Part – B Studies on isatin derivatives….. 258 A. A. Esmaeili, S. Amini and A. Bodaghi; Synlett, 2007, 9, 1452. 259 R. K. Tiwari, N. Rastogi, R. Sethi and S. Shukla; J. Ind. Chem. Soc., 2008, 85, 85. 260 O. Bekircan and H. Bektas; Molecules, 2008, 13, 2126. 261 V. Glover, J. M. Halket, P. J. Watkins, A. Clow, B. L. Goddwin and M. J. Sandler; Neurochemistry, 1988, 51, 656. 262 J. Seidel and J. Wenzel; Pol. J. Pharmacol., 1979, 35, 407. 263 I. M. Mc Intyre and T. R. Norman; J. Neural Transm., 1990, 79, 35. 264 F. D. Popp and B. E. Donigan; J. Pharm. Sci., 1979, 68, 519. 265 H. Pajouhesh, R. Parson and F. D. Popp; J. Pharm. Sci., 1983, 72, 318. 266 M. Rajopadhye and F. D. Popp; J. Het. Chem., 1984, 21, 289. 267 F. D. Popp; J. Het. Chem., 1984, 21, 1641. 268 S. K. Bhattacharya; Biog. Amines, 1988, 14, 131. 269 T. Blackburn, K. Paul and G. Smith; G.B. Pat. 9, 425, 012, 1993. (CA 122:72046e) 270 N. Karali and A. Gursoy; Farmaco, 1994, 49, 819. 271 N. Karali, G. Capan and C. N. Ergen; Sci. Pharm., 1997, 65, 277. 272 G. Galambos, B. Kiss and E. Palosi; Hun. Pat. 65, 452, 1994. (CA 123:169529y) 273 R. Jain and Bansal; Pharmazie, 1995, 50, 224. 274 A. Gursoy and N. Karali; Farmaco, 1996, 51, 437. 275 A. Ghaney and A. El-Helby; J. Pharm. Sci., 1996, 36, 343. 276 C. David, T. Marie and G. Roussel; U.S. Pat. 5, 498, 716, 12, 1996. (CA 124:343271r) 277 S. E. Smith, C. M. Man, P. K. Yip, E. Jang, A. G. Chapman and B. S. Meldrum; Br. J. Pharmacol., 1996, 119, 165. 278 J. A. Alabadi, J. L. Thibault, E. Pinard, J. Seylaz and F. Lasbennes; Brain Res., 1999, 839, 305. 279 R. Di Fabio, A. M. Capelli, N. Conti, A. Cugola, D. Donati, A. Feriani, G. Gastaldi, G. Gaviraghi, C. T. Hewkin, F. Micheli, A. Missio, M. Mugnaini, A. Pecunioso, A. M. Quaglia, E. Ratti, L. Rossi, G. Tedesco, D. G. Trist and A. Reggiani; J. Med. Chem., 1997, 40, 841. 280 H. P. Olesen and A. Kanstrup, Den. Pat. 97, 05, 137, 1997. (CA 126:212050m) 281 O. A. Sharaf; Bull. Fac. Pharm., 1997, 35, 79. 282 N. L. Reddy, M. Maillard, D. Berlove, M. David, D. Sharad and J. Graham; U.S. Pat. 9, 730, 054, 1997. (CA 127:234258h) 283 G. S. Singh, T. Singh and R. Lakhan; Indian J. Chem., 1997, 36B, 951. 284 S. K. Bhattacharya and A. Chakraborti; Indian. J. Exp. Biol., 1998, 36, 118. 285 Y. Evanno, M. Sevrin, C. Maloizel, O. Legalbudec and P. George; Fr. Pat. 9, 815, 552, 1998. (CA 128:282832h) 286 K. P. Jakobsen, F. P. Anders, H. P. Olesan, B. Lundbech and M. Jane; U.S. Pat. 5, 783, 575, 1998. (CA 129:148909f) Department of Chemistry, <strong>Saurashtra</strong> <strong>University</strong>, Rajkot-360 005 143
Part – B Studies on isatin derivatives….. 287 F. Li, W. Yue, M. Minanii, J. Zhang and Z. Liu; Yaoxue Xuebao, 1999, 34, 1. (CA 131:82850n) 288 Y. Evanno, L. Dubois, M. Sevrin, F. Marguet, J. Proissant, R. Bartsch and C. Gille; Fr. Pat. 9, 906, 406, 1999. (CA 130:168385f) 289 S. K. Srivastava, S. Srivastava and S. D. Srivastava; Indian J. Chem., 1999, 38B, 183. 290 S. N. Pandeya, I. Ponnilavarasan, A. Pandey, R. Lakhan and J. P. Stables; Pharmazie, 1999, 54, 12. 291 S. N. Pandeya, S. Smitha and J. P. Stables; Arch. Pharm. Pharm. Med. Chem., 2002, 4, 129. 292 S. N. Pandeya, A. Senthil Raja and J. P. Stables; J. Pharm. Pharm. Sci., 2002, 5, 266. 293 S. N. Pandeya, A. K. Agarwal, A. Singh and J. P. Stables; Acta Pharm., 2003, 53, 15. 294 M. Verma, S. N. Pandeya, K. Singh and J. P. Stables; Acta Pharm., 2004, 54, 49. 295 V. Shindikar, F. Khan and C. L. Viswanathan; Eur. J. Med. Chem., 2006, 41, 786. 296 K. C. Joshi, V. N. Pathak and P. Chand; J. fuer Prakt. Chemie, 1980, 322 (2), 314. 297 E. Medvedev, A. Goodwin, A. Clow, J. Halket, V. Glover and M. Sandler; Biochem. Pharmacol., 1992, 44, 590. 298 G. Palit, R. Kumar, G. K. Patnaik and S. K. Bhattacharya; Biogenic Amines, 1997, 13, 131. 299 M. Sarangapani and V. M. Reddy; Indian. J. Pharm. Sci., 1997, 59, 105. 300 L. Kennis, M. J. Edmund and C. Josephus; Bel. Pat. 9, 744, 040, 1997. (CA 28:34772e) 301 N. Hamaue, N. Yamazaki, M. Minami, T. Endo, M. Hirafugi, Y. Monma, H. Jogashi, H. Saito and S. H. Parvez; Biogenic Amines, 1999, 15, 367. 302 Y. Tozawa and A. Veki; Biochem. Pharmacol., 1998, 56, 1041. 303 R. S. Varma and W. L. Nobles; J. Med. Chem., 1967, 10, 510. 304 M. Kupinić, M. Medić-Šarić, M. Movrin and D. Maysinger; J. Pharm. Sci., 1979, 68, 459. 305 D. Maysinger, J. Ban and M. Movrin; Arzneim. Forsch., 1980, 30, 932. 306 R. W. Daisley and V. K. Shah; J. Pharm. Sci., 1984, 73, 407. 307 S. Dilber, M. Saban, A. Gelinco, L. Arsenijević, M. Bogavac and S. Pavlov; Pharmazie, 1990, 45, 800. 308 Y. Teitz, D. Ronen, A. Vansover, T. Stematsky and J. L. Riggs; Antiviral Res., 1994, 24, 305. 309 V. P. Joseph, M. Hollaway, G. Katharine and P. James; Eur. Pat. 617, 968, 05, 1994. (CA 123:198639q) 310 W. M. Foye, T. L. Lamke and D. A. Williams; Principles of Medicinal Chemistry, 4th ed., Weverly Publishers, New Delhi 1995, pp. 855. 311 F. Britcher and L. Susan; U.K. Pat. 2, 282, 808, 1995. (CA 123:143634d) Department of Chemistry, <strong>Saurashtra</strong> <strong>University</strong>, Rajkot-360 005 144
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Saurashtra University Re - Accredit
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Statement under O. Ph. D. 7 of Saur
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ACKNOWLEDGEMENT It is a moment of g
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Jignesh Lunagariya, Hitesh Sarvaiya
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CONTENT Content General Remarks 6 A
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Content 3.2 Reaction scheme 149 3.3
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MF Molecular Formula MW Molecular W
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GABA Gamma Amino Butyric Acid MES M
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PART - A STUDIES ON 2-METHYL INDOLI
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Conferences / Seminar / Workshop At