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Bulletin 2012/02 - European Patent Office

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(A61K) II.1(1)<br />

(25) En (26) En<br />

(21) 07834529.5 (22) 20.11.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 05.08.2009<br />

(86) MY 2007/000082 20.11.2007<br />

(87) WO 2008/063045 2008/22 29.05.2008<br />

(30) 21.11.2006 MY 0604536<br />

(54) • VERWENDUNG EINER ANTIKREBSVER-<br />

BINDUNG<br />

• USE OF AN ANTI-CANCER COMPOUND<br />

• UTILISATION D'UN COMPOSÉ ANTI-CAN-<br />

CER<br />

(73) Universiti Putra Malaysia, 43400 Upm Serdang,<br />

Selangor, MY<br />

(72) ABDUL, Ahmad Bustamam, 43400 UPM<br />

Serdang Selangor, MY<br />

ABDULLAH, Munammad Nazrul Hakim,<br />

43400 UPM Serdang, Selangor, MY<br />

LAJIS, Mohd Nordin, 43400 UPM Serdang<br />

Selangor, MY<br />

TAILAN, Nirmala Devi, 43400 UPM Serdang,<br />

Selangor, MY<br />

MOHD ZAIN, Zetty Nadia, 43400 UPM<br />

Serdang Selangor, MY<br />

WAHAB, Siddig Ibrahim Abdel, 43400 Serdang,<br />

MY<br />

AL-ZUBAIRI, Adel, Sharaf, 43400 Serdang,<br />

MY<br />

(74) Bates, Philip Ian, Reddie & Grose 16<br />

Theobalds Road, London WC1X 8PL, GB<br />

A61K 31/135 → (51) C07C 215/64<br />

A61K 31/135 → (51) C07C 225/22<br />

(51) A61K 31/165 (11) 1 868 595 B1<br />

A61P 3/06 A61P 3/10<br />

(25) En (26) En<br />

(21) 06784338.3 (22) 31.03.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 26.12.2007<br />

(86) US 2006/012050 31.03.2006<br />

(87) WO 2006/127133 2006/48 30.11.2006<br />

(30) 01.04.2005 US 667457 P<br />

(54) • VERBINDUNGEN ZUR BEHANDLUNG VON<br />

STOFFWECHSELSTÖRUNGEN<br />

• COMPOUNDS FOR THE TREATMENT OF<br />

METABOLIC DISORDERS<br />

• COMPOSES POUR LE TRAITEMENT DE<br />

TROUBLES METABOLIQUES<br />

(73) Wellstat Therapeutics Corporation, 930<br />

Clopper Road, Gaithersburg, MD 20878, US<br />

(72) SHARMA, Shalini, Gaithersburg, Maryland<br />

20877, US<br />

VON BORSTEL, Reid, W., Potomac, Maryland<br />

20854, US<br />

(74) MacLean, Martin Robert, Mathys & Squire<br />

LLP 120 Holborn, London EC1N 2SQ, GB<br />

(51) A61K 31/167 (11) 2 157 971 B1<br />

A61K 31/4706 A61K 31/517<br />

A61P 35/00 A61P 35/04<br />

A61P 11/06 G01N 33/574<br />

(25) En (26) En<br />

(21) 08749545.3 (22) 11.04.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 03.03.2010<br />

(86) EP 2008/054432 11.04.2008<br />

(87) WO 2008/125633 2008/43 23.10.2008<br />

(30) 13.04.2007 DK 200700547<br />

(54) • EGFR-INHIBITOREN ZUR BEHANDLUNG<br />

UND DIAGNOSE VON METASTASIEREN-<br />

DEM PROSTATAKREBS<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

• EGFR INHIBITORS FOR TREATMENT AND<br />

DIAGNOSIS OF METASTATIC PROSTATE<br />

CANCER<br />

• TRAITEMENT ET DIAGNOSTIC DU CAN-<br />

CER MÉTASTATIQUE DE LA PROSTATE<br />

PAR DES INHIBITEURS DE RÉCEPTEUR<br />

DE FACTEUR DE CROISSANCE ÉPIDER-<br />

MIQUE (EGFR)<br />

(73) Rikshospitalet- Radiumhospitalet HF,<br />

Songsvannsveien 20, 0<strong>02</strong>7 Oslo, NO<br />

PamGene B.V., Nieuwstraat 30, 5211 's<br />

Hertogenbosch, NL<br />

(72) REE, Anne Hansen, N-1344 Haslum, NO<br />

BRATLAND, Ase, N-0310 Oslo, NO<br />

BOENDER, Pieter Jacob, NL-6522 KJ Nijmegen,<br />

NL<br />

RUIJTENBEEK, Robby, NL-3524 BK Utrecht,<br />

NL<br />

(74) De Clercq, Ann G. Y., et al, De Clercq &<br />

Partners cvba Edgard Gevaertdreef 10 a,<br />

9830 Sint-Martens-Latem, BE<br />

A61K 31/18 → (51) C07C 311/29<br />

A61K 31/185 → (51) C07D 209/82<br />

A61K 31/192 → (51) A61K 31/715<br />

A61K 31/195 → (51) A61K 31/44<br />

A61K 31/197 → (51) A23B 7/<strong>02</strong><br />

A61K 31/205 → (51) A61K 38/28<br />

A61K 31/225 → (51) A61K 31/44<br />

A61K 31/27 → (51) A61K 31/44<br />

A61K 31/295 → (51) C07D 239/32<br />

A61K 31/335 → (51) A61K 31/44<br />

A61K 31/335 → (51) C07D 209/82<br />

A61K 31/35 → (51) C07D 407/04<br />

A61K 31/40 → (51) C07D 209/22<br />

A61K 31/403 → (51) C07D 209/82<br />

A61K 31/4166 → (51) C07D 233/76<br />

A61K 31/4178 → (51) C07D 401/06<br />

A61K 31/4178 → (51) C07D 409/10<br />

A61K 31/4188 → (51) C07D 487/04<br />

(51) A61K 31/4196 (11) 1 789 039 B1<br />

C07D 249/08 A61P 31/18<br />

(25) En (26) En<br />

(21) 05790722.2 (22) 25.08.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK YU<br />

(43) 30.05.2007<br />

(86) US 2005/03<strong>02</strong>59 25.08.2005<br />

(87) WO 2006/<strong>02</strong>6356 2006/10 09.03.2006<br />

(30) 25.08.2004 US 604219 P<br />

25.08.2004 US 604220 P<br />

31.05.2005 US 686351 P<br />

(54) • S-TRIAZOLYL ALPHA MERCAPTOACETA-<br />

NILIDE ALS HEMMER DER REVERSEN<br />

TRANSKRIPTASE VON HIV<br />

• S-TRIAZOLYL ALPHA -MERCAPTOACETA-<br />

NILDES AS INHIBITORS OF HIV REVERSE<br />

TRANSCRIPTASE<br />

520<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>02</strong>/<strong>2012</strong>) 11.01.<strong>2012</strong><br />

• S-TRIAZOLYL ALPHA-MERCAPTOACETA-<br />

NILDES TENANT LIEU D'INHIBITEURS DE<br />

LA TRANSCRIPTASE INVERSE VIH<br />

(73) Ardea Biosciences, Inc., 3300 Hyland Avenue,<br />

Costa Mesa, CA 92626, US<br />

(72) GIRARDET, Jean-Luc, Aliso Viejo, CA 92656,<br />

US<br />

KOH, Yung-Hyo, Irvin, CA 92620, US<br />

DE LA ROSA, Martha, Santa Ana, CA 93707,<br />

US<br />

GUNIC, Esmir, Irvine, CA 92614, US<br />

HONG, Zhi, Irvine, CA 92603, US<br />

LANG, Stanley, Valeant Research & Development,<br />

Costa Mesa, CA 92626, US<br />

KIM, Hong, Woo, Irvine, CA 92606, US<br />

(74) Cole, William Gwyn, avidity IP Merlin House<br />

Falconry Court Baker's Lane, Epping, Essex<br />

CM16 5DQ, GB<br />

(60) 09170772.9 / 2 135 608<br />

11177941.9 / 2 4<strong>02</strong> 011<br />

11184<strong>02</strong>5.2<br />

A61K 31/422 → (51) C07D 209/82<br />

A61K 31/424 → (51) C07D 487/04<br />

A61K 31/426 → (51) C07D 209/82<br />

A61K 31/427 → (51) C07D 233/50<br />

A61K 31/433 → (51) C07D 487/04<br />

A61K 31/437 → (51) C07D 471/04<br />

(51) A61K 31/44 (11) 1 9<strong>02</strong> 714 B1<br />

A61K 31/335 A61K 31/27<br />

A61K 31/225 A61K 31/195<br />

A61P 25/00 C07D 213/<strong>02</strong><br />

C07D 317/00 C07C 205/00<br />

C07C 229/00 C07C 261/00<br />

(25) En (26) En<br />

(21) 07<strong>02</strong>0763.4 (22) 11.06.20<strong>02</strong><br />

(84) AT BE CH CY DE DK ES FI FR GB GR IE IT LI<br />

LU MC NL PT SE TR<br />

(43) 26.03.2008<br />

(30) 11.06.2001 US 297521 P<br />

14.06.2001 US 298514 P<br />

19.03.20<strong>02</strong> US 366090 P<br />

(54) • Prodrugs aus GABA-Analoga, Zusammensetzungen<br />

und ihre Verwendungen<br />

• Prodrugs of gaba analogs, compositions<br />

and uses thereof<br />

• Promédicaments d'analogues gaba, compositions<br />

et leurs utilisations<br />

(73) XenoPort, Inc., 3410 Central Expressway,<br />

Santa Clara, CA 95051, US<br />

(72) Gallop, Mark A., Santa Clara CA 95015, US<br />

Cundy, Kenneth C., Redwood City CA 94062,<br />

US<br />

Zhou, Cindy X., Palo Alto CA 94303, US<br />

Yao, Fenmei, Mountain View CA 94040, US<br />

Xiang, Jia-Ning, Palo Alto CA 94303, US<br />

Ollmann, Ian R., San Jose CA 95129, US<br />

Qiu, Fayang G., Mountain View CA 94043,<br />

US<br />

(74) Wytenburg, Wilhelmus Johannes, et al,<br />

Mewburn Ellis LLP 33 Gutter Lane, London<br />

EC2V 8AS, GB<br />

(60) 09003173.3 / 2 085 087<br />

(62) <strong>02</strong>744314.2 / 1 404 324<br />

A61K 31/44 → (51) C07C 311/29<br />

(51) A61K 31/4412 (11) 1 750 703 B1<br />

A61K 31/513 A61K 31/53<br />

A61K 45/00 A61P 35/00<br />

A61K 47/22<br />

(25) En (26) En

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