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Bulletin 2009/07 - European Patent Office

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(C<strong>07</strong>D) II.1(1)<br />

(74) Hütter, Klaus, et al, Clariant Produkte<br />

(Deutschland) GmbH Group Intellectual<br />

Property Am Unisys-Park 1, 65843 Sulzbach,<br />

DE<br />

C<strong>07</strong>D 403/12 → (51) C<strong>07</strong>D 401/12<br />

C<strong>07</strong>D 417/12 → (51) C<strong>07</strong>D 401/12<br />

C<strong>07</strong>D 417/14 → (51) C<strong>07</strong>D 401/12<br />

(51) C<strong>07</strong>D 471/04 (11) 1 605 938 B1<br />

C<strong>07</strong>D 491/04 C<strong>07</strong>D 498/04<br />

C<strong>07</strong>D 513/04 C<strong>07</strong>D 519/00<br />

A61K 31/4375 A61P 31/04<br />

(25) En (26) En<br />

(21) 04758428.9 (22) 26.03.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

LT LV<br />

(43) 21.12.2005<br />

(86) US 2004/009371 26.03.2004<br />

(87) WO 2004/087145 2004/42 14.10.2004<br />

(30) 27.03.2003 US 458147 P<br />

(54) • Antibakterielle Naphthydrin- und Quinolinderivate<br />

• Antibacterial derivatives of napthydrin and<br />

quinoline<br />

• Dérivés antibacteriens de la naphthydrine<br />

et quinoline<br />

(73) GLAXO GROUP LIMITED, Glaxo Wellcome<br />

House, Berkeley Avenue, Greenford, Middlesex<br />

UB6 0NN, GB<br />

(72) HENNESSY, Alan J., Harlow, Essex CM19<br />

5AW, GB<br />

MILLER, William, Henry, Collegeville, PA<br />

19426, US<br />

SEEFELD, Mark, Andrew, Collegeville, PA<br />

19426, US<br />

(74) Valentine, Jill Barbara, et al, GlaxoSmithKline<br />

Corporate Intellectual Property (CN9.25.1)<br />

980 Great West Road, Brentford, Middlesex<br />

TW8 9GS, GB<br />

(51) C<strong>07</strong>D 471/04 (11) 1 851 217 B1<br />

A61K 31/519 A61P 35/00<br />

(25) En (26) En<br />

(21) 067<strong>07</strong>117.5 (22) 21.02.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

HR MK<br />

(43) <strong>07</strong>.11.20<strong>07</strong><br />

(86) EP 2006/001539 21.02.2006<br />

(87) WO 2006/087229 2006/34 24.08.2006<br />

(30) 21.02.2005 GB 0503506<br />

(54) • ALS MEDIKAMENTE FÜR DIE BEHAND-<br />

LUNG VON AUTOIMMUNERKRANKUNGEN<br />

GEEIGNETE SUBSTITUIERTE PYRIDO[2,3-<br />

D]PYRIMIDINDERIVATE<br />

• SUBSTITUTED PYRIDO[2,3-D]PYRIMI-<br />

DINE DERIVATIVES USEFUL AS MEDI-<br />

CINES FOR THE TREATMENT OF<br />

AUTOIMMUNE DISORDERS<br />

• DERIVES SUBSTITUES DE PYRIDO [2,3-D]<br />

PYRIMIDINE UTILES EN TANT QUE<br />

MEDICAMENTS POUR LE TRAITEMENT<br />

DES TROUBLES AUTOIMMUNS<br />

(73) 4 AZA IP NV, Kapucijnenvoer 33, 3000<br />

Leuven, BE<br />

(72) DE JONGHE, Steven, Cesar, Alfons, B-3080<br />

Tervuren, BE<br />

HERDEWIJN, Piet, André, Maurits, Maria, B-<br />

3111 Rotselaar/Wezemaal, BE<br />

GAO, Ling-Jie, B-3360 Bierbeek, BE<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(74) Weiss, Wolfgang, Weickmann & Weickmann<br />

<strong>Patent</strong>anwälte Postfach 86 08 20, 81635<br />

München, DE<br />

(51) C<strong>07</strong>D 471/04 (11) 1 853 601 B1<br />

A61K 31/551 A61P 29/00<br />

(25) En (26) En<br />

(21) 06708243.8 (22) 14.02.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

HR YU<br />

(43) 14.11.20<strong>07</strong><br />

(86) EP 2006/050906 14.02.2006<br />

(87) WO 2006/084917 2006/33 17.08.2006<br />

(30) 14.02.2005 EP 05101086<br />

(54) • NICHTSTEROIDE GLUCOCORTICOID-<br />

REZEPTORMODULATOREN<br />

• NON STEROIDAL GLUCOCORTICOID<br />

RECEPTOR MODULATORS<br />

• MODULATEURS DE RECEPTEURS GLU-<br />

COCORTICOIDES NON STEROIDIENS<br />

(73) N.V. Organon, Kloosterstraat 6, 5349 AB<br />

Oss, NL<br />

(72) PLATE, Ralf, NL-5340 BH Oss, NL<br />

ZAMAN, Guido Jenny Rudolf, NL-5340 BH<br />

Oss, NL<br />

HERMKENS, Pedro Harold Han, NL-5340 BH<br />

Oss, NL<br />

JANS, Christiaan Gerardus Johannes Maria,<br />

NL-5340 BH Oss, NL<br />

BUIJSMAN, Rogier Christian, NL-5340 BH<br />

Oss, NL<br />

DE MAN, Adrianus, Petrus, Antonius, NL-<br />

5340 BH Oss, NL<br />

CONTI, Paolo Giovanni Martino, NL-5340 BH<br />

Oss, NL<br />

LUSHER, Scott James, NL-5340 BH Oss, NL<br />

DOKTER, Willem Hendrik Abraham, NL-5340<br />

BH Oss, NL<br />

(74) van Wezenbeek, Petrus M.G.F., et al, P.O.<br />

Box 20, 5340 BH Oss, NL<br />

(51) C<strong>07</strong>D 487/04 (11) 1 370 561 B1<br />

A61K 31/4985 A61P 3/00<br />

(25) En (26) En<br />

(21) 02732459.9 (22) 06.03.2002<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

(43) 17.12.2003<br />

(86) EP 2002/002443 06.03.2002<br />

(87) WO 2002/<strong>07</strong>2584 2002/38 19.09.2002<br />

(30) 13.03.2001 GB 0106177<br />

(54) • TETRAHYDRO-PYRAZINO[1,2-A]INDOLE<br />

FÜR DIE BEHANDLUNG VON KRANKHEI-<br />

TEN DES ZENTRALNERVENSYSTEMS<br />

• TETRAHYDRO-PYRAZINO[1,2-A]INDOLES<br />

FOR THE TREATMENT OF CENTRAL NER-<br />

VOUS DISORDERS<br />

• TETRAHYDRO-PYRAZINO[1,2-A]INDOLES<br />

POUR LE TRAITEMENT DES MALADIES<br />

DU SYSTEME NERVEUX CENTRAL<br />

(73) F. Hoffmann-La Roche AG, Grenzacherstrasse<br />

124, 4<strong>07</strong>0 Basel, CH<br />

VERNALIS RESEARCH LIMITED, Oakdene<br />

Court, 613 Reading Road, Winnersh,<br />

Wokingham RG41 5UA, GB<br />

(72) HEBEISEN, Paul, CH-4052 Basle, CH<br />

MATTEI, Patrizio, CH-4125 Riehen, CH<br />

MULLER, Marc, F-68300 St. Louis, FR<br />

RICHTER, Hans, 79639 Grenzach-Wyhlen,<br />

DE<br />

ROEVER, Stephan, 79594 Inzlingen, DE<br />

TAYLOR, Sven, F-68400 Riedisheim, FR<br />

(74) Waschbüsch, Klaus, 124 Grenzacherstrasse,<br />

4<strong>07</strong>0 Basle, CH<br />

C<strong>07</strong>D 487/04 → (51) C<strong>07</strong>D 401/12<br />

540<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>07</strong>/<strong>2009</strong>) 11.02.<strong>2009</strong><br />

(51) C<strong>07</strong>D 487/08 (11) 1 819 709 B1<br />

A61K 31/4995 A61P 25/00<br />

(25) En (26) En<br />

(21) 05817438.4 (22) 29.11.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 22.08.20<strong>07</strong><br />

(86) EP 2005/056300 29.11.2005<br />

(87) WO 2006/058879 2006/23 08.06.2006<br />

(30) 30.11.2004 US 631423 P<br />

30.11.2004 DK 200401863<br />

(54) • NEUARTIGE DIAZABICYCLISCHE ARYL-<br />

DERIVATE ALS CHOLINERGE LIGANDEN<br />

• NOVEL DIAZABICYCLIC ARYL DERIVA-<br />

TIVES AS CHOLINERGY LIGANDS<br />

• NOUVEAUX DERIVES ARYLIQUES DIAZA-<br />

BICYCLIQUES UTILISES EN TANT QUE<br />

LIGANDS CHOLINERGIQUES<br />

(73) NEUROSEARCH A/S, Pederstrupvej 93, 2750<br />

Ballerup, DK<br />

(72) PETERS, Dan, DK-2750 Ballerup, DK<br />

TIMMERMANN, Daniel, B., DK-2750 Ballerup,<br />

DK<br />

OLSEN, Gunnar, M., DK-2750 Ballerup, DK<br />

NIELSEN, Elsebet, Østergaard, DK-2750<br />

Ballerup, DK<br />

JØRGENSEN, Tino, Dyhring, DK-2750 Ballerup,<br />

DK<br />

(74) Abildgren, Michael Padkjaer, et al, Neuro-<br />

Search A/S <strong>Patent</strong> Department 93 Pederstrupvej,<br />

2750 Ballerup, DK<br />

C<strong>07</strong>D 491/04 → (51) C<strong>07</strong>D 401/12<br />

C<strong>07</strong>D 491/04 → (51) C<strong>07</strong>D 471/04<br />

(51) C<strong>07</strong>D 491/14 (11) 1 685 134 B1<br />

A61P 35/00<br />

(25) De (26) De<br />

(21) 03776835.5 (22) 05.11.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 02.08.2006<br />

(86) DE 2003/003702 05.11.2003<br />

(87) WO 2005/044820 2005/20 19.05.2005<br />

(54) • NEUE CHELIDONIN-DERIVATE, VERFAH-<br />

REN ZU IHRER HERSTELLUNG UND IHRE<br />

VERWENDUNG ZUR HERSTELLUNG VON<br />

PHARMAZEUTISCHEN WIRKSTOFFEN<br />

• NOVEL CHELIDONINE DERIVATIVES,<br />

METHODS FOR THE PRODUCTION<br />

THEREOF, AND USE THEREOF FOR PRO-<br />

DUCING PHARMACEUTICAL AGENTS<br />

• NOUVEAUX DERIVES DE CHELIDONINE,<br />

LEUR PROCEDE DE PRODUCTION ET<br />

LEUR UTILISATION POUR PRODUIRE DES<br />

PRINCIPES ACTIFS PHARMACEUTIQUES<br />

(73) Salama, Zoser B. nat.rer.Dr., Ansgarstrasse<br />

13, 13465 Berlin, DE<br />

(72) Salama, Zoser B. nat.rer.Dr., 13465 Berlin,<br />

DE<br />

(74) Boeckh, Tobias, et al, HERTIN Anwaltssozietät<br />

Kurfürstendamm 54/55, 1<strong>07</strong><strong>07</strong> Berlin,<br />

DE<br />

C<strong>07</strong>D 495/04 → (51) C<strong>07</strong>D 401/12<br />

C<strong>07</strong>D 498/04 → (51) C<strong>07</strong>D 471/04<br />

C<strong>07</strong>D 513/04 → (51) C<strong>07</strong>D 401/12<br />

C<strong>07</strong>D 513/04 → (51) C<strong>07</strong>D 471/04<br />

C<strong>07</strong>D 519/00 → (51) C<strong>07</strong>D 471/04<br />

C<strong>07</strong>F 15/00 → (51) C<strong>07</strong>D 221/10

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