07.02.2013 Views

Bulletin 2011/50 - European Patent Office

Bulletin 2011/50 - European Patent Office

Bulletin 2011/50 - European Patent Office

SHOW MORE
SHOW LESS

Create successful ePaper yourself

Turn your PDF publications into a flip-book with our unique Google optimized e-Paper software.

(C07D) I.1(2)<br />

C07D 277/20 → (51) C07C 279/22<br />

C07D 277/56 → (51) C07C 279/22<br />

C07D 309/22 → (51) C07C 279/22<br />

C07D 311/22 → (51) C07B 53/00<br />

(51) C07D 401/04 (11) 2 394 997 A1<br />

C07D 211/58<br />

(25) Ja (26) En<br />

(21) 10738529.6 (22) 03.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2010/051465 03.02.2010<br />

(87) WO 2010/090198 2010/32 12.08.2010<br />

(30) 03.02.2009 JP 2009022834<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON 1-<br />

(4-PIPERIDINYL)BENZIMIDAZOLON-DERI-<br />

VATEN<br />

• PROCESS FOR PREPARING 1-(4-PIPERI-<br />

DINYL)BENZIMIDAZOLONE DERIVATIVES<br />

• PROCÉDÉ DE PRÉPARATION DE DÉRIVÉS<br />

DE 1-(4-PIPÉRIDINYL)BENZIMIDAZOLONE<br />

(71) Mitsubishi Tanabe Pharma Corporation, 2-6-<br />

18, Kitahama, Chuo-ku Osaka-shi, Osaka<br />

541-8<strong>50</strong>5, JP<br />

(72) IWAMURA, Hiroshi, Osaka-shi, Osaka 541-<br />

8<strong>50</strong>5, JP<br />

TARAO, Yoshihiro, Osaka-shi, Osaka 541-<br />

8<strong>50</strong>5, JP<br />

(74) von Kreisler Selting Werner, Deichmannhaus<br />

am Dom Bahnhofsvorplatz 1, <strong>50</strong>667 Köln,<br />

DE<br />

C07D 401/04 → (51) C07C 231/02<br />

C07D 401/04 → (51) C07D 211/22<br />

C07D 401/06 → (51) C07D 209/08<br />

(51) C07D 401/12 (11) 2 394 998 A1<br />

C07D 401/14 A61K 31/<strong>50</strong>1<br />

A61P 29/00 A61P 11/00<br />

(25) En (26) En<br />

(21) 10382155.9 (22) 31.05.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

BA ME RS<br />

(54) • 3-(5-Amino-6-oxo-1,6-dihydropyridazin-3yl)-biphenyl<br />

Derivate als PDE4 Inhibitoren<br />

• 3-(5-Amino-6-oxo-1,6-dihydropyridazin-3yl)-biphenyl<br />

derivatives as PDE4 inhibitors<br />

• Dérivés de 3-(5-Amino-6-oxo-1,6-dihydropyridazin-3-yl)-biphenyl<br />

en tant qu'inhibiteurs<br />

de la PDE4<br />

(71) Almirall, S.A., Ronda General Mitre 151,<br />

08022 Barcelona, ES<br />

(72) Gracia Ferrer, Jordi, 08980, Sant Feliu de<br />

Llobregat, ES<br />

Pages Santacana, Lluis Miquel, 08980, Sant<br />

Feliu de Llobregat, ES<br />

(74) Elzaburu Marquez, Alberto, et al, ELZABURU<br />

S.L.P. C/ Miguel Angel, 21, 2º, 28010<br />

Madrid, ES<br />

C07D 401/12 → (51) C07D 209/08<br />

C07D 401/12 → (51) C07D 413/06<br />

(51) C07D 401/14 (11) 2 394 999 A1<br />

A61K 31/497 A61K 31/<strong>50</strong>6<br />

A61P 7/00 A61P 35/02<br />

C07D 403/12 C07D 403/14<br />

C07D 413/14<br />

(25) Ja (26) En<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(21) 10738621.1 (22) 05.02.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2010/051722 05.02.2010<br />

(87) WO 2010/090290 2010/32 12.08.2010<br />

(30) 06.02.2009 JP 2009026470<br />

04.12.2009 JP 2009276133<br />

(54) • AMINOPYRAZINDERIVAT UND MEDIZIN<br />

• AMINOPYRAZINE DERIVATIVE AND MED-<br />

ICINE<br />

• DÉRIVÉ D'AMINOPYRAZINE ET MÉDICA-<br />

MENT CORRESPONDANT<br />

(71) Nippon Shinyaku Co., Ltd., 14, Kisshoin<br />

Nishinosho Monguchicho Minami-ku, Kyotoshi<br />

Kyoto 601-85<strong>50</strong>, JP<br />

(72) FUJIHARA, Hidetaka, Kyoto-shi Kyoto 601-<br />

8319, JP<br />

ASAKI, Tetsuo, Uji-shi Kyoto 611-0041, JP<br />

HORI, Katsutoshi, Kusatsu-shi Shiga 525-<br />

0033, JP<br />

NAITO, Haruna, Kyoto-shi Kyoto 602-0036,<br />

JP<br />

(74) von Uexküll - Güldenband, Alexa, et al,<br />

Vossius & Partner Siebertstrasse 4, 81675<br />

München, DE<br />

C07D 401/14 → (51) C07D 401/12<br />

(51) C07D 403/04 (11) 2 395 000 A1<br />

C07D 513/04 C07D 407/14<br />

A61K 31/4184 A61P 35/00<br />

(25) En (26) En<br />

(21) 11180160.1 (22) 30.12.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK YU<br />

(30) 30.12.2004 GB 0428554<br />

30.12.2004 GB 0428552<br />

30.12.2004 US 640597 P<br />

30.12.2004 US 640475 P<br />

(54) • Benzimidazolverbindungen, die die Aktivität<br />

von CDK, GSK und Aurora-Kinasen modulieren<br />

• Benzimidazole compounds that modulate<br />

the activity of CDK, GSK and aurora kinases<br />

• Composés de benzimidazole régulant l'<br />

activite de kinases CDK, GSK et aurora<br />

(71) Astex Therapeutics Limited, 436 Cambridge<br />

Science Park Milton Park Cambridge, Cambridgeshire<br />

CB4 0QA, GB<br />

(72) Berdini, Valerio, Cambridge, Cambridgeshire<br />

CB4 0QA, GB<br />

Carr, Maria Grazia, Cambridge, Cambridgeshire<br />

CB4 0QA, GB<br />

Gill, Adrian Liam, Cambridge, Cambridgeshire<br />

CB4 0QA, GB<br />

Howard, Steven, Cambridge, Cambridgeshire<br />

CB4 0QA, GB<br />

Navarro, Eva Figueroa, Cambridge, Cambridgeshire<br />

CB4 0QA, GB<br />

Trewartha, Gary, Cambridge, Cambridgeshire<br />

CB4 0QA, GB<br />

Rees, David Charles, Cambridge, Cambridgeshire<br />

CB4 0QA, GB<br />

Vinkovic, Mladen, Cambridge, Cambridgeshire<br />

CB04 0QA, GB<br />

Wyatt, Paul Graham, Dundee, DD1 5EH, GB<br />

(74) Cooke, Richard Spencer, Elkington and Fife<br />

LLP Prospect House 8 Pembroke Road,<br />

Sevenoaks, Kent TN13 1XR, GB<br />

(62) 05823721.5 / 1 833 819<br />

C07D 403/06 → (51) C07D 209/08<br />

C07D 403/12 → (51) C07D 209/08<br />

228<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>50</strong>/<strong>2011</strong>) 14.12.<strong>2011</strong><br />

C07D 403/12 → (51) C07D 401/14<br />

C07D 403/12 → (51) C07D 413/06<br />

(51) C07D 403/14 (11) 2 395 001 A1<br />

A61K 31/<strong>50</strong>6 A61P 35/00<br />

(25) En (26) En<br />

(21) 10163597.7 (22) 21.05.2010<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO SE SI SK SM TR<br />

BA ME RS<br />

(54) • Neue Pyrimidinderivate<br />

• Novel pyrimidine derivatives<br />

• Nouveaux dérivés de pyrimidine<br />

(71) Chemilia AB, Alfred Nobels Allè 10, 141 52<br />

Huddinge, SE<br />

(72) Dahlstedt, Emma, 115 43 Stockholm, SE<br />

Johansson, Tommy, 167 36 Bromma, SE<br />

Högberg, Marita, 146 52 Tullinge, SE<br />

(74) Lundquist, Tomas, Awapatent AB Box 4<strong>50</strong><br />

86, 104 30 Stockholm, SE<br />

C07D 403/14 → (51) C07D 401/14<br />

C07D 405/04 → (51) C07D 233/64<br />

C07D 405/06 → (51) C07D 209/08<br />

(51) C07D 405/12 (11) 2 395 002 A1<br />

A61P 11/00 A61K 31/443<br />

(25) En (26) En<br />

(21) 10192912.3 (22) 08.11.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(30) 08.11.2005 US 734<strong>50</strong>6 P<br />

27.12.2005 US 754086 P<br />

22.05.2006 US 802458 P<br />

(54) • Pharmazeutische Zusammensetzung enthaltend<br />

einen heterozyklischen Modulator<br />

von ATP-bindenden Kassettentransportern<br />

• Pharmaceutical composition containing a<br />

heterocyclic modulator of ATP-binding<br />

cassette transporters.<br />

• Composition pharmaceutique contenant un<br />

modulateur hétérocyclique de transporteurs<br />

de cassette à liaison ATP<br />

(71) Vertex Pharmaceuticals Incorporated, 130<br />

Waverly Street, Cambridge, MA 02139, US<br />

(72) Hadida Ruah, Sara, La Jolla, CA 92037, US<br />

Hamilton, Matthew, Hackettstown, NJ<br />

07840, US<br />

Miller, Mark, San Diego, CA 92109, US<br />

Grootenhuis, Peter, D., J., San Diego, CA<br />

92130, US<br />

Bear, Brian, Oceanside, CA 92057, US<br />

McCarthy, Jason, Cardiff By The Sea, CA<br />

92007, US<br />

Zhou, Jinglan, San Diego, CA 92130, US<br />

(74) Cohausz & Florack, <strong>Patent</strong>- und Rechtsanwälte<br />

Partnerschaftsgesellschaft Bleichstraße<br />

14, 40211 Düsseldorf, DE<br />

(62) 06837028.7 / 1 945 632<br />

C07D 405/12 → (51) C07D 209/08<br />

C07D 405/14 → (51) H01L 51/<strong>50</strong><br />

C07D 407/14 → (51) C07D 403/04<br />

C07D 409/04 → (51) C07D 233/64<br />

C07D 409/04 → (51) C09B 57/00<br />

C07D 409/12 → (51) C07D 209/08<br />

C07D 409/14 → (51) H01L 51/<strong>50</strong>

Hooray! Your file is uploaded and ready to be published.

Saved successfully!

Ooh no, something went wrong!