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Bulletin 2011/27 - European Patent Office

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(A61K) I.1(1)<br />

(74) Docherty, Robert Charles, et al, Symbiosis IP<br />

Limited Apollo House Eboracum Way,<br />

Heworth Green, York YO31 7RE, GB<br />

(51) A61K 9/28 (11) 2 340 018 A2*<br />

A61P 1/00<br />

(25) En (26) En<br />

(21) 09740698.7 (22) <strong>27</strong>.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) EP 2009/064166 <strong>27</strong>.10.2009<br />

(87) WO 2010/049433 2010/18 06.05.2010<br />

(88) 23.12.2010<br />

(30) <strong>27</strong>.10.2008 EP 08305740<br />

(54) • WASSERUNLÖSLICHES POLYMER: FILM-<br />

ÜBERZÜGE AUF STÄRKEBASIS FÜR DEN<br />

KOLON<br />

• WATER INSOLUBLE POLYMER: STARCH-<br />

BASED FILM COATINGS FOR COLON<br />

TARGETING<br />

• POLYMÈRE INSOLUBLE DANS L'EAU :<br />

REVÊTEMENT DE FILM À BASE D'AMIDON<br />

POUR CIBLER LE COLON<br />

(71) Roquette Freres, 62136 Lestrem, FR<br />

(72) HAEUSLER, Olaf, F-59<strong>27</strong>0 Fletre, FR<br />

WILS, Daniel, F-59190 Morbecque, FR<br />

SIEPMANN, Juergen, F-59133 Phalempin,<br />

FR<br />

KARROUT, Youness, F-59000 Lille, FR<br />

(74) Cabinet Plasseraud, 52, rue de la Victoire,<br />

75440 Paris Cedex 09, FR<br />

(51) A61K 9/28 (11) 2 340 019 A1*<br />

A61P 1/00<br />

(25) En (26) En<br />

(21) 09748748.2 (22) <strong>27</strong>.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) EP 2009/064165 <strong>27</strong>.10.2009<br />

(87) WO 2010/049432 2010/18 06.05.2010<br />

(30) <strong>27</strong>.10.2008 EP 08305740<br />

(54) • WASSERUNLÖSLICHES POLYMER:<br />

UNVERDAULICHE WASSERLÖSLICHE<br />

POLYSACCHARID-FILMÜBERZÜGE FÜR<br />

DEN KOLON<br />

• WATER INSOLUBLE POLYMER: INDIGES-<br />

TIBLE WATER-SOLUBLE POLYSACCHAR-<br />

IDE FILM COATINGS FOR COLON<br />

TARGETING<br />

• POLYMÈRE INSOLUBLE DANS L'EAU :<br />

REVÊTEMENTS EN FILM POLYSACCHA-<br />

RIDIQUE SOLUBLES DANS L'EAU ET NON<br />

DIGÉRABLES POUR UN CIBLAGE DU<br />

CÔLON<br />

(71) Roquette Freres, 62136 Lestrem, FR<br />

(72) HAEUSLER, Olaf, F-59<strong>27</strong>0 Fletre, FR<br />

WILS, Daniel, F-59190 Morbecque, FR<br />

SIEPMANN, Juergen, F-59133 Phalempin,<br />

FR<br />

KARROUT, Youness, F-59000 Lille, FR<br />

(74) Cabinet Plasseraud, 52, rue de la Victoire,<br />

75440 Paris Cedex 09, FR<br />

A61K 9/28 → (51) A61K 9/20<br />

A61K 9/70 → (51) A61K 9/00<br />

A61K 31/166 → (51) C07C 259/06<br />

A61K 31/167 → (51) C07C 311/33<br />

A61K 31/18 → (51) C07C 311/33<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

A61K 31/20 → (51) C07D <strong>27</strong>7/36<br />

A61K 31/205 → (51) A61K 9/06<br />

A61K 31/25 → (51) C07D <strong>27</strong>7/36<br />

A61K 31/352 → (51) A61K 36/534<br />

A61K 31/37 → (51) A61K 36/534<br />

(51) A61K 31/395 (11) 2 340 020 A1*<br />

C07F 13/00 C07F 15/06<br />

(25) It (26) En<br />

(21) 09811182.6 (22) 04.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) IB 2009/053859 04.09.2009<br />

(87) WO 2010/026545 2010/10 11.03.2010<br />

(30) 05.09.2008 IT FI20080173<br />

(54) • MANGAN- UND KOBALTKOMPLEXE, IHRE<br />

HERSTELLUNG UND VERWENDUNG<br />

• MANGANESE AND COBALT COMPLEXES,<br />

THEIR PREPARATION AND USE<br />

• COMPLEXES DE MANGANÈSE ET DE<br />

COBALT, LEUR SYNTHÈSE ET LEUR<br />

APPLICATION<br />

(71) Universita' Degli Studi di Firenze, Piazza San<br />

Marco, 4, 50121 Firenze, IT<br />

(72) BANI, Daniele, I-501<strong>27</strong> Firenze, IT<br />

BENCINI, Andrea, I-50019 Sesto Fiorentino,<br />

IT<br />

CANTORE, Miriam, I-51016 Montecatini<br />

Terme, IT<br />

FAILLI, Paola, I-50129 Firenze, IT<br />

GIORGI, Claudia, I-50134 Firenze, IT<br />

VALTANCOLI, Barbara, I-50019 Sesto Fiorentino,<br />

IT<br />

(74) Brighenti, Livio, NOTARBARTOLO & GER-<br />

VASI S.p.A. Corso di Porta Vittoria, 9, 20122<br />

Milano, IT<br />

(51) A61K 31/40 (11) 2 340 021 A1*<br />

A61K 31/4025 A61P 35/00<br />

C07D 207/16 C07D 401/06<br />

C07D 401/12 C07D 401/14<br />

C07D 403/06 C07D 403/12<br />

C07D 405/06 C07D 405/12<br />

C07D 409/04 C07D 409/12<br />

C07D 413/12 C07D 417/12<br />

(25) En (26) En<br />

(21) 0978<strong>27</strong>45.5 (22) 08.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) EP 2009/061610 08.09.2009<br />

(87) WO 2010/031713 2010/12 25.03.2010<br />

(30) 18.09.2008 US 97884 P<br />

15.07.2009 US 225633 P<br />

(54) • SUBSTITUIERTE PYRROLIDIN-2-CARBO-<br />

XYLAMIDE<br />

• SUBSTITUTED PYRROLIDINE-2-CARBOX-<br />

AMIDES<br />

• PYRROLIDINE-2-CARBOXAMIDES SUB-<br />

STITUÉS<br />

(71) F. Hoffmann-La Roche AG, Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

(72) DING, Qingjie, Bridgewater, NJ 08807, US<br />

JIANG, Nan, Fairfield, NJ 07004, US<br />

LIU, Jin-Jun, Warren, NJ 07059, US<br />

ROSS, Tina, Morgan, Royersford, PA 19468,<br />

US<br />

ZHANG, Jing, Parsippany, NJ 07054, US<br />

ZHANG, Zhuming, Hillsborough, NJ 08844,<br />

US<br />

31<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>27</strong>/<strong>2011</strong>) 06.07.<strong>2011</strong><br />

(74) Beyermann, Jochen Carl, F. Hoffmann-La<br />

Roche AG CLP - <strong>Patent</strong> Department Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

A61K 31/4025 → (51) A61K 31/40<br />

A61K 31/404 → (51) C07D 209/42<br />

A61K 31/405 → (51) A01N 43/50<br />

A61K 31/409 → (51) A61K 41/00<br />

A61K 31/415 → (51) A01N 43/50<br />

A61K 31/437 → (51) A61K 47/14<br />

A61K 31/437 → (51) C07D 471/04<br />

A61K 31/437 → (51) C07D 471/06<br />

(51) A61K 31/4409 (11) 2 340 022 A1*<br />

A61K 31/4709 A61K 31/496<br />

A61K 31/4965 A61K 31/5377<br />

A61K 31/541 A61K 45/06<br />

A61P 31/06<br />

(25) En (26) En<br />

(21) 09787058.8 (22) 31.08.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) IB 2009/053796 31.08.2009<br />

(87) WO 2010/026526 2010/10 11.03.2010<br />

(30) 03.09.2008 US 93879 P<br />

(54) • KOMBINATIONSTHERAPIE GEGEN<br />

TUBERKULOSE<br />

• COMBINATION THERAPY FOR TUBERCU-<br />

LOSIS<br />

• THÉRAPIE COMBINÉE POUR LA TUBER-<br />

CULOSE<br />

(71) Pfizer Inc., 235 East 42nd Street, New York,<br />

NY 10017, US<br />

The Johns Hopkins University, 3400 North<br />

Charles Street, Baltimore, MD 21218, US<br />

(72) BRICKNER, Steven Joseph, Ledyard Connecticut<br />

06339, US<br />

NUERMBERGER, Eric, Baltimore Maryland<br />

21231, US<br />

STOVER, Charles Kendall, Gaithersburg<br />

Maryland 20878, US<br />

(74) Kingsbury, Oliver William, Pfizer Limited<br />

<strong>European</strong> <strong>Patent</strong> Department Ramsgate<br />

Road, Sandwich Kent CT13 9NJ, GB<br />

(51) A61K 31/4439 (11) 2 340 023 A1*<br />

A61K 45/06 A61P 11/02<br />

(25) En (26) En<br />

(21) 09782423.9 (22) 01.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) EP 2009/061236 01.09.2009<br />

(87) WO 2010/026129 2010/10 11.03.2010<br />

(30) 02.09.2008 US 93517 P<br />

(54) • DER TRPVL-ANTAGONIST SB705498 ZUR<br />

BEHANDLUNG VON RHINITIS<br />

• THE TRPVL ANTAGONIST SB-705498 FOR<br />

TREATING RHINITIS<br />

• ANTAGONISTE SB-705498 DU RÉCEP-<br />

TEUR TRPVL POUR LE TRAITEMENT DE<br />

LA RHINITE<br />

(71) Glaxo Group Limited, Glaxo Wellcome House<br />

Berkeley Avenue Greenford, Middlesex UB6<br />

0NN, GB<br />

(72) BOUNTRA, Charanjit, Essex CM19 5AW, GB<br />

DENYER, Jane, Christina, Hertfordshire SG1<br />

2NY, GB

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