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Bulletin 2010/31 - European Patent Office

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(C07C) I.1(1)<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) GB 2008/003527 17.10.2008<br />

(87) WO 2009/050483 2009/17 23.04.2009<br />

(30) 19.10.2007 GB 0720486<br />

(54) • KATIONISCHE LIPIDE<br />

• CATIONIC LIPIDS<br />

• LIPIDES CATIONIQUES<br />

(71) The University Court Of The University of<br />

Edinburgh, Old College, South Bridge Edinburgh<br />

EH8 9YL, GB<br />

(72) UNCITI-BROCETA, Asier, Edinburgh EH9<br />

3JJ, GB<br />

BRADLEY, Mark, Edinburgh EH9 3JJ, GB<br />

(74) McNab, Donald C., et al, Marks & Clerk LLP<br />

Aurora 120 Bothwell Street, Glasgow G2<br />

7JS, GB<br />

C07C 233/20 → (51) C07C 233/18<br />

C07C 233/47 → (51) C07C 2<strong>31</strong>/12<br />

C07C 233/64 → (51) C07D 213/65<br />

(51) C07C 233/81 (11) 2 212 280 A1*<br />

A61K <strong>31</strong>/167 A61P 25/28<br />

(25) En (26) En<br />

(21) 08838993.7 (22) 14.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/079782 14.10.2008<br />

(87) WO 2009/052079 2009/17 23.04.2009<br />

(30) 19.10.2007 US 981170 P<br />

(54) • AMIDGEBUNDENE MODULATOREN VON<br />

Y-SEKRETASE<br />

• AMIDE LINKED MODULATORS OF Y-<br />

SECRETASE<br />

• MODULATEURS DE LA -SECRÉTASE LIÉS<br />

À UN AMIDE<br />

(71) Janssen Pharmaceutica, N.V., Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) HO, Chih Yung, Lansdale, Pennsylvania<br />

19446, US<br />

(74) Warner, James Alexander, Carpmaels &<br />

Ransford 43-45 Bloomsbury Square, London<br />

WC1A 2RA, GB<br />

C07C 237/22 → (51) C07C 233/18<br />

C07C 255/58 → (51) C07C 229/34<br />

C07C 257/18 → (51) C07D 257/04<br />

C07C 309/29 → (51) C07D 257/04<br />

C07C <strong>31</strong>1/29 → (51) C07D 205/04<br />

C07C 391/00 → (51) C01B 19/00<br />

(51) C07D 205/04 (11) 2 212 281 A1*<br />

C07D 207/06 C07C <strong>31</strong>1/29<br />

(25) De (26) De<br />

(21) 08803006.9 (22) 12.08.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) EP 2008/060563 12.08.2008<br />

(87) WO 2009/021945 2009/08 19.02.2009<br />

(30) 14.08.2007 PCT/EP2007/058408<br />

21.02.2008 PCT/EP2008/052157<br />

26.02.2008 EP 08102044<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(54) • ARYLSULFONAMIDE MIT ANALGETI-<br />

SCHER WIRKUNG<br />

• ARYLSULFONAMIDES WITH ANALGESIC<br />

ACTIVITY<br />

• ARYLSULFONAMIDES À EFFET ANALGÉ-<br />

SIQUE<br />

(71) Boehringer Ingelheim International GmbH,<br />

Binger Straße 173, 55216 Ingelheim am<br />

Rhein, DE<br />

(72) HAUEL, Norbert, 55216 Ingelheim am Rhein,<br />

DE<br />

CECI, Angelo, 55216 Ingelheim am Rhein,<br />

DE<br />

DOODS, Henri, 55216 Ingelheim am Rhein,<br />

DE<br />

KAUFFMANN-HEFNER, Iris, 55216 Ingelheim<br />

am Rhein, DE<br />

KONETZKI, Ingo, 55216 Ingelheim am Rhein,<br />

DE<br />

SCHULER-METZ, Annette, 55216 Ingelheim<br />

am Rhein, DE<br />

WALTER, Rainer, 55216 Ingelheim am<br />

Rhein, DE<br />

(74) Hammann, Heinz, et al, Boehringer Ingelheim<br />

GmbH CD-<strong>Patent</strong>s Binger Straße 173, 55216<br />

Ingelheim am Rhein, DE<br />

(51) C07D 207/06 (11) 2 212 282 A1*<br />

C07D 401/12 C07D 401/14<br />

C07D 403/12 C07D 405/12<br />

C07D 409/12 C07D 417/04<br />

C07D 471/04 A61K <strong>31</strong>/4025<br />

(25) En (26) En<br />

(21) 08839473.9 (22) 14.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/079760 14.10.2008<br />

(87) WO 2009/052065 2009/17 23.04.2009<br />

(30) 17.10.2007 US 980601 P<br />

(54) • SUBSTITUIERTE N-PHENYL-BIPYRROLI-<br />

DINCARBONSÄUREAMIDE UND DEREN<br />

THERAPEUTISCHE VERWENDUNG<br />

• SUBSTITUTED N-PHENYL-BIPYRROLI-<br />

DINE CARBOXAMIDES AND THERAPEUTIC<br />

USE THEREOF<br />

• CARBOXAMIDES DE N-PHÉNYL-BIPYR-<br />

ROLIDINE SUBSTITUÉS ET LEUR UTILI-<br />

SATION THÉRAPEUTIQUE<br />

(71) Sanofi-Aventis, 174 Avenue de France,<br />

75013 Paris, FR<br />

(72) CZECHTIZKY, Werngard, 65926 Frankfurt<br />

Am Main, DE<br />

GAO, Zhongli, Bridgewater, New Jersey<br />

08807, US<br />

HURST, William J., Bridgewater, New Jersey<br />

08807, US<br />

SCHWINK, Lothar, 65926 Frankfurt Am<br />

Main, DE<br />

STENGELIN, Siegfried, 65926 Frankfurt Am<br />

Main, DE<br />

(74) Rauline, Mathilde, et al, Sanofi-Aventis<br />

Département Brevets 174 Avenue de France,<br />

75013 Paris, FR<br />

(51) C07D 207/06 (11) 2 212 283 A1*<br />

C07D 401/14 C07D 403/12<br />

C07D 405/12 C07D 413/12<br />

A61K <strong>31</strong>/4025 A61P 25/00<br />

(25) En (26) En<br />

(21) 08839959.7 (22) 14.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/079757 14.10.2008<br />

(87) WO 2009/052062 2009/17 23.04.2009<br />

108<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>31</strong>/<strong>2010</strong>) 04.08.<strong>2010</strong><br />

(30) 17.10.2007 US 980599 P<br />

(54) • SUBSTITUIERTE N-PHENYL-BIPYRROLI-<br />

DINCARBONSÄUREAMIDE UND DEREN<br />

THERAPEUTISCHE VERWENDUNG<br />

• SUBSTITUTED N-PHENYL-BIPYRROLI-<br />

DINE CARBOXAMIDES AND THERAPEUTIC<br />

USE THEREOF<br />

• CARBOXAMIDES DE N-PHÉNYL-BIPYR-<br />

ROLIDINE SUBSTITUÉS ET LEUR UTILI-<br />

SATION THÉRAPEUTIQUE<br />

(71) Sanofi-Aventis, 174 Avenue de France,<br />

75013 Paris, FR<br />

(72) CZECHTIZKY, Werngard, 65926 Frankfurt<br />

Am Main, DE<br />

GAO, Zhongli, Bridgewater, New Jersey<br />

08807, US<br />

HURST, William J., Bridgewater, New Jersey<br />

08807, US<br />

SCHWINK, Lothar, 65926 Frankfurt Am<br />

Main, DE<br />

STENGELIN, Siegfried, 65926 Frankfurt Am<br />

Main, DE<br />

(74) Rauline, Mathilde, et al, Sanofi-Aventis<br />

Département Brevets 174 Avenue de France,<br />

75013 Paris, FR<br />

C07D 207/06 → (51) C07D 205/04<br />

C07D 207/335→ (51) C07D 207/48<br />

(51) C07D 207/48 (11) 2 212 284 A2*<br />

C07D 2<strong>31</strong>/12 C07D 2<strong>31</strong>/16<br />

C07D 2<strong>31</strong>/22 C07D 233/64<br />

C07D 261/08 C07D 271/06<br />

C07D 277/28 C07D 401/04<br />

C07D 207/335 A61K <strong>31</strong>/415<br />

A61K <strong>31</strong>/4164 A61K <strong>31</strong>/40<br />

A61P 7/00<br />

(25) En (26) En<br />

(21) 08839241.0 (22) 15.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/011755 15.10.2008<br />

(87) WO 2009/051718 2009/17 23.04.2009<br />

(88) 11.06.2009<br />

(30) 15.10.2007 US 998933 P<br />

(54) • CALCIUM-REZEPTOR-MODULIERENDE<br />

MITTEL<br />

• CALCIUM RECEPTOR MODULATING<br />

AGENTS<br />

• AGENTS DE MODULATION DU RÉCEP-<br />

TEUR DU CALCIUM<br />

(71) Amgen Inc., One Amgen Center Drive,<br />

Thousand Oaks, CA 91320-1799, US<br />

(72) COULTER, Thomas S., Wantage, Oxfordshire<br />

OX12 7PA, GB<br />

FOTSCH, Christopher H., Thousand Oaks<br />

California 91360, US<br />

GHIRON, Chiara, I-53041 Siena, IT<br />

HARRINGTON, Paul E., Camarillo California<br />

93012, US<br />

KELLY, Michael G., South San Francisco<br />

California 94080, US<br />

MILLER, Philip, Headington, Oxford OX3<br />

8AS, GB<br />

RISHTON, Gilbert M., Malibu California<br />

90265, US<br />

ST. JEAN, David J., Jr., Camarillo California<br />

93012, US<br />

SEMIN, David J., Thousand Oaks California<br />

91320, US<br />

(74) Grünecker, Kinkeldey, Stockmair & Schwanhäusser<br />

Anwaltssozietät, Leopoldstrasse 4,<br />

80802 München, DE<br />

C07D 209/04 → (51) C07D 403/08

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