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Bulletin 2011/27 - European Patent Office

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(C07D) I.1(1)<br />

MERGNY, Jean-Louis, F-94800 Villejuif, FR<br />

GRIERSON, David, Vancouver BC V6T 2L1,<br />

CA<br />

(74) Gallois, Valérie, Cabinet BECKER & ASS-<br />

OCIES 25, rue Louis Le Grand, 75002 Paris,<br />

FR<br />

C07D 413/14 → (51) C07D 209/42<br />

C07D 417/12 → (51) A61K 31/40<br />

C07D 417/14 → (51) C07D 209/42<br />

(51) C07D 471/04 (11) 2 340 250 A1*<br />

A61K 31/437 G01N 33/53<br />

(25) En (26) En<br />

(21) 09802332.8 (22) 31.07.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) CA 2009/001087 31.07.2009<br />

(87) WO 2010/012106 2010/05 04.02.2010<br />

(30) 01.08.2008 US 855<strong>27</strong> P<br />

(54) • SELEKTIVE GLYCOSIDASEHEMMER UND<br />

IHRE VERWENDUNG<br />

• SELECTIVE GLYCOSIDASE INHIBITORS<br />

AND USES THEREOF<br />

• INHIBITEURS SÉLECTIFS DES GLYCOSI-<br />

DASES ET LEURS UTILISATIONS<br />

(71) Simon Fraser University, Innovation <strong>Office</strong><br />

8888 University Drive Multi Tenant Facility,<br />

Burnaby BC V5A 4W9, CA<br />

(72) VOCADLO, David, Jaro, Burnaby British<br />

Columbia V5A 4B5, CA<br />

MCEACHERN, Ernest John, Burnaby British<br />

Columbia V5A 4B5, CA<br />

STUBBS, Keith, Burnaby British Columbia<br />

V5A 4B5, CA<br />

(74) Atkinson, Jennifer, et al, Barker Brettell LLP<br />

100 Hagley Road, Edgbaston Birmingham<br />

B16 8QQ, GB<br />

C07D 471/04 → (51) C07D 209/42<br />

(51) C07D 471/06 (11) 2 340 251 A1*<br />

C12R 1/04 A61K 31/437<br />

A61P 35/00<br />

(25) En (26) En<br />

(21) 09791426.1 (22) 12.08.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) US 2009/053543 12.08.2009<br />

(87) WO 2010/019659 2010/07 18.02.2010<br />

(30) 12.08.2008 US 88192 P<br />

15.12.2008 US 122449 P<br />

(54) • PYRROLO[4,3,2-DE]CHINOLIN-8-AMIN-<br />

VERBINDUNGEN UND VERFAHREN ZU<br />

IHRER HERSTELLUNG UND ANWENDUNG<br />

• PYRROLO[4,3,2-DE]QUINOLIN-8-AMINE<br />

COMPOUNDS AND METHODS OF THEIR<br />

PREPARATION AND USE<br />

• COMPOSÉS PYRROLO[4,3,2-DE]QUINO-<br />

LÉIN-8-AMINES ET LEURS PROCÉDÉS DE<br />

PRÉPARATION ET D'UTILISATION<br />

(71) Wyeth LLC, Five Giralda Farms, Madison, NJ<br />

07940, US<br />

(72) HE, Min, Congers NY 10920, US<br />

JANSO, Jeffrey, Edwin, Montclair NJ 07042,<br />

US<br />

YU, Ker, Pine Brook NJ 07058, US<br />

MCDONALD, Leonard, Alexander, Mountainside<br />

NJ 07092, US<br />

BARBIERI, Laurel, Rita, Blauvelt NY 10913,<br />

US<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

GOPALSAMY, Ariamala, Mahway NJ 07430,<br />

US<br />

(74) Lane, Graham Mark Hamilton, Pfizer Limited<br />

<strong>European</strong> <strong>Patent</strong> Department Ramsgate<br />

Road, Sandwich CT13 9NJ, GB<br />

(51) C07D 487/04 (11) 2 340 252 A1*<br />

C07D 317/44 C07D 405/04<br />

C07D 405/12<br />

(25) En (26) En<br />

(21) 09813307.7 (22) 08.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) SE 2009/050999 08.09.2009<br />

(87) WO 2010/030224 2010/11 18.03.2010<br />

(30) 09.09.2008 US 95341 P<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

[1S-[1-ALPHA, 2-ALPHA, 3-BETA<br />

(1S*,2R*)5-BETA]]-3-[7-[2-(3,4- DIF-<br />

LUORPHENYL)CYCLOPROPYLAMINO]-5-<br />

(PROPYLTHIO)-3H-1,2,3-TRIAZOLO[4,5-<br />

D] PYRIMIDIN-3-YL]-5-(2-HYDROXYE-<br />

THOXY) CYCLOPENTAN-1,2-DIOL UND<br />

ZWISCHENPRODUKTEN DAVON<br />

• A PROCESS FOR PREPARING [1S- ]1-<br />

ALPHA, 2-ALPHA, 3-BETA (1S*, 2R*) 5-<br />

BETA] ]-3- [7- [2- (3, 4-DIF LUOROPHE-<br />

NYL) -CYCLOPROPYLAMINO]- 5- (PRO-<br />

PYLTHIO) -3H-1, 2, 3-TRIAZOLO [4, 5-D]<br />

PYRIMIDIN-3-YL]-5- (2- HYDRO-<br />

XYETHOXY) CYCLOPENTANE-1, 2-DIOL<br />

AND TO ITS INTERMEDIATES<br />

• PROCÉDÉ POUR PRÉPARER LE [1S-[1-<br />

ALPHA,2-ALPHA,3-BÊTA(1S*,2R*)-5-<br />

BÊTA]]-3-[7-[2-(3,4-DIFLUOROPHÉNYL)-<br />

CYCLOPROPYLAMINO]-5-(PROPYLTHIO)-<br />

3H-1,2,3-TRIAZOLO[4,5-D]PYRIMIDIN-3-<br />

YL]-5-(2-HYDROXYÉTHOXY)CYCLOPEN-<br />

TANE-1,2-DIOL ET SES INTERMÉDIAIRES<br />

(71) AstraZeneca AB, 151 85 Södertälje, SE<br />

(72) AUFDENBLATTEN, Rhony, CH-3930 Visp, CH<br />

BOHLIN, Martin, Hans, S-151 85 Södertälje,<br />

SE<br />

HELLSTRÖM, Helena, S-151 85 Södertälje,<br />

SE<br />

JOHANSSON, Peter, W, S-151 85 Södertälje,<br />

SE<br />

LARSSON, Ulf, G, S-151 85 Södertälje, SE<br />

RECKNAGEL, Mikaela, S-151 85 Södertälje,<br />

SE<br />

WEISS, Ursula, heiress of WEISS Andreas<br />

(Deceased), CH-3939 Eggerberg, CH<br />

C07D 487/04 → (51) C07D 209/42<br />

(51) C07D 489/12 (11) 2 340 253 A2*<br />

(25) En (26) En<br />

(21) 09789384.6 (22) 29.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) US 2009/005377 29.09.2009<br />

(87) WO 2010/039222 2010/14 08.04.2010<br />

(88) 18.11.2010<br />

(30) 30.09.2008 US 194696 P<br />

(54) • VERFAHREN ZUR SELEKTIVEN AMINIE-<br />

RUNG VON KETOMORPHINANEN<br />

• PROCESSES FOR THE SELECTIVE AMI-<br />

NATION OF KETOMORPHINANS<br />

• PROCÉDÉS D'AMINATION SÉLECTIVE DE<br />

CÉTOMORPHINANES<br />

(71) Mallinckrodt Inc., 675 McDonnell Boulevard,<br />

Hazelwood, MO 63042, US<br />

(72) HUDSON, Edmund, C., Clayton Missouri<br />

63105, US<br />

64<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>27</strong>/<strong>2011</strong>) 06.07.<strong>2011</strong><br />

TERAMURA, Douglas, Valley Park Missouri<br />

63088, US<br />

GROTE, Christopher, W., Webster Groves<br />

Missouri 63119, US<br />

THOMASSON, Catherine, E., Webster Groves<br />

Missouri 63119, US<br />

CANTRELL, Gary, L., Troy Illinois 62294, US<br />

(74) Albrecht, Thomas, Kraus & Weisert <strong>Patent</strong>und<br />

Rechtsanwälte Thomas-Wimmer-Ring<br />

15, 80539 München, DE<br />

(51) C07D 491/00 (11) 2 340 254 A1*<br />

C07D 513/00 C07D 515/00<br />

(25) En (26) En<br />

(21) 09813797.9 (22) 15.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) US 2009/056988 15.09.2009<br />

(87) WO 2010/031054 2010/11 18.03.2010<br />

(30) 15.09.2008 US 96940 P<br />

02.06.2009 US 183209 P<br />

(54) • ZUSAMMENSETZUNGEN UND VERFAH-<br />

REN ZUR BEHANDLUNG VON EPILEPSIE<br />

• COMPOSITIONS AND METHODS FOR<br />

TREATING EPILEPSY<br />

• COMPOSITIONS ET PROCÉDÉS POUR<br />

TRAITER L ÉPILEPSIE<br />

(71) Biovista, Inc., 9<strong>27</strong> Raymond Road, Charlottesville,<br />

VA 22902, US<br />

(72) DEFTEREOS, Spyros, GR-15342 Athens, GR<br />

PERSIDIS, Andreas, GR-16673 Athens, GR<br />

(74) Elsy, David, Withers & Rogers LLP Goldings<br />

House 2 Hays Lane, London SE1 2HW, GB<br />

C07D 513/00 → (51) C07D 491/00<br />

C07D 515/00 → (51) C07D 491/00<br />

(51) C07F 7/28 (11) 2 340 255 A2*<br />

(25) En (26) En<br />

(21) 09817960.9 (22) 24.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) KR 2009/005442 24.09.2009<br />

(87) WO 2010/038950 2010/14 08.04.2010<br />

(88) 17.06.2010<br />

(30) 30.09.2008 KR 20080095869<br />

(54) • NEUE ÜBERGANGSMETALLKATALYSA-<br />

TORSYSTEME UND -VERFAHREN ZUR<br />

HERSTELLUNG VON ETHYLEN-HOMO-<br />

POLYMEREN ODER -COPOLYMEREN AUS<br />

ETHYLEN UND ALPHA-OLEFINEN DAMIT<br />

• NEW TRANSITION METAL CATALYTIC<br />

SYSTEMS AND METHODS FOR PREPAR-<br />

ING ETHYLENE HOMOPOLYMERS OR<br />

COPOLYMERS OF ETHYLENE AND a-<br />

OLEFINS USING THE SAME<br />

• NOUVEAUX SYSTÈMES CATALYTIQUES À<br />

BASE DE MÉTAUX DE TRANSITION ET<br />

PROCÉDÉS DE PRÉPARATION D HOMO-<br />

POLYMÈRES D ÉTHYLÈNE OU DE COPO-<br />

LYMÈRES D ÉTHYLÈNE ET D -OLÉFINES<br />

LES UTILISANT<br />

(71) SK Energy Co., Ltd., 99, Seorin-dong<br />

Jongno-gu, Seoul 110-110, KR<br />

(72) OK, Myungahn, Daejeon 305-500, KR<br />

SHIN, Dongcheol, Daejeon 305-762, KR<br />

JEONG, Jisu, Daejeon 305-712, KR<br />

HAHN, Jongsok, Daejeon 305-761, KR<br />

LEE, Hoseong, Seoul 151-050, KR<br />

SHIN, Daeho, Daejeon 305-761, KR

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