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Bulletin 2010/31 - European Patent Office

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(C07C) II.1(1)<br />

AL BA HR MK RS<br />

(43) 02.07.2008<br />

(86) GB 2006/003697 05.10.2006<br />

(87) WO 2007/039741 2007/15 12.04.2007<br />

(30) 06.10.2005 GB 0520324<br />

09.12.2005 GB 0525082<br />

11.02.2006 GB 0602800<br />

(54) • BIPHENYLOXYESSIGSÄUREDERIVATE<br />

ZUR BEHANDLUNG VON ATEMWEGSER-<br />

KRANKUNGEN<br />

• BIPHENYLOXYACETIC ACID DERIVATIVES<br />

FOR THE TREATMENT OF RESPIRATORY<br />

DISEASE<br />

• DERIVES D'ACIDE BIPHENYLOXYACE-<br />

TIQUE UTILISES POUR LE TRAITEMENT<br />

DE MALADIES RESPIRATOIRES<br />

(73) AstraZeneca AB, 151 85 Södertälje, SE<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

(72) LUKER, Timothy, Jon, Leicestershire LE11<br />

5RH, GB<br />

MOHAMMED, Rukhsana, Tasneem, Leicestershire<br />

LE11 5RH, GB<br />

DICKINSON, Mark, Leicestershire LE11 5RH,<br />

GB<br />

THOM, Stephen, Leicestershire LE11 5RH,<br />

GB<br />

C07C 323/17 → (51) C07C <strong>31</strong>7/20<br />

C07C 323/20 → (51) C07C 59/70<br />

C07C 323/20 → (51) C07D 327/02<br />

(51) C07C 323/52 (11) 1 844 008 B1<br />

A61K <strong>31</strong>/22<br />

(25) En (26) En<br />

(21) 06706426.1 (22) 26.01.2006<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC NL PL PT RO<br />

SE SI SK TR<br />

(43) 17.10.2007<br />

(86) EP 2006/000680 26.01.2006<br />

(87) WO 2006/079535 2006/<strong>31</strong> 03.08.2006<br />

(30) 26.01.2005 EP 05001498<br />

(54) • KRISTALLINE VALNEMULINSALZE MIT<br />

ORGANISCHEN SÄUREN<br />

• VALNEMULIN CRYSTALLINE SALTS WITH<br />

ORGANIC ACIDS<br />

• SELS CRISTALLINS DE VALNEMULINE<br />

CONTENANT DES ACIDES ORGANIQUES<br />

(73) Novartis AG, Lichtstrasse 35, 4056 Basel, CH<br />

(72) MACHER, Ingolf, A-6300 Wörgl, AT<br />

GEISSLER, Annett, 79576 Weil am Rhein-<br />

Haltingen, DE<br />

WIELAND-BERGHAUSEN, Susanne, Christine,<br />

79541 Lörrach, DE<br />

SCHOTE, Uwe, Thomas, CH-4055 Basel, CH<br />

RAKOCZI, Ferenc, Jozsef, CH-4132 Muttenz,<br />

CH<br />

(74) Liphardt, Bernd, et al, Novartis Animal<br />

Health, Inc. <strong>Patent</strong> and Trademark Group<br />

Werk Rosenthal, 4002 Basel, CH<br />

C07C 333/08 → (51) C07D 233/32<br />

(51) C07D 207/09 (11) 2 039 682 B1<br />

C07D 209/42 C07D 209/52<br />

C07D 217/26 C07D 233/36<br />

C07D 271/08 A61K <strong>31</strong>/385<br />

A61K <strong>31</strong>/40 A61K <strong>31</strong>/403<br />

A61K <strong>31</strong>/404 A61K <strong>31</strong>/4245<br />

A61K <strong>31</strong>/472 C07D 495/10<br />

(25) Fr (26) Fr<br />

(21) 08290885.6 (22) 19.09.2008<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HR HU IE IS IT LI LT LU LV MC MT NL<br />

NO PL PT RO SE SI SK TR<br />

Europäisches <strong>Patent</strong>blatt<br />

<strong>European</strong> <strong>Patent</strong> <strong>Bulletin</strong><br />

<strong>Bulletin</strong> européen des brevets<br />

AL BA MK RS<br />

(43) 25.03.2009<br />

(30) 21.09.2007 FR 0706629<br />

(54) • Additionssalze von Hemmern des Angiotensin<br />

konvertierenden Enzyms mit NO<br />

abgebenden Säuren, Verfahren zu ihrer<br />

Herstellung und die sie enthaltenden<br />

pharmazeutischen Zusammensetzungen<br />

• Addition salts of inhibitors of the angiotensin-conversing<br />

enzyme with NO-donor<br />

acids, method for their preparation and<br />

pharmaceutical compositions containing<br />

them<br />

• Sels d'addition d'inhibiteurs d'enzyme de<br />

conversion de l'angiotensine avec des<br />

acides donneurs de NO, leur procédé de<br />

préparation et les compositions pharmaceutiques<br />

les contenant<br />

(73) Les Laboratoires Servier, 12, Place de La<br />

Défense, 92415 Courbevoie Cedex, FR<br />

(72) de Nanteuil, Guillaume, 92150 Suresnes, FR<br />

Portevin, Bernard, 45450 Fay Aux Loges, FR<br />

Gloanec, Philippe, 78160 Marly le Roi, FR<br />

Parmentier, Jean-Gilles, 92130 Issy Les<br />

Moulineaux, FR<br />

Benoist, Alain, 95130 Franconville, FR<br />

Verbeuren, Tony, 78540 Vernouillet, FR<br />

Rupin, Alain, 37510 Savonnieres, FR<br />

Courchay, Christine, 91430 Igny, FR<br />

Simonet, Serge, 78700 Conflans Sainte<br />

Honorine, FR<br />

(74) Giudicelli, Cathy, et al, Les Laboratoires<br />

Servier Direction Brevets 35, rue de Verdun,<br />

92284 Suresnes Cedex, FR<br />

C07D 209/42 → (51) C07D 207/09<br />

C07D 209/52 → (51) C07D 207/09<br />

(51) C07D 209/88 (11) 1 756 057 B1<br />

(25) En (26) En<br />

(21) 05744187.5 (22) 19.05.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

(43) 28.02.2007<br />

(86) GB 2005/001978 19.05.2005<br />

(87) WO 2005/113502 2005/48 01.12.2005<br />

(30) 20.05.2004 GB 0411273<br />

(54) • VERFAHREN ZUR HERSTELLUNG VON<br />

CARVEDILOL<br />

• PROCESS FOR THE PREPARATION OF<br />

CARVEDILOL<br />

• PROCESSUS POUR LA PRÉPARATION DE<br />

CARVÉDILOL<br />

(73) Cipla Ltd., 289, Belasis Road, Mumbai<br />

Central, Mumbai 400 008, IN<br />

(72) KANKAN, Rajendra Narayanrao, Mumbai<br />

400076, IN<br />

RAO, Dharmaraj Ramachandra, 4/403 Garden<br />

Enclave, Mumbai 400 601, Maharashtra,<br />

IN<br />

(74) Curtis, Philip Anthony, A.A. Thornton & Co.<br />

235 High Holborn, London WC1V 7LE, GB<br />

C07D 211/22 → (51) A61K <strong>31</strong>/445<br />

(51) C07D 211/58 (11) 2 029 540 B1<br />

C07D 405/04 C07D 405/06<br />

A61K <strong>31</strong>/445 A61K <strong>31</strong>/453<br />

(25) En (26) En<br />

(21) 07795529.2 (22) <strong>31</strong>.05.2007<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU LV MC MT NL PL PT<br />

RO SE SI SK TR<br />

(43) 04.03.2009<br />

(86) US 2007/012808 <strong>31</strong>.05.2007<br />

(87) WO 2007/145834 2007/51 21.12.2007<br />

(30) 08.06.2006 US 811759 P<br />

604<br />

<strong>Patent</strong>e<br />

<strong>Patent</strong>s<br />

Brevets (<strong>31</strong>/<strong>2010</strong>) 04.08.<strong>2010</strong><br />

(54) • BENZAMIDDERIVATE UND ASSOZIIERTE<br />

VERWENDUNGEN<br />

• BENZAMIDE DERIVATIVES AND USES<br />

RELATED THERETO<br />

• DÉRIVÉS DE BENZAMIDE ET UTILISA-<br />

TIONS ASSOCIÉES À CEUX-CI<br />

(73) Amgen Inc., One Amgen Center Drive,<br />

Thousand Oaks, CA 91320-1799, US<br />

(72) POWERS, Jay, P., Pacifica, CA 94044, US<br />

REW, Yosup, Foster City, CA 94404, US<br />

YAN, Xuelei, Foster City, CA 94404, US<br />

(74) Sexton, Jane Helen, J.A. Kemp & Co. 14<br />

South Square Gray's Inn, London WC1R 5JJ,<br />

GB<br />

C07D 213/79 → (51) A61K 33/24<br />

(51) C07D 217/24 (11) 1 667 976 B1<br />

C07D 401/04 C07D 401/06<br />

A61K <strong>31</strong>/472 A61K <strong>31</strong>/4725<br />

A61P 9/06<br />

(25) En (26) En<br />

(21) 04784368.5 (22) 17.09.2004<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IT LI LU MC NL PL PT RO SE SI SK<br />

TR<br />

LT LV<br />

(43) 14.06.2006<br />

(86) US 2004/030484 17.09.2004<br />

(87) WO 2005/030726 2005/14 07.04.2005<br />

(30) 23.09.2003 US 505215 P<br />

(54) • ISOCHINOLINON-KALIUMKANALINHIBI-<br />

TOREN<br />

• ISOQUINOLINONE POTASSIUM CHANNEL<br />

INHIBITORS<br />

• INHIBITEURS DU CANAL POTASSIQUE A<br />

BASE D'ISOQUINOLINONE<br />

(73) Merck Sharp & Dohme Corp., 126 East<br />

Lincoln Avenue, Rahway, NJ 07065, US<br />

(72) DINSMORE, Christopher, J., Rahway, New<br />

Jersey 07065-0907, US<br />

BERGMAN, Jeffrey, M., Rahway, New Jersey<br />

07065-0907, US<br />

MCINTYRE, Charles, J., Rahway, New Jersey<br />

07065-0907, US<br />

ISAACS, Richard, Rahway, New Jersey<br />

07065-0907, US<br />

CLAREMON, David, A., Rahway, New Jersey<br />

07065-0907, US<br />

(74) Man, Jocelyn, et al, Merck & Co., Inc.<br />

<strong>European</strong> <strong>Patent</strong> Department Merck Sharp &<br />

Dohme Limited, Hertford Road, Hoddesdon,<br />

Hertfordshire, EN11 9BU, GB<br />

C07D 217/26 → (51) C07D 207/09<br />

C07D 221/18 → (51) C07D 295/08<br />

(51) C07D 221/28 (11) 1 747 200 B1<br />

A61K <strong>31</strong>/485<br />

(25) En (26) En<br />

(21) 05739715.0 (22) 21.04.2005<br />

(84) AT BE BG CH CY CZ DE DK EE ES FI FR GB<br />

GR HU IE IS IT LI LT LU MC NL PL PT RO SE<br />

SI SK TR<br />

(43) <strong>31</strong>.01.2007<br />

(86) EP 2005/005239 21.04.2005<br />

(87) WO 2005/103009 2005/44 03.11.2005<br />

(30) 22.04.2004 EP 04291055<br />

(54) • ALKALOIDVERBINDUNGEN UND IHRE<br />

VERWENDUNG ALS ANTIMALARIAMITTEL<br />

• ALKALOID COMPOUNDS AND THEIR USE<br />

AS ANTI-MALARIAL DRUGS<br />

• COMPOSES ALCALOIDES ET LEUR UTILI-<br />

SATION COMME MEDICAMENTS ANTIPA-<br />

LUDIQUES

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