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Bulletin 2011/27 - European Patent Office

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(C07D) II.1(1)<br />

HEITGER, Helmut, 55218 Ingelheim am<br />

Rhein, DE<br />

MEYER, Oliver, 55452 Dorsheim, DE<br />

(60) 10192561.8 / 2 322 511<br />

C07D 235/26 → (51) C09B 47/067<br />

C07D 237/14 → (51) A61P 35/00<br />

C07D <strong>27</strong>7/20 → (51) C07C 51/377<br />

C07D <strong>27</strong>7/56 → (51) C07C 51/377<br />

(51) C07D 295/073 (11) 1 853 576 B1<br />

A61K 31/495 A61P 25/18<br />

(25) En (26) En<br />

(21) 06706059.0 (22) 14.02.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK YU<br />

(43) 14.11.2007<br />

(86) DK 2006/000088 14.02.2006<br />

(87) WO 2006/086986 2006/34 24.08.2006<br />

(30) 16.02.2005 DK 200500239<br />

16.02.2005 US 653419 P<br />

(54) • KRISTALLINE BASE VON TRANS-1-((1R,<br />

3S)-6-CHLOR-3-PHENYLINDAN-1-YL)-<br />

3,3-DIMETHYLPIPERAZIN<br />

• CRYSTALLINE BASE OF TRANS-1-<br />

((1R,3S)-6-CHLORO-3-PHENYLINDAN-1-<br />

YL)-3,3-DIMETHYLPIPERAZINE<br />

• BASE CRISTALLINE DE LA TRANS-1-<br />

[(1R,3S)-6-CHLORO-3-PHENYLINDAN-1-<br />

YL]-3,3-DIMETHYLPIPERAZINE<br />

(73) H. Lundbeck A/S, Ottiliavej 9, 2500 Valby-<br />

Copenhagen, DK<br />

(72) BANG-ANDERSEN, Benny, DK-2300 Copenhagen<br />

S, DK<br />

LOPEZ DE DIEGO, Heidi, DK-2850 Nærum,<br />

DK<br />

C07D 295/088→ (51) C07C 317/22<br />

C07D 307/77 → (51) A61K 31/14<br />

(51) C07D 307/79 (11) 2 215 069 B1<br />

C07C 33/18 C07C 47/235<br />

A61K 8/49<br />

(25) En (26) En<br />

(21) 08841678.9 (22) 20.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 11.08.2010<br />

(86) IB 2008/054298 20.10.2008<br />

(87) WO 2009/053883 2009/18 30.04.2009<br />

(30) 23.10.2007 EP 07119037<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

TETRANORLABDANDERIVATEN<br />

• PROCESS FOR THE PREPARATION OF<br />

TETRANORLABDANE DERIVATIVES<br />

• PROCÉDÉ POUR LA PRÉPARATION DE<br />

DÉRIVÉS DE TÉTRANORLABDANE<br />

(73) Firmenich S.A., 1, route des Jeunes P.O. Box<br />

239, 1211 Geneva 8, CH<br />

(72) FEHR, Charles, CH-1290 Versoix, CH<br />

(74) Carina, Riccardo Filippo, et al, FIRMENICH<br />

SA Legal Dept., IP Group Route des Jeunes,<br />

1 P.O. Box 239, 1211 Geneva 8, CH<br />

(51) C07D 307/81 (11) 2 125 766 B1<br />

A01N 43/08<br />

(25) En (26) En<br />

(21) 08709831.5 (22) 08.02.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(43) 02.12.2009<br />

(86) IB 2008/000362 08.02.2008<br />

(87) WO 2008/102232 2008/35 28.08.2008<br />

(30) 21.02.2007 US 890914 P<br />

(54) • ANTIPARASITISCHE BENZOFURANMITTEL<br />

• BENZOFURAN ANTIPARASITIC AGENTS<br />

• AGENTS ANTIPARASITAIRES DE TYPE<br />

BENZOFURANE<br />

(73) Pfizer Limited, Ramsgate Road, Sandwich,<br />

Kent CT13 9NJ, GB<br />

(72) GIBSON, Stephen, Paul, Sandwich Kent<br />

CT13 9NJ, GB<br />

LAURET, Christelle, Sandwich Kent CT13<br />

9NJ, GB<br />

(74) Kingsbury, Oliver William, Pfizer Limited<br />

<strong>European</strong> <strong>Patent</strong> Department Ramsgate<br />

Road, Sandwich Kent CT13 9NJ, GB<br />

C07D 317/20 → (51) C07C 2<strong>27</strong>/04<br />

(51) C07D 401/06 (11) 2 010 519 B1<br />

C07D 403/06 C07D 405/14<br />

A61K 31/454 A61K 31/496<br />

A61P 3/00<br />

(25) En (26) En<br />

(21) 07755189.3 (22) 10.04.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 07.01.2009<br />

(86) US 2007/008832 10.04.2007<br />

(87) WO 2007/120655 2007/43 25.10.2007<br />

(30) 14.04.2006 US 791961 P<br />

(54) • SUBSTITUIERTE IMIDAZOL-4-CARBOXA-<br />

MIDE ALS CHOLECYSTOKININ-1-REZEP-<br />

TOR-MODULATOREN<br />

• SUBSTITUTED IMIDAZOLE 4-CARBOXA-<br />

MIDES AS CHOLECYSTOKININ-1 RECEP-<br />

TOR MODULATORS<br />

• IMIDAZOLE 4-CARBOXAMIDES SUBSTI-<br />

TUÉS COMME MODULATEURS DES<br />

RÉCEPTEURS DE CHOLÉCYSTOKININE 1<br />

(73) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065, US<br />

(72) BERGER, Richard, Rahway, New Jersey<br />

07065-0907, US<br />

EDMONDSON, Scott, Rahway, New Jersey<br />

07065-0907, US<br />

HANSEN, Alexa, Danville ,CA 94526, US<br />

ZHU, Cheng, Rahway, New Jersey 07065-<br />

0907, US<br />

(74) Buchan, Gavin MacNicol, et al, Merck Sharp<br />

& Dohme Limited <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

C07D 401/12 → (51) A61P 35/00<br />

C07D 401/14 → (51) C09B 5/14<br />

C07D 403/06 → (51) A61P 35/00<br />

C07D 403/06 → (51) C07D 401/06<br />

C07D 403/12 → (51) A61P 35/00<br />

C07D 405/14 → (51) C07D 401/06<br />

C07D 409/04 → (51) C07D 213/26<br />

(51) C07D 413/12 (11) 2 066 663 B1<br />

A61K 31/4155 A61P 3/10<br />

A61P 29/00 A61P 25/30<br />

(25) En (26) En<br />

(21) 07801977.5 (22) 29.08.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 10.06.2009<br />

465<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>27</strong>/<strong>2011</strong>) 06.07.<strong>2011</strong><br />

(86) EP 2007/007556 29.08.2007<br />

(87) WO 2008/025539 2008/10 06.03.2008<br />

(30) 29.08.2006 US 840912 P<br />

29.08.2006 EP 06018024<br />

(54) • HETEROCYCLISCHE FXR-BINDENDE VER-<br />

BINDUNGEN<br />

• HETEROCYCLIC FXR BINDING COM-<br />

POUNDS<br />

• COMPOSÉS DE LIAISON AU FXR HÉTÉ-<br />

ROCYCLIQUES<br />

(73) Phenex Pharmaceuticals AG, J542N, Werksgelände<br />

BASF, 67056 Ludwigshafen, DE<br />

(72) KREMOSER, Claus, 69121 Heidelberg, DE<br />

DEUSCHLE, Ulrich, 67549 Worms, DE<br />

ABEL, Ulrich, 69126 Heidelberg, DE<br />

SCHULZ, Andreas, 69118 Heidelberg, DE<br />

(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser<br />

Anwaltssozietät, Leopoldstrasse 4,<br />

80802 München, DE<br />

C07D 413/12 → (51) A61P 35/00<br />

(51) C07D 417/04 (11) 2 118 099 B1<br />

(25) En (26) En<br />

(21) 08708929.8 (22) 13.02.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 18.11.2009<br />

(86) EP 2008/051704 13.02.2008<br />

(87) WO 2008/098949 2008/34 21.08.2008<br />

(30) 13.02.2007 US 889587 P<br />

(54) • VERFAHREN ZUR SYNTHESE VON 2-<br />

AMINOTHIAZOLVERBINDUNGEN ALS<br />

KINASEINHIBITOREN<br />

• PROCESS FOR THE SYNTHESIS OF 2-<br />

AMINOTHIAZOLE COMPOUNDS AS<br />

KINASE INHIBITORS<br />

• PROCÉDÉ DE SYNTHÈSE DE COMPOSÉS<br />

2-AMINOTHIAZOLE COMME INHIBITEURS<br />

DE KINASE<br />

(73) AB Science, 3, avenue George V, 75008<br />

Paris, FR<br />

(72) MOUSSY, Alain, F-75006 Paris, FR<br />

REGINAULT, Philippe, F-21121 Fontaine-les-<br />

Dijon, FR<br />

BELLAMY, François, F-21910 Saulon Larue,<br />

FR<br />

LERMET, Anne, F-69100 Villeurbanne, FR<br />

(74) Portal, Frédéric, et al, Cabinet Beau de<br />

Loménie 158, rue de l'Université, 75340<br />

Paris Cedex 07, FR<br />

(51) C07D 475/04 (11) 2 162 456 B1<br />

(25) De (26) De<br />

(21) 08748372.3 (22) 29.05.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 17.03.2010<br />

(86) CH 2008/000242 29.05.2008<br />

(87) WO 2008/144953 2008/49 04.12.2008<br />

(30) 30.05.2007 CH 856072007<br />

(54) • Stabile kristalline (6S) -N (5) -Methyl-<br />

5,6,7,8-tetrahydrofolsäure, deren Herstellung<br />

und Verwendung<br />

• Stable crystalline (6S)-N(5)-methyl-<br />

5,6,7,8-tetrahydrofolic acid, process for its<br />

preparation and its use<br />

• Acide (6S)-N-(5)-méthyl-5,6,7,8-tétrahydrofolique<br />

stable et cristallin, procédé pour<br />

sa préparation et son utilisation<br />

(73) Cerbios-Pharma S.A., Via Pian Scairolo 6,<br />

CH-6917 Barbengo, CH<br />

(72) MANZOTTI, Raffella, I-22020 Pellio Intelvi<br />

(Como), IT<br />

MOROSOLI, Moreno, CH-6950 Tesserete, CH

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