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Bulletin 2012/02 - European Patent Office

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(C07D) I.1(2)<br />

(71) Shionogi & Co., Ltd., 1-8, Doshomachi 3chome<br />

Chuo-ku Osaka-shi, Osaka 541-0045,<br />

JP<br />

(72) SAKAGAMI, Masahiro, Osaka 553-00<strong>02</strong>, JP<br />

ARAKI, Hitomi, Osaka-shi Osaka 553-00<strong>02</strong>,<br />

JP<br />

HASHIZUME, Hiroshi, Osaka-shi Osaka 553-<br />

00<strong>02</strong>, JP<br />

YARI, Hiroshi, Osaka-shi Osaka 553-00<strong>02</strong>,<br />

JP<br />

TAKAYA, Kenji, Osaka-shi Osaka 553-00<strong>02</strong>,<br />

JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastraße 4, 81925 München, DE<br />

(51) C07D 207/404 (11) 2 404 903 A1<br />

A61K 51/00 C07B 59/00<br />

C07B 61/00<br />

(25) Ja (26) En<br />

(21) 10748713.4 (22) 01.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2010/053252 01.03.2010<br />

(87) WO 2010/101118 2010/36 10.09.2010<br />

(30) 04.03.2009 JP 2009050814<br />

(54) • VERFAHREN ZUR SYNTHESE VON [18F]<br />

SFB MITHILFE EINER MIKROSYNTHESE-<br />

TECHNIK<br />

• METHOD OF SYNTHESIZING [18F]SFB<br />

USING MICROSYNTHESIS TECHNIQUE<br />

• MÉTHODE DE SYNTHÈSE DU [18F]SFB<br />

PAR UNE TECHNIQUE DE MICROSYN-<br />

THÈSE& xA;<br />

(71) Shimadzu Corporation, 1, Nishinokyo-<br />

Kuwabaracho Nakagyo-ku, Kyoto-shi, Kyoto<br />

604-8511, JP<br />

Kyoto University, 36-1, Yoshida-honmachi,<br />

Sakyo-ku Kyoto-shi Kyoto 606-8501, JP<br />

(72) NAKANISHI Hiroaki, Kyoto-shi Kyoto 604-<br />

8511, JP<br />

SAIKI Hidekazu, Kyoto-shi Kyoto 604-8511,<br />

JP<br />

SAJI Hideo, Kyoto-shi Kyoto 606-8501, JP<br />

KIMURA Hiroyuki, Kyoto-shi Kyoto 606-<br />

8501, JP<br />

KAWASHIMA Hidekazu, Kyoto-shi Kyoto<br />

606-8501, JP<br />

TOMATSU Kenji, Kyoto-shi Kyoto 606-8501,<br />

JP<br />

KUGE Yuji, Kyoto-shi Kyoto 606-8501, JP<br />

(74) Müller-Boré & Partner <strong>Patent</strong>anwälte, Grafinger<br />

Straße 2, 81671 München, DE<br />

C07D 207/44 → (51) C07C 31/22<br />

(51) C07D 209/00 (11) 2 404 904 A1<br />

A61K 31/415 C07D 403/10<br />

C07D 471/04<br />

(25) En (26) En<br />

(21) 11171816.9 (22) 30.10.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK RS<br />

(27) 30.10.2006 PCT/US2006/042690<br />

(30) 04.11.2005 US 734030 P<br />

12.05.2006 US 747174 P<br />

23.08.2006 US 823344 P<br />

27.10.2006 US 553946<br />

(54) • Hemmer des 5-Lipoxygenase activierenden<br />

proteins (FLAP)<br />

• 5-lipoxygenase-activating protein (FLAP)<br />

inhibitors<br />

• Inhibiteurs de la proteine d'activation de la<br />

5-lipoxygenase (FLAP)<br />

(71) Amira Pharmaceuticals, Inc., 9535 Waples<br />

Street, Suite 100, San Diego, CA 92121, US<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(72) Hutchinson, John H, San Diego, California<br />

92121, US<br />

Prasit, Petpiboon Peppi, San Diego, CA<br />

California 92121, US<br />

Moran, Mark, Orinda, CA California 94563,<br />

US<br />

Evans, Jillian F, Calsbad, CA California<br />

92009, US<br />

Stearns, Brian Andrew, San Diego, CA<br />

California 92121, US<br />

Roppe, Jeffrey Roger, Temecula, CA California<br />

92592, US<br />

Li, Yiwei, San Diego, CA California 92131,<br />

US<br />

Zunic, Jasmine Eleanor, San Diego, CA<br />

California 92127, US<br />

Arruda, Jeannie M, La Jolla, CA California<br />

92037, US<br />

Stock, Nicholas Simon, San Diego, CA<br />

California 92111, US<br />

Haddach, Mustapha, San Diego, CA California<br />

92127, US<br />

(74) Price, Susanna Clare Hopley, et al, GlaxoSmithKline<br />

Corporate Intellectual Property 980<br />

Great West Road Brentford, Middlesex, TW8<br />

9GS, GB<br />

(62) 06836773.9 / 1 943 219<br />

C07D 211/14 → (51) C07D 295/18<br />

C07D 211/62 → (51) C07D 207/16<br />

(51) C07D 213/74 (11) 2 404 905 A1<br />

C07D 213/75 C07D 213/81<br />

C07D 213/82 C07D 237/20<br />

C07D 239/42 C07D 263/48<br />

C07D 277/42 C07D 401/10<br />

C07D 401/12 C07D 401/14<br />

C07D 405/12 C07D 413/10<br />

C07D 413/12 A61K 31/44<br />

A61K 31/50 A61K 31/53<br />

A61K 31/421 A61K 31/426<br />

A61K 31/4427 A61K 31/4965<br />

(25) En (26) En<br />

(21) 11158212.8 (22) 28.03.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

BA HR<br />

(27) 28.03.2007 PCT/US2007/007772<br />

(30) 31.03.2006 US 787859 P<br />

(54) • Neue Verbindungen<br />

• New compounds<br />

• Nouveaux composés<br />

(71) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(72) Serrano-Wu, Michael H, Belmont, MA <strong>02</strong>478,<br />

US<br />

Kwak, Young-Shin, Lexington, MA <strong>02</strong>421,<br />

US<br />

Liu, Wenming, Morris Plains, NJ 07950, US<br />

(74) Campbell, Lachlan Clive, Novartis Pharma AG<br />

<strong>Patent</strong> Department, 40<strong>02</strong> Basel, CH<br />

(62) 07754311.4 / 2 004 607<br />

(51) C07D 213/75 (11) 2 404 906 A1<br />

A61K 31/44 A61P 7/00<br />

(25) En (26) En<br />

(21) 11183853.8 (22) 01.11.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(30) <strong>02</strong>.11.2006 US 864145 P<br />

(54) • Verfahren zur Synthetisierung pharmazeutischer<br />

Salze aus einem Faktor XA-Hemmer<br />

• Methods of synthesizing pharmaceutical<br />

salts of a factor XA inhibitor<br />

221<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>02</strong>/<strong>2012</strong>) 11.01.<strong>2012</strong><br />

• Procédé de synthèse de sels pharmaceutiques<br />

d'un inhibiteur du facteur XA<br />

(71) Millennium Pharmaceuticals, Inc., 40 Landsdowne<br />

Street, Cambridge, MA <strong>02</strong>139, US<br />

(72) Kanter, James P., San Ramon, California<br />

94583, US<br />

Sujino, Keiko, Foster City, California 94404,<br />

US<br />

Zuberi, Sharique Sami, Folsom, California<br />

95630, US<br />

Scarborough, Robert M., ., US<br />

(74) Sexton, Jane Helen, J.A. Kemp & Co. 14<br />

South Square Gray's Inn, London WC1R 5JJ,<br />

GB<br />

(62) 07863800.4 / 2 077 995<br />

C07D 213/75 → (51) C07D 213/74<br />

C07D 213/81 → (51) C07D 213/74<br />

C07D 213/82 → (51) C07D 213/74<br />

C07D 225/<strong>02</strong> → (51) C07D 201/04<br />

C07D 233/<strong>02</strong> → (51) C07C 31/22<br />

C07D 237/20 → (51) C07D 213/74<br />

C07D 239/<strong>02</strong> → (51) A61K 31/505<br />

C07D 239/42 → (51) C07D 213/74<br />

C07D 239/47 → (51) A61K 31/505<br />

(51) C07D 239/70 (11) 2 404 907 A1<br />

A61K 31/517 A61P 35/00<br />

(25) En (26) En<br />

(21) 11169324.8 (22) 03.07.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(30) 05.07.2007 US 948147 P<br />

(54) • Pyrimidyl-Cyclopentane als AKT-Proteinkinasehemmer<br />

• Pyrimidyl cyclopentanes as AKT protein<br />

kinase inhibitors<br />

• Pyrimidyl cyclopentanes en tant qu'inhibiteurs<br />

de protéine kinase AKT<br />

(71) Array Biopharma, Inc., 3200 Walnut Street,<br />

Boulder, CO 80301, US<br />

Genentech, Inc., 1 DNA Way, South San<br />

Francisco CA 94080-4990, US<br />

(72) Bencsik, Josef, R., Longmont, CO Colorado<br />

80501, US<br />

Blake, James, F., Longmont, CO Colorado<br />

80504, US<br />

Kallan, Nicholas, C., Boulder, CO Colorado<br />

80301, US<br />

Mitchell, Ian, S., Lafayette, CO Colorado<br />

80<strong>02</strong>6, US<br />

Spencer, Keith, L., Lyons, CO Colorado<br />

80540, US<br />

Xiao, Dengming, Longmont, CO Colorado<br />

80501, US<br />

Xu, Rui, Longmont, CO Colorado 80504, US<br />

Chabot, Christine, San Mateo, CA California<br />

944<strong>02</strong>, US<br />

Liang, Jun, Palo Alto, CA California 94306,<br />

US<br />

Safina, Brian, S., Redwood City, CA California<br />

94061, US<br />

(74) Bailey, Sam Rogerson, Mewburn Ellis LLP<br />

33 Gutter Lane, London EC2V 8AS, GB<br />

(62) 08781340.8 / 2 173 723<br />

C07D 249/08 → (51) C07C 235/20

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