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Bulletin 2009/49 - European Patent Office

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(A61P) I.1(1)<br />

A61P 29/00 → (51) A61K 31/70<br />

A61P 29/00 → (51) A61K 31/7004<br />

A61P 29/00 → (51) A61K 35/74<br />

A61P 29/00 → (51) A61K 45/06<br />

A61P 29/00 → (51) A61L 27/54<br />

A61P 29/00 → (51) C07D 211/70<br />

A61P 29/00 → (51) C07D 213/61<br />

A61P 29/00 → (51) C07D 213/81<br />

A61P 29/00 → (51) C07D 231/12<br />

A61P 29/00 → (51) C07D 233/10<br />

A61P 29/00 → (51) C07D 401/12<br />

A61P 29/00 → (51) C07D 401/14<br />

A61P 29/00 → (51) C07D 403/04<br />

A61P 29/00 → (51) C07D 413/04<br />

A61P 29/00 → (51) C07D 471/04<br />

A61P 29/00 → (51) C07D <strong>49</strong>8/04<br />

A61P 29/00 → (51) C12N 15/11<br />

A61P 29/00 → (51) C12N 15/62<br />

A61P 29/02 → (51) A61K 31/195<br />

A61P 31/00 → (51) A61K 9/08<br />

A61P 31/00 → (51) A61K 9/107<br />

A61P 31/00 → (51) A61K 31/403<br />

A61P 31/00 → (51) A61K 33/16<br />

A61P 31/00 → (51) C07D 213/61<br />

A61P 31/00 → (51) C07D 471/06<br />

A61P 31/00 → (51) C07D <strong>49</strong>8/04<br />

A61P 31/02 → (51) A61K 38/04<br />

A61P 31/04 → (51) A23K 1/18<br />

A61P 31/04 → (51) A61K 31/427<br />

A61P 31/04 → (51) A61K 35/74<br />

A61P 31/04 → (51) A61K 38/04<br />

A61P 31/04 → (51) C07D 471/04<br />

A61P 31/04 → (51) C07H 17/08<br />

A61P 31/06 → (51) C07H 13/06<br />

A61P 31/10 → (51) A61K 31/137<br />

A61P 31/10 → (51) C07D 233/10<br />

A61P 31/10 → (51) C07D 401/14<br />

A61P 31/12 → (51) A61K 47/48<br />

A61P 31/12 → (51) C07H 7/00<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

A61P 31/12 → (51) C07H 21/00<br />

(51) A61P 31/14 (11) 2 125 113 A2*<br />

A61K 38/06 C07K 5/08<br />

(25) En (26) En<br />

(21) 08726107.9 (22) 26.02.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) US 2008/002524 26.02.2008<br />

(87) WO 2008/106130 2008/36 04.09.2008<br />

(88) 02.10.2008<br />

(30) 26.02.2007 US 891634 P<br />

(54) • TERTIÄRAMIN-SUBSTITUIERTE PEPTIDE<br />

ALS HCV-REPLIKATIONSHEMMER<br />

• TERTIARY AMINE SUBSTITUTED PEP-<br />

TIDES USEFUL AS INHIBITORS OF HCV<br />

REPLICATION<br />

• PEPTIDES SUBSTITUÉS PAR UNE AMINE<br />

TERTIAIRE UTILES COMME INHIBITEURS<br />

DE LA RÉPLICATION DU VIRUS DE<br />

L'HÉPATITE C<br />

(71) Achillion Pharmaceuticals, Inc., 300 George<br />

Street, New Haven, CT 06511, US<br />

(72) AGARWAL, Atul, Hamden, CT 06518, US<br />

WANG, Xiangzhu, Branford, CT 06405, US<br />

CHEN, Dawei, Middletown, CT 06457, US<br />

ZHANG, Suoming, Madison, CT 06443, US<br />

PHADKE, Avinash, Branford, CT 06405, US<br />

(74) Smaggasgale, Gillian Helen, W.P. Thompson<br />

& Co, 55 Drury Lane, London WC2B 5SQ,<br />

GB<br />

A61P 31/14 → (51) A61K 38/16<br />

A61P 31/14 → (51) C07D 257/02<br />

A61P 31/14 → (51) C07K 5/08<br />

A61P 31/14 → (51) C07K 16/10<br />

A61P 31/16 → (51) A61K 36/185<br />

A61P 31/18 → (51) C07D 401/12<br />

A61P 33/02 → (51) A61K 47/48<br />

A61P 33/06 → (51) A61K 31/52<br />

A61P 35/00 → (51) A61K 31/409<br />

A61P 35/00 → (51) A61K 31/4184<br />

A61P 35/00 → (51) A61K 31/437<br />

A61P 35/00 → (51) A61K 31/506<br />

A61P 35/00 → (51) A61K 39/395<br />

A61P 35/00 → (51) A61K 45/06<br />

A61P 35/00 → (51) A61K 47/48<br />

A61P 35/00 → (51) A61K 48/00<br />

A61P 35/00 → (51) C07C 311/37<br />

A61P 35/00 → (51) C07C 327/44<br />

A61P 35/00 → (51) C07D 209/12<br />

A61P 35/00 → (51) C07D 213/61<br />

A61P 35/00 → (51) C07D 231/40<br />

A61P 35/00 → (51) C07D 233/96<br />

A61P 35/00 → (51) C07D 239/84<br />

99<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>49</strong>/<strong>2009</strong>) 02.12.<strong>2009</strong><br />

A61P 35/00 → (51) C07D 401/04<br />

A61P 35/00 → (51) C07D 409/14<br />

A61P 35/00 → (51) C07D 417/12<br />

A61P 35/00 → (51) C07D 471/04<br />

A61P 35/00 → (51) C07D 473/34<br />

A61P 35/00 → (51) C07D 487/04<br />

A61P 35/00 → (51) C07H 21/00<br />

A61P 35/00 → (51) C07J 43/00<br />

A61P 35/00 → (51) C07K 16/00<br />

A61P 35/00 → (51) C07K 16/30<br />

A61P 35/00 → (51) C12N 5/18<br />

A61P 35/00 → (51) C12N 15/11<br />

A61P 35/00 → (51) C12N 15/62<br />

A61P 35/00 → (51) C12Q 1/68<br />

A61P 35/04 → (51) A61K 31/167<br />

A61P 37/00 → (51) A61K 31/506<br />

A61P 37/00 → (51) A61K 38/17<br />

A61P 37/00 → (51) C07D 211/06<br />

A61P 37/00 → (51) C07D 213/73<br />

A61P 37/00 → (51) C07D 403/04<br />

A61P 37/00 → (51) C07D 413/04<br />

A61P 37/00 → (51) C07D 471/04<br />

A61P 37/00 → (51) C07D 487/04<br />

A61P 37/00 → (51) C07K 16/28<br />

A61P 37/04 → (51) C12N 5/18<br />

A61P 37/06 → (51) A61K 9/08<br />

A61P 37/06 → (51) C07K 16/28<br />

A61P 37/08 → (51) A61K 31/506<br />

A61P 37/08 → (51) C07D 211/70<br />

A61P 37/08 → (51) C07D 471/04<br />

A61P 39/06 → (51) A61K 31/7004<br />

A61P 39/06 → (51) C07D <strong>49</strong>8/04<br />

A61P 43/00 → (51) A61K 31/34<br />

A61P 43/00 → (51) A61K 31/506<br />

A61P 43/00 → (51) A61K 38/21<br />

A61P 43/00 → (51) A61K 47/48<br />

A61Q 5/00 → (51) A61K 8/04<br />

A61Q 5/02 → (51) A61K 8/88<br />

A61Q 5/04 → (51) C07K 1/113

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