Bulletin 2009/07 - European Patent Office
Bulletin 2009/07 - European Patent Office
Bulletin 2009/07 - European Patent Office
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(C<strong>07</strong>D) I.1(1)<br />
• 2-PHENYL-5-AMINO-1,3,4-OXADIAZOLES<br />
AND THEIR USE AS NICOTINIC ACETYL-<br />
CHOLINE RECEPTOR LIGANDS<br />
• 2-PHÉNYL-5-AMINO-1,3,4-OXADIAZOLES<br />
ET UTILISATION DE CEUX-CI EN TANT<br />
QUE LIGANDS DU RÉCEPTEUR NICOTI-<br />
NIQUE DE L'ACÉTYLCHOLINE<br />
(71) GLAXO GROUP LIMITED, Glaxo Wellcome<br />
House, Berkeley Avenue, Greenford, Middlesex<br />
UB6 0NN, GB<br />
(72) COPPO, Frank, TeenGlaxoSmithKline, P.o.<br />
Box 5089 Collegeville, Pennsylvania 19426,<br />
US<br />
MASKELL, Emma, S. L.GlaxoSmithKline,<br />
Third Avenue Harlow Essex CM19 5AW, GB<br />
REDSHAW, SallyGlaxoSmithKline, Third<br />
AvenueHarlow Essex CM19 5AW, GB<br />
SKIDMORE, JohnGlaxoSmithKline, Third<br />
Avenue Harlow Essex CM19 5AW, GB<br />
WARD, Robert, WilliamGlaxoSmithKline,<br />
Third Avenue Harlow Essex CM19 5AW, GB<br />
WILSON, David, Matthew, Third Avenue<br />
Harlow Essex CM19 5AW, GB<br />
(74) Goddard, Carolyn Janice, GlaxoSmithKline<br />
Corporate Intellectual Property (CN925.1)<br />
980 Great West Road Brentford, Middlesex<br />
TW8 9GS, GB<br />
C<strong>07</strong>D 277/64 → (51) C<strong>07</strong>C 225/20<br />
C<strong>07</strong>D 285/06 → (51) C<strong>07</strong>C 225/20<br />
(51) C<strong>07</strong>D 3<strong>07</strong>/68 (11) 2 021 332 A2*<br />
C08G 75/00 G02F 1/361<br />
(25) En (26) En<br />
(21) <strong>07</strong>794377.7 (22) 24.04.20<strong>07</strong><br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) US 20<strong>07</strong>/010123 24.04.20<strong>07</strong><br />
(87) WO 20<strong>07</strong>/133414 20<strong>07</strong>/47 22.11.20<strong>07</strong><br />
(88) 22.05.2008<br />
(30) 03.05.2006 US 418101<br />
(54) • MERCAPTOFUNKTIONELLE HIGH-MU-<br />
BETA-EO-CHROMOPHORE UND KOVA-<br />
LENT GEBUNDENE HIGH-TG-POLYMERE<br />
MIT GERINGEM OPTISCHEN VERLUST<br />
MIT DIESEN CHROMOPHOREN SOWIE<br />
VERFAHREN ZUR SYNTHETISIERUNG<br />
VON EO-MATERIALIEN<br />
• MERCAPTOFUNCTIONAL HIGH "MU-BETA"<br />
EO CHROMOPHORES AND HIGH TG, LOW<br />
OPTICAL LOSS, COVALENTLY BONDED,<br />
POLYMERS CONTAINING SAID CHROMO-<br />
PHORES AND METHODS OF SYNTHESIZ-<br />
ING EO MATERIALS<br />
• CHROMOPHORES À BASE D'EO, DE UB<br />
ÉLEVÉ ET À FONCTION MERCAPTO ET<br />
POLYMÈRES CONTENANT DES CHROMO-<br />
PHORES À BASE D'EO, DE UB ÉLEVÉ, LIÉS<br />
DE MANIÈRE COVALENTE, DE FAIBLE<br />
PERTE OPTIQUE ET DE TV ÉLEVÉE ET<br />
PROCÉDÉS DE SYNTHÈSE DE MATÉRIAUX<br />
À BASE D'EO<br />
(71) Corning Incorporated, 1 Riverfront Plaza,<br />
Corning NY 14831, US<br />
(72) HE, Mingqian, Horseheads, New York 14845,<br />
US<br />
WANG, Jianguo, Horseheads, NY 14845, US<br />
(74) Marchant, James Ian, Elkington and Fife LLP<br />
Prospect House 8 Pembroke Road, Sevenoaks,<br />
Kent TN13 1XR, GB<br />
C<strong>07</strong>D 3<strong>07</strong>/68 → (51) C<strong>07</strong>D 233/90<br />
C<strong>07</strong>D 3<strong>07</strong>/93 → (51) C<strong>07</strong>D 213/64<br />
Europäisches <strong>Patent</strong>blatt<br />
<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />
<strong>Bulletin</strong> européen des brevets<br />
(51) C<strong>07</strong>D 309/38 (11) 2 021 333 A2*<br />
C<strong>07</strong>D 215/22 C<strong>07</strong>D 405/12<br />
C<strong>07</strong>D 4<strong>07</strong>/12 A61K 31/4704<br />
A61K 31/352<br />
(25) En (26) En<br />
(21) <strong>07</strong>789580.3 (22) 22.05.20<strong>07</strong><br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) IB 20<strong>07</strong>/002179 22.05.20<strong>07</strong><br />
(87) WO 20<strong>07</strong>/135565 20<strong>07</strong>/48 29.11.20<strong>07</strong><br />
(88) 03.04.2008<br />
(30) 22.05.2006 EP 06290821<br />
(54) • PROLIFERATIONSHEMMENDE VERBIN-<br />
DUNGEN AUS EINEM 3-ARYL-COUMARIN<br />
ODER EINEM 3-ARYL-CHINOLIN-2-ON<br />
UND ANWENDUNGEN DAVON<br />
• ANTI-PROLIFERATIVE COMPOUNDS<br />
DERIVING FROM A 3-ARYL-COUMARINE<br />
OR 3-ARYL-QUINOLIN-2-ONE AND USES<br />
THEREOF<br />
• COMPOSÉS ANTIPROLIFÉRATIFS DÉRI-<br />
VÉS DE LA 3-ARYL-COUMARINE OU DE<br />
LA 3-ARYL-QUINOLIN-2-ONE ET LEUR<br />
UTILISATIONS<br />
(71) EOS - Ethical Oncology Science S.p.A., Via<br />
Monte di Pietà, 1/A, 20121 Milano, IT<br />
(72) SCHAPIRA, Matthieu, F-69001 Lyon, FR<br />
LAMIGEON, Cyrille, F-69800 Saint Priest, FR<br />
GUTMANN, Mathieu, F-69004 Lyon, FR<br />
BARTHELAIX, Audrey, F-69009 Lyon, FR<br />
HUGO, Nicolas, F-69001 Lyon, FR<br />
COLAS, Pierre, F-69370 St Didier au Mont<br />
d'Or, FR<br />
(74) Minoja, Fabrizio, Bianchetti Bracco Minoja S.<br />
r.l. Via Plinio, 63, 20129 Milano, IT<br />
C<strong>07</strong>D 311/72 → (51) C<strong>07</strong>C 59/62<br />
C<strong>07</strong>D 311/94 → (51) G02B 5/23<br />
C<strong>07</strong>D 333/20 → (51) C<strong>07</strong>C 225/20<br />
C<strong>07</strong>D 333/78 → (51) C<strong>07</strong>D 213/64<br />
C<strong>07</strong>D 401/04 → (51) C<strong>07</strong>D 413/04<br />
(51) C<strong>07</strong>D 401/06 (11) 2 021 334 A1*<br />
C<strong>07</strong>D 2<strong>07</strong>/28 C<strong>07</strong>K 5/06<br />
A61K 31/4015 A61K 31/4425<br />
(25) En (26) En<br />
(21) <strong>07</strong>728359.6 (22) 20.04.20<strong>07</strong><br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) EP 20<strong>07</strong>/053900 20.04.20<strong>07</strong><br />
(87) WO 20<strong>07</strong>/122199 20<strong>07</strong>/44 01.11.20<strong>07</strong><br />
(30) 20.04.2006 EP 06380090<br />
(54) • SYNTHESE UND ANWENDUNGEN VON<br />
PYROGLUTAMINSÄUREDERIVATEN<br />
• SYNTHESIS AND USES OF PYROGLUTA-<br />
MIC ACID DERIVATIVES<br />
• SYNTHÈSE ET UTILISATIONS DE DÉRIVÉS<br />
D'ACIDE PYROGLUTAMIQUE<br />
(71) Prodimed, S.A., Guzman el Bueno 74, 28003<br />
Madrid, ES<br />
(72) Álvarez Builla Gomez, Julio, 28033 Madrid,<br />
ES<br />
Novella Robisco, José Luis, 28045 Madrid,<br />
ES<br />
Matia Martin, Mª Paz, 28005 Madrid, ES<br />
Serna Pereda, Sonia, 48015 Bilbao, ES<br />
(74) ABG <strong>Patent</strong>es, S.L., Avenida de Burgos 16D<br />
Edificio Euromor, 28036 Madrid, ES<br />
85<br />
Anmeldungen<br />
Applications<br />
Demandes (<strong>07</strong>/<strong>2009</strong>) 11.02.<strong>2009</strong><br />
C<strong>07</strong>D 401/06 → (51) C<strong>07</strong>D 235/08<br />
(51) C<strong>07</strong>D 401/12 (11) 2 021 335 A1*<br />
C<strong>07</strong>D 403/12 A61K 31/454<br />
A61K 31/513 A61K 31/54<br />
A61P 29/00 A61P 35/00<br />
A61P 9/00 A61P 11/00<br />
A61P 19/00 C<strong>07</strong>D 401/14<br />
C<strong>07</strong>D 4<strong>07</strong>/12 C<strong>07</strong>D 4<strong>07</strong>/14<br />
C<strong>07</strong>D 417/12 C<strong>07</strong>D 417/14<br />
(25) En (26) En<br />
(21) <strong>07</strong>760833.9 (22) 18.04.20<strong>07</strong><br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) US 20<strong>07</strong>/066860 18.04.20<strong>07</strong><br />
(87) WO 20<strong>07</strong>/124316 20<strong>07</strong>/44 01.11.20<strong>07</strong><br />
(30) 20.04.2006 US 793697 P<br />
05.01.20<strong>07</strong> US 883539 P<br />
(54) • HETEROCYCLISCHE VERBINDUNGEN ALS<br />
C-FMS-KINASEHEMMER<br />
• HETEROCYCLIC COMPOUNDS AS INHIBI-<br />
TORS OF C-FMS KINASE<br />
• COMPOSÉS HÉTÉROCYCLIQUES INHIBI-<br />
TEURS DE C-FMS KINASE<br />
(71) Janssen Pharmaceutica, N.V., Turnhoutseweg<br />
30, 2340 Beerse, BE<br />
(72) ILLIG, Carl R., Phoenixville, Pennsylvania<br />
19460, US<br />
BALLENTINE, Shelley K., Lansdale, Pennsylvania<br />
19446, US<br />
CHEN, Jinsheng, Exton, Pennsylvania 19341,<br />
US<br />
DESJARLAIS, Renee Louise, Saint Davids,<br />
Pennsylvania 19087, US<br />
MEEGALLA, Sanath K., Boothwyn, Pennsylvania<br />
19061, US<br />
WALL, Mark, Flourtown, Pennsylvania<br />
19031, US<br />
WILSON, Kenneth, Media, Pennsylvania<br />
19063, US<br />
(74) Warner, James Alexander, et al, Carpmaels &<br />
Ransford 43-45 Bloomsbury Square, London<br />
WC1A 2RA, GB<br />
(51) C<strong>07</strong>D 401/12 (11) 2 021 336 A2*<br />
C<strong>07</strong>D 2<strong>07</strong>/26 A61K 31/4015<br />
A61K 31/4025 A61P 3/10<br />
C<strong>07</strong>D 2<strong>07</strong>/50<br />
(25) En (26) En<br />
(21) <strong>07</strong>761091.3 (22) 23.04.20<strong>07</strong><br />
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />
GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />
RO SE SI SK TR<br />
AL BA HR MK RS<br />
(86) US 20<strong>07</strong>/067182 23.04.20<strong>07</strong><br />
(87) WO 20<strong>07</strong>/127688 20<strong>07</strong>/45 08.11.20<strong>07</strong><br />
(88) 21.12.20<strong>07</strong><br />
(30) 24.04.2006 US 745475 P<br />
(54) • 11-BETA-HYDROXYSTEROID-DEHYDRO-<br />
GENASE-1-HEMMER<br />
• INHIBITORS OF 11-BETA-HYDROXYSTER-<br />
OID DEHYDROGENASE 1<br />
• INHIBITEURS DE 1-BETA-HYDROXYSTÉ-<br />
ROÏDE DÉSHYDROGENASE 1<br />
(71) ELI LILLY AND COMPANY, Lilly Corporate<br />
Center, Indianapolis IN 46285, US<br />
(72) BUSH, Julie Kay, McCordsville, Indiana<br />
46055, US<br />
HANSEN, Marvin Martin, Indianapolis, Indiana<br />
46227, US<br />
LI, Renhua, Fishers, Indiana 46038, US<br />
MABRY, Thomas, Edward, Indianapolis,<br />
Indiana 46280, US<br />
SNYDER, Nancy June, Lizton, Indiana<br />
46149, US