Part – B Studies on isatin derivatives….. 312 M. Artico, S. Marsa, L. Romano, G. Anna, A. Demontis and P. Lacella; Ital. Pat. 96, 33, 171, 1995. (CA 126:187187e) 313 S. E. Webber, J. Tikhe, S. T. Worland, S. A. Fuhrman, T. F. Hendrickson, D. A. Mathews, R. A. Love and A. K. Patick; J. Med. Chem., 1996, 39, 5072. 314 S. N. Pandeya and D. Sriram; Acta. Pharm. Turc., 1998, 40, 33. 315 S. N. Pandeya, P. Yogeeswari, D. Sriram and G. Nath; Boll. Chim. Farm., 1998, 137, 321. 316 S. N. Pandeya, C. Gnana Sundari, M. Mariammal, M. Saravanan, P. Saravana Balaji, S. Senthil Kumar and D. Sriram; Indian J. Pharm. Sci., 1998, 60, 280. 317 S. N. Pandeya, D. Sriram, G. Nath and E. De Clercq; Eur. J. Pharm. Sci., 1999, 9, 25. 318 S. N. Pandeya, D. Sriram, G. Nath and E. De Clercq; Indian J. Pharm. Sci., 1999, 61, 358. 319 S. N. Pandeya, D. Sriram, G. Nath and E. De Clercq; Pharm. Acta Helv., 1999, 74, 11. 320 S. N. Pandeya, D. Sriram, G. Nath and E. De Clercq; Arzneim. Forsch., 2000, 50, 55. 321 S. N. Pandeya, D. Sriram, G. Nath and E. De Clercq; Eur. J. Med. Chem., 2000, 35, 249. 322 Z. H. Chohan, H. Pervez, A. Rauf, K. M. Khan, C. T. Supuran; J. Enz. Inhib. and Med. Chem., 2004, 19 (5), 417. 323 M. T. Makhija, R. T. Kasliwal, V. M. Kulkarni and N. Neamati; Bioorg. & Med. Chem., 2004, 12, 2317. 324 P. S. Bhasin, N. Sachdeva, S. N. Pandeya, G. Nath and S. K. Singh; Acta Pharma. Tur., 2005, 47, 21. 325 D. Sriram, T. Ratan Bal, P. Yogeeswari; J. Pharm Pharmaceut Sci., 2005, 8(3), 565. 326 V. Ravichandran, S. Mohan and K. Suresh Kumar; Arkivoc, 2007, XIV, 51. 327 A. Jarrahpour, D. Khalili, E. De Clercq, C. Salmi and J. M. Brunel; Molecules, 2007, 12, 1720. 328 A. M. Vijey, G. Shiny and V. Vaidhyalingam; Arkivoc, 2008, XI, 187. 329 W. C. Cheah, D. StC Black, W. K. Goh, Naresh Kumar; Tet. Lett., 2008, 49, 2965. 330 D. Popp and H. Pajouhesh; J. Pharm. Sci., 1983, 72, 318. 331 N. H. Eshbha and H. M. Salama; Pharmazie, 1985, 40, 320. 332 M. Rajopadhye, F. D. Popp, J. Het. Chem., 1987, 24, 1637. 333 Y. Teitz, E. Ladizensky, N. Barko and E. Burstein; Antimicrob. Agents Chem. Ther., 1993, 37, 2483. 334 A. Broadbent, H. Thomas and S. Broadbent; Curr. Med. Chem., 1998, 5, 469. 335 P. Yogeeswari, D. Sriram, R. Kavya, S. Tiwari; Biomed. & Pharmaco., 2005, 59, 501. 336 A. Beauchard, Y. Ferandin, S. Frère, O. Lozach, M. Blairvacq, L. Meijer, V. Thiéry and T. Besson; Bioorg. & Med. Chem., 2006, 14, 6434. 337 K. L. Vine, J. M. Locke, M. Ranson, S. G. Pyne and J. B. Bremner; Bioorg. & Med. Chem., 2007, 15, 931. Department of Chemistry, <strong>Saurashtra</strong> <strong>University</strong>, Rajkot-360 005 145
Part – B Studies on isatin derivatives….. 338 C.-Y. Hung, M.-H. Hsu, L.-J. Huang, C.-S. Hwang, O. Lee, C.-Y. Wu, C.-H. Chen and S.-C. Kuo; Bioorg. & Med. Chem., 2008, 16, 4222. 339 L. Matesic, J. M. Locke, J. B. Bremner, S. G. Pyne, D. Skropeta, M. Ranson and K. L. Vine; Bioorg. & Med. Chem., 2008, 16, 3118. 340 M. P. Sathisha, V. K. Revankar and K. S. R. Pai; Metal-Based Drugs, 2008, 362105. 341 I. Chiyanzu, E. Hansell, J. Gut, P. J. Rosenthal, J. H. McKerrow and K. Chibale; Bioorg. & Med. Chem. Lett., 2003, 13, 3527. 342 I. Chiyanzu, C. Clarkson, P. J. Smith, J. Lehman, J. Gut, P. J. Rosenthal and K. Chibale; Bioorg. & Med. Chem., 2005, 13, 3249. 343 R. S. Varma and R. K. Pandeya; Indian J. Pharm. Sci., 1982, 46, 132. 344 J. Collino and S. Volpe; Ital. Boll. Chim. Farm., 1982, 121, 408. 345 J. Ramachandran; Swed. Pat. 9, 944, 608, 1998. (CA 131:209113g) 346 L. Gargari, R. C. Bansal, K. Singh and A. Mahmood; Experientia, 1994, 50, 833. 347 D. Hota and S. B. Acharya; Indian J. Exp. Biol., 1994, 32, 710. 348 S. J. Shuttleworth, D. Nasturica, C. Gervais, M. A. Siddiqui, R. F. Rando and N. Lee, Bioorg. & Med. Chem. Lett., 2000, 10, 2501. 349 L.-R. Chen, Y.-C. Wang, Y. W. Lin, S.-Y. Chou, S.-F. Chen, L. T. Liu, Y.-T. Wu, C.-J. Kuo, T. S.-Shung Chen and S.-H. Juanga; Bioorg. & Med. Chem. Lett., 2005, 15, 3058. 350 A. Quattropani, J. Dorbais, D. Covini, P.-A. Pittet, V. Colovray, R. J. Thomas, R. Coxhead, S. Halazy, A. Scheer, M. Missotten, G. Ayala, C. Bradshaw, A.-M. De Raemy-Schenk, A. Nichols, R. Cirillo, E. G. Tos, C. Giachetti, L. Golzio, P. Marinelli, D. J. Church, C. Barberis, �A. Chollet and M. K. Schwarz; J. Med. Chem., 2005, 48, 7882. 351 J. Konkel, M. Packiarajan, H. Chen, U. P. Topiwala, H. Jimenez, I. J. Talisman, H. Coate and M. W. Walker; Bioorg. & Med. Chem. Lett., 2008, 16, 3950. 352 G. Bursavich, A. M. Gilbert, S. Lombardi, K. E. Georgiadis, E. Reifenberg, C. R. Flannery and Elisabeth A. Morris; Bioorg. & Med. Chem. Lett., 2007, 17, 5630. 353 R. K. Tiwari, N. Rastogi, R. Sethi and S. Shukla; J. Indian Chem. Soc., 2008, 85, 85. Department of Chemistry, <strong>Saurashtra</strong> <strong>University</strong>, Rajkot-360 005 146
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Saurashtra University Re - Accredit
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Statement under O. Ph. D. 7 of Saur
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ACKNOWLEDGEMENT It is a moment of g
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Jignesh Lunagariya, Hitesh Sarvaiya
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CONTENT Content General Remarks 6 A
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Content 3.2 Reaction scheme 149 3.3
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MF Molecular Formula MW Molecular W
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GABA Gamma Amino Butyric Acid MES M
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PART - A STUDIES ON 2-METHYL INDOLI
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Conferences / Seminar / Workshop At