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Bulletin 2010/31 - European Patent Office

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(C07D) II.1(1)<br />

• DÉRIVÉS DE PIPÉRIDINE ET D'AZÉTIDINE<br />

EN TANT QU'INHIBITEURS DE GLYT1<br />

(73) MERCK SHARP & DOHME LTD., Hertford<br />

Road, Hoddesdon, Hertfordshire EN11 9BU,<br />

GB<br />

(72) BLACKABY, Wesley Peter, Harlow Essex<br />

CM20 2QR, GB<br />

FLETCHER, Stephen Robert, Harlow Essex<br />

CM20 2QR, GB<br />

JENNINGS, Andrew, Harlow Essex CM20<br />

2QR, GB<br />

LEWIS, Richard Thomas, Harlow Essex<br />

CM20 2QR, GB<br />

NAYLOR, Elizabeth Mary, Harlow Essex<br />

CM20 2QR, GB<br />

STREET, Leslie Joseph, Harlow Essex CM20<br />

2QR, GB<br />

THOMSON, Joanne, Harlow Essex CM20<br />

2QR, GB<br />

(74) Horgan, James Michael Frederic, et al, Merck<br />

& Co., Inc. <strong>European</strong> <strong>Patent</strong> Department<br />

Hertford Road, Hoddesdon EN11 9BU, GB<br />

C07D 403/12 → (51) C07D 237/04<br />

C07D 403/12 → (51) C07D 243/14<br />

C07D 405/04 → (51) C07D 211/58<br />

C07D 405/06 → (51) C07D 211/58<br />

C07D 405/06 → (51) C07D 243/14<br />

C07D 405/12 → (51) C07D 243/14<br />

(51) C07D 413/04 (11) 2 160 391 B1<br />

(25) De (26) De<br />

(21) 08758799.4 (22) 28.05.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

(43) 10.03.<strong>2010</strong><br />

(86) EP 2008/004214 28.05.2008<br />

(87) WO 2008/155003 2008/52 24.12.2008<br />

(30) 19.06.2007 EP 07011966<br />

(54) • NICOTINAMID-DERIVATE ALS SYNTHE-<br />

SEBAUSTEINE ZUR HERSTELLUNG VON<br />

AGROCHEMISCHEN WIRKSTOFFEN UND<br />

VERFAHREN ZU DEREN HERSTELLUNG<br />

• NICOTINAMIDE DERIVATIVES AS SYNTH-<br />

ESIS UNITS FOR PRODUCING AGRO-<br />

CHEMICAL SUBSTANCES, AND METHOD<br />

FOR THE PRODUCTION THEREOF<br />

• DÉRIVÉS DE NICOTINAMIDE EN TANT<br />

QU'ÉLÉMENTS DE SYNTHÈSE PERMET-<br />

TANT LA PRODUCTION DE PRINCIPES<br />

ACTIFS AGROCHIMIQUES ET LEUR PRO-<br />

CÉDÉ DE PRÉPARATION<br />

(73) Bayer CropScience AG, Alfred-Nobel-Strasse<br />

50, 40789 Monheim, DE<br />

(72) PAZENOK, Sergii, 42699 Solingen, DE<br />

STELZER, Uwe, 51399 Burscheid, DE<br />

BLASCHKE, Harry, 42327 Wuppertal, DE<br />

NEEFF, Arnd, 51399 Burscheid, DE<br />

MULDER, Lubbertus, 58135 Hagen-Haspe,<br />

DE<br />

C07D 413/12 → (51) C07D 243/14<br />

(51) C07D 417/04 (11) 1 999 128 B1<br />

A61K <strong>31</strong>/4439 A61P 11/00<br />

(25) En (26) En<br />

(21) 07739373.4 (22) 15.03.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 10.12.2008<br />

(86) JP 2007/0559<strong>31</strong> 15.03.2007<br />

(87) WO 2007/119496 2007/43 25.10.2007<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

(30) 17.03.2006 JP 2006075307<br />

(54) • TETOMILAST-POLYMORPHE<br />

• TETOMILAST POLYMORPHS<br />

• POLYMORPHES DE TÉTOMILAST<br />

(73) OTSUKA PHARMACEUTICAL CO., LTD., 9,<br />

Kanda Tsukasamachi 2-chome, Chiyoda-ku<br />

Tokyo 101-8535, JP<br />

(72) AOKI, Satoshi, Tokushima-shi, Tokushima<br />

771-0182, JP<br />

NAKAYA, Kenji, Tokushima-shi, Tokushima<br />

771-0182, JP<br />

SOTA, Masahiro, Tokushima-shi, Tokushima<br />

771-0182, JP<br />

ISHIGAMI, Masashi, Kanzaki-gun, Saga 842-<br />

0197, JP<br />

(74) HOFFMANN EITLE, <strong>Patent</strong>- und Rechtsanwälte<br />

Arabellastrasse 4, 81925 München, DE<br />

(60) 10160007.0 / 2 206 711<br />

C07D 471/10 → (51) C07D 243/14<br />

C07D 487/04 → (51) C07D 249/08<br />

C07D 487/22 → (51) A61K <strong>31</strong>/409<br />

C07D 493/04 → (51) A61K <strong>31</strong>/03<br />

C07D 493/04 → (51) C07B 63/04<br />

(51) C07D 495/04 (11) 1 879 899 B1<br />

(25) En (26) En<br />

(21) 05818439.1 (22) 09.12.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 23.01.2008<br />

(86) GB 2005/004753 09.12.2005<br />

(87) WO 2006/061642 2006/24 15.06.2006<br />

(30) 09.12.2004 GB 0427005<br />

09.12.2004 US 634271 P<br />

(54) • THIENOPYRIDINDERIVATE ALS KALIUM-<br />

KANALINHIBITOREN<br />

• THIENOPYRIDINE DERIVATIVES AS<br />

POTASSIUM CHANNEL INHIBITORS<br />

• DERIVES DE THIENOPYRIDINE EN TANT<br />

QU'INHIBITEURS DE CANAUX POTASSI-<br />

QUES<br />

(73) Xention Limited, Iconix Park London Road,<br />

Pampisford Cambridge Cambridgeshire CB2<br />

4EF, GB<br />

(72) FORD, John, Huntingdon PE28 9BN, GB<br />

MADGE, David John, Ely, Cambridgeshire<br />

CB6 8XA, GB<br />

PALMER,Nicholas, John, Cambridge CB1<br />

3HJ, GB<br />

ATHERALL, John Frederick, Essex CB10 2LL,<br />

GB<br />

JOHN, Derek, Sawston CB2 4TA, GB<br />

(74) Hart, Deborah Mary, et al, Kilburn & Strode<br />

LLP 20 Red Lion Street, London WC1R 4PJ,<br />

GB<br />

C07D 495/10 → (51) C07D 207/09<br />

(51) C07F 7/08 (11) 1 513 850 B1<br />

(25) En (26) En<br />

(21) 03732572.7 (22) 27.05.2003<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PT RO SE SI SK<br />

TR<br />

(43) 16.03.2005<br />

(86) EP 2003/006268 27.05.2003<br />

(87) WO 2003/099828 2003/49 04.12.2003<br />

(30) 29.05.2002 GB 0212324<br />

(54) • SILIZIUMZUSAMMENSETZUNGEN<br />

• SILICON COMPOSITION<br />

• COMPOSITION DE SILICIUM<br />

(73) Dow Corning Corporation, Midland, Michigan<br />

48611, US<br />

607<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>31</strong>/<strong>2010</strong>) 04.08.<strong>2010</strong><br />

(72) DEMES, Hagen, 6<strong>31</strong>79 Obertshausen, DE<br />

FACKLER, Helmut, 89415 Lauingen, DE<br />

(74) Russell, Lindsey, et al, Elkington and Fife<br />

LLP Thavies Inn House 3-4 Holborn Circus,<br />

London EC1N 2HA, GB<br />

(51) C07F 9/09 (11) 1 045 853 B1<br />

C07F 9/12<br />

(25) En (26) En<br />

(21) 99902121.5 (22) 08.01.1999<br />

(84) AT BE CH DE DK ES FI FR GB GR IE IT LI LU<br />

NL PT SE<br />

(43) 25.10.2000<br />

(86) US 1999/000419 08.01.1999<br />

(87) WO 1999/035150 1999/28 15.07.1999<br />

(30) 09.01.1998 US 71070 P<br />

09.12.1998 US 1115<strong>31</strong> P<br />

(54) • SYNTHESE VON COMBRETASTATIN A-4<br />

PRODRUGS<br />

• SYNTHESIS OF COMBRETASTATIN A-4<br />

PRODRUGS<br />

• SYNTHESE DE PROMEDICAMENTS A<br />

BASE DE COMBRESTATINE A-4<br />

(73) ARIZONA BOARD OF REGENTS, A BODY<br />

CORPORATE OF THE STATE OF ARIZONA<br />

acting for and on behalf of ARIZONA STATE<br />

UNIVERSITY, Tempe, AZ 85287, US<br />

(72) PETTIT, George, R., Paradise Valley, AZ<br />

85253, US<br />

RHODES, Monte, R., Louisville, KY 40222,<br />

US<br />

(74) Didmon, Mark, Potter Clarkson LLP Park<br />

View House 58 The Ropewalk, Nottingham<br />

NG1 5DD, GB<br />

C07F 9/09 → (51) C07C 29/149<br />

C07F 9/12 → (51) C07F 9/09<br />

C07F 9/655 → (51) A61K <strong>31</strong>/03<br />

(51) C07F 17/02 (11) 1 844 061 B1<br />

C07B 53/00 C07B <strong>31</strong>/00<br />

(25) En (26) En<br />

(21) 06700701.3 (22) 13.01.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 17.10.2007<br />

(86) GB 2006/000114 13.01.2006<br />

(87) WO 2006/075166 2006/29 20.07.2006<br />

(30) 14.01.2005 GB 0500702<br />

(54) • AUF METALLOCEN BASIERENDE CHIRALE<br />

PHOSPHORPHOSPHINE<br />

• METALLOCENE-BASED PHOSPHORUS<br />

CHIRAL PHOSPHINES<br />

• PHOSPHINES CHIRALES DE PHOSPHORE<br />

À BASE DE MÉTALLOCÈNE<br />

(73) Solvias AG, Klybeckstrasse 191, 4057 Basel,<br />

CH<br />

(72) MCCORMACK, Peter, Phoenix Chemicals<br />

Ltd., Wirral, Merseyside CH62 3PW, GB<br />

CHEN, Weiping, Liverpool L16 3GD, GB<br />

WHITTALL, John, Hestbank, Lancaster, LA2<br />

6DF, GB<br />

(74) Maué, Paul Georg, et al, Solvias AG <strong>Patent</strong>s<br />

Erlenstrasse 1, 4058 Basel, CH<br />

(51) C07H 17/00 (11) 1 851 236 B1<br />

A61K <strong>31</strong>/7048 C07H 17/08<br />

A61P 29/00 A61K <strong>31</strong>/7052<br />

(25) En (26) En<br />

(21) 06727595.8 (22) 13.01.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

AL BA HR MK YU<br />

(43) 07.11.2007

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