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Bulletin 2009/49 - European Patent Office

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(C07D) II.1(1)<br />

(86) US 2002/035571 07.11.2002<br />

(87) WO 2003/042195 2003/21 22.05.2003<br />

(30) 13.11.2001 US 8787<br />

(54) • PHOTOCHROME OXAZINVERBINDUNGEN<br />

UND VERFAHREN ZU IHRER HERSTEL-<br />

LUNG<br />

• PHOTOCHROMIC OXAZINE COMPOUNDS<br />

AND METHODS FOR THEIR MANUFAC-<br />

TURE<br />

• COMPOSES D'OXAZINE PHOTOCHROMES<br />

ET LEURS PROCEDES DE FABRICATION<br />

(73) ESSILOR INTERNATIONAL (COMPAGNIE<br />

GENERALE D'OPTIQUE), 147, Rue de Paris,<br />

94220 Charenton-le-Pont, FR<br />

(72) ZHAO, Weili, CH-8051 Zurich, CH<br />

CARREIRA, Erick, M., CH-8124 Zumikon, CH<br />

(74) Perin, Georges, Cabinet Plasseraud 52 rue de<br />

la Victoire, 75440 Paris Cedex 09, FR<br />

(51) C07D 285/08 (11) 1 569 922 B1<br />

A01N 43/836<br />

(25) En (26) En<br />

(21) 03758967.8 (22) 28.10.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 07.09.2005<br />

(86) JP 2003/013750 28.10.2003<br />

(87) WO 2004/046125 2004/23 03.06.2004<br />

(30) 21.11.2002 JP 2002337884<br />

(54) • 1,2,4-THIADIAZOLVERBINDUNGEN UND<br />

DIESE ENTHALTENDE ZUSAMMENSET-<br />

ZUNG ZUR BEKÄMPFUNG VON ARTHRO-<br />

PODEN<br />

• 1,2,4-THIADIAZOLE COMPOUNDS AND<br />

ARTHROPOD CONTROLLING COMPOSI-<br />

TION CONTAINING THE SAME<br />

• COMPOSES A BASE DE 1,2,4-THIADIA-<br />

ZOLE ET COMPOSITION ANTI-ARTHRO-<br />

PODES LES CONTENANT<br />

(73) Sumitomo Chemical Company, Limited, 27-<br />

1, Shinkawa 2-chome, Chuo-ku, Tokyo 104-<br />

8260, JP<br />

(72) IHARA, Hideki, Osaka-shi, Osaka 556-0016,<br />

JP<br />

TAKAOKA, Daisuke, Toyonaka-shi, Osaka<br />

560-0021, JP<br />

(74) Vossius & Partner, Siebertstrasse 4, 81675<br />

München, DE<br />

C07D 295/08 → (51) C07D 295/18<br />

(51) C07D 295/18 (11) 1 <strong>49</strong>0 346 B1<br />

C07D 295/08 C07B 37/04<br />

(25) En (26) En<br />

(21) 03733842.3 (22) 27.03.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

AL LT LV MK<br />

(43) 29.12.2004<br />

(86) US 2003/009275 27.03.2003<br />

(87) WO 2003/08<strong>49</strong>42 2003/42 16.10.2003<br />

(30) 29.03.2002 US 368707 P<br />

(54) • STEREOSELEKTIVE ALKYLIERUNG VON<br />

CHIRALE 2-METHYL-4-GESCHÜTZTE<br />

PIPERAZINEN<br />

• STEREOSELECTIVE ALKYLATION OF<br />

CHIRAL 2-METHYL-4-PROTECTED PIPER-<br />

AZINES<br />

• ALKYLATION STEREOSELECTIVE DE<br />

PIPERAZINES 2-METHYL-4-PROTEGEES<br />

CHIRALES<br />

(73) Schering Corporation, 2000 Galloping Hill<br />

Road, Kenilworth, NJ 07033-0530, US<br />

(72) WU, Wenxue, West Windsor, NJ 08550, US<br />

LIAO, Hongbiao, Bridgewater, NJ 08807, US<br />

TSAI, David, J., Warren, NJ 07059, US<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

ANDREWS, David, R., Maplewood, NJ<br />

07040, US<br />

GALA, Dinesh, East Brunswick, NJ 08816,<br />

US<br />

LEE, Gary, M., Belmont, CA 94002, US<br />

SCHWARTZ, Martin, Lawrence, Morris<br />

Plains, NJ 07950, US<br />

MCALLISTER, Timothy, L., Westfield, NJ<br />

07090, US<br />

FU, Xiaoyong, Edison, NJ 08820, US<br />

MALONEY, Donal, Union, NJ 07083, US<br />

THIRUVENGADAM, T., K., Kendall Park, NJ<br />

08824, US<br />

TANN, Chou-Hang, Berkeley Heights, NJ<br />

07922, US<br />

(74) UEXKÜLL & STOLBERG, <strong>Patent</strong>anwälte<br />

Beselerstrasse 4, 22607 Hamburg, DE<br />

(60) 09013102.0<br />

09013103.8<br />

C07D 307/89 → (51) C07C 51/265<br />

C07D 311/04 → (51) C07D 409/00<br />

C07D 311/58 → (51) C07D 409/00<br />

(51) C07D 311/80 (11) 1 542 984 B1<br />

A61K 31/352 A61P 29/00<br />

(25) En (26) En<br />

(21) 03750947.8 (22) 23.09.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 22.06.2005<br />

(86) GB 2003/004078 23.09.2003<br />

(87) WO 2004/026857 2004/14 01.04.2004<br />

(30) 23.09.2002 GB 0222077<br />

(54) • METHODEN ZUR REINIGUNG VON CAN-<br />

NABINOIDEN AUS PFLANZENMATERIAL<br />

• METHODS OF PURIFYING CANNABINOIDS<br />

FROM PLANT MATERIAL<br />

• METHODES DE PREPARATION DE CAN-<br />

NABINOIDES A PARTIR DE MATIERE<br />

VEGETALE<br />

(73) GW Pharma Limited, Porton Down Science<br />

Park, Salisbury, Wiltshire SP4 OJR, GB<br />

(72) FLOCKHART, Ian Applied Analysis, Hull,<br />

Yorkshire HU17 0TB, GB<br />

WHEATLEY, Gary, William GW Pharmaceuticals<br />

plc, Salisbury, Wiltshire SP4 0JQ, GB<br />

DRING, Su Applied Analysis, Hull, Yorkshire<br />

HU17 0TB, GB<br />

ARCHER, Lesley Applied Analysis, Hull,<br />

Yorkshire HU17 0TB, GB<br />

(74) Schiller, Dominic Christopher, et al, Harrison<br />

Goddard Foote Orlando House 11 C Compstall<br />

Road Marple Bridge, Stockport SK6<br />

5HH, GB<br />

C07D 333/08 → (51) C07C 13/66<br />

(51) C07D 333/38 (11) 1 863 785 B1<br />

C07D 413/12 C07D 409/12<br />

C07D 417/12 A61K 31/435<br />

A61K 31/38 A61K 31/41<br />

A61K 31/535 A61P 29/00<br />

A61P 37/00 A61P 25/00<br />

(25) En (26) En<br />

(21) 06738277.0 (22) 14.03.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 12.12.2007<br />

(86) US 2006/009196 14.03.2006<br />

(87) WO 2006/101860 2006/39 28.09.2006<br />

(30) 16.03.2005 US 662518 P<br />

873<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>49</strong>/<strong>2009</strong>) 02.12.<strong>2009</strong><br />

(54) • NEUE THIOPHENSULFOXIMINE ZUR<br />

BEHANDLUNG VON KOMPLEMENTVER-<br />

MITTELTEN KRANKHEITEN UND LEIDEN<br />

• NOVEL THIOPHENE SULFOXIMINES FOR<br />

TREATING COMPLEMENT-MEDIATED<br />

DISEASES AND CONDITIONS<br />

• NOUVEAUX COMPOSES DE THIOPHENE<br />

SULFOXIMINE DESTINES A TRAITER DES<br />

MALADIES ET DES ETATS PATHOLOGI-<br />

QUES ASSOCIES AU COMPLEMENT<br />

(73) Janssen Pharmaceutica NV, Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) SUBASINGHE, Nalin, L., Exton, PA 19341,<br />

US<br />

BALLENTINE, Shelley, Lansdale, PA 19446,<br />

US<br />

TRAVINS, Jeremy, M., Downingtown, PA<br />

19335, US<br />

KHALIL, Ehab, M., West Chester, PA 19380,<br />

US<br />

ALI, Farah, Exton, PA 19341, US<br />

LEONARD, Kristi, A., Flourtown, PA 19031,<br />

US<br />

GUSHUE, Joan, M., Conshohcken, PA<br />

19428, US<br />

WINTERS, Michael, Peter, Morgantown, PA<br />

19543, US<br />

HUFNAGEL, Heather, Glenmoore, PA 19343,<br />

US<br />

CUMMINGS, Maxwell, David, Strafford, PA<br />

19087, US<br />

(74) Fisher, Adrian John, et al, CARPMAELS &<br />

RANSFORD 43-45 Bloomsbury Square,<br />

London WC1A 2RA, GB<br />

C07D 335/06 → (51) C07D 409/00<br />

C07D 401/00 → (51) C07D 409/00<br />

(51) C07D 401/04 (11) 1 537 097 B1<br />

(25) En (26) En<br />

(21) 03772096.8 (22) 29.07.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 08.06.2005<br />

(86) US 2003/023820 29.07.2003<br />

(87) WO 2004/011453 2004/06 05.02.2004<br />

(30) 31.07.2002 US 400356 P<br />

11.02.2003 US 446451 P<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON 3-<br />

HALOGEN-4,5-DIHYDRO-1 H-PYRAZOLEN<br />

• METHOD FOR PREPARING 3-HALO-4,5-<br />

DIHYDRO-1 I H /I -PYRAZOLES<br />

• PROCEDE D'ELABORATION DE 3-HALO-<br />

4,5-DIHYDRO-1 I H /I -PYRAZOLES<br />

(73) E.I. DU PONT DE NEMOURS AND COM-<br />

PANY, 1007 Market Street, Wilmington, DE<br />

19898, US<br />

(72) ANNIS, Gary, David, Landenberg, PA 19350,<br />

US<br />

(74) Beacham, Annabel Rose, Frank B. Dehn &<br />

Co. St Bride's House 10 Salisbury Square,<br />

London EC4Y 8JD, GB<br />

(60) 09008363.5 / 2 100 889<br />

(51) C07D 401/04 (11) 1 856 093 B1<br />

A61K 31/473 A61P 11/08<br />

(25) En (26) En<br />

(21) 06708593.6 (22) 01.03.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK YU<br />

(43) 21.11.2007<br />

(86) EP 2006/060377 01.03.2006<br />

(87) WO 2006/092422 2006/36 08.09.2006<br />

(30) 02.03.2005 EP 05101619<br />

14.09.2005 EP 05108442

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