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Bulletin 2012/02 - European Patent Office

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(C07D) I.1(1)<br />

(71) F.I.S. Fabbrica Italiana Sintetici S.p.A., Viale<br />

Milano, 26, 36075 Alte di Montecchio<br />

Maggiore, IT<br />

(72) MOTTERLE, Riccardo, I-36057 Arcugnano<br />

Vicenza, IT<br />

ARVOTTI, Giancarlo, I-36075 Montecchio<br />

Maggiore Vicenza, IT<br />

BERGANTINO, Elisabetta, I-35010 Cadoneghe<br />

Padova, IT<br />

CASTELLIN, Andrea, I-35035 Mestrino<br />

Padova, IT<br />

FOGAL, Stefano, I-31030 Altivole Treviso, IT<br />

GALVAGNI, Marco, I-37131 Verona, IT<br />

(74) Long, Giorgio, et al, Jacobacci & Partners S.<br />

p.A. Via Senato 8, <strong>2012</strong>1 Milano, IT<br />

(51) C07D 213/75 (11) 2 403 832 A1*<br />

C07D 401/12 C07D 401/14<br />

C07D 403/12 C07D 413/14<br />

C07D 417/12 C07D 417/14<br />

A61K 31/44 A61P 35/00<br />

(25) En (26) En<br />

(21) 10708670.4 (22) 01.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/<strong>02</strong>5813 01.03.2010<br />

(87) WO 2010/101849 2010/36 10.09.2010<br />

(30) <strong>02</strong>.03.2009 US 156599 P<br />

23.09.2009 US 245187 P<br />

(54) • N-(HETERO)ARYL, 2-(HETERO)ARYL-<br />

SUBSTITUIERTE ACETAMIDE ZUR VER-<br />

WENDUNG ALS MODULATOREN DER<br />

WNT-SIGNALVERMITTLUNG<br />

• N- (HETERO)ARYL, 2- (HETERO)ARYL-<br />

SUBSTITUTED ACETAMIDES FOR USE AS<br />

WNT SIGNALING MODULATORS<br />

• ACÉTAMIDES À SUBSTITUTION N-<br />

(HÉTÉRO)ARYL, 2-(HÉTÉRO)ARYLE POUR<br />

UNE UTILISATION EN TANT QUE MODU-<br />

LATEURS DE LA VOIE DE SIGNALISATION<br />

WNT<br />

(71) IRM LLC, 131 Front Street P.O. Box HM<br />

2899, Hamilton HM LX, BM<br />

(72) CHENG, Dai, San Diego, California 92130,<br />

US<br />

ZHANG, Guobao, San Diego, California<br />

92130, US<br />

HAN, Dong, San Diego California 92014, US<br />

GAO, Wenqi, San Diego California 92127, US<br />

PAN, Shifeng, San Diego California 92130,<br />

US<br />

(74) Kiddle, Simon John, et al, Mewburn Ellis LLP<br />

33 Gutter Lane, London EC2V 8AS, GB<br />

(51) C07D 215/48 (11) 2 403 833 A1*<br />

A61K 31/519 C07D 401/12<br />

A61K 31/4375 A61K 31/5377<br />

C07D 401/14 A61K 31/47<br />

A61K 31/538 C07D 413/14<br />

A61K 31/4709 A61P 3/00<br />

C07D 417/12 A61K 31/497<br />

A61P 5/50 C07D 417/14<br />

A61K 31/501 A61P 9/00<br />

C07D 487/04 A61K 31/506<br />

A61P 35/<strong>02</strong><br />

(25) En (26) En<br />

(21) 10749227.4 (22) <strong>02</strong>.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA ME RS<br />

(86) US 2010/<strong>02</strong>5963 <strong>02</strong>.03.2010<br />

(87) WO 2010/101949 2010/36 10.09.2010<br />

(30) <strong>02</strong>.03.2009 US 156749 P<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(54) • B-SUBSTITUIERTE CHINOLINE UND ANA-<br />

LOGA DAVON ALS SIRTUIN-MODULATO-<br />

REN<br />

• 8-SUBSTITUTED QUINOLINES AND<br />

RELATED ANALOGS AS SIRTUIN MODU-<br />

LATORS<br />

• QUINOLÉINES SUBSTITUÉES EN 8 ET<br />

ANALOGUES ASSOCIÉS UTILISÉS COMME<br />

MODULATEURS DE SIRTUINE<br />

(71) Sirtris Pharmaceuticals, Inc., 200 Technology<br />

Square, Suite 300, Cambridge, MA<br />

<strong>02</strong>139, US<br />

(72) VU, Chi, B., Cambridge, MA <strong>02</strong>139, US<br />

CASAUBON, Rebecca, L., Cambridge, MA<br />

<strong>02</strong>139, US<br />

(74) Valentine, Jill Barbara, GlaxoSmithKline<br />

Corporate Intellectual Property (CN9.25.1)<br />

980 Great West Road, Brentford, Middlesex<br />

TW8 9GS, GB<br />

(51) C07D 231/12 (11) 2 403 834 A1*<br />

C07D 231/20 C07D 231/38<br />

C07D 401/04 C07D 401/12<br />

C07D 401/14 C07D 403/12<br />

C07D 407/12 C07D 409/04<br />

C07D 417/12 A61K 31/4155<br />

(25) En (26) En<br />

(21) 10707187.0 (22) 03.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA ME RS<br />

(86) US 2010/<strong>02</strong>6003 03.03.2010<br />

(87) WO 2010/101973 2010/36 10.09.2010<br />

(30) 03.03.2009 US 157046 P<br />

12.<strong>02</strong>.2010 US 304053 P<br />

(54) • FUNGIZIDE PYRAZOLE<br />

• Fungicidal pyrazoles<br />

• Pyrazoles fongicides<br />

(71) E. I. du Pont de Nemours and Company,<br />

1007 Market Street, Wilmington, DE 19898,<br />

US<br />

(72) LONG, Jeffrey, Keith, Wilmington Delaware<br />

19803, US<br />

HONG, Wonpyo, Lutherville Maryland 21093,<br />

US<br />

TAGGI, Andrew, Edmund, Newark Delaware<br />

19711, US<br />

(74) Beacham, Annabel Rose, Dehns St Bride's<br />

House 10 Salisbury Square, London EC4Y<br />

8JD, GB<br />

C07D 231/20 → (51) C07D 231/12<br />

C07D 231/38 → (51) C07D 231/12<br />

(51) C07D 233/54 (11) 2 403 835 A1*<br />

C07D 401/12 C07D 403/12<br />

C07D 413/12 C07D 417/12<br />

A61K 31/41 A61P 25/00<br />

(25) En (26) En<br />

(21) 10708634.0 (22) <strong>02</strong>.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) IB 2010/050896 <strong>02</strong>.03.2010<br />

(87) WO 2010/100606 2010/36 10.09.2010<br />

(30) 03.03.2009 US 156963 P<br />

(54) • NEUE PHENYLIMIDAZOLE UND PHE-<br />

NYLTRIAZOLE ALS MODULATOREN VON<br />

GAMMA-SEKRETASE<br />

• NOVEL PHENYL IMIDAZOLES AND PHE-<br />

NYL TRIAZOLES AS GAMMA-SECRETASE<br />

MODULATORS<br />

• NOUVEAUX PHÉNYL IMIDAZOLES ET<br />

PHÉNYL TRIAZOLES EN TANT QUE<br />

MODULATEURS DE LA GAMMA SÉCRÉ-<br />

TASE<br />

83<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>02</strong>/<strong>2012</strong>) 11.01.<strong>2012</strong><br />

(71) Pfizer Inc., 235 East 42nd Street, New York,<br />

NY 10017, US<br />

(72) ALLEN, Martin, Patrick, Connecticut 06340,<br />

US<br />

AM ENDE, Christopher, William, Connecticut<br />

06340, US<br />

BRODNEY, Michael, Aaron, Connecticut<br />

06340, US<br />

DOUNAY, Amy, Beth, Connecticut 06340, US<br />

JOHNSON, Douglas, Scott, Connecticut<br />

06340, US<br />

PETTERSSON, Martin, Youngjin, Connecticut<br />

06340, US<br />

SCHWARZ, Jacob, Bradley, San Ramon<br />

California 94582, US<br />

TRAN, Tuan, Phong, Connecticut 06340, US<br />

(74) Summers, Victoria Clare, Pfizer <strong>European</strong><br />

<strong>Patent</strong> Department 23-25, avenue du Docteur<br />

Lannelongue, 75668 Paris Cedex 14, FR<br />

(51) C07D 239/10 (11) 2 403 836 A2*<br />

C09D 201/00 C08G 61/12<br />

(25) En (26) En<br />

(21) 10749167.2 (22) <strong>02</strong>.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) US 2010/<strong>02</strong>5838 <strong>02</strong>.03.2010<br />

(87) WO 2010/101863 2010/36 10.09.2010<br />

(88) 06.01.2011<br />

(30) 01.03.2010 US 714911<br />

03.03.2009 US 157058 P<br />

(54) • BÜRSTENPOLYMERBESCHICHTUNG MIT-<br />

TELS IN-SITU-POLYMERISIERUNG VON<br />

EINER LICHTREAKTIVEN OBERFLÄCHE<br />

• BRUSH POLYMER COATING BY IN SITU<br />

POLYMERIZATION FROM PHOTOREAC-<br />

TIVE SURFACE<br />

• REVÊTEMENTS POLYMÈRES À LA<br />

BROSSE PAR POLYMÉRISATION IN SITU<br />

À PARTIR D'UNE SURFACE PHOTORÉAC-<br />

TIVE<br />

(71) Innovative Surface Technologies, Inc., 1000<br />

Westgate, Drive 260, Saint Paul, MN 55114,<br />

US<br />

Wen, Jie, 8866 Belvedere Drive, Eden Prairie,<br />

MN 55347, US<br />

(72) WEN, Jie, Eden Prairie, MN 55347, US<br />

LAWIN, Laurie, R., New Brighton, MN<br />

55112, US<br />

GUIRE, Patrick, Hopkins, MN 55305-4604,<br />

US<br />

(74) Johnson, Stephen William, et al, Venner<br />

Shipley LLP Byron House Cambridge Business<br />

Park Cowley Road, Cambridge CB4<br />

0WZ, GB<br />

(51) C07D 239/88 (11) 2 403 837 A1*<br />

C07D 401/04 C07D 403/04<br />

A01N 43/54<br />

(25) En (26) En<br />

(21) 10706254.9 (22) 03.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2010/052693 03.03.2010<br />

(87) WO 2010/100189 2010/36 10.09.2010<br />

(30) 04.03.2009 US 157375 P<br />

(54) • 3-ARYLCHINAZOLIN-4-ONVERBINDUN-<br />

GEN ZUR BEKÄMPFUNG VON WIRBEL-<br />

LOSEN SCHÄDLINGEN<br />

• 3-ARYLQUINAZOLIN-4-ONE COMPOUNDS<br />

FOR COMBATING INVERTEBRATE PESTS<br />

• COMPOSÉS DE 3-ARYLQUINAZOLIN-4-<br />

ONE POUR LUTTER CONTRE LES ORGA-<br />

NISMES NUISIBLES INVERTÉBRÉS<br />

(71) BASF SE, 67056 Ludwigshafen, DE<br />

(72) GROSS, Steffen, 67063 Ludwigshafen, DE<br />

KÖRBER, Karsten, 69214 Eppelheim, DE

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