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Bulletin 2012/02 - European Patent Office

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(A01N) I.1(1)<br />

A01N 37/00 → (51) A61L 2/18<br />

A01N 41/06 → (51) A01N 57/20<br />

(51) A01N 43/04 (11) 2 403 335 A1*<br />

(25) En (26) En<br />

(21) 10749258.9 (22) 03.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/<strong>02</strong>6033 03.03.2010<br />

(87) WO 2010/101992 2010/36 10.09.2010<br />

(30) 03.03.2009 US 156922 P<br />

(54) • PHARMAZEUTISCHE ZUSAMMENSET-<br />

ZUNG ZUR VERABREICHUNG REZEPTOR-<br />

TYROSIN-KINASE-HEMMENDER VERBIN-<br />

DUNGEN INS AUGE<br />

• PHARMACEUTICAL COMPOSITION FOR<br />

DELIVERY OF RECEPTOR TYROSINE<br />

KINASE INHIBITING (RTKI) COMPOUNDS<br />

TO THE EYE<br />

• COMPOSITION PHARMACEUTIQUE POUR<br />

L'ADMINISTRATION À L' IL DE COMPO-<br />

SÉS INHIBANT LES RÉCEPTEURS TYRO-<br />

SINE KINASE (RTKI)<br />

(71) Alcon Research, Ltd., 6201 South Freeway,<br />

MS-TB4-8, Fort Worth, TX 76134-2099, US<br />

(72) KABRA, Bhagwati P., Euless, Texas 76039,<br />

US<br />

GHOSH, Malay, Fort Worth, Texas 76109, US<br />

(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser,<br />

Anwaltssozietät Leopoldstrasse 4,<br />

808<strong>02</strong> München, DE<br />

(51) A01N 43/16 (11) 2 403 336 A1*<br />

A01N 59/16 A01N 59/20<br />

A01P 3/00<br />

(25) En (26) En<br />

(21) 10709307.2 (22) 05.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

RS<br />

(86) US 2010/000688 05.03.2010<br />

(87) WO 2010/101659 2010/36 10.09.2010<br />

(30) 06.03.2009 US 158111 P<br />

10.03.2009 US 158882 P<br />

(54) • PFLANZENBEHANDLUNGSZUSAMMEN-<br />

SETZUNGEN UND VERWENDUNGSVER-<br />

FAHREN DAFÜR<br />

• PLANT TREATMENT COMPOSITIONS AND<br />

METHODS FOR THEIR USE<br />

• COMPOSITIONS DE TRAITEMENT DES<br />

PLANTES ET LEURS PROCÉDÉS D'UTILI-<br />

SATION<br />

(71) Gowan Co., 370 Main Street, Yuma, AZ<br />

85364, US<br />

(72) MAJURE, Wallace, Keith, West Monore, LA<br />

71291, US<br />

VANDERVORT, Nicholas, William, Cresco, IA<br />

52136, US<br />

DAVID, Paul, Joseph, Lititz, PA 17543, US<br />

DEETER, Brian, Duane, Auberry, CA 936<strong>02</strong>,<br />

US<br />

MELCHIOR, Gary, Joseph, Walla Walla, WA<br />

99362, US<br />

BRAZZLE, James, Richard, Sancramento, CA<br />

95829, US<br />

MUZYK, Kenneth, Roger, Brandon, FL<br />

33511, US<br />

MIRANDA, Frank, Rene, Holtville, CA 92250,<br />

US<br />

CHEUNG, Tak, Wai, Yuma, AZ 85364, US<br />

BAIN, Oakford, George, Yuma, AZ 85365, US<br />

FRIENDEN, John, Edward, Kansas City, MA<br />

64152, US<br />

MARSDEN, David, Alexander, Yuma, AZ<br />

85367, US<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

MOBERG, Olaf, Christian, New Brighton, MN<br />

55112, US<br />

OELTJEN, Susan, Toddie, Lake Elmo, MN<br />

55042, US<br />

RUEB, Christopher, John, St. Paul, MN<br />

55119, US<br />

HENDRICKSON, William, Arthur, Stillwater,<br />

OK 55082, US<br />

(74) Delaney, Jennifer, Appleyard Lees 15 Clare<br />

Road, Halifax, Yorkshire HX1 2HY, GB<br />

(51) A01N 43/42 (11) 2 403 337 A2*<br />

(25) En (26) En<br />

(21) 10749264.7 (22) 03.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/<strong>02</strong>6052 03.03.2010<br />

(87) WO 2010/1<strong>02</strong>003 2010/36 10.09.2010<br />

(88) 10.03.2011<br />

(30) 03.03.2009 US 156908 P<br />

(54) • ALKYLSULFONYL-2,3-DIHYDROSPIRO<br />

[INDEN-1,4'-PIPERIDIN]-ANALOGE ALS<br />

GLYT1-HEMMER, VERFAHREN ZU IHRER<br />

HERSTELLUNG SOWIE IHRE VERWEN-<br />

DUNG ZUR BEHANDLUNG PSYCHIATRI-<br />

SCHER ERKRANKUNGEN<br />

• ALKYLSULFONYL-2,3-DIHYDROSPIRO<br />

[INDENE-1,4'-PIPERIDINE] ANALOGS AS<br />

GLYT1 INHIBITORS, METHODS FOR<br />

MAKING SAME, AND USE OF SAME IN<br />

TREATING PSYCHIATRIC DISORDERS<br />

• ANALOGUES D'ALKYLSULFONYL-2,3-<br />

DIHYDROSPIRO[INDÈNE-1,4'-PIPÉRI-<br />

DINE] EN TANT QU'INHIBITEURS DE<br />

GLYT1, LEURS PROCÉDÉS DE FABRICA-<br />

TION ET LEUR UTILISATION DANS LE<br />

TRAITEMENT DE TROUBLES PSYCHIA-<br />

TRIQUES<br />

(71) Vanderbilt University, <strong>Office</strong> Of Technology<br />

Transfer 305 Kirkland Hall, Nashville, Tennessee<br />

37240, US<br />

(72) LINDSLEY, Craig, W., Brentwood TN 37<strong>02</strong>7,<br />

US<br />

CONN, Jeffrey, P., Brentwood TN 37<strong>02</strong>7, US<br />

WILLIAMS, Richard, Nashville TN 37221, US<br />

JONES, Carrie, K., Nashville TN 37221, US<br />

SHEFFLER, Douglas, J., Nashville TN 37205,<br />

US<br />

(74) Tostmann, Holger Carl, Wallinger Ricker<br />

Schlotter Tostmann <strong>Patent</strong>- und Rechtsanwälte<br />

Zweibrückenstrasse 5-7, 80331<br />

München, DE<br />

(51) A01N 43/50 (11) 2 403 338 A1*<br />

A01N 43/52 A61K 31/415<br />

(25) En (26) En<br />

(21) 10749107.8 (22) 22.<strong>02</strong>.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/<strong>02</strong>4871 22.<strong>02</strong>.2010<br />

(87) WO 2010/101724 2010/36 10.09.2010<br />

(30) 04.03.2009 US 157430 P<br />

10.11.2009 US 259743 P<br />

(54) • IMIDAZOLDERIVATE ALS FAAH-MODULA-<br />

TOREN UND ALS FAAH-KONTRASTMIT-<br />

TEL<br />

• IMIDAZOLE DERIVATIVES USEFUL AS<br />

MODULATORS OF FAAH AND AS FAAH<br />

IMAGING AGENTS<br />

• DÉRIVÉS D'IMIDAZOLE POUVANT ÊTRE<br />

UTILISÉS EN TANT QUE MODULATEURS<br />

DE LA FAAH ET EN TANT QU'AGENTS<br />

D'IMAGERIE DE LA FAAH<br />

(71) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907,<br />

US<br />

(72) LIU, Ping, Rahway New Jersey 07065-0907,<br />

US<br />

17<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>02</strong>/<strong>2012</strong>) 11.01.<strong>2012</strong><br />

DEVITA, Robert, J., Rahway New Jersey<br />

07065-0907, US<br />

LIN, Linus, S., Rahway New Jersey 07065-<br />

0907, US<br />

CHIODA, Marc, D., Rahway New Jersey<br />

07065-0907, US<br />

HAMILL, Terence, G., Rahway New Jersey<br />

07065-0907, US<br />

LI, Wenping, Rahway New Jersey 07065-<br />

0907, US<br />

(74) Horgan, James Michael Frederic, et al, Merck<br />

& Co., Inc. <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon Hertfordshire<br />

EN11 9BU, GB<br />

A01N 43/52 → (51) A01N 43/50<br />

A01N 43/54 → (51) C07D 239/88<br />

(51) A01N 43/58 (11) 2 403 339 A1*<br />

A61K 31/50 A61K 31/495<br />

(25) En (26) En<br />

(21) 10749110.2 (22) 23.<strong>02</strong>.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/<strong>02</strong>5<strong>02</strong>8 23.<strong>02</strong>.2010<br />

(87) WO 2010/101734 2010/36 10.09.2010<br />

(30) 06.03.2009 US 158109 P<br />

(54) • TUMORKOMBINATIONSTHERAPIE MIT<br />

EINEM AKT-HEMMER UND ANDEREN<br />

ANTUMORMITTELN<br />

• COMBINATION CANCER THERAPY WITH<br />

AN AKT INHIBITOR AND OTHER ANTIC-<br />

ANCER AGENTS<br />

• THÉRAPIE DE COMBINAISON ANTI-CAN-<br />

CER AVEC UN INHIBITEUR DE AKT ET<br />

D'AUTRES AGENTS ANTI-CANCER<br />

(71) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065-0907,<br />

US<br />

MSD K.K., Kitanomaru Square 1-13-12<br />

Kudankita, Chiyoda-ku Tokyo 1<strong>02</strong>-8667, JP<br />

(72) LAYTON, Mark, E., Rahway New Jersey<br />

07065-0907, US<br />

HIRAI, Hiroshi, Tokyo 1<strong>02</strong>-8667, JP<br />

KOTANI, Hidehito, Tokyo 1<strong>02</strong>-8667, JP<br />

(74) Hussain, Deeba, et al, Merck & Co., Inc.<br />

<strong>Patent</strong> Department Hertford Road, Hoddesdon<br />

Hertfordshire EN11 9BU, GB<br />

(51) A01N 43/82 (11) 2 403 340 A1*<br />

A61K 31/41<br />

(25) En (26) En<br />

(21) 10749400.7 (22) 05.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/<strong>02</strong>6380 05.03.2010<br />

(87) WO 2010/1<strong>02</strong>218 2010/36 10.09.2010<br />

(30) 06.03.2009 US 158080 P<br />

05.03.2009 US 157789 P<br />

05.03.2009 US 2<strong>02</strong>501 P<br />

09.10.2009 US 278649 P<br />

(54) • VERBINDUNGEN UND ZUSAMMENSET-<br />

ZUNGEN FÜR VERBESSERTE WAHRNEH-<br />

MUNG, HERSTELLUNGSVERFAHREN UND<br />

BEHANDLUNGSVERFAHREN<br />

• COMPOUNDS AND COMPOSITIONS FOR<br />

COGNITION-ENHANCEMENT, METHODS<br />

OF MAKING, AND METHODS OF TREATING<br />

• COMPOSÉS ET COMPOSITIONS POUR<br />

AMÉLIORER LA FONCTION COGNITIVE,<br />

PROCÉDÉS DE FABRICATION ET MÉTHO-<br />

DES DE TRAITEMENT<br />

(71) Mithridion, Inc., 505 Science Drive Suite C,<br />

Madison, WI 53711, US<br />

(72) TWOSE, Trevor, M., Fitchburg, WI 53711,<br />

US

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