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Bulletin 2011/27 - European Patent Office

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(C07C) II.1(1)<br />

(74) Schwarz, Albin, et al, Schwarz & Partner<br />

<strong>Patent</strong>anwälte Wipplingerstraße 30, 1010<br />

Wien, AT<br />

C07C 317/24 → (51) C07C 317/22<br />

C07C 323/19 → (51) C07C 317/22<br />

(51) C07C 323/20 (11) 1 745 014 B1<br />

C07C 59/72<br />

(25) En (26) En<br />

(21) 05742978.9 (22) 03.05.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

(43) 24.01.2007<br />

(86) EP 2005/052013 03.05.2005<br />

(87) WO 2005/105736 2005/45 10.11.2005<br />

(30) 05.05.2004 DK 200400718<br />

(54) • NEUE VERBINDUNGEN, DEREN HER-<br />

STELLUNG UND VERWENDUNG<br />

• NOVEL COMPOUNDS, THEIR PREPAR-<br />

ATION AND USE<br />

• NOUVEAUX COMPOSES, LEUR PREPA-<br />

RATION ET LEUR UTILISATION<br />

(73) High Point Pharmaceuticals, LLC, 4170<br />

Mendenhall Oaks Parkway, High Point, NC<br />

<strong>27</strong>265, US<br />

(72) POLIVKA, Zdenék, 150 00 Praha 5, CZ<br />

(74) Russell, Lindsey, et al, Elkington and Fife<br />

LLP Thavies Inn House 3-4 Holborn Circus,<br />

London EC1N 2HA, GB<br />

C07C 323/22 → (51) C07C 317/22<br />

C07C 323/25 → (51) C07C 317/22<br />

(51) C07D 201/00 (11) 1 492 765 B1<br />

(25) En (26) En<br />

(21) 0<strong>27</strong>59233.6 (22) 01.08.2002<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR IE IT LI LU MC NL PT SE SK TR<br />

AL LT LV MK RO SI<br />

(43) 05.01.2005<br />

(86) US 2002/024323 01.08.2002<br />

(87) WO 2003/014075 2003/08 20.02.2003<br />

(30) 03.08.2001 US 310013 P<br />

06.02.2002 US 355510 P<br />

(54) • GAMMA SEKRETASE INHIBITOREN<br />

• NOVEL GAMMA SECRETASE INHIBITORS<br />

• NOUVEAUX INHIBITEURS DE GAMMA-<br />

SECRETASE<br />

(73) Schering Corporation, 2000 Galloping Hill<br />

Road, Kenilworth, NJ 07033-0530, US<br />

(72) ASBEROM, Theodros, West Orange, NJ<br />

07052, US<br />

GUZIK, Henry, S., Brooklyn, NY 11204, US<br />

JOSIEN, Hubert, B., Hoboken, NJ 07030, US<br />

PISSARNITSKI, Dmitri, A., Scotch Plains, NJ<br />

07076, US<br />

(74) Buchan, Gavin MacNicol, et al, Merck & Co.,<br />

Inc. <strong>European</strong> <strong>Patent</strong> Department Hertford<br />

Road, Hoddesdon, Hertfordshire EN11 9BU,<br />

GB<br />

C07D 205/08 → (51) A61K 31/397<br />

(51) C07D 209/42 (11) 1 833 789 B1<br />

(25) En (26) En<br />

(21) 05823911.2 (22) 22.12.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 19.09.2007<br />

(86) EP 2005/014171 22.12.2005<br />

(87) WO 2006/069799 2006/<strong>27</strong> 06.07.2006<br />

(30) 28.12.2004 EP 04078542<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

ENANTIOMERENANGEREICHERTER INDO-<br />

LIN-2-CARBONSÄURE<br />

• PROCESS FOR THE PREPARATION OF<br />

ENANTIOMERICALLY ENRICHED INDO-<br />

LINE-2-CARBOXYLIC ACID<br />

• PROCÉDÉ POUR LA PRÉPARATION DE<br />

L'ACIDE 2-CARBOXYLIQUE D'INDOLE<br />

ENANTIOMÈRIQUEMENT ENRICHI<br />

(73) DSM IP Assets B.V., Het Overloon 1, 6411<br />

TE Heerlen, NL<br />

(72) DE VRIES, Andreas, Hendrikus, Maria, NL-<br />

6212 CR Maastricht, NL<br />

DE VRIES, Johannes, Gerardus, NL-6228 GZ<br />

Maastricht, NL<br />

VAN ASSEMA, Friso, Bernard, Jan, NL-6166<br />

XK Geleen, NL<br />

DE LANGE, Ben, NL-6151 GE Munstergeleen,<br />

NL<br />

MINK, Daniel, B-4700 Eupen, BE<br />

HYETT, David, John, NL-6132 TH Sittard, NL<br />

MAAS, Peter, Johannes, Dominicus, NL-<br />

6155 ND Puth, NL<br />

(74) Hoogendam, Gerrie Christine, DSM Intellectual<br />

Property P.O. Box 4, 6100 AA Echt, NL<br />

C07D 209/48 → (51) H01L 51/50<br />

(51) C07D 213/26 (11) 1 989 184 B1<br />

A01N 47/24 A01N 47/40<br />

A01N 51/00 C07D 409/04<br />

(25) En (26) En<br />

(21) 07750608.7 (22) 09.02.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 12.11.2008<br />

(86) US 2007/003781 09.02.2007<br />

(87) WO 2007/095229 2007/34 23.08.2007<br />

(30) 10.02.2006 US 772108 P<br />

07.08.2006 US 836044 P<br />

(54) • INSEKTIZIDE N-SUBSTITUIERTE (6-<br />

HALOALKYLPYRIDIN-3-YL)ALKYL-SULFO-<br />

XIMINE<br />

• INSECTICIDAL N-SUBSTITUTED (6-<br />

HALOALKYLPYRIDIN-3-YL)ALKYL SUL-<br />

FOXIMINES<br />

• (6-HALOALKYLPYRIDIN-3-YL)ALKYL<br />

SULFOXIMINES N-SUBSTITUEES INSEC-<br />

TICIDES<br />

(73) Dow AgroSciences LLC, 9330 Zionsville<br />

Road, Indianapolis IN 46268-1054, US<br />

(72) LOSO, Michael, R., Carmel, IN 46032, US<br />

NUGENT, Benjamin, M., Brownsburg, IN<br />

46112, US<br />

HUANG, Jim, X., Carmel, IN 46032, US<br />

ROGERS, Richard, B., Mobile, AL 36603, US<br />

ZHU, Yuanming, Carmel, IN 46033, US<br />

RENGA, James, M., Indianapolis, IN 46220,<br />

US<br />

HEGDE, Vidyadhar, B., Carmel, IN 46032, US<br />

DEMARK, Joseph, J., Westfield, IN 46074,<br />

US<br />

(74) Dey, Michael, et al, Weickmann & Weickmann<br />

<strong>Patent</strong>anwälte Richard-Strauss-<br />

Strasse 80, 81679 München, DE<br />

(60) 1019<strong>27</strong>86.1<br />

(51) C07D 215/18 (11) 2 077 996 B1<br />

A61K 31/4704<br />

(25) En (26) En<br />

(21) 07788281.9 (22) 07.08.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

HR RS<br />

(43) 15.07.2009<br />

(86) EP 2007/058180 07.08.2007<br />

464<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>27</strong>/<strong>2011</strong>) 06.07.<strong>2011</strong><br />

(87) WO 2008/017669 2008/07 14.02.2008<br />

(30) 09.08.2006 EP 06118690<br />

09.08.2006 US 836856 P<br />

(54) • VERFAHREN ZUR AUFREINIGUNG VON<br />

MONTELUKAST UND DESSEN AMINSAL-<br />

ZEN<br />

• PURIFICATION PROCESS OF MONTELU-<br />

KAST AND ITS AMINE SALTS<br />

• PROCEDE DE PURIFICATION DE MONTE-<br />

LUKAST ET SES SELS D'AMINES& xA;<br />

(73) ESTEVE QUIMICA, S.A., Avenida Mare de<br />

Deu de Montserrat, 12, 08024 Barcelona, ES<br />

(72) GASANZ GUILLEN, Yolanda, E-08024 Barcelona,<br />

ES<br />

MONSALVATJE LLAGOSTERA, Montserrat,<br />

E-08024 Barcelona, ES<br />

TALAVERA ESCASANY, Pedro, E-08024<br />

Barcelona, ES<br />

(74) ZBM <strong>Patent</strong>s, Zea, Barlocci & Markvardsen<br />

Plaza Catalunya, 1, 08002 Barcelona, ES<br />

(51) C07D 233/72 (11) 1 493 734 B1<br />

A61K 31/415 A61P 13/12<br />

(25) Ja (26) En<br />

(21) 03745985.6 (22) 09.04.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 05.01.2005<br />

(86) JP 2003/004497 09.04.2003<br />

(87) WO 2003/084934 2003/42 16.10.2003<br />

(30) 10.04.2002 JP 2002107533<br />

(54) • NEUE KRISTALLFORM VON 5-HYDROXY-<br />

1-METHYLHYDANTOIN<br />

• NOVEL CRYSTAL FORM OF 5-HYDROXY-<br />

1-METHYLHYDANTOIN<br />

• NOUVELLE FORME CRISTALLINE DE 5-<br />

HYDROXY-1-METHYLHYDANTOINE<br />

(73) NIPPON ZOKI PHARMACEUTICAL CO. LTD.,<br />

1-2, Hiranomachi 2-chome, Chuo-ku, Osakashi,<br />

Osaka 541-0046, JP<br />

(72) OKAMOTO, Kaoru, Nippon Zoki Pharmaceutical<br />

Co.,Ltd, Kato-gu, JP<br />

NISHIMURA, Naoharu, Nippon Zoki Pharmaceutical<br />

Co.Ltd., Kato-gu, JP<br />

ISHII, Akira, Nippon Zoki Pharmaceutical Co.<br />

Ltd., Ono-shi, Hyogo 675-1363, JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastraße 4, 81925 München, DE<br />

(60) 08015840.5 / 2 003 122<br />

(51) C07D 235/18 (11) 1 611 108 B1<br />

(25) De (26) De<br />

(21) 04739071.1 (22) 26.03.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

LT LV<br />

(43) 04.01.2006<br />

(86) EP 2004/003217 26.03.2004<br />

(87) WO 2004/087676 2004/42 14.10.2004<br />

(30) 31.03.2003 DE 10314702<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

TELMISARTAN<br />

• METHOD FOR THE PRODUCTION OF<br />

TELMISARTAN<br />

• PROCEDE DE PRODUCTION DE TELMI-<br />

SARTAN<br />

(73) Boehringer Ingelheim International GmbH,<br />

Binger Strasse 173, 55216 Ingelheim am<br />

Rhein, DE<br />

(84) AT BE BG CH CY CZ DK EE ES FI FR GB GR<br />

HU IE IT LI LU MC NL PL PT RO SE SI SK TR<br />

(73) Boehringer Ingelheim Pharma GmbH & Co.<br />

KG, Binger Strasse 173, 55216 Ingelheim am<br />

Rhein, DE<br />

(84) DE<br />

(72) HAUEL, Norbert, 88433 Schemmerhofen, DE<br />

DACH, Rolf, 55435 Gau-Algesheim, DE

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