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Bulletin 2009/49 - European Patent Office

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(C07C) I.1(1)<br />

WEISSBERG, Avi, 75577 Rishon Le Zion, IL<br />

(74) Becker Kurig Straus, <strong>Patent</strong>anwälte Bavariastrasse<br />

7, 80336 München, DE<br />

C07C 381/00 → (51) C08K 5/5398<br />

(51) C07C 381/12 (11) 2 125 713 A1*<br />

G03F 7/004 G03F 7/039<br />

(25) En (26) En<br />

(21) 07820481.5 (22) 24.09.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(86) EP 2007/060074 24.09.2007<br />

(87) WO 2008/040648 2008/15 10.04.2008<br />

(30) 04.10.2006 EP 06121699<br />

(54) • SULFONIUMSALZ-FOTOINITIATOREN<br />

• SULPHONIUM SALT PHOTOINITIATORS<br />

• PHOTOAMORCEURS A BASE DE SEL DE<br />

SULFONIUM<br />

(71) Ciba Specialty Chemicals Holding Inc.,<br />

Klybeckstrasse 141, 4057 Basel, CH<br />

(72) HAYOZ, Pascal, 4114 Hofstetten, CH<br />

BIRBAUM, Jean-Luc, 4102 Binningen, CH<br />

ILG, Stephan, 4304 Giebenach, CH<br />

C07C 403/14 → (51) C07C 69/738<br />

(51) C07D 205/04 (11) 2 125 714 A1*<br />

A61K 31/397 A61P 11/00<br />

(25) En (26) En<br />

(21) 08719316.5 (22) 06.03.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) IB 2008/000622 06.03.2008<br />

(87) WO 2008/135819 2008/46 13.11.2008<br />

(30) 16.03.2007 US 895163 P<br />

(54) • HYDROCHLORIDSALZ AUS 5-[3-(3-HYD-<br />

ROXYPHENOXY)AZETIDIN-1-YL]-5-<br />

METHYL-2,2- DIPHENYLHEXANAMID<br />

• HYDROCHLORIDE SALT OF 5-[3-(3-<br />

HYDROXYPHENOXY)AZETIDIN-1-YL]-5-<br />

METHYL-2,2- DIPHENYLHEXANAMIDE<br />

• SEL HYDROCHLORURE DE 5-[3-(3-<br />

HYDROXYPHÉNOXY)AZÉTIDIN-1-YL]-5-<br />

MÉTHYL-2,2- DIPHÉNYLHEXANAMIDE<br />

(71) Pfizer Limited, Ramsgate Road, Sandwich,<br />

Kent CT13 9NJ, GB<br />

(72) GLOSSOP, Paul, Alan, Kent, CT13 9NJ, GB<br />

JAMES, Kim, Kent CT13 9NJ, GB<br />

(74) Laurent, Claire, Pfizer Limited <strong>European</strong><br />

<strong>Patent</strong> Department Ramsgate Road, Sandwich,<br />

Kent CT13 9NJ, GB<br />

(51) C07D 205/08 (11) 2 125 715 A2*<br />

A61K 31/397 A61P 3/00<br />

(25) En (26) En<br />

(21) 08707257.5 (22) 24.01.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) EP 2008/000546 24.01.2008<br />

(87) WO 2008/089984 2008/31 31.07.2008<br />

(88) 18.09.2008<br />

(30) 24.01.2007 EP 07001537<br />

01.08.2007 EP 07015107<br />

12.10.2007 EP 07020070<br />

06.12.2007 EP 07023686<br />

17.12.2007 EP 07024430<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

EZETIMIB UND DERIVATEN DAVON<br />

• PROCESS FOR THE PREPARATION OF<br />

EZETIMIBE AND DERIVATIVES THEREOF<br />

• PROCÉDÉ DE FABRICATION DE L'ÉZÉTI-<br />

MIBE ET DE SES DÉRIVÉS<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(71) KRKA, D.d., Novo mesto Smarjeska cesta 6,<br />

8501 Novo mesto, SI<br />

(72) STIMAC, Anton, 1000 Ljubljana, SI<br />

MOHAR, Barbara, 1290 Grosuplje, SI<br />

STEPHAN, Michel, F-92170 Vanves, FR<br />

BEVC, Mojca, 8233 Mirna, SI<br />

ZUPET, Rok, 1000 Ljubljana, SI<br />

GARTNER, Andrej, 1000 Ljubljana, SI<br />

KROSELJ, Vesna, 8310 Sentjernej, SI<br />

SMRKOLJ, Matej, 1420 Trbovlje, SI<br />

KIDEMET, Davor, 42000 Varazdin, HR<br />

SEDMAK, Gregor, 1000 Ljubljana, SI<br />

BENKIC , Primo, 1000 Ljubljana, SI<br />

KLJAJIC , Alen, 3000 Celje, SI<br />

PLEVNIK, Miha, 1295 Ivancna Gorica, SI<br />

(74) Becker Kurig Straus, <strong>Patent</strong>anwälte Bavariastrasse<br />

7, 80336 München, DE<br />

C07D 207/06 → (51) C07D 211/06<br />

C07D 207/16 → (51) C07K 5/08<br />

C07D 207/32 → (51) C05D 9/02<br />

C07D 207/34 → (51) A61K 9/20<br />

(51) C07D 207/46 (11) 2 125 716 A2*<br />

C07D 209/44 C07D 211/94<br />

C07D 405/12 C07D 409/12<br />

C07D 413/06 C07D 417/12<br />

C07D 417/14 A61K 31/4535<br />

A61P 17/18<br />

(25) En (26) En<br />

(21) 08730007.5 (22) 15.02.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) US 2008/054122 15.02.2008<br />

(87) WO 2008/103613 2008/35 28.08.2008<br />

(88) 30.07.<strong>2009</strong><br />

(30) 22.02.2007 US 891140 P<br />

(54) • HYDROXYLAMINVERBINDUNGEN UND<br />

VERFAHREN ZU IHRER VERWENDUNG<br />

• HYDROXYLAMINE COMPOUNDS AND<br />

METHODS OF THEIR USE<br />

• COMPOSÉS D'HYDROXYLAMINE ET<br />

LEURS PROCÉDÉS D'UTILISATION<br />

(71) Othera Holding, Inc., 1011 Centre Road,<br />

Suite 322, Wilmington, DE 19805, US<br />

(72) PATIL, Ghanshyam, Lincoln University,<br />

Pennsylvania 19352, US<br />

(74) Portal, Gérard, et al, Cabinet Beau de<br />

Loménie 158, rue de l'Université, 75340<br />

Paris Cedex 07, FR<br />

(51) C07D 209/08 (11) 2 125 717 A2*<br />

A61P 13/02 A61P 13/08<br />

(25) En (26) En<br />

(21) 08726096.4 (22) 26.02.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) US 2008/002513 26.02.2008<br />

(87) WO 2008/106125 2008/36 04.09.2008<br />

(88) 16.10.2008<br />

(30) 26.02.2007 US 903472 P<br />

(54) • DEUTERIERTE SILODOSINDERIVATE ALS<br />

ALPHA-IA-ADRENOREZEPTOR-ANTAGO-<br />

NISTEN<br />

• DEUTERATED DERIVATIVES OF SILODO-<br />

SIN AS ALPHA IA-ADRENORECEPTOR<br />

ANTAGONISTS<br />

• DERIVES DEUTERES DE SILODOSIN EN<br />

TANT QU'ANTAGONISTES DE L'ADRENO-<br />

RECEPTEUR ALPHA IA<br />

(71) Concert Pharmaceuticals Inc., 99 Hayden<br />

Avenue, Suite 500, Lexington, MA 02421-<br />

7966, US<br />

176<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>49</strong>/<strong>2009</strong>) 02.12.<strong>2009</strong><br />

(72) LIU, Julie, F., Lexington, MA 02420, US<br />

(74) Stevens, Ian Edward, Potter Clarkson LLP<br />

Park View House 58 The Ropewalk, Nottingham<br />

NG1 5DD, GB<br />

(51) C07D 209/08 (11) 2 125 718 A2*<br />

C07D 209/42 C07D 209/88<br />

C07D 231/56 C07D 235/08<br />

C07D 277/64 C07D 333/68<br />

C07D 333/70 C07D 401/12<br />

C07C 311/21 A61K 31/404<br />

A61K 31/4162 A61K 31/4184<br />

A61K 31/381 A61K 31/423<br />

(25) En (26) En<br />

(21) 08735421.3 (22) 14.03.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) EP 2008/053087 14.03.2008<br />

(87) WO 2008/113760 2008/39 25.09.2008<br />

(88) 13.11.2008<br />

(30) 16.03.2007 DE 102007012284<br />

(54) • NEUE SUBSTITUIERTE ARYLSULPHO-<br />

NYLGLYCINE, IHRE HERSTELLUNG UND<br />

IHRE VERWENDUNG ALS PHARMAZEUTI-<br />

SCHE ZUSAMMENSETZUNGEN<br />

• NEW SUBSTITUTED ARYLSULPHONYL-<br />

GLYCINES, THE PREPARATION THEREOF<br />

AND THE USE THEREOF AS PHARMA-<br />

CEUTICAL COMPOSITIONS<br />

• NOUVELLES ARYLSULFONYL-GLYCINES<br />

SUBSTITUÉES, LEUR PRÉPARATION ET<br />

LEUR UTILISATION COMME COMPOSI-<br />

TIONS PHARMACEUTIQUES<br />

(71) Boehringer Ingelheim International GmbH,<br />

Binger Straße 173, 55216 Ingelheim am<br />

Rhein, DE<br />

(72) Wagner, Holger, 55216 Ingelheim Am Rhein,<br />

DE<br />

Langkopf, Elke, 55216 Ingelheim Am Rhein,<br />

DE<br />

Eckhardt, Matthias, 55216 Ingelheim Am<br />

Rhein, DE<br />

Streicher, Rüdiger, 55216 Ingelheim Am<br />

Rhein, DE<br />

Schoelch, Corinna, 55216 Ingelheim Am<br />

Rhein, DE<br />

Schuler-Metz, Annette, 55216 Ingelheim Am<br />

Rhein, DE<br />

Pautsch, Alexander, 55216 Ingelheim Am<br />

Rhein, DE<br />

(74) Hammann, Heinz, et al, Boehringer Ingelheim<br />

GmbH CD-<strong>Patent</strong>s Binger Straße 173, 55216<br />

Ingelheim am Rhein, DE<br />

(51) C07D 209/12 (11) 2 125 719 A1*<br />

C07F 9/572 A61K 31/404<br />

A61K 31/6615 A61P 35/00<br />

A61P 5/30 A61P 19/10<br />

(25) En (26) En<br />

(21) 08730988.6 (22) 28.02.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) US 2008/055326 28.02.2008<br />

(87) WO 2008/106600 2008/36 04.09.2008<br />

(30) 28.02.2007 US 892044 P<br />

(54) • BAZEDOXIFEN-BISPHOSPHORATE<br />

• BAZEDOXIFENE BIS-PHOSPHORATES<br />

• BIS-PHOSPHORATES DE BAZÉDOXIFÈNE<br />

(71) Wyeth, Five Giralda Farms, Madison, NJ<br />

07940, US<br />

(72) FAWZI, Mahdi, B., Morristown, NJ 07960,<br />

US<br />

ZHU, Tianmin, Monroe, NY 10950, US<br />

PAN, Weitao, Belle Mead, NJ 08502, US

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