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Bulletin 2009/49 - European Patent Office

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(C07D) I.1(2)<br />

Edlauer, Robert, 2136 Laa a.d. Thaya, AT<br />

Gaß, Josef, 2265 Drösong, AT<br />

(74) Ellmeyer, Wolfgang, Mariahilfer Strasse 50,<br />

A-1070 Wien, AT<br />

C07D 333/16 → (51) C07F 9/572<br />

C07D 333/34 → (51) C07D <strong>49</strong>5/04<br />

(51) C07D 341/00 (11) 2 128 153 A1<br />

C07B 61/00<br />

(25) Ja (26) En<br />

(21) 08703281.9 (22) 16.01.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) JP 2008/050420 16.01.2008<br />

(87) WO 2008/087967 2008/30 24.07.2008<br />

(30) 16.01.2007 JP 2007006485<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

OXIDIERTEM ZYKLISCHEM PHENOLSUL-<br />

FID<br />

• PROCESS FOR PRODUCTION OF OXI-<br />

DIZED CYCLIC PHENOL SULFIDE<br />

• PROCÉDÉ POUR LA PRODUCTION DE<br />

SULFURE DE PHÉNOL CYCLIQUE OXYDÉ<br />

(71) Hodogaya Chemical Co., Ltd., 4-1 Shibakoen<br />

2-chome Minato-ku, Tokyo 105-0011, JP<br />

(72) YASUMURA, Masateru, Tsukuba-shi, Ibaraki<br />

3050841, JP<br />

AOKI, Yoshikazu, Koriyama-shi Fukushima<br />

963-8802, JP<br />

ITO, Masami, Tsukuba-shi, Ibaraki 3050841,<br />

JP<br />

UMEKAWA, Masafumi, Motomiya-shi,<br />

Fukushima 9691104, JP<br />

TARUMOTO, Naohiro, Minato-ku Tokyo, JP<br />

(74) Sendrowski, Heiko, Eisenfuhr, Speiser &<br />

Partner Postfach 10 60 78, 28060 Bremen,<br />

DE<br />

(51) C07D 401/04 (11) 2 128 154 A1<br />

A61K 31/454 A61P 25/00<br />

A61P 25/20 A61P 25/30<br />

A61P 25/32 A61P 43/00<br />

(25) Ja (26) En<br />

(21) 08712095.2 (22) 28.02.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) JP 2008/053524 28.02.2008<br />

(87) WO 2008/105<strong>49</strong>7 2008/36 04.09.2008<br />

(30) 01.03.2007 JP 2007051842<br />

08.03.2007 JP 2007059260<br />

26.03.2007 JP 2007078845<br />

30.03.2007 JP 2007093846<br />

(54) • BENZIMIDAZOLVERBINDUNG UND DEREN<br />

PHARMAZEUTISCHE VERWENDUNG<br />

• BENZIMIDAZOLE COMPOUND AND<br />

PHARMACEUTICAL USE THEREOF<br />

• COMPOSÉ DE BENZIMIDAZOLE ET UTILI-<br />

SATION PHARMACEUTIQUE DE CELUI-CI<br />

(71) Mitsubishi Tanabe Pharma Corporation, 2-<br />

10, Dosho-machi 3-chome, Chuo-ku Osakashi<br />

Osaka 541-8505, JP<br />

(72) NAKANO, Masakazu, Osaka-shi Osaka 541-<br />

8505, JP<br />

MINOGUCHI, Masanori, Osaka-shi Osaka<br />

541-8505, JP<br />

HANANO, Tokushi, Osaka-shi Osaka 541-<br />

8505, JP<br />

ONO, Shin-ichiro, Osaka-shi Osaka 541-<br />

8505, JP<br />

HORIUCHI, Hideki, Osaka-shi Osaka 541-<br />

8505, JP<br />

TESHIMA, Koji, Osaka-shi Osaka 541-8505,<br />

JP<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(74) Weber, Thomas, <strong>Patent</strong>anwälte von Kreisler<br />

Selting Werner Deichmannhaus am Dom<br />

Bahnhofsvorplatz 1, 50667 Köln, DE<br />

C07D 401/06 → (51) C07D 231/12<br />

C07D 401/10 → (51) C07D 213/80<br />

(51) C07D 401/14 (11) 2 128 155 A1<br />

A61K 31/44 A61P 31/10<br />

(25) En (26) En<br />

(21) 09161630.0 (22) 02.06.<strong>2009</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK TR<br />

(30) 30.05.2008 JP 2008143232<br />

(54) • Triazolderivat oder Salz davon<br />

• Triazole derivative or salt thereof<br />

• Dérivé de triazole ou son sel<br />

(71) Fujifilm Finechemicals Co. Ltd., 2-3, Higashiyawata<br />

5-chome, Hiratsuka, Kanagawa<br />

254-0016, JP<br />

(72) Nagayama, Takashi, Kanagawa 254-0016, JP<br />

(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser<br />

Anwaltssozietät, Leopoldstrasse 4,<br />

80802 München, DE<br />

C07D 403/06 → (51) A61K 31/<strong>49</strong>7<br />

C07D 403/12 → (51) C07D 231/12<br />

C07D 405/12 → (51) C07D 413/12<br />

C07D 413/10 → (51) C07D 213/80<br />

(51) C07D 413/12 (11) 2 128 156 A1<br />

A61K 31/4439 A61K 31/4709<br />

A61K 31/506 A61K 31/5377<br />

A61P 9/00 A61P 9/10<br />

A61P 17/06 A61P 19/02<br />

A61P 27/02 A61P 29/00<br />

A61P 35/00 C07D 413/14<br />

C07D 417/12 C07D 417/14<br />

(25) Ja (26) En<br />

(21) 08704094.5 (22) 29.01.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) JP 2008/051312 29.01.2008<br />

(87) WO 2008/093677 2008/32 07.08.2008<br />

(30) 29.01.2007 JP 2007018059<br />

28.03.2007 JP 2007083153<br />

(54) • NEUE OXADIAZOLDERIVATE UND THIA-<br />

DIAZOLDERIVATE MIT DIE NEOVASKULA-<br />

RISIERUNG HEMMENDER WIRKUNG<br />

• NOVEL OXADIAZOLE DERIVATIVES AND<br />

THIADIAZOLE DERIVATIVES HAVING<br />

NEOVASCULARIZATION INHIBITING<br />

ACTIVITY<br />

• NOUVEAUX DÉRIVÉS D'OXADIAZOLE ET<br />

DÉRIVÉS DE THIDIAZOLE AYANT UNE<br />

ACTIVITÉ INHIBANT LA NÉOVASCULARI-<br />

SATION<br />

(71) Santen Pharmaceutical Co., Ltd, 9-19, Shimoshinjo<br />

3-chome Higashiyodogawa-ku,<br />

Osaka-shi Osaka 533-8651, JP<br />

(72) HONDA, Takahiro, Ikoma-shi Nara 630-0101,<br />

JP<br />

FUJISAWA, Koushi, Ikoma-shi Nara 630-<br />

0101, JP<br />

AONO, Hiroyuki, Ikoma-shi Nara 630-0101,<br />

JP<br />

BAN, Masakazu, Ikoma-shi Nara 630-0101,<br />

JP<br />

(74) Müller-Boré & Partner <strong>Patent</strong>anwälte, Grafinger<br />

Strasse 2, 81671 München, DE<br />

488<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>49</strong>/<strong>2009</strong>) 02.12.<strong>2009</strong><br />

(51) C07D 413/12 (11) 2 128 157 A1<br />

A61K 31/4709 A61K 31/<strong>49</strong>6<br />

A61K 31/<strong>49</strong>8 A61K 31/517<br />

A61K 31/5355 A61K 31/536<br />

A61K 31/538 A61K 31/5415<br />

C07D 405/12 C07D 417/12<br />

(25) Ja (26) En<br />

(21) 08710655.5 (22) 24.01.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) JP 2008/051471 24.01.2008<br />

(87) WO 2008/091021 2008/31 31.07.2008<br />

(30) 24.01.2007 JP 2007014372<br />

(54) • HETEROCYCLIDEN-N-(ARYL)ACETAMID-<br />

DERIVAT<br />

• HETEROCYCLIDENE-N-(ARYL)ACETAMIDE<br />

DERIVATIVE<br />

• DÉRIVÉ D'HÉTÉROCYCLIDÈNE-N-(ARYL)<br />

ACÉTAMIDE<br />

(71) MOCHIDA PHARMACEUTICAL CO., LTD., 7,<br />

Yotsuya 1-chome, Shinjuku-ku Tokyo 160-<br />

8515, JP<br />

(72) UCHIDA, Hideharu, Tokyo 160-8515, JP<br />

OGAWA, Shinichi, Tokyo 160-8515, JP<br />

MAKABE, Muneyoshi, Tokyo 160-8515, JP<br />

MAEDA, Yoshitaka, Tokyo 160-8515, JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastrasse 4, 81925 München, DE<br />

(51) C07D 413/12 (11) 2 128 158 A1<br />

A61K 31/4439 A61P 1/16<br />

A61P 3/10 A61P 7/02<br />

A61P 9/10<br />

(25) En (26) En<br />

(21) 08009576.3 (22) 26.05.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(54) • Heterocyclische Cyclopropyl-substituierte<br />

FXR-bindende Verbindungen<br />

• Heterocyclic cyclopropyl-substituted FXR<br />

binding compounds<br />

• Composés de liaison FXR substitués de<br />

cyclopropyle hétérocyclique<br />

(71) Phenex Pharmaceuticals AG, J542N, Werksgelände<br />

BASF, 67056 Ludwigshafen, DE<br />

(72) Abel, Ulrich, 69126 Heidelberg, DE<br />

Kremoser, Claus, 69121 Heidelberg, DE<br />

(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser<br />

Anwaltssozietät, Leopoldstrasse 4,<br />

80802 München, DE<br />

C07D 413/12 → (51) C07C 229/44<br />

C07D 413/12 → (51) C07D 231/12<br />

C07D 413/14 → (51) C07D 413/12<br />

C07D 417/12 → (51) C07D 413/12<br />

C07D 417/14 → (51) C07D 413/12<br />

(51) C07D 471/04 (11) 2 128 159 A1<br />

C09K 11/06 H01L 51/50<br />

(25) Ja (26) En<br />

(21) 08722028.1 (22) 13.03.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) JP 2008/054624 13.03.2008<br />

(87) WO 2008/114690 2008/39 25.09.2008<br />

(30) 15.03.2007 JP 2007066214

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