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Bulletin 2009/49 - European Patent Office

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(C07D) I.1(1)<br />

(74) Talbott, Dawn Jacqueline, Wyeth Pharmaceuticals,<br />

Huntercombe Lane South, Taplow,<br />

Maidenhead, Berkshire SL6 0PH, GB<br />

(51) C07D 209/14 (11) 2 125 720 A1*<br />

C07D 401/06 C07D 401/12<br />

C07D 403/06 A61K 31/404<br />

A61P 25/00<br />

(25) En (26) En<br />

(21) 08730955.5 (22) 28.02.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/055280 28.02.2008<br />

(87) WO 2008/109333 2008/37 12.09.2008<br />

(30) 01.03.2007 US 892330 P<br />

(54) • INDOL- UND BENZOTHIOPHENVERBIN-<br />

DUNGEN ALS MODULATOREN DES HIS-<br />

TAMIN-H3-REZEPTORS<br />

• INDOLE AND BENZOTHIOPHENE COM-<br />

POUNDS AS MODULATORS OF THE HIS-<br />

TAMINE H3 RECEPTOR<br />

• COMPOSÉS À BASE D'INDOLE ET DE<br />

BENZOTHIOPHÈNE EN TANT QUE MODU-<br />

LATEURS DU RÉCEPTEUR H3DE L'HISTAMINE<br />

(71) Janssen Pharmaceutica, N.V., Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) ALLISON, Brett, D., Del Mar, California<br />

92014, US<br />

GRICE, Cheryl, A., Carlsbad, California<br />

9<strong>2009</strong>, US<br />

MCCLURE, Kelly, J., Ramona, California<br />

92065, US<br />

SANTILLAN, JR., Alejandro, San Diego,<br />

California 92130, US<br />

(74) Warner, James Alexander, et al, Carpmaels &<br />

Ransford 43-45 Bloomsbury Square, London<br />

WC1A 2RA, GB<br />

(51) C07D 209/16 (11) 2 125 721 A1*<br />

A61K 31/404 A61P 3/04<br />

A61P 25/28<br />

(25) En (26) En<br />

(21) 08707422.5 (22) 30.01.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) EP 2008/000727 30.01.2008<br />

(87) WO 2008/092666 2008/32 07.08.2008<br />

(30) 31.01.2007 EP 07384015<br />

(54) • ARYL-SUBSTITUIERTE SULFONAMIDE<br />

ZUR BEHANDLUNG VON KOGNITIVEN<br />

STÖRUNGEN ODER MIT DER NAH-<br />

RUNGSMITTELAUFNAHME IN ZUSAM-<br />

MENHANG STEHENDEN STÖRUNGEN<br />

• ARYL-SUBSTITUTED SULFONAMIDES<br />

FOR THE TREATMENT OF COGNITIVE OR<br />

FOOD INGESTION RELATED DISORDERS<br />

• SULFONAMIDES SUBSTITUÉS PAR ARYLE<br />

POUR LE TRAITEMENT DE TROUBLES<br />

COGNITIFS OU LIÉS À L'INGESTION<br />

D'ALIMENTS<br />

(71) Laboratorios Del. Dr. Esteve, S.A., Avda Mare<br />

de Deu de Montserrat 221, 08041 Barcelona,<br />

ES<br />

(72) DIAZ-FERNÁNDEZ, José-Luis, E-08240<br />

Manresa (Barcelona), ES<br />

(74) Peters, Hajo, et al, Graf von Stosch <strong>Patent</strong>anwaltsgesellschaft<br />

mbH Prinzregentenstrasse<br />

22, 80538 München, DE<br />

(51) C07D 209/30 (11) 2 125 722 A2*<br />

A61K 31/404 A61P 11/00<br />

(25) En (26) En<br />

(21) 07732970.4 (22) 25.05.2007<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(86) GB 2007/001951 25.05.2007<br />

(87) WO 2007/138282 2007/<strong>49</strong> 06.12.2007<br />

(88) 28.02.2008<br />

(30) 26.05.2006 US 803275 P<br />

(54) • BIARYL- ODER ARYLHETEROARYL-SUB-<br />

STITUIERTE INDOLE<br />

• BI-ARYL OR ARYL-HETEROARYL SUB-<br />

STITUTED INDOLES<br />

• INDOLES SUBSTITUES PAR BIARYL OU<br />

ARYL-HETEROARYL<br />

(71) AstraZeneca AB, 151 85 Södertälje, SE<br />

(72) BONNERT, Roger, Victor, Loughborough<br />

Leicestershire LE11 5RH, GB<br />

LUKER, Timothy, Jon, Loughborough Leicestershire<br />

LE11 5RH, GB<br />

CUMMING, John, Macclesfield Cheshire<br />

SK10 4TG, GB<br />

(74) Summersell, Richard John, AstraZeneca AB,<br />

Global Intellectual Property, 151 85 Södertälje,<br />

SE<br />

(51) C07D 209/42 (11) 2 125 723 A1*<br />

C07D 405/12 C07D 405/14<br />

A61K 31/404 A61P 27/00<br />

C07D 401/06<br />

(25) En (26) En<br />

(21) 08727502.0 (22) 10.01.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) US 2008/050695 10.01.2008<br />

(87) WO 2008/089015 2008/30 24.07.2008<br />

(30) 11.01.2007 US 884470 P<br />

(54) • BIOLOGISCHE AKTIVITÄT VON 6-SUBSTI-<br />

TUIERTEN INDOL-3-CARBOXYLSÄUREA-<br />

MIDVERBINDUNGEN MIT SPHINGOSIN-1-<br />

PHOSPHATREZEPTORANTAGONISTEN<br />

• 6-SUBSTITUTED INDOLE-3-CARBOXYLIC<br />

ACID AMIDE COMPOUNDS HAVING<br />

SPHINGOSINE-1-PHOSPHATE (S1P)<br />

RECEPTOR ANTAGONIST BIOLOGICAL<br />

ACTIVITY<br />

• COMPOSÉ AMIDE D'ACIDE INDOLE-3-<br />

CARBOXYLIQUE 6-SUBSTITUÉ AYANT<br />

UNE ACTIVITÉ BIOLOGIQUE D'ANTAGO-<br />

NISTE DU RÉCEPTEUR DE SPHINGOSINE-<br />

1-PHOSPHATE (S1P)<br />

(71) ALLERGAN, INC., 2525 Dupont Drive, Irvine<br />

CA 92612, US<br />

(72) BEARD, Richard, L., Newport Beach, CA<br />

92660, US<br />

YUAN, Haiqing, Irvine, CA 92606, US<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastrasse 4, 81925 München, DE<br />

C07D 209/42 → (51) C07D 209/08<br />

C07D 209/44 → (51) C07D 207/46<br />

(51) C07D 209/64 (11) 2 125 724 A1*<br />

A61K 31/4035 A61K 31/4745<br />

C07D 471/04<br />

(25) En (26) En<br />

(21) 08733664.0 (22) 25.03.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) CA 2008/000561 25.03.2008<br />

(87) WO 2008/116304 2008/40 02.10.2008<br />

(30) 26.03.2007 US 920018 P<br />

(54) • NAPHTHALIN- UND CHINOLIN-SULFO-<br />

NYLHARNSTOFFDERIVATE ALS EP4-<br />

REZEPTORANTAGONISTEN<br />

• NAPHTHALENE AND QUINOLINE SULFO-<br />

NYLUREA DERIVATIVES AS EP4 RECEP-<br />

TOR ANTAGONISTS<br />

177<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>49</strong>/<strong>2009</strong>) 02.12.<strong>2009</strong><br />

• DÉRIVÉS DE NAPHTALÈNE ET QUINO-<br />

LÉINE SULFONYLURÉE COMME ANTAGO-<br />

NISTES DU RÉCEPTEUR EP4<br />

(71) Merck Frosst Canada Ltd., 16711 Trans-<br />

Canada Highway, Kirkland, Québec H9H 3L1,<br />

CA<br />

(72) BURCH, Jason, Kirkland, Québec H9H 3L1,<br />

CA<br />

FARAND, Julie, Kirkland, Québec H9H 3L1,<br />

CA<br />

HAN, Yongxin, Kirkland, Québec H9H 3L1,<br />

CA<br />

STURINO, Claudio, Kirkland, Québec H9H<br />

3L1, CA<br />

(74) Horgan, James Michael Frederic, et al, Merck<br />

& Co., Inc. <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

C07D 209/88 → (51) C07D 209/08<br />

(51) C07D 211/06 (11) 2 125 725 A1*<br />

C07D 211/22 C07D 207/06<br />

A61K 31/40 A61K 31/4418<br />

A61P 25/28 A61P 37/00<br />

(25) En (26) En<br />

(21) 08709133.6 (22) 20.02.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) EP 2008/052058 20.02.2008<br />

(87) WO 2008/101953 2008/35 28.08.2008<br />

(30) 22.02.2007 EP 07102910<br />

(54) • VERBINDUNGEN DER FORMEL (I) ALS<br />

SERINPROTEASE-HEMMER<br />

• COMPOUNDS OF FORMULA (I) AS SERINE<br />

PROTEASE INHIBITORS<br />

• COMPOSÉS DE LA FORMULE (I) UTILISÉS<br />

COMME INHIBITEURS DE LA SÉRINE<br />

PROTÉASE<br />

(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(72) ZIMMERMANN, Kaspar, CH-4104 Oberwil,<br />

CH<br />

BAESCHLIN, Daniel Kaspar, CH-4144 Arlesheim,<br />

CH<br />

MOUSSAOUI, Saliha, F-68870 Bartenheim,<br />

FR<br />

(74) Wiessner, Michael, Novartis Pharma AG<br />

<strong>Patent</strong> Department Postfach, CH-4002 Basel,<br />

CH<br />

(51) C07D 211/16 (11) 2 125 726 A1*<br />

C07D 471/10 C07D <strong>49</strong>1/10<br />

C07D 519/00 A61K 31/438<br />

A61K 31/5377 A61P 25/00<br />

(25) En (26) En<br />

(21) 07857529.7 (22) 13.12.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(86) EP 2007/063882 13.12.2007<br />

(87) WO 2008/077811 2008/27 03.07.2008<br />

(30) 22.12.2006 EP 06127078<br />

(54) • SPIROPIPERIDINDERIVATE<br />

• SPIRO-PIPERIDINE DERIVATIVES<br />

• DÉRIVÉS DE SPIROPIPÉRIDINE<br />

(71) F. Hoffmann-La Roche AG, Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

(72) BISSANTZ, Caterina, 68128 Village-neuf, FR<br />

GRUNDSCHOBER, Christophe, 4118<br />

Rodersdorf, CH<br />

MASCIADRI, Raffaello, 4057 Basel, CH<br />

RATNI, Hasane, 68440 Habsheim, FR<br />

ROGERS-EVANS, Mark, 4103 Bottmingen,<br />

CH<br />

SCHNIDER, Patrick, 4103 Bottmingen, CH

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