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Bulletin 2011/27 - European Patent Office

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(C07C) I.1(1)<br />

(25) De (26) De<br />

(21) 09778162.9 (22) <strong>27</strong>.08.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) EP 2009/006226 <strong>27</strong>.08.2009<br />

(87) WO 2010/022953 2010/09 04.03.2010<br />

(88) <strong>27</strong>.05.2010<br />

(30) 29.08.2008 DE 102008044993<br />

(54) • SYNTHESE VON MYRTUCOMMULON A<br />

UND MYRTUCOMMULON-ANALOGA<br />

• SYNTHESIS OF MYRTUCOMMULON A<br />

AND MYRTUCOMMULON ANALOGUES<br />

• SYNTHÈSE DE MYRTUCOMMULONE A ET<br />

D'ANALOGUES À LA MYRTUCOMMULONE<br />

(71) Universität des Saarlandes, Campus Saarbrücken,<br />

66123 Saarbrücken, DE<br />

(72) JAUCH, Johann, 66564 Ottweiler, DE<br />

(74) Samson & Partner, Widenmayerstrasse 5,<br />

80538 München, DE<br />

C07C 49/723 → (51) C07C 49/713<br />

C07C 209/00 → (51) B01J 21/12<br />

(51) C07C 213/08 (11) 2 340 240 A2*<br />

C07C 215/12<br />

(25) En (26) En<br />

(21) 09736707.2 (22) 06.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) US 2009/005476 06.10.2009<br />

(87) WO 2010/042164 2010/15 15.04.2010<br />

(88) 17.06.2010<br />

(30) 06.10.2008 US 195456 P<br />

(54) • TRANSALKOXYLIERUNG NUKLEOPHILER<br />

VERBINDUNGEN<br />

• TRANSALKOXYLATION OF NUCLEOPHILIC<br />

COMPOUNDS<br />

• TRANSALKOXYLATION DE COMPOSES<br />

NUCLEOPHILES<br />

(71) Union Carbide Chemicals & Plastics Technology<br />

LLC, 2020 Dow Center, Midland, MI<br />

48674, US<br />

(72) KING, Stephen, W., League City, Texas<br />

77573, US<br />

HOFFMAN, William, C., Dunbar, West Virginia<br />

25064, US<br />

(74) Raynor, John, Beck Greener Fulwood House<br />

12 Fulwood Place, London WC1V 6HR, GB<br />

C07C 215/12 → (51) C07C 213/08<br />

C07C 237/20 → (51) C07C 311/33<br />

(51) C07C 259/06 (11) 2 340 241 A1*<br />

C07C 321/28 C07D 211/34<br />

C07D 213/56 C07D 307/16<br />

C07D 307/81 C07D 309/22<br />

A61P 31/04 A61K 31/166<br />

(25) En (26) En<br />

(21) 09782998.0 (22) 15.09.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) EP 2009/061905 15.09.2009<br />

(87) WO 2010/031750 2010/12 25.03.2010<br />

(30) 17.09.2008 US 97664 P<br />

(54) • ORGANISCHE VERBINDUNGEN FÜR<br />

ANWENDUNGEN BEI DER BEHANDLUNG<br />

BAKTERIELLER INFEKTIONEN<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

• ORGANIC COMPOUNDS FOR APPLICA-<br />

TIONS IN BACTERIAL INFECTIONS<br />

TREATMENT<br />

• COMPOSÉS ORGANIQUES DESTINÉS À<br />

ÊTRE APPLIQUÉS DANS LE TRAITEMENT<br />

D'INFECTIONS BACTÉRIENNES<br />

(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(72) DOBLER, Markus, Rolf, Cambridge, Massachusetts<br />

02139, US<br />

LENOIR, Francois, Cambridge, Massachusetts<br />

02139, US<br />

PARKER, David, Thomas, Cambridge, Massachusetts<br />

02139, US<br />

PENG, Yunshan, Cambridge, Massachusetts<br />

02139, US<br />

PIIZZI, Grazia, CH-4002 Basel, CH<br />

WATTANASIN, Sompong, Waltham, Massachusetts<br />

02453, US<br />

(74) von Sprecher, Georg, Novartis Pharma AG<br />

<strong>Patent</strong> Department, CH-4002 Basel, CH<br />

C07C <strong>27</strong>5/14 → (51) B01D 19/04<br />

C07C 311/08 → (51) C07C 311/33<br />

(51) C07C 311/33 (11) 2 340 242 A2*<br />

C07C 311/08 C07C 311/36<br />

C07C 237/20 A61K 31/18<br />

A61K 31/167 A61P <strong>27</strong>/02<br />

(25) En (26) En<br />

(21) 09822658.2 (22) 21.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) US 2009/061545 21.10.2009<br />

(87) WO 2010/048332 2010/17 29.04.2010<br />

(88) 22.07.2010<br />

(30) 22.10.2008 US 197081 P<br />

22.10.2008 US 197082 P<br />

22.10.2008 US 197083 P<br />

22.10.2008 US 197091 P<br />

(54) • VERBINDUNGEN ZUR BEHANDLUNG VON<br />

AUGENERKRANKUNGEN UND -LEIDEN<br />

• COMPOUNDS FOR TREATING OPHTHAL-<br />

MIC DISEASES AND DISORDERS<br />

• COMPOSÉS DE TRAITEMENT DE MALA-<br />

DIES ET TROUBLES OPHTALMIQUES<br />

(71) Acucela, Inc., 21720-23rd Drive SE, Suite<br />

120, Bothell, WA 98021, US<br />

(72) SCOTT, Ian L., Monroe Washington 98<strong>27</strong>2,<br />

US<br />

KUKSA, Vladimir A., Kenmore Washington<br />

98028-6323, US<br />

HONG, Feng, Bellevue Washington 98004,<br />

US<br />

KUBOTA, Ryo, Seattle Washington 98105,<br />

US<br />

GAGE, Jennifer, Kenmore Washington<br />

98028, US<br />

(74) Sahans, Sarah Anne, et al, HLBBshaw Merlin<br />

House Falconry Court Baker's Lane, Epping,<br />

Essex CM16 5DQ, GB<br />

C07C 311/36 → (51) C07C 311/33<br />

C07C 321/28 → (51) C07C 259/06<br />

C07D 207/16 → (51) A61K 31/40<br />

(51) C07D 209/42 (11) 2 340 243 A1*<br />

C07D 401/04 C07D 401/14<br />

C07D 403/04 C07D 403/14<br />

C07D 405/12 C07D 409/04<br />

C07D 409/14 C07D 413/04<br />

C07D 413/14 C07D 417/14<br />

C07D 471/04 C07D 487/04<br />

A61K 31/404 A61P 19/10<br />

62<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>27</strong>/<strong>2011</strong>) 06.07.<strong>2011</strong><br />

(25) En (26) En<br />

(21) 09740801.7 (22) 13.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) US 2009/060436 13.10.2009<br />

(87) WO 2010/045188 2010/16 22.04.2010<br />

(30) 17.10.2008 US 106207 P<br />

(54) • ALS MMP-13-INHIBITOREN GEEIGNETE<br />

HETEROARYLSUBSTITUIERTE INDOLVER-<br />

BINDUNGEN<br />

• HETEROARYL SUBSTITUTED INDOLE<br />

COMPOUNDS USEFUL AS MMP-13 INHI-<br />

BITORS<br />

• COMPOSÉS INDOLE À SUBSTITUTION<br />

HÉTÉROARYLE UTILISÉS COMME INHIBI-<br />

TEURS DE MMP-13<br />

(71) Boehringer Ingelheim International GmbH,<br />

Binger Strasse 173, 55216 Ingelheim, DE<br />

(72) ABEYWARDANE, Asitha, Ridgefield, Connecticut<br />

06877-0368, US<br />

FARMER, Bennett, Ridgefield, Connecticut<br />

06877-0368, US<br />

FARROW, Neil Alexander, Ridgefield, Connecticut<br />

06877-0368, US<br />

GAO, Donghong A., Ridgefield, Connecticut<br />

06877-0368, US<br />

HEIM-RIETHER, Alexander, Ridgefield, Connecticut<br />

06877-0368, US<br />

KEENAN, Lana Louise Smith, Ridgefield,<br />

Connecticut 06877-0368, US<br />

MUGGE, Ingo Andreas, Ridgefield, Connecticut<br />

06877-0368, US<br />

TAYLOR, Steven John, Ridgefield, Connecticut<br />

06877-0368, US<br />

XIONG, Zhaoming, Ridgefield, Connecticut<br />

06877-0368, US<br />

YU, Yang, Ridgefield, Connecticut 06877-<br />

0368, US<br />

ZHANG, Qiang, Ridgefield, Connecticut<br />

06877-0368, US<br />

(74) Hammann, Heinz, et al, Boehringer Ingelheim<br />

GmbH CD-<strong>Patent</strong>s Binger Straße 173, 55216<br />

Ingelheim am Rhein, DE<br />

C07D 211/34 → (51) C07C 259/06<br />

C07D 213/56 → (51) C07C 259/06<br />

(51) C07D 215/00 (11) 2 340 244 A1*<br />

(25) En (26) En<br />

(21) 09821043.8 (22) 09.10.2009<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA RS<br />

(86) US 2009/060076 09.10.2009<br />

(87) WO 2010/045095 2010/16 22.04.2010<br />

(30) 14.10.2008 US 105414 P<br />

(54) • VERBINDUNGEN UND ANWENDUNGS-<br />

VERFAHREN<br />

• COMPOUNDS AND METHODS OF USE<br />

• COMPOSÉS ET PROCÉDÉS D'UTILISA-<br />

TION<br />

(71) Xi, Ning, 565 Timberwood Ave., Thousand<br />

Oaks, CA 91360, US<br />

Shenzhen Dongyangguang Industrial Development<br />

Co., Ltd., E25, District E, the<br />

Dongfang Garden, Overseas Chinese Town,<br />

Nanshan District Shnezhen Guangdong, CN<br />

(72) Xi, Ning, Thousand Oaks, CA 91360, US<br />

Shenzhen Dongyangguang Industrial Development<br />

Co., Ltd., Overseas Chinese Town,<br />

Nanshan District Shnezhen Guangdong, CN<br />

(74) Ritter, Thomas Kurt, et al, Jones Day<br />

Prinzregentenstraße 11, 80538 München, DE

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