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Bulletin 2011/50 - European Patent Office

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(C07D) II.1(1)<br />

• AZABIPHENYLAMINOBENZOIC ACID<br />

DERIVATIVES AS DHODH INHIBITORS<br />

• DÉRIVÉS D'ACIDE AZABIPHÉNYLAMINO-<br />

BENZOÏQUE COMME INHIBITEURS DE LA<br />

DHODH<br />

(73) Almirall, S.A., Ronda General Mitre 151,<br />

08022 Barcelona, ES<br />

(72) CASTRO PALOMINO LARIA, Julio, Cesar, E-<br />

08330 Premia de Mar (Barcelona), ES<br />

TERRICABRAS BELART, Emma, E-08190<br />

Sant Cugat Del Valles Barcelona, ES<br />

ERRA SOLA, Montserrat, E-08903 L' Hospitalet<br />

de Llobregat (Barcelona), ES<br />

NAVARRO ROMERO, Eloisa, E-08011 Barcelona,<br />

ES<br />

FONQUERNA POU, Silvia, E-08030 Barcelona,<br />

ES<br />

CARDUS FIGUERAS, Aranzazu, E-08780<br />

Palleja Barcelona, ES<br />

LOZOYA TORIBIO, Maria, Estrella, Barcelona,<br />

ES<br />

(74) Srinivasan, Ravi Chandran, J.A. Kemp & Co.<br />

14 South Square Gray's Inn, London WC1R<br />

5JJ, GB<br />

C07D 213/74 → (51) C07D 317/58<br />

C07D 213/81 → (51) C07D 417/12<br />

(51) C07D 221/22 (11) 2 080 755 B1<br />

(25) Ja (26) En<br />

(21) 07829480.8 (22) 10.10.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 22.07.2009<br />

(86) JP 2007/069742 10.10.2007<br />

(87) WO 2008/044702 2008/16 17.04.2008<br />

(30) 11.10.2006 JP 20062781<strong>50</strong><br />

(54) • VERFAHREN ZUR HERSTELLUNG EINES<br />

AZABICYCLOALKANOLDERIVATS<br />

• PROCESS FOR PRODUCTION OF AZABI-<br />

CYCLOALKANOL DERIVATIVE<br />

• PROCÉDÉ DE PRODUCTION D'UN DÉRIVÉ<br />

AZABICYCLOALCANOL<br />

(73) Nippon Soda Co., Ltd., 2-1 Ohtemachi 2chome,Chiyoda-ku,<br />

Tokyo, 100-8165, JP<br />

(72) OOOKA, Hirohito, Takaoka-Shi, Toyama 933-<br />

8<strong>50</strong>7, JP<br />

FUKUHARA, Shinya, Takaoka-Shi, Toyama<br />

933-8<strong>50</strong>7, JP<br />

(74) Wibbelmann, Jobst, et al, Wuesthoff &<br />

Wuesthoff <strong>Patent</strong>- und Rechtsanwälte<br />

Schweigerstrasse 2, 81541 München, DE<br />

(51) C07D 231/06 (11) 2 069 310 B1<br />

C07D 401/12 C07D 409/12<br />

C07D 513/04 C07D 417/12<br />

C07D 403/12 C07D 231/12<br />

A61K 31/415 A61K 31/4155<br />

A61P 25/00 C07D 401/04<br />

C07D 407/04<br />

(25) En (26) En<br />

(21) 07820387.4 (22) 20.09.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

HR<br />

(43) 17.06.2009<br />

(86) EP 2007/059944 20.09.2007<br />

(87) WO 2008/034863 2008/13 27.03.2008<br />

(30) 22.09.2006 US 846406 P<br />

22.09.2006 EP 06121087<br />

23.02.2007 US 902865 P<br />

23.02.2007 EP 07102965<br />

(54) • SULFONYL-PYRAZOLINYL-1-CARBOXA-<br />

MIDINDERIVATE ALS 5-HT6-ANTAGONIS-<br />

TEN<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

• SULFONYLPYRAZOLINE-1-CARBOXAMI-<br />

DINE DERIVATIVES AS 5-HT6 ANTAGO-<br />

NISTS<br />

• DÉRIVÉS SULFONYLIQUES DE PYRAZO-<br />

LINYL-1-CARBOXAMIDINE EN TANT<br />

QU'ANTAGONISTES DE 5-HT6<br />

(73) Abbott Healthcare Products B.V., C.J. van<br />

Houtenlaan 36, 1381 CP Weesp, NL<br />

(72) IWEMA BAKKER, Wouter I., 1381 CP Weesp,<br />

NL<br />

KEIZER, Hiskias G., 1381 CP Weesp, NL<br />

NEUT, VAN DER, Martina A.W., 1381 CP<br />

Weesp, NL<br />

KRUSE, Cornelis G., 1381 CP Weesp, NL<br />

LOEVEZIJN, VAN, Arnold, 1381 CP Weesp,<br />

NL<br />

ZORGDRAGER, Jan, 1381 CP Weesp, NL<br />

(74) Jansen, Cornelis Marinus, VEREENIGDE<br />

Johan de Wittlaan 7, 2517 JR Den Haag, NL<br />

C07D 231/12 → (51) C07D 231/06<br />

(51) C07D 231/18 (11) 1 948 615 B1<br />

C07D 401/12 A61K 31/415<br />

A61P 15/00<br />

(25) En (26) En<br />

(21) 06809167.7 (22) 26.10.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK RS<br />

(43) 30.07.2008<br />

(86) IB 2006/003080 26.10.2006<br />

(87) WO 2007/054770 2007/20 18.05.2007<br />

(30) 08.11.2005 US 73<strong>50</strong>91 P<br />

(54) • Zur Behandlung gynäkologischer Erkrankungen<br />

geeignete Pyrazolderivate<br />

• Pyrazole derivatives useful for the treatment<br />

of gynaecological diseases<br />

• Dérivés de pyrazole utiles pour le traitement<br />

de troubles gynécologiques<br />

(73) Pfizer Limited, Ramsgate Road, Sandwich,<br />

Kent CT13 9NJ, GB<br />

(72) BRADLEY, Paul, Anthony, Kent CT13 9NJ,<br />

GB<br />

DACK, Kevin, Neil, Kent CT13 9NJ, GB<br />

JOHNSON, Patrick, Stephen, Kent CT13 9NJ,<br />

GB<br />

SKERRATT, Sarah, Elizabeth, Kent CT13 9NJ,<br />

GB<br />

(74) Ruddock, Keith Stephen, et al, Pfizer Limited<br />

<strong>European</strong> <strong>Patent</strong> Department Ramsgate<br />

Road, Sandwich Kent CT13 9NJ, GB<br />

(51) C07D 231/54 (11) 2 089 367 B1<br />

C07D 401/04 C07D 405/04<br />

C07D 493/04 A61K 31/416<br />

A61K 31/4162 A61P 9/12<br />

(25) En (26) En<br />

(21) 07825488.5 (22) 17.10.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(43) 19.08.2009<br />

(86) IB 2007/003207 17.10.2007<br />

(87) WO 2008/053300 2008/19 08.05.2008<br />

(30) 31.10.2006 US 863606 P<br />

(54) • PYRAZOLINVERBINDUNGEN ALS MINE-<br />

RALOCORTICOIDREZEPTORANTAGONIS-<br />

TEN<br />

• PYRAZOLINE COMPOUNDS AS MINERA-<br />

LOCORTICOID RECEPTOR ANTAGONISTS<br />

• COMPOSÉS DE PYRAZOLINE EN TANT<br />

QU'ANTAGONISTES DES RÉCEPTEURS<br />

MINÉRALOCORTICOÏDES<br />

(73) Pfizer Products Inc., Eastern Point Road,<br />

Groton, CT 06340, US<br />

566<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>50</strong>/<strong>2011</strong>) 14.12.<strong>2011</strong><br />

(72) MEYERS, Marvin Jay, Chesterfield, MO<br />

63017-1732, US<br />

ARHANCET, Graciela Barbieri, Chesterfield,<br />

MO 63017-1732, US<br />

CHEN, Xiangyang, Chesterfield, MO 63017-<br />

1732, US<br />

HOCKERMAN, Susan Landis, Chesterfield,<br />

MO 63017-1732, US<br />

LONG, Scott, Allen, Chesterfield, MO 63017-<br />

1732, US<br />

MAHONEY, Matthew, William, Chesterfield,<br />

MO 63017-1732, US<br />

REITZ, David, Bruce, Chesterfield, MO<br />

63017, US<br />

RICO, Joseph Gerace, Chesterfield, MO<br />

63017-1732, US<br />

(74) Dekker, Henrike Cornelie Christine, Pfizer<br />

Limited <strong>European</strong> <strong>Patent</strong> Department Ramsgate<br />

Road, Sandwich, Kent CT13 9NJ, GB<br />

C07D 231/56 → (51) C07D 417/12<br />

(51) C07D 233/54 (11) 1 893 582 B1<br />

C07D 249/08 C07D 257/04<br />

C07D 263/32 C07D 277/24<br />

C07D 417/12 A61K 31/41<br />

A61K 31/4164 A61K 31/4196<br />

A61K 31/421 A61K 31/427<br />

A61P 3/10 A61P 3/04<br />

A61P 3/06<br />

(25) En (26) En<br />

(21) 06770714.1 (22) 18.05.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK YU<br />

(43) 05.03.2008<br />

(86) US 2006/019545 18.05.2006<br />

(87) WO 2006/127<strong>50</strong>3 2006/48 30.11.2006<br />

(30) 20.05.2005 US 683331 P<br />

17.05.2006 US 436732<br />

(54) • Verbindungen, ihre pharmazeutischen<br />

Zusammensetzungen und ihre Verwendung<br />

in der Behandlung von Stoffwechselstörungen<br />

• Compounds, their pharmaceutical compositions<br />

and their use in treating metabolic<br />

disorders<br />

• Composés, leur compositions pharmaceutiques<br />

et leur utilisation dans le traitment<br />

des troubles du métabolisme<br />

(73) Amgen, Inc, <strong>Patent</strong> Operations, M/S 28-2-C<br />

One Amgen Center Drive, Thousand Oaks,<br />

California 91320-1799, US<br />

(72) HOUZE, Jonathan, San Mateo, California<br />

94402, US<br />

LIU, Jiwen, Foster City, California 94404, US<br />

MA, Zhihua, San Mateo, California 94403,<br />

US<br />

MEDINA, Julio C., San Carlos, California<br />

94070, US<br />

SCHMITT, Michael J., Oakland, California<br />

94608, US<br />

SHARMA, Rajiv, Fremont, California 94555,<br />

US<br />

SUN, Ying, Albany, California 94706, US<br />

WANG, Yingcai, Fremont, California 94555,<br />

US<br />

ZHU, Liusheng, Burlingame, California<br />

94010, US<br />

(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser,<br />

Leopoldstrasse 4, 80802 München,<br />

DE<br />

(51) C07D 239/10 (11) 1 794 133 B1<br />

C07D 401/02 A61K 31/435<br />

A61K 31/499<br />

(25) En (26) En

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