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Bulletin 2012/02 - European Patent Office

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(C07C) I.1(2)<br />

A61K 31/20 A61K 31/23<br />

A61K 31/33<br />

(25) En (26) En<br />

(21) 11005303.0 (22) 23.12.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(30) 23.01.2003 US 441795 P<br />

(54) • Hydroxylverbindungen und -zusammensetzungen<br />

zur Steuerung des Cholesterinspiegels<br />

und verwandte Verwendungen<br />

• Hydroxyl compounds and compositions for<br />

cholesterol management and related uses<br />

• Composés d'hydroxyle et compositions<br />

pour gestion du cholestérol et utilisations<br />

associées<br />

(71) Esperion Therapeutics Inc., 695 KMS Place,<br />

3261 South State Street, Ann Arbor, Michigan<br />

48101, US<br />

(72) Dasseux, Jean-Louis, Henri, Brighton, MI<br />

48116, US<br />

Oniciu, Daniela, Carmen, Ann Arbor, MI<br />

48103, US<br />

(74) Schnappauf, Georg, et al, Dr. Volker Vossius<br />

<strong>Patent</strong>- und Rechtsanwaltskanzlei Geibelstrasse<br />

6, 81679 München, DE<br />

(62) 0380<strong>02</strong>58.0 / 1 597 223<br />

C07C 33/46 → (51) C07C 237/42<br />

C07C 43/225 → (51) C07C 235/20<br />

C07C 45/49 → (51) B01J 31/24<br />

(51) C07C 45/61 (11) 2 404 891 A1<br />

C07C 49/794 C07C 49/78<br />

(25) Zh (26) En<br />

(21) 10748283.8 (22) 22.<strong>02</strong>.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) CN 2010/00<strong>02</strong>27 22.<strong>02</strong>.2010<br />

(87) WO 2010/099693 2010/36 10.09.2010<br />

(30) 04.03.2009 CN 200910118751<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

ACYLBENZENEN<br />

• PREPARATION METHOD OF ACYLBEN-<br />

ZENES<br />

• PROCÉDÉ DE PRÉPARATION D'ACYLBEN-<br />

ZÈNES<br />

(71) DSM IP Assets B.V., Het Overloon 1, 6411<br />

TE Heerlen, NL<br />

(72) JEPHCOTE, Vincent, John, Shanghai<br />

200000, CN<br />

SHEN, Hongyan, Shanghai 200000, CN<br />

(74) Kurt, Manfred, DSM Nutritional Products AG<br />

<strong>Patent</strong> Department (241/625) Wurmisweg<br />

576, CH-4303 Kaiseraugst, CH<br />

C07C 45/74 → (51) A61K 31/122<br />

C07C 49/78 → (51) C07C 45/61<br />

C07C 49/794 → (51) C07C 45/61<br />

C07C 59/105 → (51) C07C 31/22<br />

C07C 59/245 → (51) C07C 31/22<br />

C07C 217/18 → (51) C07C 235/20<br />

(51) C07C 231/<strong>02</strong> (11) 2 404 892 A1<br />

(25) En (26) En<br />

(21) 11172262.5 (22) 30.06.2011<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

BA ME<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(30) 05.07.2010 JP 2010153161<br />

(54) • Synthese von Seltenerdmetallextraktionsmittel<br />

• Synthesis of Rare Earth Metal Extractant<br />

• Synthèse d'extraction de métaux de terres<br />

rares<br />

(71) Shin-Etsu Chemical Co., Ltd., 6-1, Otemachi<br />

2-chome, Chiyoda-ku, Tokyo, JP<br />

Nissin Chemical Industry Co., Ltd., 17-33,<br />

Kitago 2-chome, Echizen-shi, Fukui-ken<br />

Fukui, JP<br />

(72) Sakaki, Kazuaki, Fukui-ken,, Fukui, JP<br />

Sugahara, Hiroto, Fukui-ken,, Fukui, JP<br />

Ohashi, Tetsuya, Fukui-ken,, Fukui, JP<br />

Kume, Tetsuya, Fukui-ken,, Fukui, JP<br />

Ikka, Masahiko, Fukui-ken,, Fukui, JP<br />

Naganawa, Hirochika, Ibaraki,, Ibaraki 319-<br />

1195, JP<br />

Shimojo, Kojiro, Ibaraki,, Ibaraki 319-1195,<br />

JP<br />

(74) Bailey, Sam Rogerson, Mewburn Ellis LLP<br />

33 Gutter Lane, London EC2V 8AS, GB<br />

(51) C07C 231/<strong>02</strong> (11) 2 404 893 A1<br />

(25) En (26) En<br />

(21) 11172278.1 (22) 30.06.2011<br />

(84) AL AT BE BG CH CY CZ DE DK EE ES FI FR<br />

GB GR HR HU IE IS IT LI LT LU LV MC MK<br />

MT NL NO PL PT RO RS SE SI SK SM TR<br />

BA ME<br />

(30) 05.07.2010 JP 2010153175<br />

(54) • Synthese von Seltenerdmetallextraktionsmittel<br />

• Synthesis of rare earth metal extractant<br />

• Synthèse d'extraction de métaux de terres<br />

rares<br />

(71) Shin-Etsu Chemical Co., Ltd., 6-1, Otemachi<br />

2-chome, Chiyoda-ku, Tokyo, JP<br />

Nissin Chemical Industry Co., Ltd., 17-33,<br />

Kitago 2-chome, Echizen-shi, Fukui-ken, JP<br />

(72) Sakaki, Kazuaki, Fukui-ken,, Fukui, JP<br />

Sugahara, Hiroto, Fukui-ken,, Fukui, JP<br />

Ohashi, Tetsuya, Fukui-ken,, Fukui, JP<br />

Kume, Tetsuya, Fukui-ken,, Fukui, JP<br />

Ikka, Masahiko, Fukui-ken,, Fukui, JP<br />

Naganawa, Hirochika, Ibaraki,, Ibaraki 319-<br />

1195, JP<br />

Shimojo, Kojiro, Ibaraki,, Ibaraki 319-1195,<br />

JP<br />

(74) Bailey, Sam Rogerson, Mewburn Ellis LLP<br />

33 Gutter Lane, London EC2V 8AS, GB<br />

C07C 231/08 → (51) C07C 237/42<br />

(51) C07C 233/05 (11) 2 404 894 A1<br />

C07C 233/09 C07C 233/49<br />

C07C 235/06 C07C 235/74<br />

C07C 237/06 C07C 237/20<br />

C07C 237/42 C07C 323/59<br />

C07C 323/60 C07C 403/20<br />

(25) En (26) En<br />

(21) 11167097.2 (22) 26.12.20<strong>02</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR IE IT LI LU MC NL PT SE SI SK TR<br />

(30) 11.01.20<strong>02</strong> JP 20<strong>02</strong>004123<br />

11.01.20<strong>02</strong> JP 20<strong>02</strong>004131<br />

11.01.20<strong>02</strong> JP 20<strong>02</strong>004136<br />

27.09.20<strong>02</strong> JP 20<strong>02</strong>283644<br />

(54) • Mevalonsäurederivate<br />

• Mevalonic Acid Derivatives<br />

• Dérivés d'acide mévalonique<br />

(71) Ohgen Research Laboratories Ltd., Wo 80,<br />

Yatano-machi, Komatsu-shi, Ishikawa 923-<br />

0342, JP<br />

(72) Akiyama, Kiyoshi, Komatsu-shi Ishikawa<br />

923-0342, JP<br />

219<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>02</strong>/<strong>2012</strong>) 11.01.<strong>2012</strong><br />

(74) Beckmann, Claus, Kraus & Weisert <strong>Patent</strong>und<br />

Rechtsanwälte Thomas-Wimmer-Ring<br />

15, 80539 München, DE<br />

(62) <strong>02</strong>795432.0 / 1 471 052<br />

C07C 233/09 → (51) C07C 233/05<br />

C07C 233/49 → (51) C07C 233/05<br />

C07C 235/06 → (51) C07C 233/05<br />

(51) C07C 235/20 (11) 2 404 895 A1<br />

C07C 235/34 C07C 279/08<br />

C07C 217/18 C07C 43/225<br />

C07D 249/08 A61K 31/015<br />

A61K 31/135 A61K 31/216<br />

A61K 31/09 A61K 31/155<br />

A61K 31/4192 A61P 31/04<br />

A61P 35/00 A61P 43/00<br />

A61P 9/10 A61P 27/<strong>02</strong><br />

(25) En (26) En<br />

(21) 11173181.6 (22) 04.10.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(30) 04.10.2004 US 616133 P<br />

(54) • Calixaren-basierte Peptidkonformationsmimetika,<br />

Verfahren zu ihrer Verwendung und<br />

Verfahren zu ihrer Herstellung<br />

• Calixarene-based peptide conformation<br />

mimetics, methods of use, and methods of<br />

making<br />

• Mimétiques à conformation peptidique à<br />

base de calixarene, procédés d'utilisation et<br />

procédés de fabrication<br />

(71) Regents of the University of Minnesota, 1000<br />

Westgate Drive, Suite 160, St. Paul, Minnesota<br />

55114-8658, US<br />

(72) Mayo, Kevin, H., Minneapolis, MN 55413, US<br />

Hoye, Thomas, R., St. Paul, MN 55104, US<br />

Chen, Xuemei, Voorheesville, New York<br />

12186, US<br />

(74) Vossius & Partner, Siebertstrasse 4, 81675<br />

München, DE<br />

(62) 05817221.4 / 1 8<strong>02</strong> 291<br />

C07C 235/34 → (51) C07C 235/20<br />

C07C 235/74 → (51) C07C 233/05<br />

C07C 237/06 → (51) C07C 233/05<br />

C07C 237/20 → (51) C07C 233/05<br />

(51) C07C 237/24 (11) 2 404 896 A1<br />

A61K 31/167 A61K 31/275<br />

A61K 31/415 A61K 31/4184<br />

A61K 31/4192 A61K 31/42<br />

A61K 31/421 A61K 31/422<br />

A61K 31/423 A61K 31/427<br />

A61K 31/4375 A61K 31/44<br />

A61K 31/4439 A61K 31/4709<br />

A61K 31/4965 A61K 31/497<br />

A61K 31/5375 A61K 31/5377<br />

A61P 3/04 A61P 43/00<br />

(25) Ja (26) En<br />

(21) 10748840.5 (22) 05.03.2010<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MK MT<br />

NL NO PL PT RO SE SI SK SM TR<br />

(86) JP 2010/053663 05.03.2010<br />

(87) WO 2010/101247 2010/36 10.09.2010<br />

(30) 05.03.2009 JP 2009052065<br />

(54) • CYCLOHEXANDERIVAT MIT NPY-Y5-<br />

REZEPTORANTAGONISMUS<br />

• CYCLOHEXANE DERIVATIVE HAVING NPY<br />

Y5 RECEPTOR ANTAGONISM

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