc Natl Acad Sci USA 1994; 91:8042–8046; (d) Onogi T, Miniami M, Katao Y, Nakagawa T, Aoki Y, Toya T, Katsumata S, Satoh M. FEBS Lett 1995; 357:93– http://legacy.netlibrary.com/nlreader/nlReader.dll?bookid=12640&filename=Page_626.html (2 of 2) [4/9/2004 1:46:39 AM]
Document 97; (e) Fujii I, Nakamura H, Sagara T, Kanematsu K. Med Chem Res 1994; 4:424–431. Page 627 138. (a) Mouillac B, Chin B, Balestre M-N, Elands J, Trumpp-Kallmeyer S, Hoflack J, Hibert M, Jard S, Barberis C. J Biol Chem 270:25771–25777; (b) Chini B, Mouillac B, Ala Y, Balestre M-N, Trumpp- Kallmeyer S, Hoflack J, Elands J, Hibert M, Manning M, Jard S, Barberis C, EMBO J 1995; 14:2176–2182; (c) Huggins JP, Trumpp-Kallmeyer S, Hibert M, Hoflack JM, Fanger BO, Jones CR. Eur J Pharmacol 1993; 245:203–214. 139. Kyle DJ, Chakravarty S, Sinako JA, Stormann TM. J Med Chem 1994; 37:1347–1354. 140. Pang Y-P, Cusack B, Groshan K, Richelson E. J Biol Chem 1996; 271:15060–15068. 141. Haskell-Luevano C, Sawyer TK, Trumpp-Kallmeyer Bikker J, Humblet C, Gantz I, Hruby VJ. Drug Design Disc. 1996; 14:197–211. 142. (a) Rich DH, In: Sammes PG, Ed. Comprehensive Medicinal Chemistry. New York: Pergamon Press, 1990: 391–441; (b) Lawton G, Paciorek PM, Waterfall JF. Adv Drug Res 1992; 23:12–220; (c) Wyvratt MJ, Patchett AA. Med Res Rev 1985; 5:483–531. 143. James MN, and Sielecki AR. J Mol Biol 1983; 163:299–361. 144. Suguna K, Bott RR, Padlan EA, Subramanian E, Sheriff S, Cohen GH, Davis DR. J Mol Biol 1987; 196:877–900. 145. Blundell TL, Jenkins JA, Sewell BT, Pearl LH, Cooper JB, Tickle IJ, Veerpandian B, Wood SP. J Mol Biol 1990; 211:919–941. 146. Sielecki AR, Fujinaga M, Read RJ, James MN, J Mol Biol 1991; 219:671–. 147. (a) Abad-Zapatero C, Rydel TJ, Erickson J, Proteins 1990; 8:62-; (b) Cooper JB, Khan G, Taylor G, Tickle IJ, Blundell TL. J Mol Biol 1990; 214:199-; (c) Sielecki AR, Fedorov AA, Boodhoo A, Andreeva NS, James MN. J Mol Biol 1990; 214:143–170. 148. (a) Sibanda BL, Blundell T, Hobart PM, Fogliano M, Bindra JS, Dominy BW, Chirgwin JM. FEBS Lett 1984; 174:96–101; (b) Carson W, Karplus M, Haber E. Hypertension 1985; 7:13–26; (c) Akahane K, Umeyama H, Nakagawa S, Moriguchi I, Hirose S, Iizuka K, Murakami Hypertension 1985; 7:3–12; (d) Sham HL, Bolis G, Stein HH, Fesik SW, Marcotte PA, Plattner JJ, Remple CA, Greer J. J Med Chem 1988; 31:284–295. 149. (a) Abdel-Meguid SS, Med Res Rev 1993; 13:731–778; (b) Hutchins C, Greer J. Crit Rev Biochem Mol Biol 1991; 26:77–127; (c) Greenlee W. Med Res Rev 1990; 10:173–236. http://legacy.netlibrary.com/nlreader/nlReader.dll?bookid=12640&filename=Page_627.html (1 of 2) [4/9/2004 1:47:10 AM]
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netLibrary - eBook Summary Universi
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Structure-based Drug Design 14 Stru
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Page 803 and 804: Document factors, 247 Combination t
Page 805 and 806: Document Cyclotheonamide A (CtA), 2
Page 807 and 808: Document D ddI, 152 tumour necrosis
Page 809 and 810: Document antistasin peptides, 281 c
Page 811 and 812: Document fragment-based programs, 5
Page 813 and 814: Document [Human immunodeficiency vi
Page 815 and 816: Document overview, 103-104, 108-109
Page 817 and 818: Document [Inhibitors] 2-((3,4-dihyd
Page 819 and 820: Document antagonistic activity, 416
Page 821 and 822: Document [Interleukin-1] homology w
Page 823 and 824: Document Kininogen, 119 high molecu
Page 825 and 826: Document Matrix-metalloproteinase (
Page 827 and 828: Document RT inhibitor, 41, 56 Nonpe
Page 829 and 830:
Document Phosphoglycerate kinase (P
Page 831:
Document [Protease targets] serinyl
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