Bulletin 2011/50 - European Patent Office

(C07D) I.1(1)
• DÉRIVÉS HÉTÉROCYCLIQUES EN TANT
QU'ANTAGONISTES DE MGLU5
(71) Recordati Ireland Limited, Raheens East,
Ringaskiddy County Cork, IE
(72) LEONARDI, Amedeo, I-20154 Milano, IT
MOTTA, Gianni, I-20030 Barlassina, IT
RIVA, Carlo, I-21100 Varese, IT
POGGESI, Elena, I-20148 Milano, IT
GRAZIANI, Davide, I-20155 Milano, IT
(74) McKelvey, Ian Edward, et al, Serjeants 25
The Crescent King Street, Leicester LE1 6RX,
GB
(51) C07D 211/86 (11) 2 393 781 A1*
C07D 401/12 C07D 405/12
C07D 409/12 C07D 417/12
A61K 31/4422 A61K 31/47
A61P 11/00 A61P 11/06
A61P 19/02 A61P 29/00
(25) En (26) En
(21) 09768393.2 (22) 14.12.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
(86) EP 2009/067032 14.12.2009
(87) WO 2010/072599 2010/26 01.07.2010
(30) 23.12.2008 US 203467 P
(54) • DIHYDROPYRIDONHARNSTOFFE ALS
P2X7-MODULATOREN
• DIHYDROPYRIDONE UREAS AS P2X7
MODULATORS
• DIHYDROPYRIDONE URÉES EN TANT QUE
MODULATEURS DE P2X7
(71) F. Hoffmann-La Roche AG, Grenzacherstrasse
124, 4070 Basel, CH
(72) BROTHERTON-PLEISS, Christine E., Sunnyvale
California 94087, US
CAROON, Joan Marie, Mountain View California
94043, US
LOPEZ-TAPIA, Francisco Javier, Mahwah
New Jersey 07430, US
NITZAN, Dov, San Jose California 95129, US
WALKER, Keith Adrian Murray, Los Altos
Hills California 94022, US
(74) Salud, Carlos E., F. Hoffmann-La Roche AG
Grenzacherstrasse 124, 4070 Basel, CH
C07D 213/06 → (51) C07D 241/44
C07D 213/48 → (51) C07C 45/38
(51) C07D 213/61 (11) 2 393 782 A1*
C07D 213/89 A61K 31/44
A61P 11/00
(25) En (26) En
(21) 10704746.6 (22) 04.02.2010
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
AL BA RS
(86) EP 2010/000676 04.02.2010
(87) WO 2010/089107 2010/32 12.08.2010
(30) 06.02.2009 EP 09001660
(54) • BENZOESÄURE(1-PHENYL-2-PYRIDIN-4-
YL)ETHYLESTER ALS PHOSPHODIESTE-
RASE-INHIBITOREN
• BENZOIC ACID (1-PHENYL-2-PYRIDIN-4-
YL) ETHYL ESTERS AS PHOSPHODIES-
TERASE INHIBITORS
• ESTERS (1-PHÉNYL-2-PYRIDIN-4-YL)
ÉTHYLIQUES D'ACIDE BENZOÏQUE EN
TANT QU'INHIBITEURS DE LA PHOSPHO-
DIESTÉRASE
(71) Chiesi Farmaceutici S.p.A., Via Palermo, 26/
A, 43100 Parma, IT
(72) AMARI, Gabriele, I-43100 Parma, IT
ARMANI, Elisabetta, I-43100 Parma, IT
DELCANALE, Maurizio, I-43100 Parma, IT
Europäisches Patentblatt
European Patent Bulletin
Bulletin européen des brevets
(74) Minoja, Fabrizio, Bianchetti Bracco Minoja S.
r.l. Via Plinio, 63, 20129 Milano, IT
C07D 213/643→ (51) C07C 49/753
C07D 213/89 → (51) C07D 213/61
C07D 215/227→ (51) C07C 49/753
C07D 221/18 → (51) C07D 241/44
(51) C07D 221/28 (11) 2 393 783 A1*
C07D 489/02
(25) En (26) En
(21) 09760689.1 (22) 30.11.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
(86) US 2009/066067 30.11.2009
(87) WO 2010/065441 2010/23 10.06.2010
(30) 02.12.2008 US 119064 P
(54) • VERFAHREN ZUR HERSTELLUNG VON
HYDROCODON UNTER ANWENDUNG
EINER SUPERSÄURE
• PROCESS FOR PREPARING HYDROCO-
DONE USING A SUPER ACID
• PROCÉDÉ DE PRÉPARATION D'HYDRO-
CODONE À L'AIDE D'UN SUPERACIDE
(71) Mallinckrodt LLC, 675 McDonnell Boulevard,
Hazelwood, MO 63042, US
(72) WANG, Peter, X., Clarkson Valley Missouri
63005, US
JIANG, Tao, St. Louis, Missouri 63146, US
LIAO, Subo, Ballwin Missouri 63021, US
MOORE, Erin, Imperial Missouri 63052, US
(74) Albrecht, Thomas, Kraus & Weisert Patentund
Rechtsanwälte Thomas-Wimmer-Ring
15, 80539 München, DE
(51) C07D 223/16 (11) 2 393 784 A1*
A61K 31/55 A61P 9/10
A61P 9/06 A61P 9/04
(25) Fr (26) Fr
(21) 10707068.2 (22) 03.02.2010
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
AL BA RS
(86) FR 2010/000080 03.02.2010
(87) WO 2010/089475 2010/32 12.08.2010
(30) 04.02.2009 FR 0900457
(54) • NEUARTIGES VERFAHREN ZUR SYN-
THESE VON IVABRADIN UND PHARMA-
ZEUTISCH AKZEPTALEN
SÄUREADDITIONSSALZEN DARAUS
• NOVEL METHOD FOR THE SYNTHESIS OF
IVABRADINE AND THE PHARMACEUTI-
CALLY ACCEPTABLE ACID ADDITION
SALTS THEREOF
• NOUVEAU PROCEDE DE SYNTHESE DE
L'IVABRADINE ET DE SES SELS D'ADDI-
TION A UN ACIDE PHARMACEUTIQUE-
MENT ACCEPTABLE
(71) Les Laboratoires Servier, 35, rue de Verdun,
92284 Suresnes Cedex, FR
(72) PEGLION, Jean-Louis, F-78110 Le Vesinet,
FR
DESSINGES, Aimée, F-92500 Rueil-Malmaison,
FR
SERKIZ, Bernard, F-77170 Servon Brie
Comte Robert, FR
LERESTIF, Jean-Michel, F-76190 Yvetot, FR
LECOUVE, Jean-Pierre, F-76600 Le Havre,
FR
(74) Giudicelli, Cathy, Les Laboratoires Servier
Direction Brevets 35, rue de Verdun, 92284
Suresnes Cedex, FR
73
Anmeldungen
Applications
Demandes (50/2011) 14.12.2011
C07D 231/06 → (51) C07D 207/18
C07D 231/20 → (51) C07C 49/753
C07D 233/42 → (51) C07C 317/00
(51) C07D 239/00 (11) 2 393 785 A1*
C07D 403/12
(25) En (26) En
(21) 10736412.7 (22) 28.01.2010
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK SM TR
(86) US 2010/022430 28.01.2010
(87) WO 2010/088406 2010/31 05.08.2010
(30) 28.01.2009 US 206271 P
(54) • SUBSTITUIERTE 1,1,3,3-TETRAOXIDO-
BENZO[D][1,3,2]DITHIAZOLE ALS ALLOS-
TERISCHE MGLUR4-POTENTIATOREN,
ZUSAMMENSETZUNGEN UND VERFAH-
REN ZUR BEHANDLUNG NEUROLOGI-
SCHER DYSFUNKTIONEN
• SUBSTITUTED 1,1,3,3-TETRAOXIDO-
BENZO[D][1,3,2]DITHIAZOLES AS
MGLUR4 ALLOSTERIC POTENTIATORS,
COMPOSITIONS, AND METHODS OF
TREATING NEUROLOGICAL DYSFUNC-
TION
• 1,1,3,3-TÉTRAOXYDOBENZO[D][1,3,2]
DITHIAZOLES SUBSTITUÉS EN TANT QUE
POTENTIALISATEURS ALLOSTÉRIQUES
DE MGLUR4, COMPOSITIONS ET PROCÉ-
DÉS DE TRAITEMENT D'UN DYSFONC-
TIONNEMENT NEUROLOGIQUE
(71) Vanderbilt University, 305 Kirkland Hall,
Nashville, Tennessee 37240, US
(72) CONN, P. Jeffrey, Brentwood, Tennessee
37027, US
LINDSLEY, Craig W., Brentwood, Tennessee
37027, US
HOPKINS, Corey R., Nolensville, Tennessee
37135, US
WEAVER, Charles David, Franklin, Tennessee
37067, US
NISWENDER, Colleen M., Brentwood, Tennessee
37027, US
GOGLIOTTI, Rocco D., Kingston Springs,
Tennessee 37082, US
ENGERS, Darren W., Nashville, Tennessee
37221, US
(74) O'Connell, Maura, et al, FRKelly 27 Clyde
Road Ballsbridge, Dublin 4, IE
(51) C07D 239/10 (11) 2 393 786 A2*
(25) En (26) En
(21) 09839567.6 (22) 06.02.2009
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MK MT
NL NO PL PT RO SE SI SK TR
(86) IN 2009/000083 06.02.2009
(87) WO 2010/089753 2010/32 12.08.2010
(54) • NEUE POLYMORPHE AUS LOPINAVIR
• NOVEL POLYMORPHS OF LOPINAVIR
• NOUVEAUX POLYMORPHES DU LOPINA-
VIR
(71) Hetero Research Foundation, Plot No. B-
80&81 A.P.I.E., Balanagar, Hyderabad 500
018, Andhrapradesh, IN
(72) PARTHASARADHI REDDY, Bandi, Hyderabad
500 018, IN
RATHNAKAR REDDY, Kura, Hyderabad 500
018, IN
RAJI REDDY, Rapolu, Hyderabad 500 018,
IN
MURALIDHARA REDDY, Dasari, Hyderabad
500 018, IN
SUBASH CHANDER REDDY, Kesireddy,
Hyderabad 500 018, IN