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Bulletin 2009/49 - European Patent Office

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(C07D) I.1(1)<br />

• NOUVEAUX ANTIFOLATES CLASSIQUES<br />

(71) Chelsea Therapeutics, Inc., 3530 Toringdon<br />

Way Suite 200, Charlotte, NC 28277, US<br />

(72) ROBERTS, Michael, J., Charlotte, NC 28277,<br />

US<br />

PEDDER, Simon, Fort Mill, SC 29715, US<br />

(74) Noel, Chantal Odile, et al, Cabinet Orès 36,<br />

rue Saint Pétersbourg, 75008 Paris, FR<br />

(51) C07D 487/04 (11) 2 125 819 A2*<br />

A61K 31/4188 A61K 31/53<br />

A61P 35/00 A61P 37/00<br />

(25) En (26) En<br />

(21) 08732562.7 (22) 20.03.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) US 2008/057656 20.03.2008<br />

(87) WO 2008/116064 2008/39 25.09.2008<br />

(30) 21.03.2007 US 776003 P<br />

(54) • ANELLIERTE HETEROCYCLISCHE VER-<br />

BINDUNGEN ZUR BEHANDLUNG VON<br />

PROLIFERATIVEN, ALLERGISCHEN,<br />

AUTOIMMUN- UND ENTZÜNDUNGSER-<br />

KRANKUNGEN<br />

• FUSED HETEROCYCLIC COMPOUNDS<br />

USEFUL FOR THE TREATMENT OF PRO-<br />

LIFERATIVE, ALLERGIC, AUTOIMMUNE<br />

OR INFLAMMATORY DISEASES<br />

• COMPOSÉS HÉTÉROCYCLIQUES FUSION-<br />

NÉS UTILES EN TANT QUE MODULA-<br />

TEURS DE KINASES<br />

(71) Bristol-Myers Squibb Company, Route 206<br />

and Province Line Road, Princeton NJ<br />

08543-4000, US<br />

(72) LIU, Chunjian, Princeton, New Jersey 08543,<br />

US<br />

LEFTHERIS, Katerina, Princeton, New Jersey<br />

08543, US<br />

TEBBEN, Andrew, J., Princeton, New Jersey<br />

08543, US<br />

(74) Beacham, Annabel Rose, Frank B. Dehn &<br />

Co. St Bride's House 10 Salisbury Square,<br />

London EC4Y 8JD, GB<br />

(51) C07D 487/04 (11) 2 125 820 A1*<br />

C07D 473/34 C07D 471/04<br />

A61K 31/519 A61P 35/00<br />

(25) En (26) En<br />

(21) 07848737.8 (22) 20.12.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(86) GB 2007/050777 20.12.2007<br />

(87) WO 2008/075110 2008/26 26.06.2008<br />

(30) 21.12.2006 GB 0625682<br />

21.12.2006 US 871355 P<br />

25.10.2007 US 982636 P<br />

07.11.2007 US 986150 P<br />

(54) • EINE HETEROARYLAMID- ODER HETERO-<br />

ARYLPHENYLGRUPPE ENTHALTENDE<br />

SUBSTITUIERTE PIPERIDINE<br />

• SUBSTITUTED PIPERIDINES CONTAINING<br />

A HETEROARYLAMIDE OR HETEROARYL-<br />

PHENYL MOIETY<br />

• PIPÉRIDINES SUBSTITUÉES CONTENANT<br />

UN HÉTÉROARYLAMIDE OU UNE FRAC-<br />

TION HÉTÉROARYLPHÉNYLE<br />

(71) Astex Therapeutics Limited, 436 Cambridge<br />

Science Park Milton Park Cambridge, Cambridgeshire<br />

CB4 0QA, GB<br />

The Institute of Cancer Research: Royal<br />

Cancer Hospital, 123 Old Brompton Road,<br />

London SW7 3RP, GB<br />

Cancer Research Campaign Technology<br />

Limited, Sardinia House Sardinia Street,<br />

London WC2A 3NL, GB<br />

AstraZeneca AB, 151 85 Södertälje, SE<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(72) WOODHEAD, Steven John, Cambridge Cambridgeshire<br />

CB4 0QA, GB<br />

HAMLETT, Christopher, Cambridge Cambridgeshire<br />

CB4 0QA, GB<br />

VERDONK, Marinus Leendert, Cambridge<br />

Cambridgeshire CB4 0QA, GB<br />

SORE, Hannah Fiona, Cambridge Cambridgeshire<br />

CB1 3NX, GB<br />

WALKER, David Winter, Cambridge Cambridgeshire<br />

CB40QA, GB<br />

COLLINS, Ian, Sutton Surrey SM2 5NG, GB<br />

CALDWELL, John, Sutton Surrey SM2 5NG,<br />

GB<br />

DA FONSECA McHARDY, Tatiana Faria,<br />

Sutton Surrey, GB<br />

LUKE, Richard William Arthur, Macclesfield<br />

Cheshire SK10 4TG, GB<br />

MATUSIAK, Zbigniew Stanley, Macclesfield<br />

Cheshire SK10 4TG, GB<br />

CARR, Gregory Richard, Macclesfield Cheshire<br />

SK10 4TG, GB<br />

MORRIS, Jeffrey James, Macclesfield Cheshire<br />

SK10 4TG, GB<br />

CHEUNG, Kwai Ming, Sutton Surrey SM2<br />

5NG, GB<br />

(74) Brearley, Helen Rebecca, Elkington and Fife<br />

LLP Prospect House 8 Pembroke Road,<br />

Sevenoaks Kent TN13 1XR, GB<br />

(51) C07D 487/04 (11) 2 125 821 A1*<br />

(25) En (26) En<br />

(21) 07857066.0 (22) 21.12.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(86) EP 2007/011355 21.12.2007<br />

(87) WO 2008/074512 2008/26 26.06.2008<br />

(30) 21.12.2006 PCT/CN2006/003530<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

SILDENAFIL<br />

• PROCESS FOR THE PREPARATION OF<br />

SILDENAFIL<br />

• PROCÉDÉ DE PRÉPARATION DE SILDÉ-<br />

NAFIL<br />

(71) Krka Tovarna Zdravil, D.D., Novo Mesto,<br />

Smarjeska cesta 6, 8501 Novo Mesto, SI<br />

(72) TIAN, Guanghui, Shanghai 201209, CN<br />

ZHU, Yi, Shanghai 201209, CN<br />

LIU, Zheng, Shanghai 201209, CN<br />

WANG, Zhen, Shanghai 201209, CN<br />

SHEN, Jingsham, Shanghai, CH<br />

BOMBEK, Sergeja, 8000 Novo Mesto, SI<br />

STROPNIK, Tadej, 1000 Ljubljana, SI<br />

(74) UEXKÜLL & STOLBERG, <strong>Patent</strong>anwälte<br />

Beselerstrasse 4, 22607 Hamburg, DE<br />

(51) C07D 487/04 (11) 2 125 822 A1*<br />

C07D 295/135 C07D 295/155<br />

C40B 40/04 A61K 31/519<br />

A61P 35/00<br />

(25) En (26) En<br />

(21) 07857726.9 (22) 17.12.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(86) EP 2007/064096 17.12.2007<br />

(87) WO 2008/074788 2008/26 26.06.2008<br />

(30) 21.12.2006 EP 06126902<br />

08.10.2007 EP 07118039<br />

(54) • SUBSTITUIERTE PYRAZOLO-CHINAZO-<br />

LINDERIVATE, VERFAHREN ZU IHRER<br />

HERSTELLUNG UND IHRE VERWENDUNG<br />

ALS KINASEINHIBITOREN<br />

193<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>49</strong>/<strong>2009</strong>) 02.12.<strong>2009</strong><br />

• SUBSTITUTED PYRAZOLO-QUINAZOLINE<br />

DERIVATIVES, PROCESS FOR THEIR<br />

PREPARATION AND THEIR USE AS<br />

KINASE INHIBITORS<br />

• DÉRIVÉS DE PYRAZOLO-QUINAZOLINE<br />

SUBSTITUÉS, LEUR PROCÉDÉ DE PRÉ-<br />

PARATION ET LEUR UTILISATION EN<br />

TANT QU'INHIBITEURS DES KINASES<br />

(71) NERVIANO MEDICAL SCIENCES S.r.l., Viale<br />

Pasteur, 10, 20014 Nerviano (MI), IT<br />

(72) CARUSO, Michele, 20131 Milan, IT<br />

BERIA, Italo, 20014 Nerviano, IT<br />

BRASCA, Maria Gabriella, <strong>2009</strong>0 Cusago, IT<br />

FERGUSON, Ron, 21020 Casale Litta, IT<br />

POSTERI, Helena, 21028 Travedona Monate<br />

( Varese ), IT<br />

VALSASINA, Barbara, 20131 Milan, IT<br />

(51) C07D 487/04 (11) 2 125 823 A1*<br />

(25) En (26) En<br />

(21) 07859469.4 (22) 20.12.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

HR<br />

(86) IB 2007/055245 20.12.2007<br />

(87) WO 2008/078291 2008/27 03.07.2008<br />

(30) 22.12.2006 PCT/IB2006/055019<br />

(54) • 5,6,7,8-TETRAHYDRO-IMIDAZO[1,5-A]<br />

PYRAZINDERIVATE<br />

• 5,6,7,8-TETRAHYDRO-IMIDAZO[1,5-A]<br />

PYRAZINE DERIVATIVES<br />

• DÉRIVÉS DE 5,6,7,8-TÉTRAHYDRO-IMI-<br />

DAZO[1,5-A]PYRAZINE<br />

(71) Actelion Pharmaceuticals Ltd., Gewerbestrasse<br />

16, 4123 Allschwil, CH<br />

(72) AISSAOUI, Hamed, 68840 Pulversheim, FR<br />

BOSS, Christoph, 4123 Allschwil, CH<br />

GUDE, Markus, 4123 Allschwil, CH<br />

KOBERSTEIN, Ralf, 79539 Lörrach, DE<br />

SIFFERLEN, Thierry, 68220 Wentzwiller, FR<br />

(74) Ruhlmann, Eric, Actelion Pharmaceuticals<br />

Ltd Gewerbestrasse 16, 4123 Allschwil, CH<br />

C07D 487/04 → (51) C07D 217/02<br />

C07D 487/04 → (51) C07D 231/40<br />

C07D 487/04 → (51) C07D 257/02<br />

C07D 487/04 → (51) C07D 471/04<br />

C07D 487/08 → (51) C07D 217/02<br />

C07D 487/08 → (51) C07D 257/02<br />

C07D 487/12 → (51) C07D 213/73<br />

(51) C07D 489/08 (11) 2 125 824 A1*<br />

A61K 31/485<br />

(25) En (26) En<br />

(21) 08732176.6 (22) 14.03.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) US 2008/056929 14.03.2008<br />

(87) WO 2008/118654 2008/40 02.10.2008<br />

(30) 23.03.2007 US 896537 P<br />

(54) • VERBESSERTE ZUBEREITUNG VON OXY-<br />

MORPHON AUS ORIPAVIN<br />

• IMPROVED PREPARATION OF OXYMOR-<br />

PHONE FROM ORIPAVINE<br />

• PRÉPARATION AMÉLIORÉE D'OXYMOR-<br />

PHONE À PARTIR D'ORIPAVINE<br />

(71) Mallinckrodt Inc., 675 McDonnell Boulevard,<br />

Hazelwood, MO 63042, US<br />

(72) WANG, Peter, X., Chesterfield, Missouri<br />

63017, US

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