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Bulletin 2011/50 - European Patent Office

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(C07D) I.1(2)<br />

• INDOLINE DERIVATIVES<br />

• DÉRIVÉS D'INDOLINE<br />

(71) Kyoto University, 36-1, Yoshida-honmachi,<br />

Sakyo-ku Kyoto-shi Kyoto 606-8<strong>50</strong>1, JP<br />

Tokyo Institute of Technology, 2-12-1,<br />

Ookayama Meguro-ku, Tokyo 152-85<strong>50</strong>, JP<br />

(72) SUGIMOTO, Hachiro, Kyoto-shi Kyoto 606-<br />

8<strong>50</strong>1, JP<br />

TAKAHASHI, Jun, Kyoto-shi Kyoto 606-<br />

8<strong>50</strong>1, JP<br />

TAKAHASHI, Takashi, Tokyo 152-85<strong>50</strong>, JP<br />

HIJIKURO, Ichiro, Tokyo 152-85<strong>50</strong>, JP<br />

(74) Duckworth, Timothy John, et al, J.A. Kemp &<br />

Co. 14 South Square Gray's Inn, London<br />

WC1R 5JJ, GB<br />

C07D 209/08 → (51) C07D 471/04<br />

(51) C07D 209/16 (11) 2 394 991 A1<br />

(25) En (26) En<br />

(21) 11179043.2 (22) 07.06.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(30) 12.06.2006 US 804527 P<br />

30.11.2006 US 867878 P<br />

(54) • Verfahren zur Herstellung von N-Hydroxy-<br />

3-ü4-üüü2-(2-methyl-1h-indol-3-yl)ethyl¨amino¨methyl¨phenyl¨-2e-2-propenamid<br />

und Ausgangsmaterialien dafür<br />

• Process for making n-hydroxy-3-ü4-üüü2-<br />

(2-methyl-1h-indol-3-yl)ethyl¨amino¨methyl¨phenyl¨-2e-2-propenamide<br />

and<br />

starting materials therefor<br />

• Procédé de fabrication de n-hydroxy-3-ü4üüü2-(2-méthyl-1h-indol-3-yl)éthyl¨amino¨méthyl¨phényl¨-2e-2-propénamide<br />

et<br />

matériaux de départ associés<br />

(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(84) BE BG CH CY CZ DE DK EE ES FI FR GB GR<br />

HU IE IS IT LI LT LU LV MC MT NL PL PT RO<br />

SE SI SK TR<br />

(71) Novartis Pharma GmbH, Brunner Strasse 59,<br />

1230 Wien, AT<br />

(84) AT<br />

(72) Acemoglu, Murat, 4052 Basel, CH<br />

Bajwa, Joginder, S., Elmwood Park, NJ New<br />

Jersey 07407, US<br />

Parker, David, John, West Milford, NJ New<br />

Jersey 07480, US<br />

Slade, Joel, Flanders, NJ New Jersey 07836,<br />

US<br />

(74) Gruber, Markus, Novartis Pharma AG <strong>Patent</strong><br />

Department, 4002 Basel, CH<br />

(62) 077843<strong>50</strong>.6 / 2 032 533<br />

C07D 209/86 → (51) C07C 209/10<br />

(51) C07D 211/22 (11) 2 394 992 A2<br />

A61K 31/445 A61K 31/47<br />

C07D 401/04 C07D 217/22<br />

C07D 211/32 A61P 25/36<br />

(25) En (26) En<br />

(21) 11166283.9 (22) 15.06.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

AL HR LT LV MK<br />

(30) 16.06.2003 US 462<strong>50</strong>7<br />

(54) • Substituierte Piperidinverbindungen und<br />

Verfahren zu deren Verwendung<br />

• Substituted piperidine compounds and<br />

methods of their use<br />

• Composés de pipéridine substitués et leurs<br />

procédés d'utilisation<br />

(71) Adolor Corporation, 700 Pennsylvania Drive,<br />

Exton, PA 19341, US<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(72) Le Bourdonnec, Bertrand, East Fallowfield,<br />

PA 19320, US<br />

Dolle, Roland E., Pennsylvania, PA 19406,<br />

US<br />

(74) Hallybone, Huw George, Carpmaels &<br />

Ransford One Southampton Row, London<br />

WC1B 5HA, GB<br />

(62) 04755219.5 / 1 638 565<br />

C07D 211/32 → (51) C07D 211/22<br />

C07D 211/58 → (51) C07D 401/04<br />

(51) C07D 213/16 (11) 2 394 993 A2<br />

C07D 213/53<br />

(25) Ko (26) En<br />

(21) 09832072.4 (22) 04.12.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) KR 2009/007216 04.12.2009<br />

(87) WO 2010/067987 2010/24 17.06.2010<br />

(88) 10.09.2010<br />

(30) 10.12.2008 KR 20080125360<br />

(54) • NEUES 2,6-SUBSTITUIERTES 3-NITROPY-<br />

RIDINDERIVAT, VERFAHREN ZU DESSEN<br />

HERSTELLUNG UND PHARMAZEUTISCHE<br />

ZUSAMMENSETZUNG, DIE DIESES ENT-<br />

HÄLT<br />

• NOVEL 2,6-SUBSTITUTED-3-NITROPYRI-<br />

DINE DERIVATIVE, METHOD FOR PRE-<br />

PARING SAME, AND PHARMACEUTICAL<br />

COMPOSITION INCLUDING SAME<br />

• NOUVEAU DÉRIVÉ 3-NITROPYRIDINE<br />

SUBSTITUÉE EN 2,6, PROCÉDÉ DE PRÉ-<br />

PARATION DE CE COMPOSÉ ET COMPO-<br />

SITION PHARMACEUTIQUE COMPRENANT<br />

CE COMPOSÉ<br />

(71) Dong Wha Pharm. Co., Ltd., 5 Sunwhadong,<br />

Jung-gu Seoul 100-130, KR<br />

(72) RYU, Jei Man, Anyang-si Gyeonggi-do 431-<br />

817, KR<br />

LEE, Jin Soo, Yongin-si Gyeonggi-do 448-<br />

172, KR<br />

PARK, Whui Jung, Suwon-si Gyeonggi-do<br />

442-1<strong>50</strong>, KR<br />

HWANG, Yun Ha, Gunpo-si Gyeonggi-do<br />

435-040, KR<br />

KIM, Ki Yoon, Hwaseong-si Gyeonggi-do<br />

445-360, KR<br />

(74) Fabry, Bernd, IP2 <strong>Patent</strong>anwalts GmbH<br />

Bruchstrasse 13, 41352 Korschenbroich, DE<br />

C07D 213/53 → (51) C07D 213/16<br />

C07D 213/61 → (51) C07C 279/22<br />

(51) C07D 213/74 (11) 2 394 994 A1<br />

A61K 31/44<br />

(25) En (26) En<br />

(21) 11168652.3 (22) 03.06.<strong>2011</strong><br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

BA ME<br />

(30) 08.06.2010 IT MI20101015<br />

(54) • Ein-topf Verfahren zur Herstellung von<br />

Dalfampridine<br />

• One-pot process for the synthesis of<br />

dalfampridine<br />

• Procédé à pot unique pour la synthèse de<br />

la Dalfampridine<br />

(71) Procos S.p.A., Via Matteotti 249, 28062<br />

Cameri NO, IT<br />

(72) Garavaglia, Fabio, 28065 Cerano (NO), IT<br />

Barozza, Alessandro, 20020 Nosate (MI), IT<br />

Roletto, Jacopo, 10135 Torino, IT<br />

Paissoni, Paolo, 10040 Druento (TO), IT<br />

227<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>50</strong>/<strong>2011</strong>) 14.12.<strong>2011</strong><br />

(74) Minoja, Fabrizio, Bianchetti Bracco Minoja S.<br />

r.l. Via Plinio, 63, 20129 Milano, IT<br />

C07D 213/75 → (51) A61K 31/44<br />

(51) C07D 215/22 (11) 2 394 995 A1<br />

A01N 43/42 A01N 43/90<br />

A01P 13/00 C07D 471/04<br />

(25) Ja (26) En<br />

(21) 10738335.8 (22) 02.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2010/000607 02.02.2010<br />

(87) WO 2010/089993 2010/32 12.08.2010<br />

(30) 03.02.2009 JP 2009023115<br />

(54) • RINGKONDENSIERTE 2-PYRIDONDERI-<br />

VATE UND HERBIZIDE<br />

• RING-FUSED 2-PYRIDONE DERIVATIVES<br />

AND HERBICIDES<br />

• DÉRIVÉS DE 2-PYRIDONE À CYCLES<br />

CONDENSÉS ET HERBICIDES<br />

(71) Kumiai Chemical Industry CO., LTD., 4-26,<br />

Ikenohata 1-chome Taito-ku, Tokyo 110-<br />

8782, JP<br />

IHARA CHEMICAL INDUSTRY CO., LTD., 4-<br />

26, Ikenohata 1-chome, Taito-ku Tokyo 110-<br />

0008, JP<br />

(72) TAKABE, Fumiaki, Iwata-shi Shizuoka 437-<br />

1213, JP<br />

HIRANO, Yuuki, Iwata-shi Shizuoka 437-<br />

1213, JP<br />

FUNYU, Akira, Iwata-shi Shizuoka 437-1213,<br />

JP<br />

KOBAYASHI, Masami, Tokyo 110-8782, JP<br />

MITSUNARI, Takashi, Tokyo 110-8782, JP<br />

(74) Albrecht, Thomas, Kraus & Weisert <strong>Patent</strong>und<br />

Rechtsanwälte Thomas-Wimmer-Ring<br />

15, 80539 München, DE<br />

C07D 217/22 → (51) C07D 211/22<br />

C07D 231/16 → (51) C07C 231/02<br />

(51) C07D 233/64 (11) 2 394 996 A1<br />

A61K 31/4164 A61K 31/4178<br />

A61P 3/04 A61P 3/06<br />

A61P 9/10 A61P 43/00<br />

C07D 405/04 C07D 409/04<br />

(25) Ja (26) En<br />

(21) 10738531.2 (22) 03.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2010/051469 03.02.2010<br />

(87) WO 2010/090200 2010/32 12.08.2010<br />

(30) 04.02.2009 JP 2009023793<br />

09.11.2009 JP 2009255980<br />

(54) • PHENYLIMIDAZOLVERBINDUNGEN<br />

• PHENYLIMIDAZOLE COMPOUNDS<br />

• COMPOSÉS DE PHÉNYLIMIDAZOLE<br />

(71) Otsuka Pharmaceutical Factory, Inc., 115<br />

Aza-Kuguhara Tateiwa Muya-cho, Narutoshi,<br />

Tokushima 772-8601, JP<br />

(72) SHIBUTANI, Tadao, Naruto-shi Tokushima<br />

772-8601, JP<br />

IWATA, Koushi, Naruto-shi Tokushima 772-<br />

8601, JP<br />

KIDO, Satoshi, Naruto-shi Tokushima 772-<br />

8601, JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastraße 4, 81925 München, DE<br />

C07D 249/08 → (51) C07C 209/10<br />

C07D 265/14 → (51) C07C 231/02<br />

C07D 265/26 → (51) C07C 231/02

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