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Bulletin 2011/50 - European Patent Office

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(C07C) I.1(1)<br />

• PROCEDE DE SYNTHESE D'UN OMEGA-<br />

AMINOACIDE OU ESTER A PARTIR D'UN<br />

ACIDE OU ESTER GRAS MONO-INSATURE<br />

(71) Arkema France, 420, rue d'Estienne d'Orves,<br />

92700 Colombes, FR<br />

(72) DUBOIS, Jean-Luc, F-69390 Millery, FR<br />

(74) Sauvageot, Olivier Roger, Arkema France<br />

DPI/DRD 420, rue d'Estienne d'Orves, 92705<br />

Colombes Cedex, FR<br />

(51) C07C 227/16 (11) 2 393 774 A1*<br />

C07C 229/22<br />

(25) En (26) En<br />

(21) 10705791.1 (22) 03.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2010/000654 03.02.2010<br />

(87) WO 2010/089094 2010/32 12.08.2010<br />

(30) 05.02.2009 EP 09001609<br />

05.02.2009 US 1<strong>50</strong>095 P<br />

(54) • VERFAHREN ZUR HERSTELLUNG EINES<br />

FETTSÄUREN-/CARNITINDERIVATS<br />

• PROCESS FOR THE PRODUCTION OF A<br />

FATTY ACID/L-CARNITINE DERIVATIVE<br />

• PROCÉDÉ DE PRODUCTION D'UN DÉRIVÉ<br />

D'ACIDE GRAS/L CARNITINE<br />

(71) Lonza Ltd, Lonzastrasse, 3930 Visp, CH<br />

(72) SMIDA, Donya, 2070 La Marsa, Tunis, TN<br />

C07C 227/40 → (51) B01D 61/58<br />

C07C 229/08 → (51) C07C 227/06<br />

C07C 229/22 → (51) C07C 227/16<br />

C07C 231/02 → (51) A61K 9/00<br />

C07C 233/18 → (51) A61K 9/00<br />

C07C 249/02 → (51) C10L 1/22<br />

(51) C07C 249/12 (11) 2 393 775 A2*<br />

C07C 251/38<br />

(25) En (26) En<br />

(21) 10701692.5 (22) 01.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) EP 2010/051144 01.02.2010<br />

(87) WO 2010/089267 2010/32 12.08.2010<br />

(88) 13.10.<strong>2011</strong><br />

(30) 05.02.2009 EP 08172487<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON 2-<br />

HALOGENMETHYLPHENYLESSIGSÄURE-<br />

DERIVATEN<br />

• METHOD FOR PRODUCING 2-HALOGEN-<br />

OMETHYLPHENYL ACETIC ACID DERIVA-<br />

TIVES<br />

• PROCÉDÉ DE PRODUCTION DES DÉRIVÉS<br />

D'ACIDE ACÉTIQUE 2-HALOGÉNOMÉ-<br />

THYLPHENYL<br />

(71) BASF SE, 67056 Ludwigshafen, DE<br />

(72) KORTE, Alexander, 67433 Neustadt, DE<br />

KEARNS, Mark, Alan, Wake Forest, NC<br />

27587, US<br />

SMITH, Jonathan, O., Quincy, IL 62301, US<br />

LIPOWSKY, Gunter, 68526 Ladenburg, DE<br />

BIECHE, Willi, 67167 Erpolzheim, DE<br />

C07C 251/38 → (51) C07C 249/12<br />

C07C 253/22 → (51) C07C 227/06<br />

C07C 253/30 → (51) C07C 227/06<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(51) C07C 317/00 (11) 2 393 776 A1*<br />

C07D 233/42 C07D 295/00<br />

(25) En (26) En<br />

(21) 10738989.2 (22) 29.01.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/022560 29.01.2010<br />

(87) WO 2010/090954 2010/32 12.08.2010<br />

(30) 06.02.2009 US 1<strong>50</strong>575 P<br />

(54) • NEUER TRIFLUORMETHYLSULFONAMID-<br />

GAMMA-SEKRETASEHEMMER<br />

• NOVEL TRIFLUOROMETHYLSULFONA-<br />

MIDE GAMMA SECRETASE INHIBITOR<br />

• NOUVEAU TRIFLUOROMÉTHYLSULFONA-<br />

MIDE INHIBITEUR DE LA GAMMA-<br />

SÉCRÉTASE<br />

(71) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907,<br />

US<br />

(72) DANIELS, Matthew, Rahway New Jersey<br />

07065-0907, US<br />

HUBBS, Jed, Rahway New Jersey 07065-<br />

0907, US<br />

MILLER, Thomas, Rahway New Jersey<br />

07065-0907, US<br />

(74) Buchan, Gavin MacNicol, Merck Sharp &<br />

Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

(51) C07D 207/18 (11) 2 393 777 A1*<br />

C07D 231/06 C07D 261/04<br />

C07D 263/08 C07D 277/08<br />

C07D 401/04 C07D 413/04<br />

C07D 417/04 A01N 35/00<br />

(25) En (26) En<br />

(21) 10721058.5 (22) 05.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2010/052109 05.02.2010<br />

(87) WO 2010/090344 2010/32 12.08.2010<br />

(30) 06.02.2009 JP 2009025839<br />

(54) • HYDRAZIDVERBINDUNG UND IHRE VER-<br />

WENDUNG ZUR SCHÄDLINGSBEKÄMP-<br />

FUNG<br />

• HYDRAZIDE COMPOUND AND USE OF<br />

THE SAME IN PEST CONTROL<br />

• COMPOSÉS HYDRAZIDES ET LEUR UTI-<br />

LISATION DANS LA PROTECTION PHY-<br />

TOSANITAIRE<br />

(71) Sumitomo Chemical Company, Limited, 27-<br />

1, Shinkawa 2-chome Chuo-ku, Tokyo 104-<br />

8260, JP<br />

(72) IHARA, Hideki, Osaka-shi Osaka 556-0016,<br />

JP<br />

KUMAMOTO, Koji, Toyonaka-shi Osaka 560-<br />

0021, JP<br />

(74) Vossius & Partner, Siebertstrasse 4, 81675<br />

München, DE<br />

(51) C07D 209/34 (11) 2 393 778 A1*<br />

A61K 31/4045 A61P 25/18<br />

(25) En (26) En<br />

(21) 10707659.8 (22) 05.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) HU 2010/000014 05.02.2010<br />

(87) WO 2010/089616 2010/32 12.08.2010<br />

(30) 06.02.2009 HU 0900071<br />

(54) • OPTISCH AKTIVE 3-[(PHENYLPIPERAZIN-<br />

1-YL)ALKYL]-3-ALKYLOXINDOLDERIVATE<br />

MIT ZNS-AKTIVITÄT<br />

72<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>50</strong>/<strong>2011</strong>) 14.12.<strong>2011</strong><br />

• Optically active 3-[(phenylpiperazin-1-yl)<br />

alkyl]-3- alkyl-oxindole derivatives having<br />

cns activity<br />

• Dérivés de 3 [(phénylpipérazine-1-yl)alkyl]-<br />

3-alkyl-oxindole optiquement actifs possédant<br />

une activité sur le snc<br />

(71) Egis Gyógyszergyár Nyilvánosan M Köd<br />

Részvénytársaság, Keresztúri út 30-38, 1106<br />

Budapest, HU<br />

(72) VOLK, Balázs, H -1165 Budapest, HU<br />

BARKÓCZY, József, H -1016 Budapest, FR<br />

GACSALYI, István, H -1201 Budapest, HU<br />

FOGASSY, Elemér, H -2030 Érd, HU<br />

SCHINDLER, József, H - 2151 Fót, HU<br />

GIGLER, Gábor, H - 1119 Budapest, FR<br />

KOMPAGNE, Hajnalka, H -1221 Budapest,<br />

HU<br />

NAGYNÉ GYÖNÖS, Ildikó, H -1192 Budapest,<br />

HU<br />

PALLAGI, Katalin, H -1054 Budapest, HU<br />

PORCS-MAKKAY, Márta, H -2013 Pomáz,<br />

HU<br />

SZÉNÁSI, Gábor, H-2096 Üröm, HU<br />

MEZEI, Tibor, H -1221 Budapest, HU<br />

LUKÁCS, Gyula, H - 1163 Budapest, HU<br />

LÉVAY, György, H - 2092 Budakeszi, HU<br />

EGYED, András, H - 1145 Budapest, HU<br />

HÁRSING, László Gábor, H - 1071 Budapest,<br />

HU<br />

(74) Beszédes, Stephan G., <strong>Patent</strong>anwalt Münchener<br />

Strasse 80a, 85221 Dachau, DE<br />

(51) C07D 209/56 (11) 2 393 779 A2*<br />

(25) En (26) En<br />

(21) 10738292.1 (22) 04.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) IN 2010/000066 04.02.2010<br />

(87) WO 2010/089778 2010/32 12.08.2010<br />

(88) 14.10.2010<br />

(30) 05.02.2009 IN MU02342009<br />

(54) • VERFAHREN ZUR SYNTHESE VON CLEIS-<br />

TANTHIN<br />

• PROCESS FOR THE SYNTHESIS OF<br />

CLEISTANTHIN<br />

• PROCÉDÉ DE SYNTHÈSE DE CLEISTAN-<br />

THINE<br />

(71) Godavari Biorefineries Ltd., Somaiya Bhavan<br />

45/47 Mahatma Gandhi Road, Fort Mumbai<br />

400 001 Maharashtra, IN<br />

(72) SINGH, Om, Vir, Thane West 400 610<br />

Maharashtra, IN<br />

TAPADIYA, Sarika, Madhusudan, Thane<br />

West 400 610 Maharashtra, IN<br />

DESHMUKH, Rahul, Ganpat, Thane West 400<br />

610 Maharashtra, IN<br />

(74) Kilger, Ute, Forrester & Boehmert Pettenkoferstrasse<br />

20-22, 80336 München, DE<br />

(51) C07D 211/70 (11) 2 393 780 A1*<br />

C07D 401/04 C07D 401/14<br />

C07D 409/04 C07D 471/04<br />

A61K 31/4523 A61K 31/4535<br />

A61K 31/4545 A61K 31/454<br />

A61K 31/445 A61P 13/00<br />

(25) En (26) En<br />

(21) 10703620.4 (22) 04.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2010/000695 04.02.2010<br />

(87) WO 2010/089119 2010/32 12.08.2010<br />

(30) 04.02.2009 US 206863 P<br />

(54) • HETEROCYCLISCHE DERIVATE ALS M-<br />

GLU5-ANTAGONISTEN<br />

• HETEROCYCLIC DERIVATIVES AS M-GLU5<br />

ANTAGONISTS

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