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Bulletin 2009/49 - European Patent Office

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(C07D) II.1(1)<br />

(30) 23.08.2002 US 405823 P<br />

06.09.2002 US 408589 P<br />

01.11.2002 US 423129 P<br />

20.03.2003 US 456159 P<br />

28.03.2003 US 402004<br />

09.05.2003 US 435408<br />

21.08.2003 US <strong>49</strong>6741 P<br />

(54) • Synthese von Epothilonen, Zwischenprodukte<br />

davon, Analoga und ihre Verwendung<br />

• Synthesis of epothilones, intermediates<br />

thereto, analogues and uses thereof<br />

• Synthèse d'épothilones, intermédiaires,<br />

analogues et leurs utilisations<br />

(73) Sloan-Kettering Institute For Cancer<br />

Research, 1275 York Avenue, New York,<br />

New York 10021, US<br />

(72) Danishefsky, Samuel J., Engelwood NJ<br />

07631, US<br />

Rivkin, Alexey, Hoboken NJ 07030, US<br />

Yoshimura, Fumihiko, Kita-ku Sapporo, JP<br />

Gabarda Ortega, Ana Esther, New York , NY<br />

10021, US<br />

Cho, Young Shin, Cambridge, MA 02141, US<br />

Chou, Ting-Chao, Paramus NJ 10028, US<br />

Dong, Huajin, Beijing 100850, CN<br />

(74) Harris, Jennifer Lucy, et al, Kilburn & Strode<br />

LLP 20 Red Lion Street, London WC1R 4PJ,<br />

GB<br />

(62) 03793304.1 / 1 506 203<br />

(51) C07D 451/04 (11) 1 663 220 B1<br />

A61K 31/439 C07D 453/02<br />

A61P 31/04<br />

(25) En (26) En<br />

(21) 04782599.7 (22) 30.08.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

HR LT LV<br />

(43) 07.06.2006<br />

(86) US 2004/028159 30.08.2004<br />

(87) WO 2005/023257 2005/11 17.03.2005<br />

(30) 03.09.2003 US <strong>49</strong>9781 P<br />

(54) • NEUES VERFAHREN ZUR HERSTELLUNG<br />

VON PLEUROMUTILINDERIVATEN<br />

• NOVEL PROCESS FOR THE PREPARATION<br />

OF PLEUROMUTILIN DERIVATIVES<br />

• NOUVEAU PROCEDE POUR LA FABRICA-<br />

TION DE DERIVES DE LA PLEUROMUTI-<br />

LINE<br />

(73) GLAXO GROUP LIMITED, Glaxo Wellcome<br />

House, Berkeley Avenue, Greenford, Middlesex<br />

UB6 ONN, GB<br />

(72) BREEN, Gary, Francis, GlaxoSmithKline,<br />

Tonbridge, Kent TN11 9AW, GB<br />

FORTH, Michael, Anthony, GlaxoSmithKline,<br />

Tonbridge, Kent TN11 9AW, GB<br />

KOPELMAN, Susan, ShuMei, Hu, King of<br />

Prussia, PA 19406, US<br />

MULLER, Francis, Xavier, King of Prussia,<br />

PA 19406, US<br />

SANDERSON, Francis, Dominic, GlaxoSmithKline,<br />

Harlow, Essex CM19 5AW, GB<br />

(74) Hambleton, Bernadette Angelina, et al, GlaxoSmithKline<br />

C.I.P. (CN925.1) 980 Great<br />

West Road, Brentford, Middlesex TW8 9GS,<br />

GB<br />

C07D 453/02 → (51) C07D 451/04<br />

C07D 471/00 → (51) C09K 11/06<br />

(51) C07D 471/04 (11) 1 737 859 B1<br />

A61K 31/4709 A61P 31/04<br />

(25) De (26) De<br />

(21) 05716236.4 (22) 19.03.2005<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

HR<br />

(43) 03.01.2007<br />

(86) EP 2005/002953 19.03.2005<br />

(87) WO 2005/097789 2005/42 20.10.2005<br />

(30) 01.04.2004 DE 102004015981<br />

(54) • NEUE KRISTALLINE FORM VON 8-CYAN-1-<br />

CYCLOPROPYL-7-(1S,6S-2,8-DIAZABI-<br />

CYCLO¬4.3.0 NONAN-8-YL)-6-FLUOR-1,4-<br />

DIHYDRO-4-OXO-3-CHINOLINCARBON-<br />

SÄURE<br />

• NOVEL CRYSTALLINE FORM OF 8-CYANO-<br />

1-CYCLOPROPYL-7-(1S,6S-2,8-DIAZABI-<br />

CYCLO¬4.3.0 NONAN-8-YL)-6-FLUORO-<br />

1,4-DIHYDRO-4-OXO-3-QUINOLINE CAR-<br />

BOXYLIC ACID<br />

• NOUVELLE FORME CRISTALLINE D'ACIDE<br />

8-CYAN-1-CYCLOPROPYL-7-(1S,6S-2,8-<br />

DIAZABICYCLO¬4.3.0 NONAN-8-YL)-6-<br />

FLUOR-1,4-DIHYDRO-4-OXO-3-CHINOLIN-<br />

CARBOXYLIQUE<br />

(73) Bayer Animal Health GmbH, 51368 Leverkusen,<br />

DE<br />

(72) RAST, Hubert, 51381 Leverkusen, DE<br />

HEEP, Iris, 50859 Köln, DE<br />

GRUNENBERG, Alfons, 41539 Dormagen,<br />

DE<br />

HALLENBACH, Werner, 40789 Monheim, DE<br />

BENET-BUCHHOLZ, Jordi, 43893 Altafulla,<br />

ES<br />

(51) C07D 471/04 (11) 2 054 412 B1<br />

(25) De (26) De<br />

(21) 07765222.0 (22) 18.07.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 06.05.<strong>2009</strong><br />

(86) EP 2007/006360 18.07.2007<br />

(87) WO 2008/014888 2008/06 07.02.2008<br />

(30) 02.08.2006 DE 102006036023<br />

(54) • IMINO-IMIDAZO-PYRIDINDERIVATE MIT<br />

ANTITHROMBOTISCHER AKTIVITÄT<br />

• IMINO-IMIDAZO-PYRIDINE DERIVATIVES<br />

HAVING ANTITHROMBOTIC ACTIVITY<br />

• DÉRIVÉ DE IMINO-IMIDAZO-PYRIDINE<br />

PRÉSENTANT UNE ACTIVITÉ ANTI-<br />

THROMBOTIQUE<br />

(73) Sanofi-Aventis, 174 Avenue de France,<br />

75013 Paris, FR<br />

(72) HEINELT, Uwe, 65926 Frankfurt am Main, DE<br />

HOFMEISTER, Armin, 65926 Frankfurt am<br />

Main, DE<br />

CZECH, Joerg, 65926 Frankfurt am Main, DE<br />

(74) Then, Johann, et al, Sanofi-Aventis<br />

Deutschland GmbH <strong>Patent</strong>- und Lizenzabteilung<br />

Industriepark Höchst Gebäude K 801,<br />

65926 Frankfurt am Main, DE<br />

C07D 471/04 → (51) A61K 31/4439<br />

C07D 471/04 → (51) C07D 215/22<br />

C07D 471/04 → (51) C07D 401/12<br />

C07D 471/08 → (51) A61K 31/551<br />

C07D 471/10 → (51) C07D 207/16<br />

(51) C07D 471/20 (11) 1 694 677 B1<br />

C07D <strong>49</strong>5/20 A01N 43/40<br />

(25) En (26) En<br />

(21) 04806330.9 (22) 09.12.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

(43) 30.08.2006<br />

876<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>49</strong>/<strong>2009</strong>) 02.12.<strong>2009</strong><br />

(86) IB 2004/004083 09.12.2004<br />

(87) WO 2005/061500 2005/27 07.07.2005<br />

(30) 12.12.2003 GB 0328905<br />

(54) • SPIROPIPERIDINDERIVATE ZUR<br />

BEKÄMPFUNG VON SCHÄDLINGEN<br />

• SPIROPIPERIDINE DERIVATIVES FOR<br />

CONTROLLING PESTS<br />

• DÉRIVÉS DE SPIROPIPÉRIDINE POUR<br />

LUTTER CONTRE LES NUISIBLES<br />

(73) Syngenta Participations AG, Schwarzwaldallee<br />

215, 4058 Basel, CH<br />

(72) MOLLEYRES, Louis-Pierre, Schwarzwaldallee<br />

215, CH-4058 Basel, CH<br />

CASSAYRE, Jerome, Schwarzwaldallee 215,<br />

CH-4058 Basel, CH<br />

CEDERBAUM, Fredrik, Schwarzwaldallee<br />

215, CH-4058 Basel, CH<br />

MAIENFISCH, Peter, Schwarzwaldallee 215,<br />

CH-4058 Basel, CH<br />

(74) Waterman, John Richard, et al, Syngenta<br />

Limited - IP Department Jealott's Hill International<br />

Research Centre P.O. Box 3538,<br />

Bracknell Berkshire RG42 6YA, GB<br />

C07D 487/04 → (51) C09K 11/06<br />

C07D 487/10 → (51) C07D 207/16<br />

(51) C07D <strong>49</strong>1/22 (11) 1 664 054 B1<br />

(25) En (26) En<br />

(21) 04762302.0 (22) 24.08.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

HR<br />

(43) 07.06.2006<br />

(86) CZ 2004/000050 24.08.2004<br />

(87) WO 2005/019223 2005/09 03.03.2005<br />

(30) 26.08.2003 CZ 20032305<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON 7-<br />

ETHYL-10-[4-(1-PIPERIDINO)-1-PIPERI-<br />

DINO]-CARBONYLOXYCAMPTOTHECIN<br />

• METHOD OF MANUFACTURING OF 7-<br />

ETHYL-10-[4-(1-PIPERIDINO)-1-PIPERI-<br />

DINO]-CARBONYLOXYCAMPTOTHECIN<br />

• PROCEDE D'ELABORATION DE 7-ETHYL-<br />

10-[4-(1-PIPERIDINO)–1- PIPERIDINO]-<br />

CARBONYLOXYCAMPTOTHECINE<br />

(73) Pliva-Lachema A.S., Karásek 1, 621 33 Brno,<br />

CZ<br />

(72) DOBROVOLNY, Petr, 674 01 Brno, CZ<br />

(74) Pavlica, Tomas, et al, Traplová, Hakr, Kubát<br />

Law and <strong>Patent</strong> <strong>Office</strong>s Pristavni 24, 170 00<br />

Praha 7, CZ<br />

C07D <strong>49</strong>3/04 → (51) C07D 419/06<br />

C07D <strong>49</strong>5/04 → (51) C07D 215/22<br />

(51) C07D <strong>49</strong>5/06 (11) 1 626 050 B1<br />

C07D 513/06 C07D 221/14<br />

A61K 31/473 A61K 31/4743<br />

A61K 31/4745 A61P 35/00<br />

(25) Zh (26) En<br />

(21) 04730460.5 (22) 30.04.2004<br />

(84) DE FR GB<br />

(43) 15.02.2006<br />

(86) CN 2004/000442 30.04.2004<br />

(87) WO 2004/101570 2004/48 25.11.2004<br />

(30) 30.04.2003 CN 03116709<br />

(54) • SCHWEFELHALTIGE NAPHTHOYLIMID-<br />

DERIVATE<br />

• SULFUR-CONTAINING NAPHTHOYLIMIDE<br />

DERIVATIVES<br />

• DERIVES DE NAPHTHOYLIMIDE CONTE-<br />

NANT DU SOUFRE<br />

(73) East China University of Science and Technology,<br />

P.O. Box 289 No. 130 MeiLong<br />

Road, Shanghai 200237, CN

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