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Bulletin 2010/31 - European Patent Office

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(C07D) I.1(1)<br />

C07D 261/12 → (51) C07D 257/04<br />

C07D 271/06 → (51) C07D 207/48<br />

C07D 271/113→ (51) C07D 413/10<br />

C07D 277/28 → (51) C07D 207/48<br />

C07D 295/155→ (51) C07D 211/18<br />

(51) C07D 305/00 (11) 2 212 305 A1*<br />

(25) En (26) En<br />

(21) 08845661.1 (22) 30.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/081857 30.10.2008<br />

(87) WO 2009/059046 2009/19 07.05.2009<br />

(30) <strong>31</strong>.10.2007 US 984<strong>31</strong>3 P<br />

(54) • BETA-LAKTONVERBINDUNGEN<br />

• BETA-LACTONE COMPOUNDS<br />

• COMPOSÉS DE BÊTA-LACTONE<br />

(71) Burnham Institute for Medical Research,<br />

10901 N. Torrey Pines Road, La Jolla, CA<br />

92037, US<br />

The Texas A&M University System, Mail Stop<br />

3369, College Station, TX 77843-3369, US<br />

(72) SMITH, Jeffrey, W., La Jolla CA 92037, US<br />

ROMO, Daniel, College Station TX 77843-<br />

3369, US<br />

MA, Gil, College Station TX 77843-3369, US<br />

ZANCANELLA, Manuel, College Station TX<br />

77843-3369, US<br />

(74) Coles, Andrea Birgit, Kilburn & Strode LLP<br />

20 Red Lion Street, GB-London WC1R 4PJ,<br />

GB<br />

C07D 305/00 → (51) A61K 9/70<br />

C07D 307/14 → (51) C07D 209/42<br />

C07D 307/60 → (51) B01J 27/14<br />

C07D 307/68 → (51) C07D 209/42<br />

C07D 307/78 → (51) C07D 453/00<br />

C07D 307/85 → (51) C07D 209/42<br />

(51) C07D 307/92 (11) 2 212 306 A1*<br />

(25) En (26) En<br />

(21) 08840902.4 (22) 20.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) IB 2008/054299 20.10.2008<br />

(87) WO 2009/053884 2009/18 30.04.2009<br />

(30) 23.10.2007 EP 07119038<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

TETRANORLABDANDERIVATEN<br />

• PROCESS FOR THE PREPARATION OF<br />

TETRANORLABDANE DERIVATIVES<br />

• PROCÉDÉ DE PRÉPARATION DE DÉRIVÉS<br />

DE TÉTRANORLABDANE<br />

(71) Firmenich S.A., 1, route des Jeunes P.O. Box<br />

239, 1211 Geneva 8, CH<br />

(72) FEHR, Charles, CH-1290 Versoix, CH<br />

(74) Carina, Riccardo Filippo, Firmenich SA 1,<br />

route des Jeunes P.O. Box 239, 1211 Genève<br />

8, CH<br />

(51) C07D 307/92 (11) 2 212 307 A1*<br />

(25) En (26) En<br />

(21) 08842543.4 (22) 22.10.2008<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) US 2008/080699 22.10.2008<br />

(87) WO 2009/055416 2009/18 30.04.2009<br />

(30) 24.10.2007 US 164<br />

(54) • HOCHREINES SYNTHETISCHES VERFAH-<br />

REN ZUR HERSTELLUNG VON DODECA-<br />

HYDRONAPHTHOFURANYLCARBAMIN-<br />

SÄUREESTERZWISCHENPRODUKTEN<br />

• HIGH PURITY SYNTHETIC PROCESS FOR<br />

THE PREPARATION OF DODECAHYDRO-<br />

NAPTHO-FURANYL-CARBAMIC ACID<br />

ESTER INTERMEDIATES<br />

• PROCÉDÉ DE SYNTHÈSE HAUTE PURETÉ<br />

POUR LA PRÉPARATION DE PRODUITS<br />

INTERMÉDIAIRES D'ESTER D'ACIDE<br />

DODÉCAHYDRO-NAPHTO-FURANYL-CAR-<br />

BAMIQUE<br />

(71) Schering Corporation, 2000 Galloping Hill<br />

Road, Kenilworth, NJ 07033-0530, US<br />

(72) LIAO, Jing, Livingston New Jersey 07039,<br />

US<br />

WANG, Tao, Springfield NewJersey 07081,<br />

US<br />

(74) Quelle-Fontijn, Monique, et al, P.O. Box 20,<br />

5340 BH Oss, NL<br />

C07D 309/04 → (51) C07D 209/42<br />

C07D 309/14 → (51) C07D 209/42<br />

C07D <strong>31</strong>1/58 → (51) C07D 209/42<br />

(51) C07D <strong>31</strong>1/92 (11) 2 212 308 A1*<br />

C07D 493/04 C09K 19/34<br />

(25) De (26) De<br />

(21) 08855468.8 (22) 03.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) EP 2008/009242 03.11.2008<br />

(87) WO 2009/068152 2009/23 04.06.2009<br />

(30) 27.11.2007 DE 102007057028<br />

(54) • BENZO[F]CHROMEN- UND PYRANO[3, 2-<br />

F]CHROMEN-DERIVATE ZUR ANWEN-<br />

DUNG IN FLÜSSIGKRISTALLINEN MEDIEN<br />

• BENZO[F]CHROME AND PYRANO[3,2-F]<br />

CHROME DERIVATIVES FOR USE IN<br />

LIQUID CRYSTAL MEDIA<br />

• DÉRIVÉS DE BENZO[F]CHROMÈNE ET DE<br />

PYRANO[3,2-F]CHROMÈNE DESTINÉS À<br />

ÊTRE EMPLOYÉS DANS DES SUBSTAN-<br />

CES DE CRISTAUX LIQUIDES<br />

(71) Merck <strong>Patent</strong> GmbH, Frankfurter Strasse<br />

250, 64293 Darmstadt, DE<br />

(72) JANSEN, Axel, 64293 Darmstadt, DE<br />

KLASEN-MEMMER, Melanie, 67259 Heuchelheim,<br />

DE<br />

C07D <strong>31</strong>1/92 → (51) C07D 209/42<br />

C07D <strong>31</strong>3/08 → (51) C07D 209/42<br />

C07D 333/36 → (51) C07D 209/42<br />

C07D 333/70 → (51) C07D 209/42<br />

C07D 335/02 → (51) C07D 209/42<br />

(51) C07D 401/04 (11) 2 212 309 A1*<br />

A61K <strong>31</strong>/4196 A61P 25/00<br />

(25) En (26) En<br />

(21) 08839205.5 (22) 15.10.2008<br />

112<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>31</strong>/<strong>2010</strong>) 04.08.<strong>2010</strong><br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) EP 2008/063845 15.10.2008<br />

(87) WO 2009/050186 2009/17 23.04.2009<br />

(30) 18.10.2007 EP 07118825<br />

(54) • TRISUBSTITUIERTE 1,2,4-TRIAZOLE<br />

• TRISUBSTITUTED 1,2,4-TRIAZOLES<br />

• 1,2,4-TRIAZOLES TRISUBSTITUÉS<br />

(71) Janssen Pharmaceutica N.V., Turnhoutseweg<br />

30, 2340 Beerse, BE<br />

(72) THURING, Johannes Wilhelmus John F., B-<br />

2018 Antwerpen, BE<br />

DINKLO, Theodorus, CH-4125 Riehen, CH<br />

LESAGE, Anne, Simone, Josephine, B-2340<br />

Beerse, BE<br />

DE BRUYN, Marcel, Frans, Leopold, B-2330<br />

Wortel, BE<br />

ZHUANG, Wei, B-2340 Beerse, BE<br />

(74) Quaghebeur, Luc, Janssen Pharmaceutica N.<br />

V. <strong>Patent</strong> Department, Turnhoutseweg 30,<br />

2340 Beerse, BE<br />

(51) C07D 401/04 (11) 2 212 <strong>31</strong>0 A2*<br />

C07D 401/14 C07D 215/12<br />

C07D 241/04<br />

(25) En (26) En<br />

(21) 08839611.4 (22) 06.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(86) IN 2008/000643 06.10.2008<br />

(87) WO 2009/050734 2009/17 23.04.2009<br />

(88) 07.01.<strong>2010</strong><br />

(30) 15.10.2007 IN MU20532007<br />

(54) • FÜR DIE GROSSTECHNISCHE DURCH-<br />

FÜHRUNG GEEIGNETES VERFAHREN ZUR<br />

HERSTELLUNG VON BISCHINOLINDERI-<br />

VATEN UNTER VERWENDUNG VON IM<br />

WESENTLICHEN REINEN N-MONOSUBS-<br />

TITUIERTEN PIPERAZINEN<br />

• AN INDUSTRIALLY FEASIBLE PROCESS<br />

FOR THE MANUFACTURE OF BISQUINO-<br />

LINE DERIVATIVES BY USING SUBSTAN-<br />

TIALLY PURE N-MONOSUBSTITUTED<br />

PIPERAZINES<br />

• PROCÉDÉ POUVANT ÊTRE MIS EN OEU-<br />

VRE À L'ÉCHELLE INDUSTRIELLE POUR<br />

LA FABRICATION DE DÉRIVÉS DE BIS-<br />

QUINOLINE AU MOYEN DE PIPÉRAZINES<br />

N-MONOSUBSTITUÉES SENSIBLEMENT<br />

PURES<br />

(71) Elder Pharmaceuticals Ltd, Elder House, Plot<br />

No. C/9 Dalia Indl. Estate Off. New Link<br />

Road, Andheri (W) Mumbai 400 058, IN<br />

(72) SAKHARDANDE, Rajiv, Mumbai 400 057, IN<br />

NIMBALKAR, Manmohan, Prabhadevi Mumbai<br />

400 025, IN<br />

PATIL, Subarao, Kamothe Navi-Mumbai 410<br />

209, IN<br />

BHALEKAR, Santosh, Pin 414 306, IN<br />

PATIL, Rajendra, Sector -3$New Panvel<br />

$Raigad 410 203, IN<br />

MHASKE, Rohidas, Nerul Navi-Mumbai 400<br />

706, IN<br />

(74) Brand, Thomas Louis, W.P. Thompson & Co.<br />

55 Drury Lane, London WC2B 5SQ, GB<br />

C07D 401/04 → (51) C07D 207/48<br />

C07D 401/06 → (51) C07D 211/18<br />

C07D 401/06 → (51) C07D 241/08<br />

C07D 401/10 → (51) C07D 211/18<br />

C07D 401/10 → (51) C07D 241/08

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