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Bulletin 2010/31 - European Patent Office

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(C07D) II.1(1)<br />

(21) 0381<strong>31</strong>26.4 (22) 16.12.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 21.09.2005<br />

(86) EP 2003/014274 16.12.2003<br />

(87) WO 2004/054990 2004/27 01.07.2004<br />

(30) 18.12.2002 DE 10259672<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

ALKOXYCARBONYLAMINO-TRIAZINEN<br />

• METHOD FOR THE PRODUCTION OF<br />

ALKOXYCARBONYLAMINO TRIAZINES<br />

• PROCÉDÉ DE PRODUCTION D' ALCOXY-<br />

CARBONYLAMINOTRIAZINES<br />

(73) BASF SE, 67056 Ludwigshafen, DE<br />

(72) SCHNEIDER, Jörg, 69469 Weinheim, DE<br />

SCHERR, Günter, 67065 Ludwigshafen, DE<br />

SCHUPP, Hans, 67549 Worms, DE<br />

EICHFELDER, Andreas, 67133 Maxdorf, DE<br />

ROBERT, Alain, 67150 Niederkirchen, DE<br />

REIF, Martin, 67354 Römerberg, DE<br />

C07D 257/04 → (51) C07D 233/32<br />

C07D 261/02 → (51) C07D 233/32<br />

C07D 261/04 → (51) C07D 233/32<br />

C07D 261/18 → (51) C07D 233/32<br />

C07D 265/02 → (51) C07D 233/32<br />

C07D 271/08 → (51) C07D 207/09<br />

C07D 277/46 → (51) C07D 233/32<br />

(51) C07D 277/56 (11) 1 474 407 B1<br />

A01N 43/78<br />

(25) De (26) De<br />

(21) 03737263.8 (22) 22.01.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT SE SI SK TR<br />

RO<br />

(43) 10.11.2004<br />

(86) EP 2003/000589 22.01.2003<br />

(87) WO 2003/066610 2003/33 14.08.2003<br />

(30) 04.02.2002 DE 10204391<br />

(54) • DIFLUORMETHYL THIAZOLYL CARBOXA-<br />

NILIDE<br />

• DIFLUOROMETHYL THIAZOLYL CARBOX-<br />

ANILIDES<br />

• DIFLUOROMETHYL THIAZOLYL CARBO-<br />

XANILIDES<br />

(73) Bayer CropScience AG, Alfred-Nobel-Straße<br />

50, 40789 Monheim, DE<br />

(72) ELBE, Hans-Ludwig, 42329 Wuppertal, DE<br />

RIECK, Heiko, 69110 Ste. Foy-lès-Lyon, FR<br />

DUNKEL, Ralf, 40789 Monheim, DE<br />

WACHENDORFF-NEUMANN, Ulrike, 56566<br />

Neuwied, DE<br />

KUCK, Karl-Heinz, 40764 Langenfeld, DE<br />

MAULER-MACHNIK, Astrid, 42799 Leichlingen,<br />

DE<br />

KUGLER, Martin, 42799 Leichlingen, DE<br />

JAETSCH, Thomas, 50668 Köln, DE<br />

WACHTLER, Peter, 47800 Krefeld, DE<br />

C07D 285/08 → (51) C07D 233/32<br />

(51) C07D 295/08 (11) 1 709 021 B1<br />

C07D <strong>31</strong>1/78 C07D 335/04<br />

C07D 221/18 A61K <strong>31</strong>/4453<br />

A61K <strong>31</strong>/4523 A61K <strong>31</strong>/55<br />

A61P 15/12<br />

(25) En (26) En<br />

(21) 05704874.6 (22) 18.01.2005<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

AL BA HR LV MK YU<br />

(43) 11.10.2006<br />

(86) US 2005/000020 18.01.2005<br />

(87) WO 2005/073204 2005/32 11.08.2005<br />

(30) 22.01.2004 US 538442 P<br />

22.01.2004 US 538342 P<br />

(54) • SELEKTIVE MODULATOREN DES ÖSTRO-<br />

GENREZEPTORS ZUR BEHANDLUNG VON<br />

VASOMOTORISCHEN SYMPTOMEN<br />

• SELECTIVE ESTROGEN RECEPTOR MOD-<br />

ULATORS FOR THE TREATMENT OF<br />

VASOMOTOR SYMPTOMS<br />

• MODULATEURS SELECTIFS DU RECEP-<br />

TEUR DES OESTROGENES POUR LE<br />

TRAITEMENT DE SYMPTOMES VASOMO-<br />

TEURS<br />

(73) ELI LILLY AND COMPANY, Lilly Corporate<br />

Center, Indianapolis, IN 46285, US<br />

(72) DALLY, Robert, Dean, Carmel, Indiana<br />

46033, US<br />

DODGE, Jeffrey, Alan, Indianapolis, Indiana<br />

46256, US<br />

FRANK, Scott, Alan, Indianapolis, Indiana<br />

46220, US<br />

HINKLIN, Ronald, Jay, Longmont, Colorado<br />

80503, US<br />

SHEPHERD, Timothy, Alan, Indianapolis,<br />

Indiana 46217, US<br />

WALLACE, Owen, Brendan, Zionsville, Indiana<br />

46077, US<br />

(74) Burnside, Ivan John, Eli Lilly and Company<br />

Limited Lilly Research Centre Erl Wood<br />

Manor Sunninghill Road, Windlesham Surrey<br />

GU20 6PH, GB<br />

C07D 295/12 → (51) C07C 275/54<br />

C07D 295/20 → (51) C07D 233/32<br />

C07D 307/14 → (51) C07D 233/32<br />

C07D 307/20 → (51) C07B 63/04<br />

C07D <strong>31</strong>1/30 → (51) A61K <strong>31</strong>/03<br />

C07D <strong>31</strong>1/74 → (51) A61K <strong>31</strong>/03<br />

C07D <strong>31</strong>1/76 → (51) A61K <strong>31</strong>/03<br />

C07D <strong>31</strong>1/78 → (51) C07D 295/08<br />

C07D <strong>31</strong>7/22 → (51) C07C 59/70<br />

C07D <strong>31</strong>9/20 → (51) C07C 59/70<br />

(51) C07D 327/02 (11) 2 089 374 B1<br />

C07C 323/20<br />

(25) Fr (26) Fr<br />

(21) 07870250.3 (22) 06.11.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

BA HR MK RS<br />

(43) 19.08.2009<br />

(86) FR 2007/0018<strong>31</strong> 06.11.2007<br />

(87) WO 2008/068403 2008/24 12.06.2008<br />

(30) 08.11.2006 FR 0609815<br />

(54) • VERFAHREN ZUR SYNTHESE VON N-[3-<br />

[(2-METHOXYPHENYL)SULFANYL-2-<br />

METHYLPROPYL-3,4-DIHYDRO-2H-1,5-<br />

BENZOXATHIEPIN-3-AMIN<br />

• METHOD FOR THE SYNTHESIS OF N- [3- [<br />

(2-METHOXYPHENYL) SULFANYL] -2-<br />

METHYLPROPYL]-3,4-DIHYDRO-2H-1,5-<br />

BENZOXATHIEPIN-3-AMINE<br />

606<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>31</strong>/<strong>2010</strong>) 04.08.<strong>2010</strong><br />

• PROCEDE DE SYNTHESE DU N- [3- [ (2-<br />

METHOXYPHENYL) SULFANYL] -2-<br />

METHYLPROPYL] -3,4-DIHYDRO-2H-1,5-<br />

BENZOXATHIEPIN-3-AMINE<br />

(73) Pierre Fabre Medicament, 45 Place Abel<br />

Gance, 92100 Boulogne-Billancourt, FR<br />

(72) VACHER, Bernard, 81100 Castres, FR<br />

BRUNEL, Yves, 81150 Marssac-Sur-Tarn, FR<br />

MAUREL, Jean-Louis, 81100 Burlats, FR<br />

(74) Rousseau, Pierrick Edouard, et al, Pierre<br />

Fabre SA Direction Propriété Intellectuelle 17,<br />

Avenue Jean Moulin, F-81106 Castres Cedex,<br />

FR<br />

C07D 333/38 → (51) C07D 233/32<br />

C07D 335/04 → (51) C07D 295/08<br />

C07D 335/06 → (51) A61K <strong>31</strong>/03<br />

C07D 401/04 → (51) C07D 217/24<br />

C07D 401/06 → (51) C07D 217/24<br />

C07D 401/06 → (51) C07D 243/14<br />

(51) C07D 401/12 (11) 2 118 090 B1<br />

(25) En (26) En<br />

(21) 08708696.3 (22) 05.02.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 18.11.2009<br />

(86) EP 2008/051397 05.02.2008<br />

(87) WO 2008/095928 2008/33 14.08.2008<br />

(30) 06.02.2007 EP 07101822<br />

(54) • VERFAHREN ZUR HERSTELLUNG EINES<br />

BENZIMIDAZOL-DERIVATS<br />

• PROCESS FOR THE PREPARATION OF A<br />

BENZIMIDAZOLE DERIVATIVE<br />

• PROCÉDÉ DE PRÉPARATION D'UN<br />

DÉRIVÉ DE BENZIMIDAZOLE<br />

(73) Boehringer Ingelheim International GmbH,<br />

Binger Straße 173, 55216 Ingelheim am<br />

Rhein, DE<br />

(72) BROEDER, Wolfgang, 55216 Ingelheim Am<br />

Rhein, DE<br />

SOBOTTA, Rainer, 55216 Ingelheim Am<br />

Rhein, DE<br />

(74) Hammann, Heinz, et al, Boehringer Ingelheim<br />

GmbH CD-<strong>Patent</strong>s Binger Straße 173, 55216<br />

Ingelheim am Rhein, DE<br />

C07D 401/12 → (51) C07D 243/14<br />

C07D 401/12 → (51) C07D 403/12<br />

C07D 401/14 → (51) C07D 243/14<br />

C07D 403/06 → (51) C07D 243/14<br />

(51) C07D 403/12 (11) 1 8<strong>31</strong> 201 B1<br />

C07D 401/12 A61K <strong>31</strong>/4545<br />

A61K <strong>31</strong>/4178 A61K <strong>31</strong>/4439<br />

A61P 25/18<br />

(25) En (26) En<br />

(21) 05821636.7 (22) 21.12.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 12.09.2007<br />

(86) GB 2005/050258 21.12.2005<br />

(87) WO 2006/067529 2006/26 29.06.2006<br />

(30) 21.12.2004 GB 0427987<br />

21.12.2004 GB 0427989<br />

(54) • PIPERIDIN- UND AZETIDINDERIVATE ALS<br />

GLYT1-INHIBITOREN<br />

• PIPERIDINE AND AZETIDINE DERIVA-<br />

TIVES AS GLYT1 INHIBITORS

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