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Bulletin 2012/02 - European Patent Office

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(C07D) I.1(1)<br />

(71) Generics [UK] Limited, Albany Gate Darkes<br />

Lane, Potters Bar Hertfordshire EN6 1AG, GB<br />

(72) GORE, Vinayak Govind, District Raigad<br />

Maharashtra 41<strong>02</strong>08, IN<br />

SHUKLA, Vinay Kumar, District Raigad<br />

Maharashtra 41<strong>02</strong>08, IN<br />

BHANDARI, Sheryas, District Raigad Maharashtra<br />

41<strong>02</strong>08, IN<br />

HASBE, Suresh, District Raigad Maharashtra<br />

41<strong>02</strong>08, IN<br />

(74) Gillard, Richard Edward, Elkington and Fife<br />

LLP Thavies Inn House 3-4 Holborn Circus,<br />

London EC1N 2HA, GB<br />

C07D 401/04 → (51) C07D 231/12<br />

C07D 401/04 → (51) C07D 239/88<br />

(51) C07D 401/10 (11) 2 403 846 A1*<br />

C07D 401/14 C07D 403/14<br />

C07D 413/14 A61K 31/4412<br />

A61K 31/444 A61K 31/497<br />

A61K 31/501 A61P 19/<strong>02</strong><br />

A61P 29/00<br />

(25) En (26) En<br />

(21) 10705373.8 (22) 25.<strong>02</strong>.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2010/052394 25.<strong>02</strong>.2010<br />

(87) WO 2010/100070 2010/36 10.09.2010<br />

(30) <strong>02</strong>.03.2009 US 209<strong>02</strong>1 P<br />

01.<strong>02</strong>.2010 US 300064 P<br />

(54) • HEMMER DER BRUTON-TYROSINKINASE<br />

• INHIBITORS OF BRUTON'S TYROSINE<br />

KINASE<br />

• INHIBITEURS DE LA TYROSINE KINASE<br />

DE BRUTON<br />

(71) F. Hoffmann-La Roche AG, Grenzacherstrasse<br />

124, 4070 Basel, CH<br />

(72) BERTHEL, Steven Joseph, Mendham Township<br />

New Jersey 07945, US<br />

FIROOZNIA, Fariborz, Florham Park New<br />

Jersey 07932, US<br />

FISHLOCK, Daniel, Verona New Jersey<br />

07044, US<br />

HONG, Jun-Bae, Ridgewood New Jersey<br />

07450, US<br />

LOU, Yan, San Jose California 95130, US<br />

LUCAS, Matthew C., Verona New Jersey<br />

07044, US<br />

OWENS, Thimothy D., Mountain View California<br />

94040, US<br />

SARMA, Keshab, Kinnelon New Jersey<br />

07405, US<br />

SWEENEY, Zachary Kevin, Redwood City<br />

California 94062, US<br />

TAYGERLY, Joshua Paul Gergely, San Francisco<br />

California 94131, US<br />

(74) Sauer, Frank, F. Hoffmann-La Roche AG<br />

<strong>Patent</strong> Department, CH-4070 Basel, CH<br />

C07D 401/12 → (51) C07D 213/75<br />

C07D 401/12 → (51) C07D 215/48<br />

C07D 401/12 → (51) C07D 231/12<br />

C07D 401/12 → (51) C07D 233/54<br />

(51) C07D 401/14 (11) 2 403 847 A1*<br />

A61K 31/47 A61P 9/00<br />

(25) En (26) En<br />

(21) 10706035.2 (22) <strong>02</strong>.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA ME RS<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(86) GB 2010/000361 <strong>02</strong>.03.2010<br />

(87) WO 2010/100405 2010/36 10.09.2010<br />

(30) 06.03.2009 GB 0903949<br />

07.09.2009 GB 0915586<br />

(54) • TRIAZINDERIVATE ALS KINASEINHIBITO-<br />

REN<br />

• TRIAZINE DERIVATIVES AS KINASE INHI-<br />

BITORS<br />

• DÉRIVÉS DE TRIAZINE EN TANT QU'IN-<br />

HIBITEURS DE KINASES<br />

(71) UCB Pharma, S.A., 60, allée de la Recherche,<br />

1070 Brussels, BE<br />

(72) ALLEN, Daniel, Rees, Essex CB10 1XL, GB<br />

BÜRLI, Roland, Essex CB10 1XL, GB<br />

HAUGHAN, Alan, Findlay, Essex CB10 1XL,<br />

GB<br />

MACDONALD, Jonathan, David, Leeds LS2<br />

9JT, GB<br />

MATTEUCCI, Mizio, Essex CB10 1XL, GB<br />

NASH, David, John, Essex CB10 1XL, GB<br />

OWENS, Andrew, Pate, Essex CB10 1XL, GB<br />

RAPHY, Gilles, Essex CB10 1XL, GB<br />

SAVILLE-STONES, Elizabeth, Anne, Essex<br />

CB10 1XL, GB<br />

SHARPE, Andrew, Essex CB10 1XL, GB<br />

(74) Thompson, John, UCB Celltech, 208 Bath<br />

Road, Slough, Berkshire SL1 3WE, GB<br />

C07D 401/14 → (51) C07D 213/75<br />

C07D 401/14 → (51) C07D 215/48<br />

C07D 401/14 → (51) C07D 231/12<br />

C07D 401/14 → (51) C07D 401/10<br />

C07D 403/04 → (51) C07D 239/88<br />

C07D 403/04 → (51) C07D 265/06<br />

C07D 403/12 → (51) C07D 213/75<br />

C07D 403/12 → (51) C07D 231/12<br />

C07D 403/12 → (51) C07D 233/54<br />

C07D 403/14 → (51) C07D 401/10<br />

C07D 405/04 → (51) C07D 401/04<br />

(51) C07D 405/10 (11) 2 403 848 A1*<br />

C07D 405/12 C07D 405/14<br />

C07D 413/14 A61K 31/397<br />

A61K 31/4<strong>02</strong>5 A61K 31/4523<br />

A61K 31/41 A61K 31/422<br />

A61P 9/10<br />

(25) En (26) En<br />

(21) 10706272.1 (22) 05.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) EP 2010/052821 05.03.2010<br />

(87) WO 2010/10<strong>02</strong>55 2010/36 10.09.2010<br />

(30) 06.03.2009 EP 09154496<br />

07.10.2009 EP 09172395<br />

(54) • PHARMAZEUTISCHE HYPOCHOLESTER-<br />

INEMISCHE ZUSAMMENSETZUNGEN<br />

• PHARMACEUTICAL HYPOCHOLESTERO-<br />

LEMIC COMPOSITIONS<br />

• COMPOSITIONS PHARMACEUTIQUES<br />

HYPOCHOLESTÉROLÉMIQUES<br />

(71) Lipideon Biotechnology AG, ETH Hönggerberg<br />

HCI-D151 Wolfgang Pauli-Strasse 10,<br />

8093 Zürich, CH<br />

(72) FESSARD, Thomas, 1003 Lausanne, CH<br />

LI, Dong-Bo, CH-8052 Zürich, CH<br />

BARBARAS, Damien, CH-1007 Lausanne, CH<br />

WOLFRUM, Susanne, 8104 Weiningen, CH<br />

85<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>02</strong>/<strong>2012</strong>) 11.01.<strong>2012</strong><br />

CARREIRA, Erick, CH-8126 Zumikon, CH<br />

(74) Carreira-Staubli, Andrea, Isler & Pedrazzini<br />

AG Gotthardstrasse 53 Postfach 1772, 8<strong>02</strong>7<br />

Zürich, CH<br />

C07D 405/12 → (51) C07D 405/10<br />

C07D 405/14 → (51) C07D 405/10<br />

C07D 407/04 → (51) C07D 321/00<br />

C07D 407/12 → (51) C07D 231/12<br />

C07D 409/04 → (51) C07D 231/12<br />

(51) C07D 413/04 (11) 2 403 849 A1*<br />

C07D 413/14 A61K 31/4245<br />

A61P 37/00 A61P 29/00<br />

(25) En (26) En<br />

(21) 10705889.3 (22) <strong>02</strong>.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

AL BA ME RS<br />

(86) EP 2010/052613 <strong>02</strong>.03.2010<br />

(87) WO 2010/100142 2010/36 10.09.2010<br />

(30) 03.03.2009 EP 09154174<br />

03.03.2009 US 156985 P<br />

(54) • ALS S1P1-REZEPTOR-AGONISTEN<br />

GEEIGNETE OXAZOLPYRIDINDERIVATE<br />

• OXAZOLE PYRIDINE DERIVATIVES USE-<br />

FUL AS S1P1 RECEPTOR AGONISTS<br />

• DÉRIVÉS D'OXAZOLE PYRIDINE UTILES<br />

EN TANT QU'AGONISTES DU RÉCEPTEUR<br />

S1P1<br />

(71) Merck Serono S.A., Centre Industriel, 1267<br />

Coinsins, CH<br />

(72) QUATTROPANI, Anna, CH-1207 Geneva, CH<br />

GERBER, Patrick, CH-1163 Etoy, CH<br />

DORBAIS, Jerome, F-74000 Annecy, FR<br />

(74) Merck Serono SA - Geneva Intellectual<br />

Property, 9, chemin des Mines, 12<strong>02</strong><br />

Geneva, CH<br />

(51) C07D 413/12 (11) 2 403 850 A1*<br />

A61K 31/423 A61P 25/00<br />

(25) En (26) En<br />

(21) 10710897.9 (22) 01.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) HU 2010/000<strong>02</strong>3 01.03.2010<br />

(87) WO 2010/100512 2010/36 10.09.2010<br />

(30) 03.03.2009 HU 0900130<br />

(54) • NEUES KRISTALLINES HYDRAT, AMOR-<br />

PHE UND POLYMORPHE FORMEN EINES<br />

DIHYDRO-BENZOXAZOL-6-YL-ACETAMID-<br />

DERIVATS UND VERFAHREN ZU IHRER<br />

HERSTELLUNG<br />

• NOVEL CRYSTALLINE HYDRATE, AMOR-<br />

PHOUS AND POLYMORPHIC FORMS OF<br />

DIHYDRO-BENZOXAZOLE-6-YL-ACETA-<br />

MIDE DERIVATIVE AND PROCESSES FOR<br />

THEIR PREPARATION<br />

• NOUVELLES FORMES CRISTALLINES,<br />

AMORPHES ET POLYMORPHES HYDRA-<br />

TÉES D'UN DÉRIVÉ DE DIHYDROBENZO-<br />

XAZOL-6-YLACÉTAMIDE ET LEURS<br />

PROCÉDÉS DE PRÉPARATION<br />

(71) Richter Gedeon Nyrt., Gyömröi út 19-21.,<br />

1103 Budapest, HU<br />

(72) DEMETER, Adam, Egyenes u. 8. A/61., HU<br />

NEMET, Zoltan, Balkan u. 6.V/16., HU<br />

NEMES, Andras, H-1<strong>02</strong>5 Budapest, HU<br />

SEBOK, Ferenc, Fay A. u. 67., HU<br />

BARTANE, SZALAI, Gizella, Avarszallas u.<br />

38., HU<br />

CZIBULA, Laszló, Gergely u. 48., HU

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