Chapter – 5 Synthesis and Characterization….. 5.16 REFERENCES 1 R. Anschutz; Liebigs Ann. Chem., 1909, 367, 204. 2 S. Checchi, L. P. Vettori and M. B. Alberti; Gazz. Chim. Ital., 1967, 97, 1749. 3 V. A. Zagorevskii and N. V. Dudykina; Zh. Obshch. Khim., 1962, 32, 2384. 4 D. P. Spalding, H. S. Mosher and F. C. Whitemore; J. Am. Chem. Soc., 1950, 72, 5338. 5 O. H. Hismat, A. K. M. Gohar, M. R. Shahlash and I. Ismail; Pharm. Acta. Helv., 1977, 52, 252. 6 V. A. Zagorevskii, V. L. Savel’ev and N. V. Dudykina; Zh. Org. Khim., 1968, 4, 2041. (CA 70:28767z) 7 V. A. Zagorevskii, V. L. Savelév and L. M. Meshcheriakova; Khim. Geterotsikl. Soedin., 1970, 8, 1019. (CA 74:76279c) 8 H. Harnisch and A. Brack; CA 88:106760e. 9 K. Tabaković, I. Tabaković, N. Ajdini and O. Leci; Synthesis, 1987, 3, 308. 10 A. Mustafa, O. H. Hishmat, M. I. Ali, M. E. Wassef, E. M. Khalil and A. K. M. Gohar; Justus Liebigs Annalen der Chemie, 1968, 712, 107. 11 O. S. Wolfbeis; Monatshefte fuer Chemie, 1977, 108(3), 499. 12 K. Tabaković, I. Tabaković, M. Trkovnik, A. Jurić and N. Trinajstić; J. Het. Chem., 1980, 17(4), 801. 13 J. L. Asherson, O. Bilgic and D. W. Young; J. Chem. Soc., Perk. Trans., 1980, 2, 522. 14 G. M. Conlin and J. R. Gear; J. Nat. Prod., 1993, 56(8), 1402. 15 Z. Stunic, M. Trkovnik, M. Lacan and R. J. Jankovic; J. Het. Chem., 1981, 18, 511. 16 N. S. Bhatt; Ph. D. Thesis, <strong>Saurashtra</strong> <strong>University</strong>, 1983. 17 S. D. Joshi, V. D. Sakhardance and S. Sheshadri; Ind. J. Chem., 1984, 23B, 206. 18 T. Berghaus; Ph. D. Thesis, <strong>University</strong> of Keli, 1989. 19 S. B. Reddy and M. Darbarwar; J. Ind. Chem. Soc., 1985, 62(5), 377. 20 M. M. Bardan, A. K. El Ansari and S. El Meligie; Revue Roumaine de Chimie, 1990, 35(6), 777. 21 C. Ivanov, S. K. Karaziosov and I. Manolov; Arch. Pharm., 1991, 324, 61. 22 M. A. Kirpichenok, L. Yu. Fomina and I. I. Grandberg; Khimiya Geterotsiklicheskikh Soedinenii, 1991, 5, 609. 23 K. Tabaković, and I. Tabaković, J. Het. Chem., 1992, 29, 383. 24 M. Hamdi, O. Grech, R. Sakellariou and V. Spéziale; J. Het. Chem., 1994, 31(2), 509. 25 I. Papousis, S. Spyroudis and A. Varvoglis; J. Het. Chem., 1996, 33(3), 579. 26 M. Hamdi, S. Cottet, C. Tedeschi and V. Speziale; J. Het. Chem., 1997, 34, 1821. 27 A. Sabatié, D. Végh, A. Loupy and Ľ. Floch; ARKIVOC, 2001, (vi), 122. 28 M. Kováč, A. Sabatié and Ľ. Floch; ARKIVOC, 2001, (vi), 100. 29 E. V. Stoyanov and I. C. Ivanov; Molecules, 2004, 9(8), 627. Department of Chemistry, <strong>Saurashtra</strong> <strong>University</strong>, Rajkot – 360 005 323
Chapter – 5 Synthesis and Characterization….. 30 S. S. Soman; Ind. J. Chem., 2004, 43B (3), 624. 31 A. P. Chavan; J. Chem. Res., 2006, 3, 179. 32 V. Shcherbakov, Y. V. Burgart, V. I. Saloutin and O. N. Chupakhin; Heterocycles, 2006, 69, 319. 33 V. Shcherbakov, Y. V. Burgart and V. I. Saloutin; Russ. Chem. Bull., 2006, 55(7), 1215. 34 T. Ghosh, R. K. Sur and C. Bandyopadhyay; J. Chem. Res., 2006, 10, 651. 35 O. G. Ganina, I. S. Veselov, G. V. Grishina, A. Yu. Fedorov and I. P. Beletskaya; Russ. Chem. Bull., 2006, 55(9), 1642. 36 I. Strakova, M. Petrova and A. Strakov; Latvijas Kimijas Zurnals, 2006, 4, 345. 37 L. Zhang, T. Meng, R. Fan, and J. Wu; J. Org. Chem. 2007, 72, 7279. 38 K. Haruo and I. Ruchiro; Yakugagu Zassi, 1983, 83, 1169. 39 G. L. Bechmann; CA 76:72404. 40 S. Govori, V. Rapic, O. Leci, M. Cacic and I. Tobaković; J. Het. Chem., 1996, 33, 351. 41 D. Leurquin; CA 82:72791z. 42 V. A. Zagorevskii and V. L. Savelév; CA 80:36999. 43 V. A. Zagorevskii and V. L. Savelév; Khim. Farm. Zh., 1975, 9, 10. 44 T. G. Zagorevskii; Khim. Geterotsikl. Soedin, 1982, 7, 896. 45 M. M. Bardan, A. K. El Ansari and S. El Meligie; Egypt. J. Pharma. Sci., 1989, 30(1- 4), 379. 46 A. J. Barker; EP 602 851, 1993. 47 Osherov and A. Levitzki; Eur. J. Biochem., 1994, 225, 1947. 48 D. Thaker; Ph. D. Thesis, <strong>Saurashtra</strong> <strong>University</strong>, 1996. 49 B. Desai; Ph. D. Thesis, <strong>Saurashtra</strong> <strong>University</strong>, 2000. 50 V. Vora; Ph. D. Thesis, <strong>Saurashtra</strong> <strong>University</strong>, 2000. 51 A. Parecha; Ph. D. Thesis, <strong>Saurashtra</strong> <strong>University</strong>, 2002. 52 G. Patel; Ph. D. Thesis, <strong>Saurashtra</strong> <strong>University</strong>, 2002. 53 K. Dholaria; Ph. D. Thesis, <strong>Saurashtra</strong> <strong>University</strong>, 2002. 54 M. G. Popovic, S. E. Read and R. C. Gallo; Detection, Isolation and continuous production of cytopathic rretroviruses (HTLV-III) from patients with AIDS and pre- AIDS, Science, 1984, 224, 497. 55 F. Clavel, M. Guyaer, D. Guetard, M. Salle, L. Montagnier and H. Alizon; Molecular cloning and polymorphism of the human immunodeficiency virus type 2, Nature, 1986, 324, 691. 56 N. Hamdi, C. Lidrissi, M. Saoud, R. A. Nievas and H. Zarrouk; Chem. Het. Compds., 2006, 42(3), 320. 57 M. D. Braccio, G. Grossi, G. Roma, C. Marzano, F. Baccichetti, M. Simonato and F. Bordin; Farmaco, 2003, 58(11), 1083. 58 M. Chavda, A. Shah, S. Bhatt, K. Deo and P. Kundu, Ind. J. Chem., 2003, 42B (6), 1502. Department of Chemistry, <strong>Saurashtra</strong> <strong>University</strong>, Rajkot – 360 005 324
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ACKNOWLEDGEMENT It is a moment of g
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Jignesh Lunagariya, Hitesh Sarvaiya
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CONTENT Content General Remarks 6 A
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Content 3.2 Reaction scheme 149 3.3
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MF Molecular Formula MW Molecular W
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GABA Gamma Amino Butyric Acid MES M
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