Bulletin 2009/07 - European Patent Office
Bulletin 2009/07 - European Patent Office
Bulletin 2009/07 - European Patent Office
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(C<strong>07</strong>D) I.1(1)<br />
(54) • POLYMORPHE FORMEN VON (2S)-(4E)-N-<br />
METHYL-5-(3-ISOPROPOXYPYRIDIN)-[L]-<br />
4-PENTEN-2-AMIN ZUR BEHANDLUNG<br />
VON ERKRANKUNGEN DES ZENTRALEN<br />
NERVENSYSTEMS<br />
• POLYMORPH FORMS OF (2S) - (4E) -N-<br />
METHYL-5- (3-ISOPROPOXYPYRIDIN)<br />
YL]-4-PENTEN-2-AMINE FOR THE TREAT-<br />
MENT OF CENTRAL NERVOUS SYSTEM<br />
DISORDERS<br />
• FORMES POLYMORPHES DE (2S) - (4E)<br />
-N-MÉTHYL-5- (3-ISOPROPOXYPYRI-<br />
DINE) YL¨-4-PENTEN-2-AMINE DESTI-<br />
NÉES AU TRAITEMENT DE TROUBLES DU<br />
SYSTÈME NERVEUX CENTRAL<br />
(71) Targacept, Inc., 200 East First Street, Suite<br />
300, Winston-Salem, NC 27101-4165, US<br />
(72) DULL, Gary, Maurice, Lewisville, NC 27023,<br />
US<br />
MUNOZ, Julio, A., Walnut Cove, NC 27052,<br />
US<br />
(74) Bramley, Sarah Jane, et al, Kilburn & Strode<br />
20 Red Lion Street, London WC1R 4PJ, GB<br />
(51) C<strong>07</strong>D 213/64 (11) 2 021 327 A2*<br />
C<strong>07</strong>C 62/34 C<strong>07</strong>D 3<strong>07</strong>/93<br />
A61K 31/343 C<strong>07</strong>D 333/78<br />
A61K 31/351 C<strong>07</strong>D 405/04<br />
A61K 31/427 C<strong>07</strong>D 4<strong>07</strong>/12<br />
A61K 31/4412 C<strong>07</strong>D 413/12<br />
A61K 31/381 C<strong>07</strong>D 417/12<br />
A61P 1/18<br />
(25) En (26) En<br />
(21) <strong>07</strong>794762.0 (22) 11.05.20<strong>07</strong><br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) US 20<strong>07</strong>/011372 11.05.20<strong>07</strong><br />
(87) WO 20<strong>07</strong>/136573 20<strong>07</strong>/48 29.11.20<strong>07</strong><br />
(88) 27.03.2008<br />
(30) 15.05.2006 US 800542 P<br />
08.08.2006 US 836308 P<br />
(54) • ANTIDIABETISCHE BICYCLISCHE VERBIN-<br />
DUNGEN<br />
• ANTIDIABETIC BICYCLIC COMPOUNDS<br />
• COMPOSÉS BICYCLIQUES ANTIDIABÉTI-<br />
QUES<br />
(71) Merck & Co., Inc., 126 East Lincoln Avenue,<br />
Rahway, NJ <strong>07</strong>065-09<strong>07</strong>, US<br />
(72) GE, Min, Rahway, New Jersey <strong>07</strong>065-09<strong>07</strong>,<br />
US<br />
HE, Jiafang, Rahway, New Jersey <strong>07</strong>065-<br />
09<strong>07</strong>, US<br />
LAU, Fiona Wai Yu, Rahway, New Jersey<br />
<strong>07</strong>065-09<strong>07</strong>, US<br />
LIANG, Gui-Bai, Rahway, New Jersey <strong>07</strong>065-<br />
09<strong>07</strong>, US<br />
LIN, Songnian, Rahway, New Jersey <strong>07</strong>065-<br />
09<strong>07</strong>, US<br />
LIU, Weiguo, Rahway, New Jersey <strong>07</strong>065-<br />
09<strong>07</strong>, US<br />
WALSH, Shawn, P., Rahway, New Jersey<br />
<strong>07</strong>065-09<strong>07</strong>, US<br />
YANG, Lihu, Rahway, New Jersey <strong>07</strong>065-<br />
09<strong>07</strong>, US<br />
(74) Buchan, Gavin MacNicol, Merck & Co., Inc.<br />
<strong>European</strong> <strong>Patent</strong> Department Merck Sharp &<br />
Dohme Limited, Hertford Road, Hoddesdon,<br />
Hertfordshire, EN11 9BU, GB<br />
(51) C<strong>07</strong>D 213/75 (11) 2 021 328 A2*<br />
(25) En (26) En<br />
(21) <strong>07</strong>761921.1 (22) 04.05.20<strong>07</strong><br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
Europäisches <strong>Patent</strong>blatt<br />
<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />
<strong>Bulletin</strong> européen des brevets<br />
(86) US 20<strong>07</strong>/068292 04.05.20<strong>07</strong><br />
(87) WO 20<strong>07</strong>/131201 20<strong>07</strong>/46 15.11.20<strong>07</strong><br />
(88) 06.03.2008<br />
(30) 05.05.2006 US 797949 P<br />
(54) • VERBINDUNGEN UND ZUSAMMENSET-<br />
ZUNGEN ALS HEDGEHOG-WEGMODULA-<br />
TOREN<br />
• COMPOUNDS AND COMPOSITIONS AS<br />
HEDGEHOG PATHWAY MODULATORS<br />
• COMPOSÉS ET COMPOSITIONS MODU-<br />
LANT LE MÉCANISME D'ACTION DE LA<br />
HEDGEHOG<br />
(71) IRM LLC, Hurst Holme, 12 Trott Road,<br />
Hamilton, HM 11, BM<br />
(72) GAO, Wenqi, San Diego, California 92127,<br />
US<br />
JIANG, Jiqing, San Diego, California 92129,<br />
US<br />
WAN, Yongqin, Irvine, California 92612, US<br />
CHENG, Dai, San Diego, California 92126,<br />
US<br />
HAN, Dong, San Diego, California 92014, US<br />
WU, Xu, San Diego, California 92130, US<br />
PAN, Shifeng, San Diego, California 92130,<br />
US<br />
(74) Kiddle, Simon John, et al, Mewburn Ellis LLP<br />
33 Gutter Lane, London EC2V 8AS, GB<br />
C<strong>07</strong>D 215/22 → (51) C<strong>07</strong>D 309/38<br />
C<strong>07</strong>D 233/54 → (51) C08F 4/645<br />
(51) C<strong>07</strong>D 233/90 (11) 2 021 329 A1*<br />
C<strong>07</strong>D 235/16 C<strong>07</strong>D 3<strong>07</strong>/68<br />
C<strong>07</strong>D 401/12 C<strong>07</strong>D 403/12<br />
C<strong>07</strong>D 4<strong>07</strong>/12 A61K 31/4178<br />
A61P 11/00 A61P 25/00<br />
A61P 35/00<br />
(25) En (26) En<br />
(21) <strong>07</strong>760837.0 (22) 18.04.20<strong>07</strong><br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) US 20<strong>07</strong>/066864 18.04.20<strong>07</strong><br />
(87) WO 20<strong>07</strong>/124318 20<strong>07</strong>/44 01.11.20<strong>07</strong><br />
(30) 20.04.2006 US 793694 P<br />
21.12.2006 US 871171 P<br />
(54) • INHIBITOREN VON C-FMS-KINASE<br />
• INHIBITORS OF C-FMS KINASE<br />
• INHIBITEURS DE LA C-FMS KINASE<br />
(71) Janssen Pharmaceutica, N.V., Turnhoutseweg<br />
30, 2340 Beerse, BE<br />
(72) ILLIG, Carl R., Phoenixville, Pennsylvania<br />
19460, US<br />
BALLENTINE, Shelley K., Lansdale, Pennsylvania<br />
19446, US<br />
CHEN, Jinsheng, Exton, Pennsylvania 19341,<br />
US<br />
DESJARLAIS, Renee Louise, Saint Davids,<br />
Pennsylvania 19087, US<br />
MEEGALLA, Sanath K., Boothwyn, Pennsylvania<br />
19061, US<br />
WALL, Mark, Flourtown, Pennsylvania<br />
19031, US<br />
WILSON, Kenneth, Media, Pennsylvania<br />
19063, US<br />
(74) Warner, James Alexander, et al, Carpmaels &<br />
Ransford 43-45 Bloomsbury Square, London<br />
WC1A 2RA, GB<br />
(51) C<strong>07</strong>D 235/08 (11) 2 021 330 A2*<br />
C<strong>07</strong>D 401/06 C<strong>07</strong>D 403/06<br />
A61K 31/4184 A61K 31/4706<br />
A61P 29/00<br />
(25) En (26) En<br />
(21) <strong>07</strong>76<strong>07</strong>46.3 (22) 17.04.20<strong>07</strong><br />
84<br />
Anmeldungen<br />
Applications<br />
Demandes (<strong>07</strong>/<strong>2009</strong>) 11.02.<strong>2009</strong><br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) US 20<strong>07</strong>/066748 17.04.20<strong>07</strong><br />
(87) WO 20<strong>07</strong>/13<strong>07</strong>80 20<strong>07</strong>/46 15.11.20<strong>07</strong><br />
(88) 14.02.2008<br />
(30) 03.05.2006 US 797504 P<br />
(54) • VR1-BENZIMIDAZOLMODULATOREN<br />
• BENZIMIDAZOLE MODULATORS OF VR1<br />
• MODULATEURS DES RÉCEPTEURS VR1<br />
DÉRIVÉS DU BENZIMIDAZOLE<br />
(71) Janssen Pharmaceutica, N.V., Turnhoutseweg<br />
30, 2340 Beerse, BE<br />
(72) CALVO, Raul, L., Royersford, Pennsylvania<br />
09468, US<br />
PLAYER, Mark, R., Phoenixville, Pennsylvania<br />
19460, US<br />
DAX, Scott, L., Landenberg, Pennsylvania<br />
09350, US<br />
PARSONS, William, H., Belle Mead, New<br />
Jersey 08502, US<br />
BRANDT, Michael, Flemington, New Jersey<br />
08822, US<br />
PATEL, Sharmila, Jamison, Pennsylvania<br />
18929, US<br />
LIU, Jian, Manalapan, New Jersey <strong>07</strong>726, US<br />
CHEUNG, Wing, S., Plainsboro, New Jersey<br />
08536, US<br />
JETTER, Michele, C., Norristown, Pennsylvania<br />
19403, US<br />
LEE, Yu-kai, Exton, Pennsylvania 19341, US<br />
YOUNGMAN, Mark, A., Warminster, Pennsylvania<br />
18974, US<br />
PAN, Wenxi, Glenmoore, Pennsylvania<br />
19343, US<br />
WELLS, Kenneth, M., Hillsborough, New<br />
Jersey 08844, US<br />
BEAUCHAMP, Derek, A., Watchung, New<br />
Jersey <strong>07</strong>069, US<br />
(74) Warner, James Alexander, et al, Carpmaels &<br />
Ransford 43-45 Bloomsbury Square, London<br />
WC1A 2RA, GB<br />
C<strong>07</strong>D 235/16 → (51) C<strong>07</strong>D 233/90<br />
C<strong>07</strong>D 239/34 → (51) C<strong>07</strong>D 209/20<br />
C<strong>07</strong>D 239/52 → (51) C<strong>07</strong>D 209/20<br />
C<strong>07</strong>D 239/60 → (51) C<strong>07</strong>D 209/20<br />
C<strong>07</strong>D 249/14 → (51) C<strong>07</strong>C 225/20<br />
C<strong>07</strong>D 261/14 → (51) C<strong>07</strong>D 209/20<br />
C<strong>07</strong>D 271/06 → (51) C<strong>07</strong>D 413/04<br />
C<strong>07</strong>D 271/10 → (51) C<strong>07</strong>D 413/04<br />
(51) C<strong>07</strong>D 271/113 (11) 2 021 331 A1*<br />
C<strong>07</strong>D 413/12 C<strong>07</strong>D 471/08<br />
A61K 31/4245 A61P 25/00<br />
(25) En (26) En<br />
(21) <strong>07</strong>729582.2 (22) 29.05.20<strong>07</strong><br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) EP 20<strong>07</strong>/055159 29.05.20<strong>07</strong><br />
(87) WO 20<strong>07</strong>/138033 20<strong>07</strong>/49 06.12.20<strong>07</strong><br />
(30) 30.05.2006 GB 0610657<br />
05.10.2006 GB 0619710<br />
(54) • 2-PHENYL-5-AMINO-1,3,4-OXADIAZOLE<br />
UND IHRE VERWENDUNG ALS LIGANDEN<br />
AM NIKOTINISCHEN ACETYLCHOLINRE-<br />
ZEPTOR