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Bulletin 2009/49 - European Patent Office

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(C07D) I.1(1)<br />

(51) C07D 471/06 (11) 2 125 813 A2*<br />

C07D 519/00 A61K 31/437<br />

A61K 31/436 A61K 31/<strong>49</strong>5<br />

A61P 31/00<br />

(25) En (26) En<br />

(21) 08718070.9 (22) 20.03.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) EP 2008/053350 20.03.2008<br />

(87) WO 2008/116815 2008/40 02.10.2008<br />

(88) 11.12.2008<br />

(30) 23.03.2007 GB 0705672<br />

(54) • VERBINDUNGEN<br />

• COMPOUNDS<br />

• COMPOSÉS<br />

(71) Glaxo Group Limited, Glaxo Wellcome House<br />

Berkeley Avenue, Greenford Middlesex UB6<br />

0NN, GB<br />

(72) BROWN, Pamela, Stevenage Hertfordshire<br />

SG1 2NY, GB<br />

DABBS, Steven, Stevenage Hertfordshire<br />

SG1 2NY, GB<br />

DAVIES, David, Thomas, Stevenage Hertfordshire<br />

SG1 2NY, GB<br />

PEARSON, Neil, David, Collegeville, Pennsylvania<br />

19426, US<br />

(74) Valentine, Jill Barbara, GlaxoSmithKline<br />

Corporate Intellectual Property (CN9.25.1)<br />

980 Great West Road, Brentford, Middlesex<br />

TW8 9GS, GB<br />

C07D 471/10 → (51) C07D 211/16<br />

C07D 471/10 → (51) C07D 213/16<br />

C07D 471/14 → (51) C07D 213/73<br />

(51) C07D 473/00 (11) 2 125 814 A1*<br />

(25) En (26) En<br />

(21) 07857990.1 (22) 20.12.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

BA HR RS<br />

(86) EP 2007/064371 20.12.2007<br />

(87) WO 2008/074874 2008/26 26.06.2008<br />

(30) 21.12.2006 EP 06126797<br />

21.12.2006 US 871347 P<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

ABACAVIR<br />

• PROCESS FOR THE PREPARATION OF<br />

ABACAVIR<br />

• PROCÉDÉ POUR LA PRÉPARATION<br />

D'ABACAVIR<br />

(71) Esteve Química, S.A., Av. Mare de Déu de<br />

Montserrat 12, 08024 Barcelona, ES<br />

(72) MEDRANO RUPÉREZ, Jorge, 08024 Barcelona,<br />

ES<br />

CAMPON PARDO, Julio, 08024 Barcelona,<br />

ES<br />

ELÍAS RIUS, Laia, 08024 Barcelona, ES<br />

BERENGUER MAIMÓ, Ramón, 08024 Barcelona,<br />

ES<br />

(74) Jané Bonet, Montserrat, ZBM <strong>Patent</strong>s, S.L.<br />

Balmes, 114, 4°, 08008 Barcelona, ES<br />

C07D 473/16 → (51) A61K 31/52<br />

C07D 473/18 → (51) A61K 31/52<br />

(51) C07D 473/34 (11) 2 125 815 A2*<br />

A61K 31/52 A61P 35/00<br />

(25) En (26) En<br />

(21) 08744161.4 (22) 21.03.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

AL BA MK RS<br />

(86) US 2008/057771 21.03.2008<br />

(87) WO 2008/116129 2008/39 25.09.2008<br />

(88) 12.02.<strong>2009</strong><br />

(30) 21.03.2007 US 919300 P<br />

(54) • IMIDAZOLOPYRIMIDINANALOGA UND<br />

IHRE VERWENDUNG ALS PI3-KINASE-<br />

UND MTOR-HEMMER<br />

• IMIDAZOLOPYRIMIDINE ANALOGS AND<br />

THEIR USE AS PI3 KINASE AND MTOR<br />

INHIBITORS<br />

• ANALOGUES D'IMIDAZOLOPYRIMIDINE<br />

ET LEUR UTILISATION COMME INHIBI-<br />

TEURS DE PI3 KINASE ET DE MTOR<br />

(71) Wyeth, Five Giralda Farms, Madison, NJ<br />

07940, US<br />

(72) BURSAVICH, Matthew, Gregory, Sandy, UT<br />

84070, US<br />

VENKATESAN, Aranapakam, Mudumbai,<br />

Rego Park, NY 11374, US<br />

NOWAK, Pawel, Wojciech, Montvale, NJ<br />

07645, US<br />

LOMBARDI, Sabrina, New Haven, CT 06511,<br />

US<br />

GILBERT, Adam, Matthew, Congers, NY<br />

10920, US<br />

DEHNHARDT, Christoph, Martin, New York,<br />

NY 10028, US<br />

DOS SANTOS, Osvaldo, Astoria, NY 11106,<br />

US<br />

DELOS SANTOS, Efren, Guillermo, Nanuet,<br />

NY 10954, US<br />

BROOIJMANS, Natasja, New York, NY<br />

10021, US<br />

AYRAL-KALOUSTIAN, Semiramis, Tarrytown,<br />

NY 10591, US<br />

CHEN, Zecheng, New City, NY 10956, US<br />

VERHEIJEN, Jeroen, Cunera, Highland Mills,<br />

NY 10930, US<br />

KAPLAN, Joshua, Nyack, NY 10960, US<br />

ZASK, Arie, New York, NY 10128, US<br />

(74) Fletcher, Rodney Justin, Wyeth Pharmaceuticals<br />

Huntercombe Lane South, Taplow,<br />

Maidenhead Berkshire SL6 0PH, GB<br />

C07D 473/34 → (51) A61K 31/52<br />

C07D 473/34 → (51) C07D 471/04<br />

C07D 473/34 → (51) C07D 487/04<br />

(51) C07D 487/02 (11) 2 125 816 A2*<br />

C07D <strong>49</strong>8/02 A61P 19/00<br />

A61K 31/5365 A61K 31/5355<br />

(25) En (26) En<br />

(21) 08726687.0 (22) 07.03.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/003191 07.03.2008<br />

(87) WO 2008/109177 2008/37 12.09.2008<br />

(88) 22.01.<strong>2009</strong><br />

(30) 07.03.2007 US 905565 P<br />

(54) • METALLOPROTEASEHEMMER MIT EINEM<br />

HETEROCYCLISCHEN TEIL<br />

• METALLOPROTEASE INHIBITORS CON-<br />

TAINING A HETEROCYCLIC MOIETY<br />

• INHIBITEURS DE MÉTALLOPROTÉASE<br />

CONTENANT UNE FRACTION HÉTÉROCY-<br />

CLIQUE<br />

(71) Alantos Pharmaceuticals Holding, Inc., One<br />

Amgen Center Drive, Thousand Oaks, CA<br />

91320, US<br />

(72) GEGE, Christian, 69256 Mauer, DE<br />

TAVERAS, Arthur, Southborough, MA<br />

01772, US<br />

192<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>49</strong>/<strong>2009</strong>) 02.12.<strong>2009</strong><br />

(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser<br />

Anwaltssozietät, Leopoldstrasse 4,<br />

80802 München, DE<br />

C07D 487/02 → (51) C07D 213/73<br />

(51) C07D 487/04 (11) 2 125 817 A1*<br />

(25) En (26) En<br />

(21) 08723315.1 (22) 07.03.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) KR 2008/001278 07.03.2008<br />

(87) WO 2008/117943 2008/40 02.10.2008<br />

(30) 23.03.2007 KR 20070028620<br />

(54) • 7-(3',4'-DIALKOXYPHENYL)-[1,2,4]-TRIA-<br />

ZOL-[1,5-A]-PYRIMIDIN-VERBINDUNGEN,<br />

VERFAHREN ZU IHRER HERSTELLUNG<br />

UND PHARMAZEUTISCHE ZUSAMMEN-<br />

SETZUNG DAMIT ZUR BEHANDLUNG<br />

ODER VERHINDERUNG VON ASTHMA,<br />

CHRONISCHER OBSTRUKTIVER LUNGEN-<br />

ERKRANKUNG, ARTHRITIS, ATOPISCHER<br />

DERMATITIS, TUMOREN UND DEGENE-<br />

RATIVEN HIRNERKRANKUNGEN<br />

• 7-(3',4'-DIALKOXYPHENYL)-[1,2,4]-TRIA-<br />

ZOLO[1,5-A]PYRIMIDINE COMPOUNDS,<br />

PROCESS FOR PREPARING THEREOF,<br />

AND PHARMACEUTICAL COMPOSITION<br />

FOR TREATING OR PREVENTING<br />

ASTHMA, CHRONIC OBSTRUCTIVE PUL-<br />

MONARY DISEASE, ARTHRITIS, ATOPIC<br />

DERMATITIS, TUMOR AND DEGENERA-<br />

TIVE BRAIN DISEASES COMPRISING THE<br />

SAME<br />

• COMPOSÉS {7-(3 ', 4 '-DIALKOXYPHÉ-<br />

NYL) - [1,2,4]-TRIAZOLO [1,5-A]PYRIMI-<br />

DINE LEUR PROCÉDÉ DE PRÉPARATION<br />

ET COMPOSITIONS PHARMACEUTIQUES<br />

LES CONTENANT, POUR LE TRAITEMENT<br />

OU LA PREVENTION DE L'ASTHME, DE LA<br />

BRONCHOPNEUMOPATHIE CHRONIQUE<br />

OBSTRUCTIVE, DE L'ARTHRITE, DE LA<br />

DERMATITE ATOPIQUE,<br />

(71) Korea Research Institute of Chemical Technology,<br />

100, Jang-dong, Yuseong-gu, Daejeon<br />

305-600, KR<br />

(72) JEON, Dong Ju, Daejeon 305-707, KR<br />

NO, Zaesung, Chungcheongnam-do 339-<br />

831, KR<br />

SONG, Jong Hwan, Chungcheongbuk-do<br />

373-806, KR<br />

LEE, Gehyeong, Daejeon 305-755, KR<br />

KIM, Ikyon, Daejeon 305-761, KR<br />

PARK, Chang Min, Gimcheon-si Gyeongsangbuk-do<br />

740-983, KR<br />

CHEON, Hyae Gyeong, Daejeon 305-772, KR<br />

CHO, Young Sik, Daejeon 305-308, KR<br />

SONG, Jin Sook, Daejeon 305-509, KR<br />

BAE, Myung Ae, Daejeon 305-752, KR<br />

YOO, Sung-eun, Gongju-si Chungcheongnam-do<br />

314-911, KR<br />

(74) Scheele, Friedrich, et al, Stolmár Scheele &<br />

Partner <strong>Patent</strong>anwälte Blumenstrasse 17,<br />

80331 München, DE<br />

(51) C07D 487/04 (11) 2 125 818 A1*<br />

A61K 31/519 A61P 35/00<br />

(25) En (26) En<br />

(21) 08727890.9 (22) 18.01.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/051408 18.01.2008<br />

(87) WO 2008/089390 2008/30 24.07.2008<br />

(30) 19.01.2007 US 885719 P<br />

(54) • NEUE KLASSISCHE ANTIFOLATE<br />

• NEW CLASSICAL ANTIFOLATES

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