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Bulletin 2009/49 - European Patent Office

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(C07D) II.1(1)<br />

(25) En (26) En<br />

(21) 037959<strong>49</strong>.1 (22) 22.12.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 12.10.2005<br />

(86) EP 2003/014720 22.12.2003<br />

(87) WO 2004/060870 2004/30 22.07.2004<br />

(30) 02.01.2003 EP 03000003<br />

(54) • CB 1 REZEPTOR INVERSAGONISTEN<br />

• CB 1 RECEPTOUR INVERSE AGONISTS<br />

• AGONISTES INVERSES DU RECEPTEUR<br />

CB 1<br />

(73) F. Hoffmann-La Roche AG, Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

(72) MAYWEG, Alexander, CH-4051 Basel, CH<br />

MARTY, Hans, Peter, CH-4055 Basel, CH<br />

MUELLER, Werner, CH-4147 Aesch, CH<br />

NARQUIZIAN, Robert, F-68300 St. Louis, FR<br />

NEIDHART, Werner, F-68220 Hagenthal-le-<br />

Bas, FR<br />

PFLIEGER, Philippe, F-68130 Schwoben, FR<br />

ROEVER, Stephan, 79594 Inzlingen, DE<br />

(74) Klostermeyer-Rauber, Dörte, et al, Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

C07D 209/02 → (51) C07D 409/00<br />

(51) C07D 209/30 (11) 1 551 802 B1<br />

A61K 31/405 A61P 11/00<br />

(25) En (26) En<br />

(21) 03764279.0 (22) 15.07.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

AL LT LV MK<br />

(43) 13.07.2005<br />

(86) SE 2003/001216 15.07.2003<br />

(87) WO 2004/007451 2004/04 22.01.2004<br />

(30) 17.07.2002 SE 0202241<br />

13.12.2002 SE 0203713<br />

(54) • INDOL-3-SCHWEFELDERIVATE<br />

• INDOLE-3-SULPHUR DERIVATIVES<br />

• DERIVES D'INDOLE-3-SOUFRE<br />

(73) AstraZeneca AB, 151 85 Södertälje, SE<br />

(72) BONNERT, Roger AstraZeneca R & D<br />

Charnwood, Leicestershire LE11 5RH, GB<br />

DICKINSON, Mark AstraZeneca R & D<br />

Charnwood, Leicestershire LE11 5RH, GB<br />

MOHAMMED, Rukhsana AstraZeneca R & D<br />

Charnwood, Loughborough Leicestershire<br />

LE11 5RH, GB<br />

SANGANEE, Hitesh AstraZeneca R & D<br />

Charnwood, Leicestershire LE11 5RH, GB<br />

TEAGUE, Simon AstraZeneca R & D Charnwood,<br />

Leicestershire LE11 5RH, GB<br />

C07D 209/48 → (51) C07D 403/04<br />

C07D 211/40 → (51) G01N 33/50<br />

(51) C07D 211/46 (11) 1 546 102 B1<br />

C09D 167/08 C09K 3/30<br />

C08G 18/32 C09D 7/02<br />

C09B 67/00 C08G 18/64<br />

C09D 17/00 C08G 18/79<br />

C08J 7/04 C09D 167/00<br />

C08L 57/00 A61K 9/28<br />

(25) En (26) En<br />

(21) 0378<strong>49</strong>86.6 (22) 08.08.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 29.06.2005<br />

(86) US 2003/024714 08.08.2003<br />

(87) WO 2004/014858 2004/08 19.02.2004<br />

(30) 10.08.2002 US 402859 P<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(54) • AN KUNSTSTOFF ANHAFTENDE AERO-<br />

SOLFARBZUSAMMENSETZUNG<br />

• AEROSOL PAINT COMPOSITION FOR<br />

ADHERENCE TO PLASTIC<br />

• COMPOSITION DE PEINTURE EN AERO-<br />

SOL DESTINEE A ADHERER AU PLAS-<br />

TIQUE<br />

(73) The Sherwin-Williams Company, 101 W.<br />

Prospect Avenue, Cleveland, OH 44115, US<br />

(72) REDDING, Patricia, L., South Euclid, OH<br />

44124, US<br />

(74) Morf, Jan Stefan, et al, Abitz & Partner<br />

<strong>Patent</strong>anwälte Postfach 86 01 09, 81628<br />

München, DE<br />

(51) C07D 211/58 (11) 1 434 765 B1<br />

C07D 405/12 C07D 401/12<br />

C07D 413/12 C07D 409/12<br />

A61K 31/4545 A61P 3/04<br />

(25) En (26) En<br />

(21) 02764567.0 (22) 11.09.2002<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR IE IT LI LU MC NL PT SE SK TR<br />

(43) 07.07.2004<br />

(86) DK 2002/000594 11.09.2002<br />

(87) WO 2003/02<strong>49</strong>29 2003/13 27.03.2003<br />

(30) 14.09.2001 DK 200101344<br />

(54) • SUBSTITUIERTE PIPERIDINEN MIT<br />

SELEKTIVER BINDUNGSFÄHIGKEIT ZU<br />

HISTAMIN H3-REZEPTOREN<br />

• SUBSTITUTED PIPERIDINES WITH<br />

SELECTIVE BINDING TO HISTAMINE H3-<br />

RECEPTOR<br />

• PIPERIDINES SUBSTITUEES AVEC LIAI-<br />

SON SELECTIVE AU RECEPTEUR H3 DE<br />

L'HISTAMINE<br />

(73) High Point Pharmaceuticals, LLC, 4170<br />

Mendenhall Oaks Parkway, High Point, NC<br />

27265, US<br />

(72) DÖRWALD, Florencio, Zaragoza, DK-2750<br />

Ballerup, DK<br />

(74) Bailey, Lindsey, et al, Elkington and Fife LLP<br />

Thavies Inn House 3-4 Holborn Circus,<br />

London EC1N 2HA, GB<br />

C07D 211/58 → (51) C07D 401/14<br />

(51) C07D 211/94 (11) 1 515 950 B1<br />

C07D 241/08 C07F 9/38<br />

C08F 2/00<br />

(25) En (26) En<br />

(21) 03740262.5 (22) 17.06.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 23.03.2005<br />

(86) EP 2003/006370 17.06.2003<br />

(87) WO 2004/000809 2004/01 31.12.2003<br />

(30) 24.06.2002 EP 02405520<br />

(54) • KATIONISCHE ALKOXYAMINEN ZUR VER-<br />

WENDUNG IN DER HERSTELLUNG VON<br />

NANOPARTIKELN VON NATÜRLICHEN<br />

ODER SYNTHETISCHEN CLAYS<br />

• CATIONIC ALKOXYAMINES AND THEIR<br />

USE IN PRODUCING NANO PARTICLES<br />

FROM NATURAL OR SYNTHETIC CLAYS<br />

• ALKOXYAMINES CATIONIQUES ET UTILI-<br />

SATION DANS LA PRODUCTION DE<br />

NANOPARTICULES A PARTIR D'ARGILES<br />

NATURELLES OU SYNTHETIQUES<br />

(73) BASF SE, 67056 Ludwigshafen, DE<br />

(72) MÜHLEBACH, Andreas, CH-5070 Frick, CH<br />

NESVADBA, Peter, CH-1723 Marly, CH<br />

KRAMER, Andreas, CH-3280 Meyriez, CH<br />

C07D 213/38 → (51) A61K 31/5375<br />

C07D 213/75 → (51) A61K 31/5375<br />

871<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>49</strong>/<strong>2009</strong>) 02.12.<strong>2009</strong><br />

C07D 213/80 → (51) A61K 31/5375<br />

C07D 213/82 → (51) A61K 31/5375<br />

(51) C07D 215/22 (11) 1 520 855 B1<br />

C07D 471/04 C07D <strong>49</strong>5/04<br />

A61K 31/47 A61K 31/435<br />

A61P 15/00 A61P 35/00<br />

(25) En (26) En<br />

(21) 04078019.9 (22) 11.12.2001<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

(43) 06.04.2005<br />

(30) 12.12.2000 US 254827 P<br />

14.11.2001 US 992785<br />

(54) • Thieno¬2,3-B pyridin-derivate als Antagonisten<br />

des Gonadotropin-freisetzenden<br />

Hormons<br />

• Thieno(2,3-b)pyridine derivatives useful as<br />

antagonists of gonadotropin releasing<br />

hormone<br />

• Derivés de thieno¬2,3 pyridine comme<br />

antagonistes de l'hormone de liberation de<br />

gonadotropine<br />

(73) Ortho-McNeil-Janssen Pharmaceuticals, Inc.,<br />

1125 Trenton-Harbourton Road, Titusville,<br />

NJ 08560, US<br />

(72) Sui, Zhihua, Flemington NJ 08822, US<br />

Macielag, Mark, Branchburg NJ 08876, US<br />

Lanter, James C., Flemington NJ 08822, US<br />

(74) Mercer, Christopher Paul, et al, Carpmaels &<br />

Ransford 43-45 Bloomsbury Square, London<br />

WC1A 2RA, GB<br />

(62) 01990166.9 / 1 345 907<br />

(51) C07D 215/26 (11) 1 622 875 B1<br />

A61K 31/4704 A61P 11/06<br />

(25) En (26) En<br />

(21) 04751604.2 (22) 07.05.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

LT LV<br />

(43) 08.02.2006<br />

(86) US 2004/014302 07.05.2004<br />

(87) WO 2004/101525 2004/48 25.11.2004<br />

(30) 08.05.2003 US 468810 P<br />

(54) • KRISTALLINE FORMEN EINES ARYLANI-<br />

LIN-BETA-2-ADRENERGENREZEPTOR-<br />

AGONISTS<br />

• CRYSTALLINE FORMS OF AN ARYLANI-<br />

LINE BETA-2 ADRENERGIC RECEPTOR<br />

AGONIST<br />

• FORMES CRISTALLINES D'UN AGONISTE<br />

ARYLANILINE DU RÉCEPTEUR ADRÉNER-<br />

GIQUE BÊTA-2<br />

(73) Theravance, Inc., 901 Gateway Boulevard,<br />

South San Francisco, CA 94080, US<br />

(72) AXT, Sabine, Sunnyvale, CA 94085, US<br />

STERGIADES, Ioanna, San Francisco, CA<br />

94109, US<br />

(74) Scott, Susan Margaret, et al, Abel & Imray 20<br />

Red Lion Street, London WC1R 4PQ, GB<br />

(51) C07D 215/26 (11) 1 791 820 B1<br />

C07D 251/26<br />

(25) En (26) En<br />

(21) 05770221.9 (22) 21.06.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

AL BA HR LV MK YU<br />

(43) 06.06.2007<br />

(86) EP 2005/006686 21.06.2005<br />

(87) WO 2005/123684 2005/52 29.12.2005<br />

(30) 22.06.2004 GB 0413960

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