31.12.2012 Views

Bulletin 2012/02 - European Patent Office

Bulletin 2012/02 - European Patent Office

Bulletin 2012/02 - European Patent Office

SHOW MORE
SHOW LESS

You also want an ePaper? Increase the reach of your titles

YUMPU automatically turns print PDFs into web optimized ePapers that Google loves.

(C07D) II.1(1)<br />

(74) Motion, Keith Robert, et al, Pfizer <strong>European</strong><br />

<strong>Patent</strong> Department 23-25, avenue du Docteur<br />

Lannelongue, 75668 Paris Cedex 14, FR<br />

(51) C07D 487/04 (11) 1 991 549 B1<br />

C07D 513/04 C07D 498/04<br />

A61K 31/4188 A61K 31/433<br />

A61K 31/4985 A61K 31/424<br />

A61P 5/24<br />

(25) En (26) En<br />

(21) 07756561.2 (22) 01.<strong>02</strong>.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 19.11.2008<br />

(86) US 2007/061438 01.<strong>02</strong>.2007<br />

(87) WO 2007/095423 2007/34 23.08.2007<br />

(30) 10.<strong>02</strong>.2006 US 772168 P<br />

(54) • BIZYKLISCHE IMIDAZOL- ODER THIADIA-<br />

ZOL-HETEROZYKLEN ALS SELEKTIVE<br />

ANDROGEN-REZEPTOR-MODULATOREN<br />

• BICYCLIC IMIDAZOLE OR THIADIAZOLE<br />

HETEROCYCLES USEFUL AS SELECTIVE<br />

ANDROGEN RECEPTOR MODULATORS<br />

• IMIDAZOLE OU THIADIAZOLE BICY-<br />

CLIQUE SERVANT DE MODULATEUR<br />

SELECTIF DE RECEPTEUR D'ANDROGENE<br />

(73) Janssen Pharmaceutica N.V., Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) SUI, Zhihua, Exton, Pennsylvania 19341, US<br />

ZHANG, Xuqing, 665 Stockton Drive Exton,<br />

PA 19341, US<br />

(74) Warner, James Alexander, et al, Carpmaels &<br />

Ransford One Southampton Row, London<br />

WC1B 5HA, GB<br />

(51) C07D 487/04 (11) 2 152 712 B1<br />

(25) En (26) En<br />

(21) 08737600.0 (22) 05.05.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(43) 17.<strong>02</strong>.2010<br />

(86) IB 2008/001125 05.05.2008<br />

(87) WO 2008/139293 2008/47 20.11.2008<br />

(30) 11.05.2007 US 917333 P<br />

(54) • AMINOHETEROCYCLISCHE VERBINDUN-<br />

GEN<br />

• AMINO-HETEROCYCLIC COMPOUNDS<br />

• COMPOSÉS AMINO-HÉTÉROCYCLIQUES<br />

(73) Pfizer Inc., 235 East 42nd Street, New York,<br />

NY 10017, US<br />

(72) VERHOEST, Patrick, Robert, Groton, CT<br />

06340, US<br />

PROULX-LAFRANCE, Caroline, Groton, CT<br />

06340, US<br />

(74) Summers, Victoria Clare, Pfizer <strong>European</strong><br />

<strong>Patent</strong> Department 23-25, avenue du Docteur<br />

Lannelongue, 75668 Paris Cedex 14, FR<br />

C07D 487/04 → (51) C07D 471/04<br />

(51) C07D 491/06 (11) 2 009 015 B1<br />

(25) En (26) En<br />

(21) 08010868.1 (22) 16.06.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 31.12.2008<br />

(30) 18.06.2007 IN CH12572007<br />

(54) • Herstellungsprozess für Galantaminhydrobromid<br />

• Process for the preparation of galantamine<br />

hydrobromide<br />

• Procédé pour la préparation de bromhydrate<br />

de galantamine<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(73) Aurobindo Pharma Limited, Plot No. 2, Maitri<br />

Vihar Ameerpet, Hyderabad 500 038, IN<br />

(72) Koilpillai, Joseph Prabahar, Hyderabad 500<br />

038, Andhra Pradesh, IN<br />

Ganala, Naga Trinadhachari, Hyderabad 500<br />

038, Andhra Pradesh, IN<br />

Podila, Naveen Kumar, Hyderabad 500 038,<br />

Andhra Pradesh, IN<br />

Upputuri, Venkata lakshmi, Hyderabad 500<br />

038, Andhra Pradesh, IN<br />

Dandala, Ramesh, Hyderabad 500 038,<br />

Andhra Pradesh, IN<br />

Meenakshisunderam, Sivakumaran, Hyderabad<br />

500 038, Andhra Pradesh, IN<br />

(74) Wittkopp, Alexander, Maiwald <strong>Patent</strong>anwalts<br />

GmbH Jungfernstieg 38, 20354 Hamburg,<br />

DE<br />

(51) C07D 491/12 (11) 1 945 647 B1<br />

C07D 498/06<br />

(25) En (26) En<br />

(21) 06844315.9 (22) 08.11.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 23.07.2008<br />

(86) US 2006/043718 08.11.2006<br />

(87) WO 2007/056550 2007/20 18.05.2007<br />

(30) 08.11.2005 US 734330 P<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

MAYTANSINOL<br />

• PROCESSES FOR PREPARATION OF<br />

MAYTANSINOL<br />

• PROCEDES DE PREPARATION DE MAY-<br />

TANSINOL<br />

(73) Immunogen, Inc., 830 Winter Street, Waltham,<br />

MA <strong>02</strong>451, US<br />

(72) CHARI, Ravi, V.J., Newton, Massachusetts<br />

<strong>02</strong>461, US<br />

WIDDISON, Wayne, C., Belmont, MA <strong>02</strong>478,<br />

US<br />

(74) McNab, Donald C., Marks & Clerk LLP<br />

Aurora 120 Bothwell Street, Glasgow G2<br />

7JS, GB<br />

C07D 493/10 → (51) C07D 407/04<br />

C07D 498/04 → (51) C07D 217/24<br />

C07D 498/04 → (51) C07D 487/04<br />

C07D 498/06 → (51) C07D 491/12<br />

(51) C07D 498/08 (11) 2 189 462 B1<br />

A61K 31/553<br />

(25) En (26) En<br />

(21) 08169901.9 (22) 25.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 26.05.2010<br />

(54) • Bicyclische Peptidomimetikum-Inhibitoren<br />

von Aspartylproteasen zur Behandlung von<br />

Infektionskrankheiten<br />

• Bicyclic peptidomimetic inhibitors of<br />

aspartyl-proteases for the treatment of<br />

infectious diseases<br />

• Inhibiteurs peptidomimétiques bicycliques<br />

de protéases d'aspartyl pour le traitement<br />

des maladies infectieuses<br />

(73) Universita' Degli Studi di Firenze, Piazza San<br />

Marco, 4, 50121 Firenze, IT<br />

Instituto Superiore Di Sanita', Viale Regina<br />

Elena 299, 00161 Roma, IT<br />

(72) Cassone, Antonio, 00147 Roma, IT<br />

De Bernardis, Flavia, 00194 Roma, IT<br />

Garaci, Enrico, 00198 Roma, IT<br />

Trabocchi, Andrea, 50142 Firenze, IT<br />

Guarna, Antonio, 50019 Sesto Fiorentino, IT<br />

570<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>02</strong>/<strong>2012</strong>) 11.01.<strong>2012</strong><br />

(74) Gervasi, Gemma, et al, Notarbartolo &<br />

Gervasi S.p.A. Corso di Porta Vittoria 9,<br />

<strong>2012</strong>2 Milano, IT<br />

C07D 513/04 → (51) C07D 217/24<br />

C07D 513/04 → (51) C07D 487/04<br />

(51) C07F 1/00 (11) 1 084 128 B1<br />

C07C 51/41<br />

(25) En (26) En<br />

(21) 99927208.1 (22) 04.06.1999<br />

(84) AT BE CH DE DK ES FI FR GB IT LI LU NL PT<br />

SE<br />

(43) 21.03.2001<br />

(86) US 1999/012448 04.06.1999<br />

(87) WO 1999/062913 1999/49 09.12.1999<br />

(30) 05.06.1998 US 88266 P<br />

28.05.1999 US 322684<br />

(54) • PULVERIGE, FESTE SELTERDEN-CARBO-<br />

XYLATE MIT VERBESSERTER LÖSLICH-<br />

KEIT<br />

• POWDERY, SOLID RARE EARTH CAR-<br />

BOXYLATES WITH IMPROVED SOLUBI-<br />

LITY<br />

• CARBOXYLATES DES TERRES RARES<br />

SOLIDES, PULVERANTS, A SOLUBILITE<br />

AMELIOREE<br />

(73) Rhodia Rare Earths, Inc., 3 Enterprise Drive,<br />

Shelton, Connecticut 06484, US<br />

(72) KEYER, Julie, Lynn, Shreeve, East Windsor,<br />

NJ 08520, US<br />

YUNLU, Kenan, Princeton, NJ 08540, US<br />

FORGERON, Anne, Nadine, Bedford, Nova<br />

Scotia, CA<br />

CUIF, Jean-Pierre, F-17000 La Rochelle, FR<br />

MORIN, Anne-Gaelle, Simi Valley, CA 93063,<br />

US<br />

(74) Petraz, Gilberto Luigi, et al, GLP S.r.l.<br />

Piazzale Cavedalis 6/2, 33100 Udine, IT<br />

(51) C07F 7/12 (11) 1 915 384 B1<br />

C07F 7/18 C07F 7/20<br />

C07D 279/20<br />

(25) En (26) En<br />

(21) 06782753.5 (22) 09.08.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 30.04.2008<br />

(86) JP 2006/316075 09.08.2006<br />

(87) WO 2007/<strong>02</strong>0932 2007/08 22.<strong>02</strong>.2007<br />

(30) 19.08.2005 JP 2005238465<br />

(54) • VERFAHREN ZUR HERSTELLUNG EINER<br />

ORGANISCHEN SILICIUMVERBINDUNG,<br />

DIE EINE METHACRYLOXYGRUPPE ODER<br />

EINE ACRYLOXYGRUPPE ENTHÄLT<br />

• A METHOD OF MANUFACTURING AN<br />

ORGANIC SILICON COMPOUND THAT<br />

CONTAINS A METHACRYLOXY GROUP OR<br />

AN ACRYLOXY GROUP<br />

• PROCEDE DE PREPARATION D'UN COM-<br />

POSE ORGANOSILICIE CONTENANT UN<br />

GROUPE METHACRYLOXY OU UN<br />

GROUPE ACRYLOXY<br />

(73) Dow Corning Toray Co., Ltd., 4th Floor, AIG<br />

Building, 1-1-3, Marunouchi Chiyoda-ku,<br />

Tokyo 100-0005, JP<br />

(72) WAKITA, Keiji, Ichihara-shi, Chiba 299-0108,<br />

JP<br />

(74) Gillard, Richard Edward, Elkington and Fife<br />

LLP Thavies Inn House 3-4 Holborn Circus,<br />

London EC1N 2HA, GB<br />

(51) C07F 7/18 (11) 1 791 849 B1<br />

(25) En (26) En<br />

(21) 05793252.7 (22) 09.09.2005

Hooray! Your file is uploaded and ready to be published.

Saved successfully!

Ooh no, something went wrong!