Bulletin 2009/49 - European Patent Office

(A61K) I.1(1)
(71) IRM LLC, 131 Front Street PO Box HM 2899,
Hamilton HM LX, BM
The Scripps Research Institute, 10550 North
Torrey Pines Road, La Jolla, CA 92037, US
(72) WINZELER, Elizabeth, San Diego, California
92130, US
GRAY, Nathanael S., Boston, Massachusetts
02130, US
HAN, Dong, San Diego, California 92014, US
CHENG, Dai, San Diego, California 92126,
US
(74) Kiddle, Simon John, et al, Mewburn Ellis LLP
33 Gutter Lane, London EC2V 8AS, GB
A61K 31/52 → (51) C07D 471/04
A61K 31/52 → (51) C07D 473/34
(51) A61K 31/53 (11) 2 124 955 A2*
G01N 33/573 G01N 33/68
A61P 9/04 A61P 9/10
A61P 9/12
(25) De (26) De
(21) 07818641.8 (22) 02.10.2007
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HU IE IS IT LI LT LU LV MC MT NL PL PT
RO SE SI SK TR
(86) EP 2007/008561 02.10.2007
(87) WO 2008/043461 2008/16 17.04.2008
(88) 28.08.2008
(30) 14.10.2006 DE 102006048693
(54) • INHIBITION DER PDE2A
• INHIBITION OF PDE2A
• INHIBITION DE LA PDE2A
(71) Bayer Schering Pharma Aktiengesellschaft,
Müllerstrasse 178, 13353 Berlin, DE
(72) ELLINGHAUS, Peter, 42113 Wuppertal, DE
WILMEN, Andreas, 50676 Köln, DE
HENDRIX, Martin, 51519 Odenthal, DE
TERSTEEGEN, Adrian, 42111 Wuppertal, DE
A61K 31/53 → (51) A61K 45/06
A61K 31/53 → (51) C07D 487/04
A61K 31/535 → (51) C07C 311/37
A61K 31/5355 → (51) C07D 487/02
A61K 31/5365 → (51) C07D 487/02
A61K 31/5375 → (51) A61K 31/135
A61K 31/5375 → (51) C07D 498/04
A61K 31/5377 → (51) A61K 31/52
A61K 31/5377 → (51) C07D 211/16
A61K 31/5377 → (51) C07D 217/24
A61K 31/5383 → (51) C07D 498/04
(51) A61K 31/5415 (11) 2 124 956 A1*
A61P 13/00
(25) Fr (26) Fr
(21) 07858150.1 (22) 26.12.2007
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HU IE IS IT LI LT LU LV MC MT NL PL PT
RO SE SI SK TR
AL BA HR MK RS
(86) EP 2007/064553 26.12.2007
(87) WO 2008/080924 2008/28 10.07.2008
(30) 28.12.2006 FR 0656002
Europäisches Patentblatt
European Patent Bulletin
Bulletin européen des brevets
(54) • VERWENDUNG VON 10-[(3R)-1-AZABI-
CYCLO[2.2.2]OCT-3-YLMETHYL]-10H-
PHENOTHIAZIN FÜR DIE ZUBEREITUNG
EINES WIRKSTOFFES MIT SELEKTIVER
HEMMUNG DER MUSKARIN-REZEPT-
OREN M1, M2 UND M3
• USE OF 10-[(3R)-1-AZABICYCLO[2.2.2]
OCT-3-YLMETHYL]-10H-PHENOTHIAZINE
FOR THE PREPARATION OF A DRUG
HAVING A SELECTIVE INHIBITION OF
MUSCARINIC M1, M2 AND M3 RECEP-
TORS
• UTILISATION DU 10-[(3R)-1-AZABICY-
CLO]2.2.2]OCT-3-YLMÉTHYL]-10H-PHÉ-
NOTHIAZINE POUR LA PRÉPARATION
D'UN MÉDICAMENT EXERÇANT UNE
INHIBITION SÉLECTIVE DES RÉCEPTEURS
MUSCARINIQUES M1, M2 ET M3
(71) Pierre Fabre Medicament, 45 Place Abel
Gance, 92100 Boulogne-Billancourt, FR
(72) CLERC, Thierry, F-31320 Vigoulet Auzil, FR
TISNE-VERSAILLES, Jacky, F-81100 Castres,
FR
PRZYBYLSKI, Christophe, F-31290 Villefranche
De Lauragais, FR
(74) Ahner, Francis, et al, Cabinet Régimbeau 20,
rue de Chazelles, 75847 Paris cedex 17, FR
A61K 31/545 → (51) A61K 9/08
A61K 31/545 → (51) A61K 31/403
A61K 31/546 → (51) A61K 31/403
A61K 31/55 → (51) A01N 43/00
A61K 31/55 → (51) A61K 31/135
A61K 31/55 → (51) A61K 31/52
A61K 31/551 → (51) A61K 31/506
A61K 31/5513 → (51) A61K 31/52
A61K 31/553 → (51) A61K 31/52
(51) A61K 31/554 (11) 2 124 957 A1*
(25) En (26) En
(21) 08732646.8 (22) 21.03.2008
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HR HU IE IS IT LI LT LU LV MC MT NL
NO PL PT RO SE SI SK TR
(86) US 2008/057808 21.03.2008
(87) WO 2008/116144 2008/39 25.09.2008
(30) 22.03.2007 US 896481 P
(54) • VERFAHREN ZUR BEHANDLUNG VON
GEMÜTSERKRANKUNGEN
• METHODS OF TREATING MOOD DISOR-
DERS
• PROCÉDÉS DE TRAITEMENT DE TROU-
BLES DE L'HUMEUR
(71) AstraZeneca AB, Global Intellectual Property,
151 85 Södertälje, SE
(72) CHRISTOPH, Greg, Wilmington, DE 19850-
5437, US
GRIMM, Scott, W., Wilmington, DE 19850-
5437, US
WIDZOWSKI, Dan, Wilmington, DE 19850-
5437, US
(74) Sternas, Ann-Sofie, et al, AstraZeneca AB
Global Intellectual Property, Patents, 151 85
Södertälje, SE
A61K 31/555 → (51) A61K 9/08
A61K 31/557 → (51) A61K 9/00
A61K 31/557 → (51) A61K 39/106
75
Anmeldungen
Applications
Demandes (49/2009) 02.12.2009
(51) A61K 31/56 (11) 2 124 958 A2*
(25) En (26) En
(21) 07865244.3 (22) 05.12.2007
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HU IE IS IT LI LT LU LV MC MT NL PL PT
RO SE SI SK TR
(86) US 2007/086517 05.12.2007
(87) WO 2008/070728 2008/24 12.06.2008
(88) 07.08.2008
(30) 05.12.2006 US 634347
(54) • BEHANDLUNG FÜR TROCKENEN AUGEN
MITTELS TESTOSTERON UND PROGES-
TAGEN
• TREATMENT FOR DRY EYE USING TES-
TOSTERONE AND PROGESTAGEN
• TRAITEMENT DU SYNDROME DE L' IL
SEC EN EMPLOYANT UNE TESTOSTÉ-
RONE ET UNE PROGESTAGÈNE
(71) Southern College Of Optometry, 1245 Madison
Avenue, Memphis TN 38104, US
(72) CONNOR, Charles G., Germantown, TN
38138, US
HAINE, Charles, Memphis, TN 38104, US
(74) Duckett, Anthony Joseph, et al, Mathys &
Squire LLP 120 Holborn, London EC1N 2SQ,
GB
A61K 31/565 → (51) A61K 31/203
A61K 31/566 → (51) A61K 31/203
A61K 31/567 → (51) A61K 31/203
(51) A61K 31/569 (11) 2 124 959 A1*
A61K 9/14 A61P 9/12
(25) En (26) En
(21) 07845436.0 (22) 21.12.2007
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HU IE IS IT LI LT LU LV MC MT NL PL PT
RO SE SI SK TR
(86) AU 2007/001998 21.12.2007
(87) WO 2008/074098 2008/26 26.06.2008
(30) 21.12.2006 AU 2006907173
(54) • PHARMAZEUTISCHE ZUSAMMENSET-
ZUNG
• PHARMACEUTICAL COMPOSITION
• COMPOSITION PHARMACEUTIQUE
(71) Alphapharm PTY LTD, 15 Garnet Street,
Carole Park, QLD 4300, AU
Generics (UK) Limited, Albany Gate Darkes
Lanes, Potters Bar, Hertfordshire EN6 1AG,
GB
(72) MOONEY, Brett Antony, Mt Ommaney,
Queensland 4074, AU
OWUSU-GYAMFI, Erwin, Potters Bar Hertfordshire
EN6 1AG, GB
(74) Faivre Petit, Frédérique, et al, Cabinet
Regimbeau 20, rue de Chazelles, 75847 Paris
Cedex 17, FR
A61K 31/569 → (51) A61K 31/203
(51) A61K 31/57 (11) 2 124 960 A1*
A61K 8/63 A61P 17/00
A61P 17/08 A61P 17/10
A61P 17/14
(25) De (26) De
(21) 07856867.2 (22) 19.12.2007
(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB
GR HU IE IS IT LI LT LU LV MC MT NL PL PT
RO SE SI SK TR
(86) EP 2007/011144 19.12.2007
(87) WO 2008/077542 2008/27 03.07.2008
(30) 22.12.2006 DE 102006062120
(54) • 3-HYDROXY-CHLORMADINONACETAT
ZUR TOPISCHEN BEHANDLUNG VON
ANDROGEN-ABHÄNGIGEN HAUTERKRAN-
KUNGEN