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Bulletin 2010/31 - European Patent Office

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(C07C) I.1(2)<br />

C07C 211/07 → (51) C07C 47/04<br />

C07C 211/51 → (51) C07C 209/84<br />

(51) C07C 211/55 (11) 2 213 650 A1<br />

C07C 211/56 A61K <strong>31</strong>/136<br />

A61P <strong>31</strong>/18<br />

(25) Zh (26) En<br />

(21) 08840721.8 (22) 07.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) CN 2008/001699 07.10.2008<br />

(87) WO 2009/049491 2009/17 23.04.2009<br />

(30) 12.10.2007 CN 200710163958<br />

(54) • SUBSTITUIERTE DIPHENYLAMINE ALS<br />

INHIBITOREN DER REVERSEN TRANS-<br />

KRIPTASE, VERFAHREN ZU DEREN HER-<br />

STELLUNG UND ANWENDUNG DAVON<br />

• SUBSTITUTED DIPHENYLAMINES AS<br />

INHIBITORS OF REVERSE TRANSCRIP-<br />

TASE, PROCESS OF PREPARING THEM<br />

AND USE THEREOF<br />

• DIPHÉNYLAMINES SUBSTITUÉES EN<br />

TANT QU'INHIBITEURS DE LA TRAN-<br />

SCRIPTASE INVERSE, LEUR PROCÉDÉ DE<br />

PRÉPARATION ET LEUR UTILISATION<br />

(71) Institute Of Pharmacology And Toxicology<br />

Academy Of Military Medical Sciences P.L.A.<br />

China, No. 27 Taiping Road, Haidian District<br />

Beijing 100-850, CN<br />

(72) XIE, Lan, Beijing 100850, CN<br />

QIN, Bingjie, Beijing 100850, CN<br />

LEE, Kou-hsiung, Chapel Hill, NC 27514, US<br />

(74) Dey, Michael, et al, Weickmann & Weickmann<br />

<strong>Patent</strong>anwälte Richard-Strauss-<br />

Strasse 80, 81679 München, DE<br />

C07C 211/56 → (51) C07C 211/55<br />

C07C 213/08 → (51) C07C 217/54<br />

(51) C07C 217/54 (11) 2 213 651 A1<br />

C07C 213/08 C07D 223/16<br />

(25) Zh (26) En<br />

(21) 08800667.1 (22) 10.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) CN 2008/001711 10.10.2008<br />

(87) WO 2009/062377 2009/21 22.05.2009<br />

(30) 16.11.2007 CN 200710188301<br />

19.05.2008 CN 200810093266<br />

(54) • OPTISCHE TRENNUNG VON 4,5-DIME-<br />

THOXY-1-(METHYLAMINOMETHYL)BEN-<br />

ZOCYCLOBUTAN<br />

• RESOLUTION OF 4,5-DIMETHOXY-1-<br />

(METHYLAMINOMETHYL)-BENZOCYCLO-<br />

BUTANE<br />

• RÉSOLUTION DE 4,5-DIMÉTHOXY-1-<br />

(MÉTHYLAMINOMÉTHYL)-BENZOCYCLO-<br />

BUTANE<br />

(71) Jiangsu Hengrui Medicine Co., Ltd., No. 145<br />

Renmin East Road Xinpu District, Lianyungang,<br />

Jiangsu 222002, CN<br />

(72) SUN, Piaoyang, Jiangsu 222002, CN<br />

CHEN, Yongjiang, Jiangsu 222002, CN<br />

YU, Guangliang, Jiangsu 222002, CN<br />

(74) Dilg, Haeusler, Schindelmann <strong>Patent</strong>anwaltsgesellschaft<br />

mbH, Leonrodstraße 58,<br />

80636 München, DE<br />

(51) C07C 217/80 (11) 2 213 652 A1<br />

A61K <strong>31</strong>/135<br />

(25) En (26) En<br />

(21) 10161604.3 (22) 19.12.2005<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK YU<br />

(30) 17.12.2004 US 636696 P<br />

02.06.2005 US 686395 P<br />

(54) • Stilbenderivate und ihre Verwendung zum<br />

Binden und Abbilden von Amyloidplaques<br />

• Stilbene derivatives and their use for<br />

binding and imaging amyloid plaques<br />

• Dérivés de stilbène et leur utilisation pour<br />

l'imagerie des plaques amyloïdes et leur<br />

liaison<br />

(71) The Trustees of The University of Pennsylvania,<br />

<strong>31</strong>60 Chestnut Street, Suite 200,<br />

Philadelphia, Pennsylvania 19104-6283, US<br />

(72) Kung, Hank F., Wynnewood, PA 19096, US<br />

Kung, Mei-Ping, Wynnewood, PA 19096, US<br />

Zhuang, Zhi-Ping, Philadelphia, PA 19104,<br />

US<br />

(74) Dörries, Hans Ulrich, df-mp Fünf Höfe<br />

Theatinerstrasse 16, 80333 München, DE<br />

(62) 05854410.7 / 1 841 465<br />

(51) C07C 227/32 (11) 2 213 653 A2<br />

(25) Es (26) En<br />

(21) 08852208.1 (22) 19.11.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) ES 2008/000724 19.11.2008<br />

(87) WO 2009/065987 2009/22 28.05.2009<br />

(88) 30.07.2009<br />

(30) 19.11.2007 ES 20070<strong>31</strong>12<br />

(54) • VERFAHREN ZUR STEREOSELEKTIVEN<br />

HERSTELLUNG VON AMINOSÄUREDER-<br />

IVATEN<br />

• METHOD FOR THE STEREOSELECTIVE<br />

PREPARATION OF AMINO ACID DERIVA-<br />

TIVES<br />

• PROCEDE DE PREPARATION STEREOSE-<br />

LECTIVE DE DERIVES D'ACIDES AMINES<br />

(71) BCN Peptides, S.A., Polígono Industrial Els<br />

Vinyets Els Fogars 2, Carretera Comarcal C-<br />

244 Km 22, 08777 Sant Quinti de Mediona-<br />

Barcelona, ES<br />

(72) RAFECAS JANE, Llorenç, Tarragona, ES<br />

RIERA ESCALE, Antoni, 08005 Barcelona, ES<br />

RAMON ALBALATE, Rosario, Barcelona, ES<br />

ALONSO XALMA, Monica, 08024 Barcelona,<br />

ES<br />

(74) Carvajal y Urquijo, Isabel, et al, Clarke, Modet<br />

& Co. Goya 11, 28001 Madrid, ES<br />

C07C 229/08 → (51) C07C 327/22<br />

C07C 2<strong>31</strong>/02 → (51) C07C 327/22<br />

(51) C07C 2<strong>31</strong>/12 (11) 2 213 654 A1<br />

C07C 233/65<br />

(25) En (26) En<br />

(21) 10002063.5 (22) 18.12.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(30) 21.12.2006 US 876394 P<br />

21.02.2007 US 902465 P<br />

(54) • Verfahren zur herstellung von 2-amino-5bromobenzamid<br />

derivaten<br />

• Process for preparing 2-amino-5-bromobenzamide<br />

derivatives<br />

• Procede de preparation de derives de 2amino-5-bromobenzamide<br />

(71) E. I. Du Pont de Nemours and Company,<br />

1007 Market Street, Wilmington, DE 19898,<br />

US<br />

(72) Bruening, Joerg, Wilmington 19803, US<br />

288<br />

Anmeldungen<br />

Applications<br />

Demandes (<strong>31</strong>/<strong>2010</strong>) 04.08.<strong>2010</strong><br />

(74) Beacham, Annabel Rose, Dehns St Bride's<br />

House 10 Salisbury Square, London EC4Y<br />

8JD, GB<br />

(62) 07867794.5 / 2 094 644<br />

C07C 2<strong>31</strong>/12 → (51) C07C 237/26<br />

C07C 2<strong>31</strong>/16 → (51) C07B 53/00<br />

C07C 2<strong>31</strong>/24 → (51) C07C 237/26<br />

C07C 233/05 → (51) C07C 327/22<br />

C07C 233/43 → (51) C07D 239/70<br />

C07C 233/65 → (51) C07C 2<strong>31</strong>/12<br />

(51) C07C 237/26 (11) 2 213 655 A1<br />

C07C 2<strong>31</strong>/12 C07C 2<strong>31</strong>/24<br />

A61K <strong>31</strong>/65<br />

(25) En (26) En<br />

(21) 10152023.7 (22) 28.04.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(30) 27.04.2007 US 926461<br />

(54) • Verfahren zur Reinigung von Aminoalkyl-<br />

Tetracyclinverbindungen<br />

• Methods For Purifying Aminoalkyl Tetracycline<br />

Compounds<br />

• Procédés de purification de composés<br />

d'aminoalkyle de tétracycline<br />

(71) Paratek Pharmaceuticals, Inc., 75 Kneeland<br />

Street, Boston, MA 02111, US<br />

(72) Johnston, Sean, Doylestown, PA 18902, US<br />

Warchol, Tedeusz, Northborough, MA<br />

01532, US<br />

(74) Nash, David Allan, Haseltine Lake LLP Redcliff<br />

Quay 120 Redcliff Street, Bristol BS1<br />

6HU, GB<br />

(62) 08754132.2 / 2 144 870<br />

(51) C07C 253/00 (11) 2 213 656 A1<br />

C07C 67/08 C07C 69/675<br />

C07C 255/16 C07C 255/36<br />

C07B 61/00<br />

(25) Ja (26) En<br />

(21) 08840797.8 (22) 21.10.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

AL BA MK RS<br />

(86) JP 2008/068998 21.10.2008<br />

(87) WO 2009/054356 2009/18 30.04.2009<br />

(30) 23.10.2007 JP 2007275696<br />

(54) • VERFAHREN ZUR HERSTELLUNG EINER<br />

CYANOHYDRINVERBINDUNG UND VER-<br />

FAHREN ZUR HERSTELLUNG EINER<br />

ALPHA-HYDROXYESTERVERBINDUNG<br />

• PROCESS FOR PRODUCTION OF CYANO-<br />

HYDRIN COMPOUND, AND PROCESS FOR<br />

PRODUCTION OF ALPHA-HYDROXYESTER<br />

COMPOUND<br />

• PROCÉDÉ DE FABRICATION D'UN COM-<br />

POSÉ DE CYANHYDRINE ET PROCÉDÉ DE<br />

FABRICATION D'UN COMPOSÉ ALPHA-<br />

HYDROXYESTER<br />

(71) Nippoh Chemicals Co., Ltd, 3-3-3, NIhonbashi-muromachi,<br />

Chuo-ku, Tokyo 103-0022,<br />

JP<br />

(72) FUJIWARA, Naoki, Chiba 298-0104, JP<br />

NAKAGAWA, Kazuya, Toyama 939-8046, JP<br />

KINOSHITA, Yuichiro, Chiba 298-0104, JP<br />

MIDORIKAWA, Koji, Chuo-ku, Tokyo103-<br />

0022, JP

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