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Bulletin 2012/02 - European Patent Office

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(C07D) II.1(1)<br />

MATSUMOTO, Toshifumi MITSUBISHI<br />

PHARMA CORP. , Tokyo 103-8405, JP<br />

EGI, Y., MITSUBISHI PHARMA CORP.,<br />

Tokyo Off., Tokyo 103-8405, JP<br />

TAKAHASHI, T., MITSUBISHI PHARMA<br />

CORP., Tokyo Off., Tokyo 103-8405, JP<br />

(74) von Kreisler Selting Werner, Deichmannhaus<br />

am Dom Bahnhofsvorplatz 1, 50667 Köln,<br />

DE<br />

(51) C07D 217/26 (11) 2 150 534 B1<br />

C07D 401/06 C07D 403/06<br />

A61K 31/472 A61K 31/4725<br />

A61P 25/18<br />

(25) En (26) En<br />

(21) 08734547.6 (22) 24.04.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(43) 10.<strong>02</strong>.2010<br />

(86) DK 2008/050092 24.04.2008<br />

(87) WO 2008/131779 2008/45 06.11.2008<br />

(30) 26.04.2007 DK 200700620<br />

(54) • ISOCHINOLINONDERIVATE ALS NK3-<br />

ANTAGONISTEN<br />

• ISOQUINOLINONE DERIVATIVES AS NK3<br />

ANTAGONISTS<br />

• DÉRIVÉS D'ISOQUINOLINONE UTILISÉS<br />

EN TANT QU'ANTAGONISTES DE NK3<br />

(73) H. Lundbeck A/S, Ottiliavej 9, 2500 Valby, DK<br />

(72) SIMONSEN, Klaus, Bæk, DK-5230 Odense M,<br />

DK<br />

KEHLER, Jan, DK-2800 Kgs. Lyngby, DK<br />

JUHL, Karsten, DK-2670 Greve, DK<br />

KHANZHIN, Nikolay, DK-3050 Humlebæk, DK<br />

NIELSEN, Søren, Møller, DK-3400 Hillerød,<br />

DK<br />

C07D 223/10 → (51) C01B 39/46<br />

(51) C07D 233/50 (11) 1 960 369 B1<br />

C07D 263/28 C07D 277/18<br />

A61K 31/427 A01N 43/78<br />

A61P 33/00<br />

(25) En (26) En<br />

(21) 06819493.5 (22) 15.11.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK RS<br />

(43) 27.08.2008<br />

(86) EP 2006/068482 15.11.2006<br />

(87) WO 2007/060121 2007/22 31.05.2007<br />

(30) 25.11.2005 US 739730 P<br />

(54) • INDANYL- UND<br />

TETRAHYDRONAPHTHYLAMINO-<br />

AZOLINVERBINDUNGEN ZUR BEKÄMP-<br />

FUNG TIERISCHER SCHÄDLINGE<br />

• INDANYL-AND TETRAHYDRONAPHTHYL-<br />

AMINO-AZOLINE COMPOUNDS FOR<br />

COMBATING ANIMAL PESTS<br />

• COMPOSES INDANYLE ET TETRAHYDRO-<br />

NAPHTHYL-AMINO-AZOLINE UTILES<br />

POUR LUTTER CONTRE LES PARASITES<br />

DES ANIMAUX<br />

(73) BASF SE, 67056 Ludwigshafen, DE<br />

(72) KORDES, Markus, 67240, Bobenheim-Roxheim,<br />

DE<br />

KORADIN, Christopher, 67067 Ludwigshafen,<br />

DE<br />

CULBERTSON, Deborah L., Fuquay Varina,<br />

NC 27526, US<br />

(51) C07D 233/58 (11) 1 896 426 B1<br />

(25) En (26) En<br />

(21) 06772447.6 (22) 07.06.2006<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 12.03.2008<br />

(86) US 2006/<strong>02</strong>2154 07.06.2006<br />

(87) WO 2006/135640 2006/51 21.12.2006<br />

(30) 09.06.2005 US 688976 P<br />

(54) • VERFAHREN ZUR SYNTHESE ORGANI-<br />

SCHER VERBINDUNGEN<br />

• PROCESS FOR THE SYNTHESIS OF<br />

ORGANIC COMPOUNDS<br />

• PROCEDE DE SYNTHESE DE COMPOSES<br />

ORGANIQUES<br />

(73) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

Novartis Pharma GmbH, Brunner Strasse 59,<br />

1230 Wien, AT<br />

(84) AT<br />

(72) ABEL, Stephan, 79576 Weil am Rhein, DE<br />

ACEMOGLU, Murat, CH-4052 Basel, CH<br />

ERB, Bernhard, CH-5073 Gipf-Oberfrick, CH<br />

KRELL, Christoph, CH-4057 Basel, CH<br />

SCLAFANI, Joseph, Ledgewood, NJ 07852,<br />

US<br />

MEISENBACH, Mark, F-68480 Durmenach,<br />

FR<br />

PRASHAD, Mahavir, Montville, NJ 07045, US<br />

SHIEH, Wen-Chung, Berkeley Heights, NJ<br />

07922, US<br />

XUE, Song, Parsippany, NJ 07054, US<br />

(74) Roth, Peter Richard, Novartis AG Corporate<br />

Intellectual Property, 40<strong>02</strong> Basel, CH<br />

(60) 10171941.7 / 2 266 961<br />

10171942.5 / 2 292 607<br />

(51) C07D 233/76 (11) 2 057 127 B1<br />

C07D 233/78 C07D 401/06<br />

C07D 401/14 A61K 31/4166<br />

A61K 31/454 A61P 31/04<br />

(25) En (26) En<br />

(21) 07811615.9 (22) 29.08.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

AL BA HR MK RS<br />

(43) 13.05.2009<br />

(86) US 2007/019063 29.08.2007<br />

(87) WO 2008/<strong>02</strong>7466 2008/10 06.03.2008<br />

(30) 31.08.2006 US 841883 P<br />

(54) • HYDANTOIN-DERIVATE ALS ANTIBAK-<br />

TERIELLE WIRKSTOFFE<br />

• HYDANTOIN DERIVATIVES USEFUL AS<br />

ANTIBACTERIAL AGENTS<br />

• DERIVES D'HYDANTOINE UTILES EN<br />

TANT QU'AGENTS ANTIBACTERIENS<br />

(73) Schering Corporation, 2000 Galloping Hill<br />

Road, Kenilworth, NJ 07033, US<br />

(72) MANSOOR, Umar Faruk, Framingham, Massachusetts<br />

017<strong>02</strong>, US<br />

REDDY, Panduranga Adulla P., Walpole,<br />

Massachusetts <strong>02</strong>081, US<br />

SIDDIQUI, M. Arshad, Newton, Massachusetts<br />

<strong>02</strong>464, US<br />

(74) Horgan, James Michael Frederic, Merck &<br />

Co., Inc. <strong>European</strong> <strong>Patent</strong> Department Merck<br />

Sharpe & Dohme Limited Hertford Road,<br />

Hoddesdon Hertfordshire EN11 9BU, GB<br />

C07D 233/78 → (51) C07D 233/76<br />

C07D 239/26 → (51) C07D 239/52<br />

C07D 239/30 → (51) C07D 239/52<br />

(51) C07D 239/32 (11) 1 458 687 B1<br />

C07D 239/38 C07D 239/47<br />

C07D 239/50 C07D 239/52<br />

C07D 239/56 C07D 279/06<br />

A61K 31/506 A61K 31/295<br />

566<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>02</strong>/<strong>2012</strong>) 11.01.<strong>2012</strong><br />

A61P 29/00 C07D 401/06<br />

(25) En (26) En<br />

(21) <strong>02</strong>804468.3 (22) 27.11.20<strong>02</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR IE IT LI LU MC NL PT SE SK TR<br />

(43) 22.09.2004<br />

(86) US 20<strong>02</strong>/038161 27.11.20<strong>02</strong><br />

(87) WO 2003/047516 2003/24 12.06.2003<br />

(30) 30.11.2001 US 742<br />

10.07.20<strong>02</strong> US 192347<br />

(54) • PYRIMIDINVERBINDUNGEN ALS INTER-<br />

LEUKIN-12 (IL-12) INHIBITOREN<br />

• PYRIMIDINE COMPOUNDS AS INTER-<br />

LEUKIN-12 (IL-12) INHIBITORS<br />

• COMPOSES DE PYRIMIDINE EN TANT<br />

QU'INHIBITEURS DE L'INTERLEUKINE-12<br />

(IL-12)<br />

(73) Synta Pharmaceuticals Corporation, 45<br />

Hartwell Avenue, Lexington, MA <strong>02</strong>421, US<br />

(72) ONO, Mitsunori, Lexington, MA <strong>02</strong>421, US<br />

SUN, Lijun, Harvard, MA 01451, US<br />

PRZEWLOKA, Teresa, Tewksbury, MA<br />

01876, US<br />

ZHANG, Shijie, Nashua, NII 03062, US<br />

KOSTIK, Elena, Arlington, MA <strong>02</strong>474, US<br />

YING, Weiwen, Ayer, MA 01432, US<br />

WADA, Yumiko, Billerica, MA 01862, US<br />

KOYA, Keizo, Chestnut Hill, MA <strong>02</strong>467, US<br />

WU, Yaming, Lexington, MA <strong>02</strong>420, US<br />

ZHOU, Dan, Lexington, MA <strong>02</strong>421, US<br />

TATSUTA, Noriaki, Lexington, MA <strong>02</strong>420, US<br />

(74) Schnappauf, Georg, Dr. Volker Vossius<br />

<strong>Patent</strong>- und Rechtsanwaltskanzlei Geibelstrasse<br />

6, 81679 München, DE<br />

C07D 239/38 → (51) C07D 239/32<br />

C07D 239/42 → (51) C07D 239/52<br />

C07D 239/47 → (51) C07D 239/32<br />

C07D 239/50 → (51) C07D 239/32<br />

(51) C07D 239/52 (11) 1 334 968 B1<br />

C07D 239/26 C07D 239/42<br />

C07D 239/30 C07D 403/04<br />

C07C 243/22<br />

(25) Ja (26) En<br />

(21) 01976689.8 (22) 15.10.2001<br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

(43) 13.08.2003<br />

(86) JP 2001/009040 15.10.2001<br />

(87) WO 20<strong>02</strong>/032882 20<strong>02</strong>/17 25.04.20<strong>02</strong><br />

(30) 17.10.2000 JP 2000316345<br />

09.<strong>02</strong>.2001 JP 2001034216<br />

(54) • VERFAHREN ZUR HERSTELLUNG SUB-<br />

STITUIERTER ANILINVERBINDUNGEN<br />

• PROCESS FOR PRODUCING SUBSTI-<br />

TUTED ANILINE COMPOUND<br />

• PROCEDE DE PRODUCTION DE COMPOSE<br />

ANILINE SUBSTITUEE<br />

(73) IHARA CHEMICAL INDUSTRY CO., LTD., 4-<br />

26, Ikenohata 1-chome, Taito-ku, Tokyo 110-<br />

0008, JP<br />

(72) HIYOSHI, Hidetaka, c/o IHARA CHEMICAL<br />

IND. CO. LTD, Ihara-gun, Shizuoka 421-<br />

3306, JP<br />

OGAWA, Mahito, c/o IHARA CHEMICAL IND.<br />

CO. LTD., Ihara-gun, Shizuoka 421-3306, JP<br />

(74) Laufhütte, Dieter, et al, Lorenz-Seidler-Gossel<br />

Widenmayerstrasse 23, 80538 München,<br />

DE<br />

(60) 08017752.0 / 2 <strong>02</strong>5 665<br />

C07D 239/52 → (51) C07D 239/32<br />

C07D 239/56 → (51) C07D 239/32

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