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Bulletin 2011/50 - European Patent Office

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(C07D) I.1(1)<br />

(71) Biotium Inc., 3423 Investment Boulevard,<br />

Suite 8, Hayward, CA 94545, US<br />

(72) MAO, Fei, Fremont, CA 94555, US<br />

LEUNG, Wai-Yee, San Ramon, CA 94583, US<br />

CHEUNG, Ching-Ying, San Ramon, CA<br />

94583, US<br />

(74) Wytenburg, Wilhelmus Johannes, et al,<br />

Mewburn Ellis LLP 33 Gutter Lane, London<br />

EC2V 8AS, GB<br />

C07D 405/04 → (51) C07D 487/04<br />

C07D 405/06 → (51) C07D 303/08<br />

C07D 405/12 → (51) C07C 49/753<br />

C07D 405/12 → (51) C07D 211/86<br />

C07D 405/12 → (51) C07D 309/32<br />

C07D 405/14 → (51) C07D 295/15<br />

C07D 405/14 → (51) C07D 401/12<br />

(51) C07D 409/04 (11) 2 393 806 A1*<br />

C07D 409/14 C07D 471/04<br />

A61K 31/381 A61K 31/4192<br />

A61K 31/4196 A61K 31/427<br />

C07D 413/04 C07D 413/14<br />

C07D 417/04 C07D 417/14<br />

C07D 487/04<br />

(25) En (26) En<br />

(21) 10704662.5 (22) 05.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/023404 05.02.2010<br />

(87) WO 2010/091310 2010/32 12.08.2010<br />

(30) 06.02.2009 US 207126 P<br />

21.09.2009 US 244390 P<br />

(54) • INHIBITOREN DER JUN-N-TERMINALEN<br />

KINASE<br />

• INHIBITORS OF JUN N-TERMINAL KINASE<br />

• INHIBITEURS DE L'ENZYME JUN N-TER-<br />

MINAL KINASE<br />

(71) Elan Pharmaceuticals Inc., 800 Gateway<br />

Boulevard, South San Francisco, CA 94080,<br />

US<br />

(72) SHAM, Hing, L., Palo Alto CA 94306, US<br />

KONRADI, Andrei, W., Burlingame CA<br />

94010, US<br />

HOM, Roy, K., San Francisco CA 94102, US<br />

PROBST, Gary, D., San Francisco CA 94102,<br />

US<br />

BOWERS, Simeon, Oakland CA 94619, US<br />

TRUONG, Anh, Burlingame CA 94010, US<br />

NEITZ, R., Jeffrey, San Francisco CA 94116,<br />

US<br />

SEALY, Jennifer, Oakland CA 94602, US<br />

TOTH, Gergely, Palo Alto CA 94304, US<br />

(74) MacLean, Martin Robert, Mathys & Squire<br />

LLP 120 Holborn, London EC1N 2SQ, GB<br />

C07D 409/04 → (51) C07D 211/70<br />

C07D 409/12 → (51) C07D 211/86<br />

C07D 409/12 → (51) C07D 401/14<br />

C07D 409/14 → (51) C07D 409/04<br />

C07D 413/04 → (51) C07D 207/18<br />

C07D 413/04 → (51) C07D 409/04<br />

C07D 413/06 → (51) C07D 261/18<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(51) C07D 413/10 (11) 2 393 807 A1*<br />

C07D 417/10 A61K 31/5355<br />

A61P 3/00<br />

(25) En (26) En<br />

(21) 10701883.0 (22) 03.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2010/051262 03.02.2010<br />

(87) WO 2010/089303 2010/32 12.08.2010<br />

(30) 04.02.2009 US 206818 P<br />

(54) • CYCLISCHE 11ß -HYDROXYSTEROID-<br />

DEHYDROGENASE-1-HEMMER<br />

• CYCLIC INHIBITORS OF 11 -HYDROXYS-<br />

TEROID DEHYDROGENASE 1<br />

• INHIBITEURS CYCLIQUES DE LA 11<br />

-HYDROXYSTÉROÏDE DÉSHYDROGÉNASE<br />

DE TYPE 1<br />

(71) Boehringer Ingelheim International GmbH,<br />

Binger Strasse 173, 55216 Ingelheim am<br />

Rhein, DE<br />

(72) ECKHARDT, Matthias, 55216 Ingelheim am<br />

Rhein, DE<br />

HIMMELSBACH, Frank, 55216 Ingelheim am<br />

Rhein, DE<br />

(74) Hammann, Heinz, Boehringer Ingelheim<br />

Pharma GmbH CD-<strong>Patent</strong>s Binger Straße<br />

173, 55216 Ingelheim am Rhein, DE<br />

C07D 413/10 → (51) C07D 403/10<br />

C07D 413/12 → (51) C07D 261/18<br />

(51) C07D 413/14 (11) 2 393 808 A1*<br />

A61K 31/675 A61P 31/04<br />

(25) En (26) En<br />

(21) 10703403.5 (22) 03.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/023122 03.02.2010<br />

(87) WO 2010/091131 2010/32 12.08.2010<br />

(30) 03.02.2009 US 149402 P<br />

(54) • KRISTALLINE FORM VON R)-3-(4-(2-(2-<br />

METHYLTETRAZOL-5-YL)PYRIDIN-5-YL)-<br />

3-FLUOROPHENYL)-5-HYDROXYMETHY-<br />

LOXAZOLIDIN-2-ON-DIHYDROGENPHOS-<br />

PHAT<br />

• CRYSTALLINE FORM OF R)-3-(4-(2-(2-<br />

METHYLTETRAZOL-5-YL)PYRIDIN-5-YL)-<br />

3-FLUOROPHENYL)-5-HYDROXYMETHYL<br />

OXAZOLIDIN-2-ONE DIHYDROGEN PHOS-<br />

PHATE<br />

• FORME CRISTALLINE DU DIHYDROGÉ-<br />

NOPHOSPHATE DE (R)-3-(4-(2-(2-<br />

MÉTHYLTÉTRAZOL-5-YL)PYRIDIN-5-YL)-<br />

3-FLUOROPHÉNYL)-5-HYDROXYMÉTHYL<br />

OXAZOLIDIN-2-ONE<br />

(71) Trius Therapeutics, 6310 Nancy Ridge Drive,<br />

Suite 101, San Diego, CA 92121, US<br />

(72) PHILLIPSON, Douglas, Del Mar, CA 92014,<br />

US<br />

REICHENBACHER, Katharina, 4125 Riehen,<br />

CH<br />

DUGUID, Robert J., Glenmont, NY 12077,<br />

US<br />

WARE, Jacqueline, A., Virginia Beach VA<br />

23455, US<br />

(74) Brand, Thomas Louis, W.P. Thompson & Co.<br />

55 Drury Lane, London WC2B 5SQ, GB<br />

(51) C07D 413/14 (11) 2 393 809 A2*<br />

C07D 417/14 A61K 31/438<br />

A61P 37/00 A61P 29/00<br />

A61P 1/00 A61P 25/00<br />

A61P 9/00 A61P 35/00<br />

A61P 31/00<br />

(25) Fr (26) Fr<br />

(21) 10708283.6 (22) 04.02.2010<br />

77<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>50</strong>/<strong>2011</strong>) 14.12.<strong>2011</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) FR 2010/0<strong>50</strong>183 04.02.2010<br />

(87) WO 2010/089510 2010/32 12.08.2010<br />

(88) 30.09.2010<br />

(30) 05.02.2009 FR 0900493<br />

(54) • DERIVATE VON AZASPIRANYLALKYL-<br />

CARBAMATEN 5-GLIEDRIGER HETERO-<br />

CYCLISCHER VERBINDUNGEN, DEREN<br />

HERSTELLUNG UND DEREN THERAPEU-<br />

TISCHE VERWENDUNG<br />

• DERIVATIVES OF AZASPIRANYL-ALKYL-<br />

CARBAMATES OF 5-MEMBER HETERO-<br />

CYCLIC COMPOUNDS, PREPARATION<br />

THEREOF AND THERAPEUTIC USE<br />

THEREOF<br />

• DÉRIVÉS D'AZASPIRANYL-ALKYLCARBA-<br />

MATES D'HÉTÉROCYCLES À 5 CHAÎNONS,<br />

LEUR PRÉPARATION ET LEUR APPLICA-<br />

TION EN THÉRAPEUTIQUE<br />

(71) SANOFI, 174, Avenue de France, 7<strong>50</strong>13<br />

Paris, FR<br />

(72) ABOUABDELLAH, Ahmed, F-7<strong>50</strong>13 Paris, FR<br />

CHEREZE, Nathalie, F-7<strong>50</strong>13 Paris, FR<br />

FAYOL, Aude, F-7<strong>50</strong>13 Paris, FR<br />

LOCHEAD, Alistair, F-7<strong>50</strong>13 Paris, FR<br />

SAADY, Mourad, F-7<strong>50</strong>13 Paris, FR<br />

VACHE, Julien, F-7<strong>50</strong>13 Paris, FR<br />

YAICHE, Philippe, F-7<strong>50</strong>13 Paris, FR<br />

(74) Tinel, Marie-Line, et al, Sanofi Département<br />

Brevets 174, avenue de France, 7<strong>50</strong>13 Paris,<br />

FR<br />

C07D 413/14 → (51) C07D 401/12<br />

C07D 413/14 → (51) C07D 409/04<br />

C07D 417/04 → (51) C07D 207/18<br />

C07D 417/04 → (51) C07D 409/04<br />

C07D 417/10 → (51) C07D 413/10<br />

(51) C07D 417/12 (11) 2 393 810 A1*<br />

C07D 417/14 C07D 487/04<br />

A61K 31/<strong>50</strong> A61P 3/10<br />

(25) En (26) En<br />

(21) 10703404.3 (22) 04.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/023190 04.02.2010<br />

(87) WO 2010/091176 2010/32 12.08.2010<br />

(30) 05.02.2009 US 1<strong>50</strong>165 P<br />

(54) • PHTHALAZINHALTIGE ANTIDIABETISCHE<br />

VERBINDUNGEN<br />

• PHTHALAZINE-CONTAINING ANTIDIA-<br />

BETIC COMPOUNDS<br />

• COMPOSÉS ANTIDIABÉTIQUES CONTE-<br />

NANT DE LA PHTALAZINE<br />

(71) Schering Corporation, 2000 Galloping Hill<br />

Road, Kenilworth, NJ 07033, US<br />

(72) DAVIS, Jason, L., Albany, NY 12210, US<br />

MAYER, Michael, John, Altamont, NY 12009,<br />

US<br />

JOSIEN, Hubert, B., Jersey City, NJ 07302,<br />

US<br />

(74) Jaap, David Robert, et al, Merck & Co., Inc.<br />

<strong>Patent</strong> Department Hertford Road, Hoddesdon,<br />

Herts EN11 9BU, GB<br />

C07D 417/12 → (51) C07D 211/86<br />

C07D 417/12 → (51) C07D 309/32<br />

C07D 417/14 → (51) C07D 409/04

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