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Bulletin 2009/49 - European Patent Office

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(C07C) I.1(2)<br />

(74) Wilhelms · Kilian & Partner <strong>Patent</strong>anwälte,<br />

Eduard-Schmid-Straße 2, 81541 München,<br />

DE<br />

(51) C07C 303/44 (11) 2 128 131 A1<br />

C07C 309/20<br />

(25) Ja (26) En<br />

(21) 07860162.2 (22) 26.12.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(86) JP 2007/07<strong>49</strong>33 26.12.2007<br />

(87) WO 2008/078767 2008/27 03.07.2008<br />

(30) 27.12.2006 JP 2006351663<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

VINYLSULFONSÄURE<br />

• PROCESS FOR PRODUCING VINYLSUL-<br />

FONIC ACID<br />

• PROCÉDÉ SERVANT À PRODUIRE DE<br />

L'ACIDE VINYLSULFONIQUE<br />

(71) Asahi Kasei Finechem Co., Ltd., 8-7 Fukumachi<br />

1-chome, Nishiyodogawa-ku Osakashi<br />

Osaka 555-0034, JP<br />

(72) AKIKAZE, Hiroshi, Osaka-shi Osaka 555-<br />

0034, JP<br />

MIYAI, Takehiko, Nobeoka-shi Miyazaki 882-<br />

0861, JP<br />

(74) Kuhnen & Wacker, <strong>Patent</strong>- und Rechtsanwaltsbüro<br />

Prinz-Ludwig-Strasse 40A, 85354<br />

Freising, DE<br />

C07C 303/44 → (51) C07C 303/28<br />

C07C 309/00 → (51) H01L 31/032<br />

C07C 309/20 → (51) C07C 303/44<br />

C07C 309/65 → (51) C07C 303/28<br />

C07C 317/14 → (51) A01N 43/56<br />

C07C 319/12 → (51) C04B 41/51<br />

(51) C07C 323/47 (11) 2 128 132 A1<br />

C07D 209/88 C08F 2/50<br />

G03F 7/031<br />

(25) Ja (26) En<br />

(21) 07859948.7 (22) 21.12.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(86) JP 2007/074668 21.12.2007<br />

(87) WO 2008/078686 2008/27 03.07.2008<br />

(30) 27.12.2006 JP 2006351995<br />

(54) • OXIMESTERVERBINDUNG UND FOTO-<br />

POLYMERISATIONSINITIATOR MIT DER<br />

VERBINDUNG<br />

• OXIME ESTER COMPOUND AND PHOTO-<br />

POLYMERIZATION INITIATOR COMPRIS-<br />

ING THE COMPOUND<br />

• COMPOSÉ ESTER D'OXIME ET INITIA-<br />

TEUR DE PHOTOPOLYMÉRISATION COM-<br />

PRENANT LE COMPOSÉ<br />

(71) Adeka Corporation, 2-35, Higashiogu 7chome<br />

Arakawa-ku, Tokyo 116-8554, JP<br />

(72) SAWAMOTO, Daisuke, Tokyo 116-8554, JP<br />

KIMIJIMA, Koichi, Tokyo 116-8554, JP<br />

(74) Forstmeyer, Dietmar, et al, BOETERS &<br />

LIECK Oberanger 32, 80331 München, DE<br />

(51) C07D 205/08 (11) 2 128 133 A1<br />

(25) En (26) En<br />

(21) 08156895.8 (22) 26.05.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(54) • Ezetiminverfahren und -zusammensetzung<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

• Ezetimibe process and composition<br />

• Procédé et composition d'ézétimibe<br />

(71) Lek Pharmaceuticals D.D., Verovskova 57,<br />

1526 Ljubljana, SI<br />

(72) Selic, Lovro, 3000, Celje, SI<br />

(74) Kunic, Barbara, C/o Sandoz International<br />

GmbH Global <strong>Patent</strong>s Department Industriestrasse<br />

25, 83607 Holzkirchen, DE<br />

C07D 207/04 → (51) C07C 235/40<br />

(51) C07D 209/08 (11) 2 128 134 A1<br />

A61K 31/4418 A61K 31/451<br />

A61K 31/<strong>49</strong>5 A61K 31/<strong>49</strong>6<br />

A61K 31/5377 A61K 31/551<br />

A61P 1/02 A61P 19/02<br />

A61P 27/02 A61P 29/00<br />

A61P 31/12 A61P 31/18<br />

A61P 35/00 A61P 35/04<br />

A61P 43/00 C07D 209/86<br />

C07D 211/96 C07D 213/81<br />

C07D 215/20<br />

(25) Ja (26) En<br />

(21) 07830926.7 (22) 31.10.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(86) JP 2007/071192 31.10.2007<br />

(87) WO 2008/053913 2008/19 08.05.2008<br />

(30) 02.11.2006 JP 2006298795<br />

20.03.2007 JP 2007072150<br />

31.08.2007 JP 2007225075<br />

(54) • ZUR SELEKTIVEN INHIBIERUNG VON<br />

MMP-13 FÄHIGE SULFONYLHARNSTOFF-<br />

DERIVATE<br />

• SULFONYLUREA DERIVATIVE CAPABLE<br />

OF SELECTIVELY INHIBITING MMP-13<br />

• DÉRIVÉ DE SULFONYLURÉE CAPABLE<br />

D'INHIBER SÉLECTIVEMENT MMP-13<br />

(71) Shionogi&Co., Ltd., 1-8, Doshomachi 3chome<br />

Chuo-ku, Osaka-shi, Osaka 5410045,<br />

JP<br />

(72) ENDOH, Takeshi, Osaka-shi Osaka 5530002,<br />

JP<br />

FUJII, Yasuhiko, Osaka-shi Osaka 5530002,<br />

JP<br />

KOJIMA, Eiichi, Osaka-shi Osaka 5530002,<br />

JP<br />

TADANO, Genta, Osaka-shi Osaka 5530002,<br />

JP<br />

YAMAGUCHI, Naoko, Osaka-shi Osaka<br />

5530002, JP<br />

ADACHI, Yo, Osaka-shi Osaka 5530002, JP<br />

TAGASHIRA, Sachie, Osaka-shi Osaka<br />

5530002, JP<br />

TACHIBANA, Yuki, Osaka-shi Osaka<br />

5530002, JP<br />

ONODERA, Naohiro, Osaka-shi Osaka<br />

5530002, JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastrasse 4, 81925 München, DE<br />

C07D 209/28 → (51) C07C 229/42<br />

C07D 209/86 → (51) C07D 209/08<br />

C07D 209/88 → (51) C07C 323/47<br />

(51) C07D 211/74 (11) 2 128 135 A1<br />

C07D 211/94 C07D 221/20<br />

C07D <strong>49</strong>1/20 C07D <strong>49</strong>5/20<br />

A61K 51/00<br />

(25) Ja (26) En<br />

(21) 08710831.2 (22) 30.01.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) JP 2008/051899 30.01.2008<br />

485<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>49</strong>/<strong>2009</strong>) 02.12.<strong>2009</strong><br />

(87) WO 2008/093881 2008/32 07.08.2008<br />

(30) 31.01.2007 JP 2007022042<br />

(54) • VERFAHREN ZUR SYNTHESE VON NIT-<br />

ROXYLRADIKALEN<br />

• METHOD FOR SYNTHESIS OF NITROXYL<br />

RADICAL<br />

• PROCÉDÉ POUR LA SYNTHÈSE D'UN<br />

RADICAL NITROXYLE<br />

(71) Kyushu University, National University Corporation,<br />

10-1, Hakozaki 6-chome, Higashiku<br />

Fukuoka-shi Fukuoka 812-8581, JP<br />

(72) UTSUMI, Hideo, Fukuoka-shi Fukuoka 812-<br />

8581, JP<br />

SAKAI, Kiyoshi, Fukuoka-shi Fukuoka 812-<br />

8581, JP<br />

YAMADA, Kenichi, Fukuoka-shi Fukuoka<br />

812-8581, JP<br />

(74) Woods, Geoffrey Corlett, J.A. KEMP & CO.<br />

14 South Square, Gray's Inn London WC1R<br />

5JJ, GB<br />

C07D 211/94 → (51) C07D 211/74<br />

C07D 211/96 → (51) C07D 209/08<br />

(51) C07D 213/80 (11) 2 128 136 A1<br />

A61K 31/455 A61K 31/55<br />

A61P 3/06 A61P 19/06<br />

A61P 43/00 C07D 401/10<br />

C07D 413/10<br />

(25) Ja (26) En<br />

(21) 07850<strong>49</strong>8.2 (22) 12.12.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(86) JP 2007/073947 12.12.2007<br />

(87) WO 2008/072658 2008/25 19.06.2008<br />

(30) 12.12.2006 JP 2006334021<br />

(54) • 2-PHENYLNICOTINSÄUREDERIVAT<br />

• 2-PHENYLNICOTINIC ACID DERIVATIVE<br />

• DÉRIVÉ DE L'ACIDE 2-PHÉNYLNICOTI-<br />

NIQUE<br />

(71) Nippon Zoki Pharmaceutical Co., Ltd., 1-2<br />

Hiranomachi 2-chome Chuo-ku, Osaka-shi<br />

Osaka 541-0046, JP<br />

(72) MENJO, Nobuo, Kato-shi Hyogo 673-1461,<br />

JP<br />

OOKUBO, Tomohiro, Kato-shi Hyogo 673-<br />

1461, JP<br />

HASEGAWA, Taisuke, Kato-shi Hyogo 673-<br />

1461, JP<br />

FURUKAWA, Kazuhito, Kato-shi Hyogo 673-<br />

1461, JP<br />

FUJITA, Akihiro, Kato-shi Hyogo 673-1461,<br />

JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastrasse 4, 81925 München, DE<br />

C07D 213/81 → (51) C07D 209/08<br />

C07D 213/81 → (51) G21C 19/46<br />

C07D 215/20 → (51) C07D 209/08<br />

C07D 221/20 → (51) C07D 211/74<br />

(51) C07D 221/22 (11) 2 128 137 A1<br />

A61K 31/439 A61P 25/16<br />

(25) Zh (26) En<br />

(21) 07816770.7 (22) 07.11.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(86) CN 2007/003158 07.11.2007<br />

(87) WO 2008/080290 2008/28 10.07.2008<br />

(30) 30.12.2006 CN 200610171579<br />

(54) • SELEKTIVER M4-REZEPTORANTAGONIST<br />

UND DESSEN MEDIZINISCHE VERWEN-<br />

DUNG

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