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Bulletin 2011/50 - European Patent Office

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(C07D) II.1(1)<br />

(74) Weber, Joachim, Hoefer & Partner <strong>Patent</strong>anwälte<br />

Pilgersheimer Strasse 20, 81543<br />

München, DE<br />

(51) C07D 207/16 (11) 1 712 547 B1<br />

C07D 405/12 A61K 31/40<br />

A61K 31/4025 A61P 3/10<br />

A61P 43/00<br />

(25) Ja (26) En<br />

(21) 05704327.5 (22) 01.02.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

AL BA HR LV MK YU<br />

(43) 18.10.2006<br />

(86) JP 2005/001377 01.02.2005<br />

(87) WO 2005/075421 2005/33 18.08.2005<br />

(30) 05.02.2004 JP 2004029856<br />

(54) • BICYCLOESTERDERIVAT<br />

• BICYCLOESTER DERIVATIVE<br />

• DERIVE DE BICYCLOESTER<br />

(73) Kyorin Pharmaceutical Co., Ltd., 5, Kandasurugadai<br />

2-chome, Chiyoda-ku, Tokyo 101-<br />

8311, JP<br />

(72) FUKUDA, Yasumichi, 3290207, JP<br />

ASAHINA, Yoshikazu, Shimotsuga-gun,<br />

Tochigi 3290101, JP<br />

OHATA, Kohei, Oyama-shi, Tochigi 3290207,<br />

JP<br />

YOKOTA, Kazuya, Shimotsuga-gun, Tochigi<br />

3290101, JP<br />

MURAKAMI, Koji, 3290207, JP<br />

MATSUI, Toshiyuki, Jousou-shi, Ibaraki 300-<br />

2706, JP<br />

(74) Vossius & Partner, Siebertstrasse 4, 81675<br />

München, DE<br />

(51) C07D 209/08 (11) 2 134 682 B1<br />

(25) En (26) En<br />

(21) 08734883.5 (22) 29.03.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 23.12.2009<br />

(86) EP 2008/002519 29.03.2008<br />

(87) WO 2008/125207 2008/43 23.10.2008<br />

(30) 13.04.2007 EP 07007585<br />

(54) • ÜBERGANGSMETALLKATALYSIERTE<br />

SYNTHESE VON N-AMINOINDOLEN<br />

• A TRANSITION METAL CATALYZED<br />

SYNTHESIS OF N-AMINOINDOLES<br />

• SYNTHÈSE DE N-AMINOINDOLES CATA-<br />

LYSÉE PAR MÉTAL DE TRANSITION<br />

(73) SANOFI, 174, Avenue de France, 7<strong>50</strong>13<br />

Paris, FR<br />

(72) HALLAND, Nis, 65926 Frankfurt am Main, DE<br />

NAZARE, M, 65926 Frankfurt am Main, DE<br />

LINDENSCHMIDT, Andreas, 65926 Frankfurt<br />

am Main, DE<br />

RKYEK, Omar, Tangier, MA<br />

URMANN, Matthias, 65926 Frankfurt am<br />

Main, DE<br />

ALONSO, Jorge, 65926 Frankfurt am Main,<br />

DE<br />

(74) Then, Johann, et al, Sanofi-Aventis<br />

Deutschland GmbH <strong>Patent</strong>- und Lizenzabteilung<br />

Industriepark Höchst Gebäude K 801,<br />

65926 Frankfurt am Main, DE<br />

(51) C07D 209/14 (11) 2 257 526 B1<br />

C07D 471/04 A61K 31/437<br />

A61P 25/04<br />

(25) De (26) De<br />

(21) 09725570.7 (22) 25.03.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

(43) 08.12.2010<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(86) EP 2009/002180 25.03.2009<br />

(87) WO 2009/118169 2009/40 01.10.2009<br />

(30) 27.03.2008 EP 08005804<br />

(54) • SPIRO(5.5)UNDECAN DERIVATE<br />

• SPIRO(5.5)UNDECANE DERIVATIVES<br />

• DÉRIVÉS DE SPIRO(5.5)UNDÉCANE<br />

(73) Grünenthal GmbH, Zieglerstrasse 6, 52078<br />

Aachen, DE<br />

(72) ZEMOLKA, Saskia, 52066 Aachen, DE<br />

SCHUNK, Stefan, 52070 Aachen, DE<br />

LINZ, Klaus, 53343 Wachtberg, DE<br />

SCHRÖBER, Wolfgang, 52074 Aachen, DE<br />

ENGLBERGER, Werner, 52223 Stolberg, DE<br />

THEIL, Fritz, 12247 Berlin, DE<br />

ROLOFF, Birgit, 12587 Berlin, DE<br />

(74) Bülle, Jan, et al, Kutzenberger & Wolff<br />

<strong>Patent</strong>anwaltssozietät Theodor-Heuss-Ring<br />

23, <strong>50</strong>668 Köln, DE<br />

(51) C07D 209/20 (11) 2 021 324 B1<br />

C07D 239/34 C07D 239/52<br />

C07D 239/60 C07D 261/14<br />

C07D 401/12 C07D 401/14<br />

C07D 403/12 C07D 405/04<br />

C07D 405/06 C07D 413/12<br />

C07D 417/04 A61K 31/40<br />

A61K 31/41 A61K 31/435<br />

(25) En (26) En<br />

(21) 07729447.8 (22) 23.05.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(43) 11.02.2009<br />

(86) EP 2007/05<strong>50</strong>12 23.05.2007<br />

(87) WO 2007/137980 2007/49 06.12.2007<br />

(30) 29.05.2006 EP 06114617<br />

(54) • NITRIERTE HETEROCYCLISCHE VERBIN-<br />

DUNGEN ALS ENDOTHELINREZEPTORAN-<br />

TAGONISTEN<br />

• NITRATED HETEROCYCLIC COMPOUNDS<br />

AS ENDOTHELIN RECEPTOR ANTAGONIST<br />

• COMPOSÉS HÉTÉROCYCLIQUES NITRÉS<br />

EN TANT QU'ANTAGONISTES DE RÉCEP-<br />

TEUR DE L'ENDOTHÉLINE<br />

(73) Nicox S.A., Taissounières HB4 1681 route<br />

des Dolines, BP 313, 06560 Sophia Antipolis<br />

- Valbonne, FR<br />

(72) ALMIRANTE, Nicoletta, 20155 Milano, IT<br />

BIONDI, Stefano, 20016 Pero (Milano), IT<br />

ONGINI, Ennio, 20090 Segrate, IT<br />

(74) Barchielli, Giovanna, et al, Nicox Research<br />

Institute S.r.l., <strong>Patent</strong> Department, Via<br />

Ariosto, 21, 20091 Bresso (Milano), IT<br />

(51) C07D 209/86 (11) 2 149 555 B1<br />

C07D 401/12 C09K 11/06<br />

(25) En (26) En<br />

(21) 09251918.0 (22) 30.07.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(43) 03.02.2010<br />

(30) 30.07.2008 KR 20080074713<br />

(54) • Aminbasierte Verbindung, organische<br />

lichtemittierende Vorrichtung mit der<br />

aminbasierten Verbindung und Flachbildschirmanzeigenvorrichtung<br />

mit der organischen<br />

lichtemittierenden Vorrichtung<br />

• Amine-based compound, organic light<br />

emitting device comprising the aminebased<br />

compound, and flat panel display<br />

device including the organic light emitting<br />

device<br />

565<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>50</strong>/<strong>2011</strong>) 14.12.<strong>2011</strong><br />

• Composé à base d'amine, dispositif électroluminescent<br />

organique comprenant le<br />

composé à base d'amine, et dispositif à<br />

écran plat incluant le dispositif électroluminescent<br />

organique<br />

(73) Samsung Mobile Display Co., Ltd., San<br />

No.24 Nongseo-Dong Giheung-Gu, Yongincity,<br />

Gyunggi-do 446-711, KR<br />

(72) Hwang, Seok-Hwan, Yongin-city, Gyunggido<br />

446-711, KR<br />

Kawk, Yoon-Hyun, Yongin-city, Gyunggi-do<br />

446-711, KR<br />

Kim, Young-Kook, Yongin-city, Gyunggi-do<br />

446-711, KR<br />

Yi, Jeoung-In, Yongin-city, Gyunggi-do 446-<br />

711, KR<br />

Lee, Jong-Hyuk, Yongin-city, Gyunggi-do<br />

446-711, KR<br />

(74) Taor, Simon Edward William, Marks & Clerk<br />

LLP 90 Long Acre, London WC2E 9RA, GB<br />

(51) C07D 209/96 (11) 1 794 123 B1<br />

A61K 31/537 A61P 1/00<br />

(25) Fr (26) Fr<br />

(21) 05805585.6 (22) 07.09.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK YU<br />

(43) 13.06.2007<br />

(86) FR 2005/002219 07.09.2005<br />

(87) WO 2006/030105 2006/12 23.03.2006<br />

(30) 09.09.2004 FR 0451997<br />

(54) • 3-SPIRO-INDOLIN-2-ONDERIVATE ALS<br />

LIGANDEN DES VASOPRESSINREZEP-<br />

TORS<br />

• 3-SPIRO-INDOLIN-2-ONE DERIVATIVES<br />

AS VASOPRESSIN RECEPTOR LIGAND<br />

• DERIVES DE 3-SPIRO-INDOLIN-2-ONE<br />

COMME LIGAND DES RECEPTEURS DE LA<br />

VASOPRESSINE<br />

(73) SANOFI, 174, Avenue de France, 7<strong>50</strong>13<br />

Paris, FR<br />

(72) BRASSEUR, Denis, F-91380 Chilly Mazarin,<br />

FR<br />

SERRADEIL-LE GAL, Claudine, F-317<strong>50</strong><br />

Escalquens, FR<br />

SHACKLETON, Gareth, Tyne and Wear,<br />

NE26ITF, GB<br />

(74) Kugel, Dominique, et al, Sanofi-Aventis<br />

Département Brevets 174 Avenue de France,<br />

7<strong>50</strong>13 Paris, FR<br />

C07D 211/96 → (51) C07D 317/58<br />

C07D 213/42 → (51) C07D 317/58<br />

(51) C07D 213/74 (11) 2 178 840 B1<br />

C07D 239/42 C07D 401/04<br />

C07D 401/10 A61K 31/44<br />

A61K 31/<strong>50</strong>6 A61P 19/00<br />

A61P 17/00 A61P 35/00<br />

A61P 37/00 A61P 31/00<br />

C07D 413/10<br />

(25) En (26) En<br />

(21) 08785465.9 (22) 08.08.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(43) 28.04.2010<br />

(86) EP 2008/006573 08.08.2008<br />

(87) WO 2009/021696 2009/08 19.02.2009<br />

(30) 10.08.2007 ES 200702261<br />

13.03.2008 EP 0838<strong>2011</strong><br />

(54) • AZABIPHENYLAMINOBENZOESÄUREDER-<br />

IVATE ALS DHODH-INHIBITOREN

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