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Bulletin 2009/07 - European Patent Office

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(C<strong>07</strong>D) I.1(1)<br />

(54) • POLYMORPHE FORMEN VON (2S)-(4E)-N-<br />

METHYL-5-(3-ISOPROPOXYPYRIDIN)-[L]-<br />

4-PENTEN-2-AMIN ZUR BEHANDLUNG<br />

VON ERKRANKUNGEN DES ZENTRALEN<br />

NERVENSYSTEMS<br />

• POLYMORPH FORMS OF (2S) - (4E) -N-<br />

METHYL-5- (3-ISOPROPOXYPYRIDIN)<br />

YL]-4-PENTEN-2-AMINE FOR THE TREAT-<br />

MENT OF CENTRAL NERVOUS SYSTEM<br />

DISORDERS<br />

• FORMES POLYMORPHES DE (2S) - (4E)<br />

-N-MÉTHYL-5- (3-ISOPROPOXYPYRI-<br />

DINE) YL¨-4-PENTEN-2-AMINE DESTI-<br />

NÉES AU TRAITEMENT DE TROUBLES DU<br />

SYSTÈME NERVEUX CENTRAL<br />

(71) Targacept, Inc., 200 East First Street, Suite<br />

300, Winston-Salem, NC 27101-4165, US<br />

(72) DULL, Gary, Maurice, Lewisville, NC 27023,<br />

US<br />

MUNOZ, Julio, A., Walnut Cove, NC 27052,<br />

US<br />

(74) Bramley, Sarah Jane, et al, Kilburn & Strode<br />

20 Red Lion Street, London WC1R 4PJ, GB<br />

(51) C<strong>07</strong>D 213/64 (11) 2 021 327 A2*<br />

C<strong>07</strong>C 62/34 C<strong>07</strong>D 3<strong>07</strong>/93<br />

A61K 31/343 C<strong>07</strong>D 333/78<br />

A61K 31/351 C<strong>07</strong>D 405/04<br />

A61K 31/427 C<strong>07</strong>D 4<strong>07</strong>/12<br />

A61K 31/4412 C<strong>07</strong>D 413/12<br />

A61K 31/381 C<strong>07</strong>D 417/12<br />

A61P 1/18<br />

(25) En (26) En<br />

(21) <strong>07</strong>794762.0 (22) 11.05.20<strong>07</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(86) US 20<strong>07</strong>/011372 11.05.20<strong>07</strong><br />

(87) WO 20<strong>07</strong>/136573 20<strong>07</strong>/48 29.11.20<strong>07</strong><br />

(88) 27.03.2008<br />

(30) 15.05.2006 US 800542 P<br />

08.08.2006 US 836308 P<br />

(54) • ANTIDIABETISCHE BICYCLISCHE VERBIN-<br />

DUNGEN<br />

• ANTIDIABETIC BICYCLIC COMPOUNDS<br />

• COMPOSÉS BICYCLIQUES ANTIDIABÉTI-<br />

QUES<br />

(71) Merck & Co., Inc., 126 East Lincoln Avenue,<br />

Rahway, NJ <strong>07</strong>065-09<strong>07</strong>, US<br />

(72) GE, Min, Rahway, New Jersey <strong>07</strong>065-09<strong>07</strong>,<br />

US<br />

HE, Jiafang, Rahway, New Jersey <strong>07</strong>065-<br />

09<strong>07</strong>, US<br />

LAU, Fiona Wai Yu, Rahway, New Jersey<br />

<strong>07</strong>065-09<strong>07</strong>, US<br />

LIANG, Gui-Bai, Rahway, New Jersey <strong>07</strong>065-<br />

09<strong>07</strong>, US<br />

LIN, Songnian, Rahway, New Jersey <strong>07</strong>065-<br />

09<strong>07</strong>, US<br />

LIU, Weiguo, Rahway, New Jersey <strong>07</strong>065-<br />

09<strong>07</strong>, US<br />

WALSH, Shawn, P., Rahway, New Jersey<br />

<strong>07</strong>065-09<strong>07</strong>, US<br />

YANG, Lihu, Rahway, New Jersey <strong>07</strong>065-<br />

09<strong>07</strong>, US<br />

(74) Buchan, Gavin MacNicol, Merck & Co., Inc.<br />

<strong>European</strong> <strong>Patent</strong> Department Merck Sharp &<br />

Dohme Limited, Hertford Road, Hoddesdon,<br />

Hertfordshire, EN11 9BU, GB<br />

(51) C<strong>07</strong>D 213/75 (11) 2 021 328 A2*<br />

(25) En (26) En<br />

(21) <strong>07</strong>761921.1 (22) 04.05.20<strong>07</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(86) US 20<strong>07</strong>/068292 04.05.20<strong>07</strong><br />

(87) WO 20<strong>07</strong>/131201 20<strong>07</strong>/46 15.11.20<strong>07</strong><br />

(88) 06.03.2008<br />

(30) 05.05.2006 US 797949 P<br />

(54) • VERBINDUNGEN UND ZUSAMMENSET-<br />

ZUNGEN ALS HEDGEHOG-WEGMODULA-<br />

TOREN<br />

• COMPOUNDS AND COMPOSITIONS AS<br />

HEDGEHOG PATHWAY MODULATORS<br />

• COMPOSÉS ET COMPOSITIONS MODU-<br />

LANT LE MÉCANISME D'ACTION DE LA<br />

HEDGEHOG<br />

(71) IRM LLC, Hurst Holme, 12 Trott Road,<br />

Hamilton, HM 11, BM<br />

(72) GAO, Wenqi, San Diego, California 92127,<br />

US<br />

JIANG, Jiqing, San Diego, California 92129,<br />

US<br />

WAN, Yongqin, Irvine, California 92612, US<br />

CHENG, Dai, San Diego, California 92126,<br />

US<br />

HAN, Dong, San Diego, California 92014, US<br />

WU, Xu, San Diego, California 92130, US<br />

PAN, Shifeng, San Diego, California 92130,<br />

US<br />

(74) Kiddle, Simon John, et al, Mewburn Ellis LLP<br />

33 Gutter Lane, London EC2V 8AS, GB<br />

C<strong>07</strong>D 215/22 → (51) C<strong>07</strong>D 309/38<br />

C<strong>07</strong>D 233/54 → (51) C08F 4/645<br />

(51) C<strong>07</strong>D 233/90 (11) 2 021 329 A1*<br />

C<strong>07</strong>D 235/16 C<strong>07</strong>D 3<strong>07</strong>/68<br />

C<strong>07</strong>D 401/12 C<strong>07</strong>D 403/12<br />

C<strong>07</strong>D 4<strong>07</strong>/12 A61K 31/4178<br />

A61P 11/00 A61P 25/00<br />

A61P 35/00<br />

(25) En (26) En<br />

(21) <strong>07</strong>760837.0 (22) 18.04.20<strong>07</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(86) US 20<strong>07</strong>/066864 18.04.20<strong>07</strong><br />

(87) WO 20<strong>07</strong>/124318 20<strong>07</strong>/44 01.11.20<strong>07</strong><br />

(30) 20.04.2006 US 793694 P<br />

21.12.2006 US 871171 P<br />

(54) • INHIBITOREN VON C-FMS-KINASE<br />

• INHIBITORS OF C-FMS KINASE<br />

• INHIBITEURS DE LA C-FMS KINASE<br />

(71) Janssen Pharmaceutica, N.V., Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) ILLIG, Carl R., Phoenixville, Pennsylvania<br />

19460, US<br />

BALLENTINE, Shelley K., Lansdale, Pennsylvania<br />

19446, US<br />

CHEN, Jinsheng, Exton, Pennsylvania 19341,<br />

US<br />

DESJARLAIS, Renee Louise, Saint Davids,<br />

Pennsylvania 19087, US<br />

MEEGALLA, Sanath K., Boothwyn, Pennsylvania<br />

19061, US<br />

WALL, Mark, Flourtown, Pennsylvania<br />

19031, US<br />

WILSON, Kenneth, Media, Pennsylvania<br />

19063, US<br />

(74) Warner, James Alexander, et al, Carpmaels &<br />

Ransford 43-45 Bloomsbury Square, London<br />

WC1A 2RA, GB<br />

(51) C<strong>07</strong>D 235/08 (11) 2 021 330 A2*<br />

C<strong>07</strong>D 401/06 C<strong>07</strong>D 403/06<br />

A61K 31/4184 A61K 31/4706<br />

A61P 29/00<br />

(25) En (26) En<br />

(21) <strong>07</strong>76<strong>07</strong>46.3 (22) 17.04.20<strong>07</strong><br />

84<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>07</strong>/<strong>2009</strong>) 11.02.<strong>2009</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(86) US 20<strong>07</strong>/066748 17.04.20<strong>07</strong><br />

(87) WO 20<strong>07</strong>/13<strong>07</strong>80 20<strong>07</strong>/46 15.11.20<strong>07</strong><br />

(88) 14.02.2008<br />

(30) 03.05.2006 US 797504 P<br />

(54) • VR1-BENZIMIDAZOLMODULATOREN<br />

• BENZIMIDAZOLE MODULATORS OF VR1<br />

• MODULATEURS DES RÉCEPTEURS VR1<br />

DÉRIVÉS DU BENZIMIDAZOLE<br />

(71) Janssen Pharmaceutica, N.V., Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) CALVO, Raul, L., Royersford, Pennsylvania<br />

09468, US<br />

PLAYER, Mark, R., Phoenixville, Pennsylvania<br />

19460, US<br />

DAX, Scott, L., Landenberg, Pennsylvania<br />

09350, US<br />

PARSONS, William, H., Belle Mead, New<br />

Jersey 08502, US<br />

BRANDT, Michael, Flemington, New Jersey<br />

08822, US<br />

PATEL, Sharmila, Jamison, Pennsylvania<br />

18929, US<br />

LIU, Jian, Manalapan, New Jersey <strong>07</strong>726, US<br />

CHEUNG, Wing, S., Plainsboro, New Jersey<br />

08536, US<br />

JETTER, Michele, C., Norristown, Pennsylvania<br />

19403, US<br />

LEE, Yu-kai, Exton, Pennsylvania 19341, US<br />

YOUNGMAN, Mark, A., Warminster, Pennsylvania<br />

18974, US<br />

PAN, Wenxi, Glenmoore, Pennsylvania<br />

19343, US<br />

WELLS, Kenneth, M., Hillsborough, New<br />

Jersey 08844, US<br />

BEAUCHAMP, Derek, A., Watchung, New<br />

Jersey <strong>07</strong>069, US<br />

(74) Warner, James Alexander, et al, Carpmaels &<br />

Ransford 43-45 Bloomsbury Square, London<br />

WC1A 2RA, GB<br />

C<strong>07</strong>D 235/16 → (51) C<strong>07</strong>D 233/90<br />

C<strong>07</strong>D 239/34 → (51) C<strong>07</strong>D 209/20<br />

C<strong>07</strong>D 239/52 → (51) C<strong>07</strong>D 209/20<br />

C<strong>07</strong>D 239/60 → (51) C<strong>07</strong>D 209/20<br />

C<strong>07</strong>D 249/14 → (51) C<strong>07</strong>C 225/20<br />

C<strong>07</strong>D 261/14 → (51) C<strong>07</strong>D 209/20<br />

C<strong>07</strong>D 271/06 → (51) C<strong>07</strong>D 413/04<br />

C<strong>07</strong>D 271/10 → (51) C<strong>07</strong>D 413/04<br />

(51) C<strong>07</strong>D 271/113 (11) 2 021 331 A1*<br />

C<strong>07</strong>D 413/12 C<strong>07</strong>D 471/08<br />

A61K 31/4245 A61P 25/00<br />

(25) En (26) En<br />

(21) <strong>07</strong>729582.2 (22) 29.05.20<strong>07</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(86) EP 20<strong>07</strong>/055159 29.05.20<strong>07</strong><br />

(87) WO 20<strong>07</strong>/138033 20<strong>07</strong>/49 06.12.20<strong>07</strong><br />

(30) 30.05.2006 GB 0610657<br />

05.10.2006 GB 0619710<br />

(54) • 2-PHENYL-5-AMINO-1,3,4-OXADIAZOLE<br />

UND IHRE VERWENDUNG ALS LIGANDEN<br />

AM NIKOTINISCHEN ACETYLCHOLINRE-<br />

ZEPTOR

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